Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
05/2002
05/09/2002US20020055526 Modulators of SKCa, IKCa and BKCa channels.
05/09/2002US20020055525 Aminosulfonyl- or alkylsulfonylphenyl-heterocyclylalkylhydroxyamic acid or hydroxyurea derivatives; treating asthma and arthritis
05/09/2002US20020055522 Treatment of thrombotic diseases, asthma, emphysema, cirrhosis, arthritis, carcinoma, melanoma, restenois, atheroma, trauma, shock and reperfusion injury.
05/09/2002US20020055181 Light generating compound for use in the detection of preferential particles in sample
05/08/2002EP1203767A1 Heterocyclic-substituted alkylamide acat inhibitors
05/08/2002EP1202990A2 Neurotrophic pyrrolidines and piperidines, and related compositions containing them
05/08/2002EP1202981A1 Substituted heteroaryloxyacetanilides and their use as herbicides
05/08/2002EP1202980A1 2-arylimino-2,3-dihydrothiazoles, and their use thereof as somatostatin receptor ligands
05/08/2002EP1202979A1 Process for the preparation of thiazole derivatives
05/08/2002EP1202968A2 Antibacterial agents
05/08/2002EP1202731A2 Method for treating chronic pain using mek inhibitors
05/08/2002EP1202718A2 Substituted guanidines for the treatment of cancer and pain
05/08/2002EP1202626A1 Alpha-hydroxy-gamma-[[(carbocyclic-or heterocyclic-substituted)amino]carbonyl]alkanamide derivatives and uses thereof
05/08/2002CN1348446A Heterocyclic carboxamide-containing thiourea inhibitors of herpes viruses containing phenylenediamine group
05/08/2002CN1348370A Cyclic protein tyrosine kinase inhibitors
05/08/2002CN1347693A Noval compound, its synthetizing process and therapeutic use
05/08/2002CN1084330C Cydic amide derivatives
05/08/2002CA2361226A1 Process for the production of dithiazolyl disulfides
05/07/2002US6384230 2,6-dimethyl-5-((4-ethoxyphenyl)-methoxy)-7-(2-methylthiazol-4-yl)hepta -2,6-dienoic acid ethyl ester from malic acid, wittig reaction with 2-methyl-4-thiazolylmethyl triphenyl phosphonium bromide; intermediates for epothilone a or b
05/07/2002US6384220 Antidiabetic agents increasing the expression of glucokinase (gk) to improve glucose tolerance; increase in glucose exposure coupled through gk in beta-cells to increase insulin secretion and in hepatocytes to increase glycogen deposition
05/07/2002US6384075 Treating diseases in which mast cell dysfunction is involved
05/07/2002US6384065 Spiro compounds or salts thereof and preventives/remedies for autoimmune diseases and AP-1 inhibitors containing the same
05/07/2002US6384062 Pharmaceutical composition
05/07/2002US6384056 Cognition activators and nerve and vision disorders
05/07/2002US6384036 Bis-sulfonamide hydroxyethylamino retroviral protease inhibitors
05/07/2002US6384035 Heterocycles useful in the treatment of benign prostatic hyperplasia
05/07/2002CA2052263C Herbicides
05/02/2002WO2002034734A1 Process for the manufacture of thiazole derivatives with pesticidal activity
05/02/2002WO2002034711A1 Biaryl compounds as serine protease inhibitors
05/02/2002WO2002034265A1 Use of 2-hydrazino-1,3-thiazoles as antioxidants
05/02/2002WO2002034243A2 Method for the treatment of neurological and neuropsychological disorders
05/02/2002WO2002034242A2 Method for the treatment of neurological and neuropsychological disorders
05/02/2002WO2001090074A3 BENZOPHENONES AS INHIBITORS OF IL-1β AND TNF-$g(a)
05/02/2002WO2001081298A3 Cyclic carboxylic acids as integrin antagonists
05/02/2002WO2001024828A3 MODULATORS OF CYTOKINE MEDIATED SIGNALLING PATHWAYS AND INTEGRIN αVβ3 RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY
05/02/2002US20020052512 Diaminopropionic acid derivatives
05/02/2002US20020052417 Factor VIIa inhibitory (thio)urea derivatives, their preparation and their use
05/02/2002US20020052401 Benzophenones and sulfones as inhibitors of glycine uptake
05/02/2002US20020052399 In particular as inhibitors of HIV protease.
05/02/2002US20020052392 Have utility as, inter alia, hypoglycemic, and anti-obesity agents.
