Patents
Patents for C07D 277 - Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings (33,621)
01/2003
01/09/2003WO2003002546A1 Supported condensation reactants and method for the production thereof
01/09/2003WO2003002540A1 Cyclic diamine compound having five-membered cyclic group
01/09/2003WO2003002532A1 Cyclic diamine compounds having fused-ring groups
01/09/2003WO2003002531A2 Fluoropyrrolidines as dipeptidyl peptidase inhibitors
01/09/2003WO2003002530A2 Pyrrolidines as dipeptidyl peptidase inhibitors
01/09/2003WO2003002519A1 Phenol derivatives and their use in medicaments
01/09/2003WO2003001913A1 Thiazines and thiazoles for use as material protective agents
01/09/2003US20030009033 Substituted condensation products of N-benzyl-3-indenylacent amides with heterocyclic aldehydes for neoplasia
01/09/2003US20030008996 Utilized for image forming materials, for example, stereolithography, holography, lithographic printing plate precursors, color proofs, photoresists and color filters, and photosetting resin materials such as ink, paint, adhesive
01/09/2003US20030008915 Acylated 6,7,8,9-tetrahydro-5H-benzocycloheptenyl amines and their use as pharmaceutical agents
01/09/2003US20030008907 Intermediates for the synthesis of benzimidazole derivatives and a process for the preparation thereof
01/09/2003US20030008906 Administering benzothiazole compound for therapy, prophylaxis of disease
01/09/2003US20030008905 Increasing the capacity of insulin providing cells in an animal by administering to animal a dose of at least one Dipeptidyl-peptidase (DP IV) enzyme activity effector
01/09/2003US20030008895 Prostaglandin agonists
01/09/2003US20030008884 Fungicidal phenyl (thio) urea and phenyl (thio) carbamate derivatives
01/09/2003US20030008829 For therapy and prophylaxis of inflammatory diseases associated with the respiratory tract, such as asthma and allergic rhinitis, immunomediated inflammatory disorders, such as rheumatoid arthritis, conjunctivitis, psoriasis
01/09/2003US20030008234 Optical data carrier comprising a cyanine dye as light-absorbent compound in the information layer
01/09/2003US20030007941 Method of treating hair loss using thyromimetic compounds
01/09/2003CA2450722A1 Fluoropyrrolidines as dipeptidyl peptidase inhibitors
01/09/2003CA2424645A1 New use of dipeptidyl peptidase iv inhibitors
01/09/2003CA2418543A1 New dipeptidyl peptidase iv inhibitors and their uses as anti-cancer agents
01/08/2003EP1273572A1 Thiophene substituted piperazines useful in the treatment of benign prostatic hyperplasia
01/08/2003EP1273298A2 Ritonavir in combination with an additional HIV protease inhibitor for treating aids
01/08/2003EP1272469A1 Naphthalene derivatives and their pharmaceutical use
01/08/2003EP1272459A1 7- and 9-carbamate, urea, thiourea, thiocarbamate, and heteroaryl-amino substituted tetracycline compounds
01/08/2003EP1272456A1 Hydrazide and alkoxyamide angiogenesis inhibitors
01/08/2003EP1124819B1 Method of lithiating five-membered heterocycles
01/08/2003EP1123284B1 Method for the preparation of citalopram
01/08/2003EP1121364B1 Method for producing epothilone b and derivatives thereof
01/08/2003EP0996439B1 Beta-alkoxyacrylates against malaria
01/08/2003EP0988296B1 Naphthothiazolone derivatives active on the d 3 dopaminergic receptor
01/08/2003EP0889033B1 Alpha-substituted benzyl heterocyclic derivatives, intermediates for producing the same, and pesticides containing the same as active ingredient
01/08/2003EP0833839B1 Peptidyl heterocycles useful in the treatment of thrombin related disorders
01/08/2003CN1390206A Inhibitors of factor Xa
01/08/2003CN1390204A Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/08/2003CN1390196A Novel derivatives of dicarboxylic acid having pharmaceutical properties
01/08/2003CN1390193A Novel dicarboxylic acid derivatives with pharmaceutical properties
01/08/2003CN1389458A P-methylsulfonyl phenylacrylate derivative and its prepn process and anti-inflammatory effect
01/08/2003CN1389203A Method for treating hair-dropping using thyromimetic compound
01/07/2003US6504031 Enzyme inhibitor such as 6-(2-(1-isopropyl-1,2,3,4-tetrahydro -7-isoquinolinyl)ethenyl)-2-naphthalenecarboximidamide, used as angiogenesis inhibitors; antiarthritic, antiinflammatory and antitumor agents
01/07/2003US6503949 Glucagon antagonists/inverse agonists
01/07/2003US6503935 Imidazoles and related compounds as α1A agonists
01/07/2003US6503929 Nitrate salt of anti-ulcer medicine
01/07/2003US6503725 Composition and device for detecting leukocytes in urine
01/07/2003CA2143208C Sulfonamide inhibitors of hiv-aspartyl protease
01/03/2003WO2003000668A1 Oxa(thia)zolidine compounds, process for preparation thereof and anti-inflammatory agents
01/03/2003WO2003000262A1 Vinyl phenyl derivatives as glk activators
01/03/2003WO2003000260A1 Thiazolyl amides and their use as antiviral drugs
01/03/2003WO2003000259A1 Topical application of thiazolyl amides
01/03/2003WO2003000247A1 Carbamates of 2-heterocyclic-1,2-ethanediols
