Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550) |
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04/29/2003 | US6555711 Reacting an N-allylimino nitrobenzene compound with a diamino-dinucleophile to form an alpha-amino-N- allylamidino-nitrobenzene compound; chemical intermediate for a pyrazolo(1,5-b)(1,2,4)triazole color photographic coupler |
04/29/2003 | US6555539 For treating cancer and other disease states associated with unwanted angiogenesis and/or cellular proliferation such as diabetic retinopathy, neovascular glaucoma, rheumatoid arthritis, psoriasis |
04/29/2003 | US6555339 Altering human G protein-coupled receptors (GPCRs) by point mutation; use in drug screening |
04/29/2003 | US6554871 Oxidative hair dye precursor compositions containing 4-5-diaminopyrazole, 5-amino-2-methylphenol and m-phenylenediamine compounds and method of dyeing hair |
04/29/2003 | CA2269721C 1-phenylpyrazole compounds and medicinal application thereof |
04/24/2003 | WO2003033499A2 Inhibitors of cyclin-dependent kinases, compositions and uses related thereto |
04/24/2003 | WO2003033484A1 Substituted piperazine cyclohexane carboxilic acid amides and the use thereof |
04/24/2003 | WO2003032972A1 5’-carbamoyl-1,1-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors |
04/24/2003 | WO2003016282A3 Substituted 1h-dihydropyrazoles, their preparation and use |
04/24/2003 | WO2002102376A8 ORALLY DELIVERABLE PHARMACEUTICAL COMPOSITION COMPRISING AN ACTIVE COMPOUND HAVING AN AMINOSULFONYL GROUP (cox-2 INHIBITOR), A POLYETHYLENE GLYCOL AND A FREE-RADICAL SCAVENGING ANTIOXIDANT |
04/24/2003 | WO2002058690A3 Methods for the treatment of diseases using malonyl-coa decarbox ylase inhibitors |
04/24/2003 | US20030078431 Biheterocyclic compounds having high anticoagulant activity, used as inhibitors of factor Xa |
04/24/2003 | US20030078287 For controlling plant and animal pests |
04/24/2003 | US20030078266 Powder of 30-90% a water-soluble cycloxygenase inhibitor, 5-60% of a buffer and 0-10% of other excipients |
04/24/2003 | US20030078261 Prostaglandin agonists |
04/24/2003 | CA2463571A1 Inhibitors of cyclin-dependent kinases, compositions and uses related thereto |
04/24/2003 | CA2463426A1 Substituted piperazine cyclohexane carboxilic acid amides and the use thereof |
04/23/2003 | EP1304325A1 5-(m-cyanobenzylamino)pyrazole derivatives |
04/23/2003 | EP1304110A2 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors |
04/23/2003 | EP1303509A1 Beta3 adrenergic agonists |
04/23/2003 | EP1303493A1 Method for the production of n,n'-carbonyldiazoles and azolide salts |
04/23/2003 | EP1303483A1 Novel thiourea derivatives and the pharmaceutical compositions containing the same |
04/23/2003 | EP1303308A2 Aldosterone antagonist and cyclooxygenase-2 inhibitor combination therapy to prevent or treat inflammation-related cardiovascular disorders |
04/23/2003 | EP1303271A1 Ophthalmic formulation of a selective cyclooxygenase-2 inhibitory drug |
04/23/2003 | EP0980236B1 Colourant and method for producing temporary hair colours |
04/23/2003 | EP0915846B1 2- and 2,5-substituted phenylketoenols |
04/23/2003 | EP0854723B1 Substituted pyrazolyl benzenesulfonamides for use in veterinary therapies as antiinflammatory agents |
04/23/2003 | CN1413207A 5-membered ring heterocyclic compounds with nitrogen |
04/23/2003 | CN1106399C Process for preparing sildenafil |
04/23/2003 | CN1106386C Parasiticidal pyrazole compound |
04/23/2003 | CN1106385C Substituted 4-benzoyl-pyrazoles |
04/22/2003 | US6552062 For therapy of central nervous system disorders; damage to the central nervous system; cardiovascular disorders; gastrointestinal disorders; diabetes insipidus, and sleep apnea, and obesity |
04/22/2003 | US6552018 As antitumor agents |
04/22/2003 | US6552008 Administering effective amount of a selected azo-pyrazole derivative for therapy of thrombocytopenia |
04/17/2003 | WO2003031437A1 Propylcarbamate derivatives as inhibitors of serine and cysteine proteases |
04/17/2003 | WO2003031435A1 Pyrazole derivatives as glycine transporter inhibitors |
04/17/2003 | WO2003031418A1 3,4-dihydro-1h-naphthalene derivatives as a highly selective cyclooxygenase-2 inhibitor |
04/17/2003 | WO2003013484A3 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents |
04/17/2003 | WO2003006454A3 Heterocyclic carboxamides and their use as fungicides |
04/17/2003 | WO2003005999A3 Methods of treating cytokine mediated diseases |
04/17/2003 | US20030073853 Cationic aminoanthraquinones, their use for dyeing keratinous fibers, dyeing compositions containing them and methods of dyeing |
04/17/2003 | US20030073849 Cyclopropylindole derivatives as selective serotonin reuptake inhibitors |
04/17/2003 | US20030073847 Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production |
04/17/2003 | US20030073836 Heteroarylcarboxylic acid amides, the preparation thereof and their use as pharmaceutical compositions |
04/17/2003 | US20030073832 Novel aminophenyl ketone derivatives |
04/17/2003 | US20030073722 Pyrazole substituted hydroxamic acid derivatives as cyclooxygenase-2 and 5-lipoxygenase inhibitors |
04/17/2003 | US20030073712 Antiinflamamtory agents; antiischemic agents |
04/17/2003 | US20030073686 Anticarcinogenic agents |
04/16/2003 | EP1301829A1 Radiation sensitive compositions containing image quality and profile enhancement additives |
04/16/2003 | EP1301787A2 Method for detecting uracil biosynthesis inhibitors and their use as herbicides |
04/16/2003 | EP1301464A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments |
04/16/2003 | EP1086682B1 Utilization of aryl(or heteroaryl)azolylcarbinol derivatives in the preparation of a medicament for the treatment of neurogenic inflammation |
04/16/2003 | CN1411448A Pyrazole derivatives which modulate human 5-serotonin receptors |
04/16/2003 | CN1411447A Polymorphic crystalline forms of celecoxib |
04/16/2003 | CN1105709C 3-thiocarbamoylpyrazole derivatives as pesticides |
04/16/2003 | CN1105708C 1-Phenylpyrazole compounds and medicinal application thereof |
04/16/2003 | CN1105707C Pyrazole derivative |
04/15/2003 | US6548547 Sulfonylamino carboxylic acid N-arylamides as guanylate cyclase activators |
04/15/2003 | US6548529 Heterocyclic containing biphenyl aP2 inhibitors and method |
04/15/2003 | US6548525 Nitrogen containing heteroaromatics with ortho-substituted P1's as factor Xa inhibitors |
04/15/2003 | US6548512 Nitrogen containing heteroaromatics as factor Xa inhibitors |
04/15/2003 | CA2290843C Cationic aminoanthraquinones, their use in the dyeing of keratin fibres, dyeing compositions containing them and dyeing processes |
04/10/2003 | WO2003029226A1 Heterocyclyl substituted phenoxyalkyl-, phenylthioalkyl-, phenylaminoalkyl- and phenylalkyl-sulfamoylcarboxamides |
04/10/2003 | WO2003029224A1 6-membered unsaturated heterocyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | WO2003029223A1 Substituted n-(1,4,5,6-tetrahydrocyclopentapyrazol-3-yl) derivatives and the use of the same for the treatment of cancer |
04/10/2003 | WO2003029222A1 Insecticidal and acaricidal 3-substituted pyrazoles |
04/10/2003 | WO2003029218A1 Novel nitrogenous compound and use thereof |
04/10/2003 | WO2003029216A1 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | WO2003029211A1 Difluoroalkene derivative, pest control agent containing the same, and intermediate therefor |
04/10/2003 | WO2003028729A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | WO2003028720A1 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them |
04/10/2003 | WO2002071827A3 Retinoid x receptor modulators |
04/10/2003 | US20030069422 Process for preparation of pyrazolo[4,3-d]pyrimidin-7-ones and intermediates thereof |
04/10/2003 | US20030069292 Central nervous system disorders; anticonvulsants |
04/10/2003 | US20030069287 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors |
04/10/2003 | US20030069284 Anticancer agent |
04/10/2003 | US20030069267 Modulators of protein tyrosine phosphatases (PTPases) |
04/10/2003 | US20030069258 Novel guanidine mimics factor Xa inhibitors |
04/10/2003 | US20030069242 3-arylphenyl sulfide derivative and insecticide and miticide |
04/10/2003 | US20030069241 Analgesics; central nervous system disorders; gastrointestinal disorder; therapy for drug abruse ; antiinflammatory agents |
04/10/2003 | US20030069240 Skin disorders; food allergies |
04/10/2003 | US20030069222 Used as anti-viral agents against the HIV-1 and HIV-2 viruses. |
04/10/2003 | US20030066988 Electroconductivity coloring |
04/10/2003 | CA2462647A1 6-membered unsaturated heterocyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | CA2462601A1 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | CA2462305A1 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade |
04/10/2003 | CA2460906A1 Insecticidal and acaricidal 3-substituted pyrazoles |
04/09/2003 | EP1299389A1 A process for preparing pyrazolopyrimidinone derivatives for the treatment of impotence |
04/09/2003 | EP1299361A1 Pyrazole derivatives |
04/09/2003 | EP1299123A2 Use of cox-2 inhibitors in the treatment and prevention of ocular cox-2 mediated disorders |
04/09/2003 | EP0829474B1 Indazole derivatives having monocyclic amino group |
04/08/2003 | US6545161 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them |
04/08/2003 | US6545054 Alkenyl and alkynyl compounds as inhibitors of factor Xa |
04/08/2003 | US6545033 GABA receptor inhibitors |
04/08/2003 | US6545031 Carboxyalkenylpyrazolylbenzene derivatives, such as (E)-alpha-((5-(2-((2-carboxyphenyl)methoxy)-4-methoxyphenyl) -1-ethyl-1H-pyrazol-4-yl)methylene)-6-methoxy-1,3-benzodioxole -5-propanoic acid |
04/08/2003 | US6545030 1-heterocycle substituted diarylamines |
04/08/2003 | CA2123548C Piperazine derivatives |
04/03/2003 | WO2003027075A2 Substituted pyrazolyl benzenesulfamide compounds for the treatment of inflammation |
04/03/2003 | WO2003027074A1 Pyrazole derivatives useful in the treatment of hyper-proliferative disorders |
04/03/2003 | WO2003027068A2 Substituted amines for the treatment of neurological disorders |