Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
03/2003
03/12/2003EP0787016B1 Secretory leukocyte protease inhibitor (slpi) as an inhibitor of tryptase
03/12/2003EP0672031B1 Catechol diethers as selective pde iv inhibitors
03/12/2003CN1402730A Thiazolo (4,5-D) pyrimidine compounds
03/12/2003CN1402716A Substd. oxazoles and thiazoles derivs. as HPPAR alpha activators
03/12/2003CN1401634A 4-guanidinobenzamides antifertility compounds
03/11/2003US6531612 Nitrile derivatives that inhibit cathepsin K
03/11/2003US6531610 Intermediate acylating carbonate
03/11/2003US6531604 Useful as medicines having an osteogenesis promoting effect and chondrogensis promoting effect.
03/11/2003US6531485 Prostaglandin agonists
03/11/2003US6531479 Anti-cancer compounds
03/11/2003US6531241 Anions of equal number to cations to maintain charge neutrality, are disclosed. These spacer groups may be organic or inorganic in origin and may vary in length. The spacer groups may be saturated, containing single bonds, or may have
03/10/2003CA2401358A1 Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
03/06/2003WO2003018571A1 M-aminophenol derivatives and colouring agents containing them
03/06/2003WO2003018553A1 Oral antidiabetic agents
03/06/2003WO2003018535A2 Novel aminobenzoephenones
03/06/2003WO2003018515A2 Prime ring substituted thyroid receptor antagonists for the treatment of cardiac and metabolic disorders
03/06/2003WO2003018135A1 Method of using 5-(arylsulfonyl)-,5-(arylsulfinyl), and 5-(arylsulfanyl)-thiazolidine-2,4-diones for inhibition of farnesyl-protein transferase
03/06/2003WO2003018011A1 5-(substituted)-5-(substitutedsulfonyl or sulfanyl)thiazolidine-2,4-diones useful for inhibition of farnesyl-protein transferase
03/06/2003WO2003018010A1 Preventive and/or remedial agent for disease attributable to arteriosclerotic activity
03/06/2003WO2003018008A1 Apo ai expression accelerating agent
03/06/2003WO2003017946A2 Non-oxidatively metabolized compounds and compositions, synthetic pathways therefor, and uses thereof
03/06/2003WO2003017764A1 Substituted propargylamines
03/06/2003WO2002100844A3 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
03/06/2003WO2002099097A8 Novel compounds for chemiluminescense procedures
03/06/2003WO2002094770A3 Aminoalcohol derivatives
03/06/2003US20030045755 Polyamine analogues as cytotoxic agents
03/06/2003US20030045581 4-substituted-1- (arylmethylidene) thiosemicarbazide, 4-substituted-1- (arylcarbonyl) thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof
03/06/2003US20030045558 Such as 2-(4-(2-(2-(4-(3,5-dimethyl-isoxazol-4-yl)-phenyl)-5-methyloxazol-4-yl) -ethyoxy)-phenoxy)-2-methylpropionic acid for treatment of diabetes (lowering serum triglycerides)
03/06/2003US20030045545 Immunomodulators, induce cytokine biosynthesis, and antineoplastic agents
03/06/2003CA2458681A1 M-aminophenol derivatives and colouring agents containing them
03/06/2003CA2458621A1 Oral antidiabetic agents
03/06/2003CA2457836A1 Preventive and/or remedial agent for disease attributable to arteriosclerotic activity
03/06/2003CA2457532A1 Non-oxidatively metabolized compounds and compositions, synthetic pathways therefor, and uses thereof
03/06/2003CA2449515A1 Prime ring substituted thyroid receptor antagonists for the treatment of cardiac and metabolic disorders
03/05/2003EP1288207A1 Process for the preparation of 4,5-dihydro-1,3-thiazoles
03/05/2003EP1287018A2 Thrombin inhibitors
03/05/2003EP1286978A1 Cyclohexyl derivatives and their use as therapeutic agents
03/05/2003EP1286976A1 Method for producing 2-chloro-5-chloromethyl-1,3-thiazole
03/05/2003EP1286975A1 Biclyclic cyclohexylamines and their use as nmda receptor antagonists
03/05/2003EP1286964A1 Heterocyclic inhibitors of glycogen synthase kinase gsk-3
03/05/2003EP1286673A2 Ligands of integrin receptors
03/05/2003EP1286670A2 Use of therapeutic benzamide derivatives
03/05/2003EP0939628B1 Thiol sulfone metalloprotease inhibitors
03/05/2003EP0853610B1 Synthesis and use of retinoid compounds having negative hormone and/or antagonist activities
03/05/2003CN1400899A Use of 2-methyl thiazolidin-2, 4-dicarboxylic acid and/or physiologically compatible salts thereof for producing a medicament for treating cancers
03/05/2003CN1102596C 5H-thiazole [3,2-a] pyrmidine derivatives
03/05/2003CN1102595C Penems and their derivatives
03/05/2003CN1102593C N-[4(heteroarylmethyl)phenyl]-heteroarylamines compound