01/03/2003WO2003000180A2 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/03/2003WO2002083656A3 5-membered heterocycles, preparation and use thereof as mao inhibitors and lipid peroxidation inhibitors, preparation thereof and use thereof as medicaments
01/03/2003WO2002064577A3 Method for preparing compounds derived from thiazolidinedione, oxazolidinedione
01/03/2003CA2451543A1 Thiazolyl amides and their use as antiviral drugs
01/03/2003CA2450579A1 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/02/2003US20030004339 Therapy for benign prostatic hyperplasia
01/02/2003US20030004212 Cyclohexylamine derivatives as subtype selective N-Methyl-D-Aspartate antagonists
01/02/2003US20030004196 Antiinflamamtory agents; autoimmune disease
01/02/2003US20030004181 Disubstituted bicyclic heterocycles, the preparation thereof, and their use as pharmaceutical compositions
01/02/2003US20030004138 Hypoglycemic agents; antidiabetic agents; dietetics
01/02/2003US20030004136 IL-8 receptor ligands-drugs for inflammatory and autoimmune diseases
01/02/2003US20030003396 Reflection, protective or covering layers which can be written on or read by blue, red or infrared light
01/02/2003EP1270562A2 Cyclic alpha-amino-gamma-hydroxy-amides, process for their preparation and pharmaceutical compositions thereof
01/02/2003EP1268443A1 2-hydroxy-mutilin carbamate derivatives for antibacterial use
01/02/2003EP1268430A1 Chemical complex compprising a pyridine carboxy derivative and an h2 histamine receptor antagonist
01/02/2003EP1268429A1 Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same
01/02/2003EP1268412A1 Sulphonamido-substituted bridged bicycloalkyl derivatives
01/02/2003EP1268401A1 Process for the selective n-formylation of n-hydroxylamines
01/02/2003EP1268096A1 Extrusion die
01/02/2003EP1073654A4 2,3-olefinic epothilone derivatives
01/02/2003EP1073648A4 12,13-modified epothilone derivatives
01/02/2003EP1073647A4 12,13-cyclopropane epothilone derivatives
01/02/2003EP0751939B9 Naphthylamides as central nervous system agents
01/01/2003CN1387849A Use of thiazolidinedione for preventing or retaining non-insulin-dependent diabets mellitus (NIDDM) attack
01/01/2003CN1387848A Use of thiazolidinedione for preventing or retaining non-insulin-dependent diabets mellitus (NIDDM) attack
12/2002
12/31/2002US6500832 Administering enzyme inhibitors as viricides for prophylaxis of viral diseases such as aquired immune deficiency syndrome
12/31/2002US6500817 Thiazolyl urea derivatives and their utilization as antiviral agents
12/31/2002US6500812 Gastrointestinal disorders; antiinflammatory agents
12/31/2002US6500804 Administering a dipeptidyl aminopeptidase effector which is selected from the group consisting of n-(n-substituted glycyl)2-cyanopyrrolidones, n-aminoacyl thiazolidines, n-aminoacyl pyrrolidines
12/31/2002US6500803 Factor VIIa inhibitors
12/26/2002US20020198243 Cyclizing the tert-butyl-thiourea derivative to form the end product
12/26/2002US20020198242 Administering to an animal an effective dose of atleast an enzyme Dipeptidyl Peptidase (DP IV) enzyme activity effector to increase the capacity of insulin producing cells
12/26/2002US20020198241 Inhibiting bacterial growth in humans and nonhuman mammals by administering to the patient an antibacterially effective dose of hydroxamic acid derivatives containing carbamoyl groups
12/26/2002US20020198207 Novel Hexanoic acid derivatives
12/26/2002US20020198200 Alpha-acyl- and alpha-heteroatom-substituted benzene acetamide glucokinase activators
12/26/2002US20020198184 Matrix metalloproteinase inhibitor is useful as an anticancer agent, angiogenesis inhibitor, a tumor cell infiltration inhibitor or a tumor metastasis inhibitor; inflammatory diseases, osteoarthritis, rheumatoid arthritis
12/26/2002US20020195930 Organic electroluminescent materials
12/25/2002CN1387519A 2-imino-1,3-thiazine derivs.
12/25/2002CN1387518A Heterocyclic substd, diphenyl leukotriene antagonists
12/25/2002CN1097049C Processes for preparing intermediate product used in method of diastereoselective synthesis of nucleosides
12/24/2002US6498275 Use of compounds for the elevation of pyruvate dehydrogenase activity
12/24/2002US6498265 3-amino-2-mercaptobenzoic acid derivatives and processes for their preparation
12/24/2002US6498257 2,3-olefinic epothilone derivatives
12/24/2002US6498190 Bicyclic amino derivatives and PGD2 antagonist containing the same
12/24/2002US6498177 Alpha 2 adrenergic receptor agonist; analgesic, sedative and anaesthetic agents
12/24/2002US6498174 Agonists to peroxisome proliferator-activated receptors; modulating blood glucose and lipid levels; reducing dyslipidemia and hyperinsulinemia associated with impaired glucose tolerance or metabolic syndrome
12/24/2002US6498172 Prostaglandin agonists and their use to treat bone disorders
12/24/2002US6498004 Silver halide light sensitive emulsion layer having enhanced photographic sensitivity
12/24/2002CA2150812C Catechol diethers as selective pde iv inhibitors
12/19/2002WO2002100977A1 Organic electroluminescence device and luminance material