Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
07/2003
07/29/2003US6599943 Preventive treatment, related to the radical generating nature of the xanthine dehydrogenase/xanthine oxidase
07/29/2003CA2114136C Gallium (iii) complexes, process for their obtention and pharmaceutical compositions containing them
07/24/2003WO2003059888A1 4,5-diaminopyrazole derivatives in dimeric form and their use in oxidation dyeing of keratinous fibers
07/24/2003WO2003059887A1 Substituted pyrazolines for use as pesticides
07/24/2003WO2003059886A1 Acyl sulfonamide derivative
07/24/2003WO2003059346A1 Beta-secretase inhibitors
07/24/2003WO2003059265A2 Compositions and methods for treating heart failure
07/24/2003US20030139463 Anticancer agents; antiarthritic agents
07/24/2003US20030139407 Efficient synthesis of 5-heteroatom-containing -pyrazoles
07/24/2003US20030139405 6-Membered heterocyclic compounds useful for selective inhibition of the coagulation cascade
07/24/2003US20030139404 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents
07/24/2003US20030139402 Antiinflammatory agents; Alzheimer's disease; cardiovascular disorders
07/24/2003CA2473441A1 Beta-secretase inhibitors
07/23/2003EP1329160A2 4-acylaminopyrazole derivatives
07/23/2003EP0984688B1 Fungicidal mixtures
07/23/2003EP0888278B1 Antidiabetic agents
07/23/2003CN1432002A Process for prepn. of pesticidal compounds
07/23/2003CN1431941A 挤压模 Extrusion die
07/22/2003US6596873 2-and 2,5-substituted phenylketoenols
07/22/2003US6596863 Matrix metalloproteinase inhibitor is useful as an anticancer agent, angiogenesis inhibitor, a tumor cell infiltration inhibitor or a tumor metastasis inhibitor; inflammatory diseases, osteoarthritis, rheumatoid arthritis
07/22/2003US6596772 Relates to trifluoromethyl sulfonyl and trifluoromethyl sulfonamido compounds and the physiologically acceptable salts and the prodrugs thereof. These compounds are expected to modulate the activity of protein tyrosine enzymes which are
07/22/2003US6596746 Cyclic protein tyrosine kinase inhibitors
07/22/2003US6596741 Compounds of formula I exhibit activity as serotonin, norepinephrine, and dopamine reuptake inhibitors and can be used in the treatment of central nervous system and other disorders.
07/17/2003WO2003057674A1 4-sulfide / sulfoxide / sulfonyl-1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
07/17/2003WO2003057673A1 1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
07/17/2003WO2003057225A2 Phosphate transport inhibitors
07/17/2003WO2003057213A2 Cyclohexano- and cycloheptapyrazole derivative compounds, for use in diseases associated with the 5-ht2c receptor
07/17/2003US20030135057 5-amino- and 5-thio- substituted; prepared from a methylenedithietane intermediate
07/17/2003US20030134888 Substituted diaminopyrazoles; treating diseases, such as cancer, inflammatory disorders, restenosis, and cardiovascular disease. coatings for implantable medical devices, such as prostheses, artificial valves, etc.
07/17/2003US20030134859 Substituted 2-chloro-5-nitrobenzamides; treating retrograde osteoporosis and diabetes mellitus
07/17/2003CA2471885A1 4-sulfide / sulfoxide / sulfonyl-1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
07/17/2003CA2471880A1 1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
07/16/2003EP1326861A1 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists
07/16/2003EP1326843A1 Pyrazole derivatives for the treatment of viral diseases
07/16/2003EP1326831A1 Substituted fused pyrroleimines and pyrazoleimines
07/16/2003EP1326827A2 Insecticidal 1,8-naphthalenedicarboxamides
07/16/2003EP1261587B1 Stilbene derivatives, their preparation and their use as antiviral agents
07/16/2003CN1430602A Ary-and heteroaryl sulfonates compounds
07/16/2003CN1429816A New method of preparing Granisetron intermediate
07/15/2003USRE38188 Ethylene derivatives and pesticides containing said derivatives
07/15/2003US6593477 Synthesis of 3-acylaminopyrazoles
07/15/2003US6593357 Treating disease states in mammals that are alleviated by a protein kinase inhibitor, particularly diseases such as cancer, inflammatory disorders, restenosis, and cardiovascular disease.
07/15/2003US6593356 The present invention relates to the synthesis of a new class of indeno(1,2-c)pyrazol-4-ones of formula (I): that are potent inhibitors of the class of enzymes known as cyclin dependent kinases, which relate to the catalytic subunits cdk1-7 and the
07/14/2003WO2003059878A2 Thieno (3, 2-b) pyridones as antiviral compounds
07/14/2003CA2472960A1 Thieno (3, 2-b) pyridones as antiviral compounds
07/10/2003WO2003055860A1 3,4-diarylpyrazoles and their use in the therapy of cancer
07/10/2003WO2003055848A2 Urea derivatives as vr1- antagonists
07/10/2003WO2003055484A1 Urea derivatives
07/10/2003WO2001096297A3 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
07/10/2003US20030130542 Chlorination of an aniline in a hydrofluoric medium
07/10/2003US20030130309 Antiinflammatory agents; rheumatic diseases
07/10/2003US20030130232 Amidine derivatives, the preparation and use thereof as medicaments with LTB4 antagonistic effect
07/10/2003US20030127129 Charge transfer material, and photoelectric conversion device and photoelectric cell using same, and pyridine compound
07/10/2003CA2471236A1 Urea derivatives
07/10/2003CA2469967A1 Urea derivatives as vr1- antagonists
07/09/2003EP1325671A1 Organometallic compounds and emission-shifting organic electrophosphorescence
07/09/2003EP1324987A1 Indazoles with thyroid hormon like activity, a process for its preparation and its use in pharmaceutical compositions
07/09/2003EP1324986A1 Nitrogen-containing compounds and their use as glycine transport inhibitors
07/09/2003EP1324970A2 Retinoids for the treatment of emphysema
07/09/2003EP1235810B1 Process of making substituted pyrazoles
07/09/2003EP0966490B1 Catalyst compositions for the polymerization of olefins
07/09/2003EP0960100B1 Substituted 4-benzoyl-pyrazoles
07/09/2003EP0871426B1 Agent and method for dyeing keratin fibres
07/09/2003CN1429210A Substituted thioacetamides
07/09/2003CN1429199A Insecticidal 1,8-naphthalenedicarboxamides
07/09/2003CN1113895C Growth hormone secretagogues
07/09/2003CN1113875C Substituted aromatic thiocarboxylic acid amides and their use as herbicides
07/08/2003US6589974 Pyrazolyl benzyl ether derivatives containing a fluoromethoxyimino group and use thereof as pesticides
07/08/2003US6589970 6-(aryl-amido or aryl-amidomethyl)-naphthalen-2-yloxy-acidic derivatives as inhibitors of plasminogen activator inhibitor type-1 (PAI-1)
07/08/2003US6589914 Dihalopropene compounds, insecticidal/acaridcidal agents containing same, and intermediates for their production
07/08/2003CA2272640C Guanidinyl heterocycle compounds useful as alpha-2 adrenoceptor agonists
07/03/2003WO2003054237A1 4-(alpha branched)acyl- (3h)-pyrazol-3-ones for use in the extraction of metals, especially copper, from solution
07/03/2003WO2003053937A1 Novel substituted pyrazole derivative, process for producing the same, and herbicidal composition containing the same
07/03/2003WO2003053927A1 Piperazine derivative
07/03/2003WO2003053917A1 Guanidine compounds and pest controllers
07/03/2003WO2003053912A1 α-(N-SULPHONAMIDO)ACETAMIDE DERIVATIVES AS β-AMYLOID INHIBITORS
07/03/2003WO2003053895A2 Copper deposition using copper formate complexes
07/03/2003WO2003053885A1 Method for forming a carbon-carbon or carbon-heteroatom linkage
07/03/2003WO2003053435A1 Broadspectrum heterocyclic substituted phenyl containing sulfonamide hiv protease inhibitors
07/03/2003WO2003053368A2 Chalcone derivatives and their use to treat diseases
07/03/2003WO2003053358A2 Fused heterocyclic compounds and analogs thereof: modulators of nuclear hormone receptor function
07/03/2003US20030125361 1H-benzo(g)indazole compounds as anticarcinogenic agents and also treat arthritis
07/03/2003US20030125354 Aromatic compounds containing urea or thiourea groups are useful for terating cytokine mediated diseases
07/03/2003US20030125325 Fungicides
07/03/2003US20030125324 Alpha 4 beta 1 integrin and CD49d/ CD29 (vla-4); antiinflammatory agents
07/03/2003CA2470964A1 Broadspectrum heterocyclic substituted phenyl containing sulfonamide hiv protease inhibitors
07/03/2003CA2470931A1 Chalcone derivatives and their use to treat diseases
07/03/2003CA2470808A1 Piperazine derivative
07/03/2003CA2470141A1 Method for forming a carbon-carbon or carbon-heteroatom linkage
07/02/2003EP1322674A2 Control agents for living-type free radical polymerization, methods of polymerizing, emulsions and polymers with same
07/02/2003EP1322654A1 Platinum complexes as antitumor agents
07/02/2003EP1322598A1 Nitroso diphenylamine derivatives
07/02/2003EP1322309A2 High affinity small molecule c5a receptor modulators
07/02/2003EP0913392B1 Ethylene derivatives and pest controlling agents
07/02/2003CN1427859A Dimethyl pyrazole-blocked isocyanate mixtures
07/02/2003CN1112923C Indazole carboxamides
07/01/2003US6586603 Forming 4-(5-(4-chlorophenyl)-3-trifluoromethyl)-1H-pyrazol-1 -yl)benzenesulfonamide used as antiinflammatory agents; side effect reduction
07/01/2003CA2256227C Method of treating psychiatric conditions
06/2003
06/26/2003WO2003051906A2 Compounds and methods
06/26/2003WO2003051847A1 (1-h-indazol-3-yl) -amide derivatives as gsk-3 inhibitors