03/05/2003CN1102583C Cationic polypeptide condensing agent of thiazole,its synthesizing process and its application
03/05/2003CN1102580C Arylethenesulfonamide derivatives and drug composition containing the same
03/04/2003US6528652 Composition and device for detecting leukocytes in urine
03/04/2003US6528651 Ring cleavage deamination of a triazacylclohexane derivative with hydrogen chloride
03/04/2003US6528543 Glucokinase activating for treating type II diabetes; acylurea compound, phenylacetyl-substituted; 1-(2-(3-chloro-phenyl)-3cyclopentyl-propionyl)-3-methyl-urea
03/04/2003US6528533 Treating or preventing neuronal damage associated with neurological diseases; hydrazide based compounds containing the group -N-N-CO-X- where X is C,O,S,or N
03/04/2003US6528528 Thiourea and benzamide compounds, compositions and methods of treating or preventing inflammatory diseases and atherosclerosis
03/04/2003US6528525 Amidocarboxylic acid derivatives
03/04/2003US6528510 HIV protease inhibitors
02/2003
02/28/2003CA2399927A1 Process for preparing 4,5-dihydro-1,3-thiazoles
02/27/2003WO2003016291A1 ACTIVATOR FOR PEROXISOME PROLIFERATOR-RESPONSIVE RECEPTOR δ
02/27/2003WO2003016288A1 Fxr nr1h4 nuclear receptor binding compounds
02/27/2003WO2003016280A1 Nr1h4 nuclear receptor binding compounds
02/27/2003WO2003016270A2 Selective estrogen receptor modulators
02/27/2003WO2003016266A1 β-KETOAMIDE COMPOUNDS AND MEDICINAL USE THEREOF
02/27/2003WO2003016265A1 Cyclic compound and ppar agonist
02/27/2003WO2003015778A1 Tyrosine kinase inhibitors
02/27/2003WO2003015777A1 Nr1h4 nuclear receptor binding compounds
02/27/2003WO2003015776A1 2,4,5-trisubstituted thiazolyl derivatives and their antiinflammatory activity
02/27/2003WO2003015775A1 New dipeptidyl peptidase iv inhibitors and their uses for lowering blood pressure levels
02/27/2003WO2003015774A1 Compounds effecting glucokinase
02/27/2003WO2003015773A2 2-amino-4,5-trisubstituted thiazolyl derivatives and their use against autoimmune diseases
02/27/2003WO2003015772A1 Inhibitors of polyq-aggregation
02/27/2003WO2003015717A2 Tyrosine kinase inhibitors
02/27/2003WO2002096884A3 Substituted benzoylketones as herbicidal agents for use as plant treatment agent
02/27/2003WO2002089749A3 Arylsulfonamide ethers, and methods of use thereof
02/27/2003WO2002060374A3 Benz-1,3-azole derivatives and their uses as heparanase inhibitors
02/27/2003US20030040533 For use as hypoglycaemic and hypolipidaemic agents
02/27/2003US20030040525 Inhibition of human telomerase by a G-quadruplex-interaction compound
02/27/2003CA2456868A1 Inhibitors of polyq-aggregation
02/27/2003CA2423025A1 New dipeptidyl peptidase iv inhibitors and their uses for lowering blood pressure levels
02/26/2003EP1285914A1 Nr1h4 nuclear receptor binding compounds
02/26/2003EP1285911A2 Arylsulfonanilide ureas
02/26/2003EP1284730A1 Aralkyl ester soft drugs
02/26/2003EP0885187B1 Diphenylethers, process and intermediate products for their preparation, and their use
02/26/2003EP0832068B1 Stable reagents for the preparation of radiopharmaceuticals
02/25/2003US6525220 Intermediates for the synthesis of benzimidazole derivatives and a process for the preparation thereof
02/25/2003US6525211 Herbicidal sulphonylamino(thio)carbonyl compounds
02/25/2003US6525099 N-substituted sulfonamide derivatives
02/25/2003US6525080 Thiazoline acid derivatives
02/25/2003US6525042 Sulfonyl derivatives
02/25/2003US6525036 Compounds and compositions as protease inhibitors
02/20/2003WO2003014096A1 Process of production of n-alkyl-2-benzthiazolylsulfeneimides, device for their production and method of their purification
02/20/2003WO2003014095A1 Acylaminothiazole derivatives, their preparation and therapeutic use
02/20/2003WO2003014072A1 Disulfide and thiosulfonate ligands and libraries comprising these ligands
02/20/2003WO2003013520A1 Pramipexole for the treatment of adhd
02/20/2003WO2003013519A1 Pramipexol as an anticonvulsive agent
02/20/2003WO2003013484A2 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents
02/20/2003WO2002096516A8 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
02/20/2003WO2002024635A3 Aminoalcohol derivatives
02/20/2003US20030036558 Useful in the treatment of chronic complications arising from diabetes, such as neuropathy; may also contain an angiotensin converting enzyme inhibitor.
02/20/2003US20030036532 Treatment of infections caused by parasites, especially malaria.