05/02/2002US20020052378 Novel compounds and compositions as protease inhibitors
05/02/2002US20020052349 p-(sulfonyl) aryl and heteroarylamines as anti-inflammatory agents
05/02/2002US20020052007 Diarylmethylbenzylpiperazines and corresponding halobenzyl derivatives
05/02/2002EP1201666A2 Epothilones with a modified side chain
05/02/2002EP1201662A1 Preparation of thiazoles
05/02/2002EP1201650A2 Ionic malonitril derivatives and their uses
05/02/2002EP1201648A1 Carbamate derivatives and agricultural/horticultural bactericides
05/02/2002EP1200420A1 Process for making n-alkyl bis(thiazolyl)sulfenimides
05/02/2002EP1200419A1 Aminothiazole derivatives and their use as crf receptor ligands
05/02/2002EP1200418A1 Nematicidal trifluorobutenes
05/02/2002EP1200411A2 Novel process for synthesis of heteroaryl-substituted urea compounds
05/02/2002EP1200398A1 3-arylsulfonyl-2-(substituted methyl)propanoic acid derivates as matrix metalloproteinase inhibitors
05/02/2002EP1200395A1 Urea derivatives as inhibitors of ccr-3 receptor
05/02/2002EP1146875A4 Myt1 kinase inhibitors
05/02/2002DE10052590A1 Verwendung von 2-Hydrazino-1,3-thiazolen als Antioxidantien Use of 2-hydrazino-1,3-thiazoles as antioxidants
05/02/2002CA2689012A1 Method for the treatment of neurological and neuropsychological disorders
05/02/2002CA2426430A1 Biaryl compounds as serine protease inhibitors
05/02/2002CA2424475A1 Method for the treatment of neurological and neuropsychological disorders
05/01/2002CN1083715C Use of insulin sensitisers for treating renal diseases
04/2002
04/30/2002US6380395 Anticancer agents
04/30/2002US6380258 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
04/30/2002US6380255 Treatment for dermal skin atrophy using thyroid hormone compounds or thyroid hormone-like compounds
04/30/2002US6380235 Useful as progesterone receptor agonists and antagonists, used for contraception, in therapy of fibroids, endometriosis, breast, uterine, ovarian and prostate cancer, and post menopausal hormone replacement therapy
04/30/2002US6380230 For therapy of dyskinesia, obesity, irritable bowel syndrome, diseases whose treatment requires stimulation of the cholecystokinin cck-a receptors
04/30/2002US6380229 Useful for therapy and prophylaxis of hyperlipidemia and related complications
04/30/2002US6380223 For therapy of diseases, such as obesity, diabetes, inflammation
04/30/2002US6380213 Compounds useful as neuro-protective agents
04/30/2002US6380191 Arylthiazolidinedione and aryloxazolidinedione derivatives
04/30/2002US6380190 Nonnucleoside inhibitors of reverse transcriptase, composite binding pocket and methods for use thererof
04/30/2002US6380188 For inhibiting human immunodeficiency virus protease
04/30/2002US6380187 Fungicides
04/30/2002US6380186 Psychotherapeutic agents
04/25/2002WO2002032897A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
04/25/2002WO2002032889A1 Aromatic and heterocyclic thiazolyl thiourea compounds and use
04/25/2002WO2002032886A1 A process for the preparation of bis-benzazolyl compounds
04/25/2002WO2002032883A1 Novel 4-benzyloxyphenyl derivative and use thereof
04/25/2002WO2002032872A1 Nitrogenous aromatic ring compounds
04/25/2002WO2002032844A2 Epothilone synthesis components iii and iv: asymmetrically substituted acyloins and acyloin derivatives, method for the production thereof and method for the production of epithilone b, d and epothilone derivatives
04/25/2002WO2001097810A3 Use of therapeutic benzamide derivatives
04/25/2002WO2001058891A3 Piperazine and piperidine derivatives for treatment or prevention of neuronal damage
04/25/2002US20020049344 New vitamin d derivatives with carbo-or heterocyclic substituents at c-25, a process for their production, intermediate products and their use for producing medicaments
04/25/2002US20020049316 Protease inhibitors
04/25/2002US20020049241 Conformationally rigid bicyclic and adamantane derivatives useful as alpha2-adrenergic blocking agents
04/25/2002US20020049240 Novel compounds
04/25/2002US20020049239 Novel indole and benzothiazole derivatives
04/25/2002US20020049236 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
04/25/2002US20020049228 2-Sulfamoylbenzoic acid derivatives
04/25/2002US20020049215 Pyrazole-thiazole compounds, pharmaceutical compositions containing them, and methods of their use for inhibiting cyclin-dependent kinases
04/25/2002US20020049214 Aralkyl and aralkylidene heterocyclic lactams and imides as selective agonists and antagonists of serotonin 1 (5-HT1) recepor, used in treating hypertension and all forms of depression
04/25/2002US20020049211 Combination treatment for depression and anxiety
04/25/2002US20020049210 Heteroaryl amines as novel acetylcholinesterase inhibitors
04/25/2002US20020049201 Sulfonamide inhibitors of aspartyl protease
04/25/2002US20020049165 Inhibiting the enzymatic activity of HIV protease
04/25/2002CA2426148A1 Aromatic and heterocyclic thiazolyl thiourea compounds and use
04/25/2002CA2423792A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
04/25/2002CA2324194A1 Novel antifungal agents
04/24/2002EP1199306A1 Biarylurea derivatives
04/24/2002EP1198451A2 Substituted phenoxyacetic acids
04/24/2002EP0830353B1 Process for the preparation of an hiv protease inhibiting compound
04/24/2002CN1083450C Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides