Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
04/2002
04/24/2002CN1083447C Process for preparation of benzothiazolone compounds
04/24/2002CN1083446C Process for preparing 2-chlorothiazole compounds
04/24/2002CN1083432C Process for preparing amine compound and its salt
04/23/2002US6376671 2-sulfamoylbenzoic acid derivatives
04/23/2002US6376538 Antiinflammatory agents; autoimmune diseases
04/23/2002US6376502 Osteoporosis compounds
04/23/2002US6376495 Antidiabetic piperazine derivatives, processes for their preparation and compositions containing them
04/23/2002US6376494 Cycloalkyl-substituted aryl-piperazines, piperidines and tetrahydropyridines as serotonergic agents
04/23/2002US6376492 Compounds and methods for inhibition of HIV and related viruses
04/23/2002US6376428 Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production
04/18/2002WO2002030875A1 Beta-amino acid derivatives as integrin receptor antagonists
04/18/2002WO2002030358A2 Modulation of ccr4 function
04/18/2002WO2002030357A2 Compounds and methods for modulating ccr4 function
04/18/2002WO2002030356A2 Synthesis of epothilones and relates analogs
04/18/2002WO2002012210A9 Biphenyl derivatives and their use as ppar-gamma receptor activators
04/18/2002WO2002012166A3 Triamine derivative melanocortin receptor ligands and methods of using same
04/18/2002WO2001087830A3 Substituted thioacetamides
04/18/2002WO2001062709A3 Use of 2-phenylene diamine derivatives for the treatment of infections
04/18/2002WO2001026656A3 5-membered heterocycle derivatives and use thereof as monoamine oxidase inhibitors
04/18/2002US20020045753 E.g., (S)-N-(4-(4-((3,4-dihydro-6-hydroxy-2,5,7,8-tetramethyl-2H-1-benzopyran-2 -yl)-carbonyl)-1-piperazinyl)phenyl)-2-thiophenecarboximidamide , or a salt thereof.
04/18/2002US20020045654 Sulfonylbenzene compounds as anti-inflammatory/analgesic agents
04/18/2002US20020045641 Multiple heteroatom containing heterocyclic ring compounds substituted with carboxylic acids and isosteres thereof
04/18/2002US20020045629 Sleep, eating and brain disorders, wakefulness promoters; Parkinson's disease, antiischemic agents, stroke, chronic fatigue syndrome; antidepressants; schizophrenia, nervous system disorders; multiple sclerosis, cognition activators
04/18/2002US20020045620 Readily metabolized by the metabolic drug detoxification systems; metabolized by serum or intracellular hydrolases and esterases; shorthalf-life; noninsulin-dependent diabetes mellitus (NIDDM) (Type II); side effect reduction
04/18/2002US20020045615 Benzothiazole derivatives with activity as adenosine receptor ligands
04/18/2002US20020045065 Novel organometallic luminescent materials and organic electroluminescent device containing same
04/18/2002US20020045064 Metal sulfonates of metal complexes of hydroxy- and mercapto-quinolines, benzoxazoles, benzothiazoles, benzotriazoles, benzoselenazoles, benzotellurazoles and phenanthridines
04/18/2002US20020045063 Metal sulfonates of metal complexes of hydroxy- and mercapto-quinolines, benzoxazoles, benzothiazoles, benzotriazoles, benzoselenazoles, benzotellurazoles and phenanthridines
04/18/2002DE10122447A1 Biphenylcarboxamide Biphenylcarboxamides
04/18/2002DE10051136A1 New alpha-hydroxy-ketone derivatives, useful as intermediates for biologically active polyketides, terpenoids, epothilones and their derivatives
04/18/2002DE10046934A1 Verfahren zur fermentativen Herstellung von nicht-proteinogenen L-Aminosäuren A process for the fermentative production of non-proteinogenic L-amino acids
04/18/2002CA2425828A1 Synthesis of epothilones and related analogs
04/18/2002CA2425259A1 Modulation of ccr4 function
04/18/2002CA2424951A1 Beta-amino acid derivatives as integrin receptor antagonists
04/17/2002EP1197211A1 Preventive and therapeutic agents for cancer
04/17/2002EP1196402A1 Method for producing 4-cyano-2-aminomethylthiazol
04/17/2002EP1196401A1 Method for producing 2-aminomethyl-4-cyano-thiazol
04/17/2002EP1196400A1 Amino-alkyl derivatives
04/17/2002EP1196397A1 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
04/17/2002EP1196388A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
04/17/2002EP1196387A1 Azo amino acid derivatives for the treatment of neurological diseases
04/17/2002EP1196384A1 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
04/17/2002EP1196371A1 Quaternary bis-ammonium salt precursors and their uses as prodrugs having an antiparasitic activity
04/17/2002EP0934290B1 Aminothiazole derivatives, method of preparation and pharmaceutical compositions containing same
04/17/2002EP0871362B1 Synergistic insecticide mixtures
04/17/2002CN1345308A Acetylenic alpha-amino acid based sulfonamide hydroxamic acid TACE inhibitors
04/17/2002CN1344801A Method for production of non-proteinogen L-amino acid by fermentation
04/17/2002CN1082958C Alternate crystal form of tazofelone
04/17/2002CN1082957C New L-2-ketothiazolidine-4-carboxylic derivatives and use for treating skin
04/17/2002CN1082956C Micacocidin derivatives
04/17/2002CN1082945C Alkoxiyimino acetamide
04/16/2002US6372913 Process for preparing 2-substituted 5-formylthiazoles
04/16/2002US6372912 Process for ring cleavage of thiazolidine derivatives
04/16/2002US6372778 Sulfonamide inhibitors of aspartyl protease
04/16/2002US6372769 Applying fungicides to rice
04/16/2002US6372750 Heterocyclic compounds, process for their preparation and pharmaceutical compounds containing them and their use in the treatment of diabetes and related diseases
04/16/2002US6372742 Telomerase enzyme inhibitors and anticancer agents
04/11/2002WO2002028841A2 Reagents for labeling biomolecules having aldehyde or ketone moieties
04/11/2002WO2002028835A1 Benzamide compounds as apo b secretion inhibitors
04/11/2002WO2002028829A2 Peptide deformylase inhibitors
04/11/2002WO2002028827A1 5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation
04/11/2002WO2002028820A1 Nitroso diphenylamine derivatives
04/11/2002WO2002028815A1 Pharmaceutical compounds
04/11/2002WO2002028810A2 Retinoids for the treatment of emphysema
04/11/2002WO2002028434A2 Use of a ppar delta activator for treating inflammatory conditions
04/11/2002WO2002028433A2 Use of a ppar delta activator in the treatment of diseases related to no inhibit ion or tnf inhibition
04/11/2002WO2001094317A3 Method for synthesis of substituted azole libraries
04/11/2002WO2000012493A9 Thiazoline acid derivatives
04/11/2002US20020042520 Method for synthesis of substituted azole libraries
04/11/2002US20020042519 By selective reduction of the exocyclic double bond in a benzylidene thiazolidine-2,4-dione moiety by complex hydride reducing agents such as lithium tri-sec-butyl borohydride
04/11/2002US20020042512 Alpha-acyl- and alpha-heteroatom-substituted benzene acetamide glucokinase activators
04/11/2002US20020042511 New derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
04/11/2002US20020042434 Pharmaceutical composition
04/11/2002US20020042109 Enzymatically degrading certain epothilone compounds to form ring-open structures containing a carboxyl which is esterified, the hydroxyl groups on the moiety protected and the resulting compound oxidized by, e.g. ozone,
04/11/2002US20020042085 Produce light energy when decomposed; stable at room temperature
04/11/2002CA2425097A1 Benzamide compounds as apo b secretion inhibitors
04/11/2002CA2424684A1 Nitroso diphenylamine derivatives
04/11/2002CA2424300A1 Reagents for labeling biomolecules having aldehyde or ketone moieties
04/11/2002CA2419777A1 Pharmaceutical compounds
04/10/2002EP1195375A1 Benzamide derivatives, insecticides for agricultural and horticultural use and usage thereof
04/10/2002EP1194421A1 Selective npy (y5) antagonists
04/10/2002EP1194147A1 Arylthiazolidinedione and aryloxazolidinedione derivatives
04/10/2002EP1194146A1 Arylthiazolidinedione and aryloxazolidinedione derivatives
04/10/2002CN1344263A Polycyclic 2-aimino-thiazole systems, method for prodn. thereof and medicament contg. said compounds
04/10/2002CN1344247A Multicyclic compounds which inhibit beukocyte adhesion mediated by VLA-4
04/10/2002CN1344160A Heterocyclic aromatic compounds useful as growth hormone secretagogues
04/10/2002CN1082508C antivirally active heterocyclic azahexane derivatives
04/09/2002USRE37650 Aryl and heteroaryl quinazoline compounds which inhibit CSF-1R receptor tyrosine kinase
04/09/2002US6369234 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
04/09/2002US6369233 Multistage reaction to form halosubstituted thiazoles with chlorination
04/09/2002US6369232 Antidiabetic agents
04/09/2002US6369071 Treatment of angina pectoris
04/09/2002US6369042 Radical-scavenging functions which counteract pathophysiological disorders especially connected with aging processes; also antidotes against organophosphorous compounds; vitamin b6 antagonists; wound healing promoters
04/04/2002WO2002026737A1 Novel polymorphic forms of 5-[4-[2-[n-methyl-n-(2-pyridyl)amino]ethoxy]benzyl] thiazolidine-2,4-dione maleate and process for their preparation
04/04/2002WO2002004407A3 7-substituted tetracycline compounds
04/04/2002WO2001094301A3 Factor viia inhibitory (thio)urea derivatives, their preparation and their use
04/04/2002WO2001090717A3 Linker arms for nanocrystals and compounds thereof
04/04/2002WO2001090716A3 Linker arms for nanocrystals and compounds thereof
04/04/2002WO2001047898A3 Substituted piperazine derivatives and their use as inhibitors of the microsomal triglyceride transfer protein (mtp)
04/04/2002US20020040157 3-amino-2-mercaptobenzoic acid derivatives and processes for their preparation