Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
12/2002
12/27/2002CA2449212A1 Alkylidene pyrazolidinedione derivatives and use for treating diabetes and obesity
12/27/2002CA2444356A1 Orally deliverable pharmaceutical composition comprising an active compound having an aminosulfonyl group (cox-2 inhibitor), a polyethylene glycol and a free-radical scavenging antioxidant
12/26/2002US20020198184 Matrix metalloproteinase inhibitor is useful as an anticancer agent, angiogenesis inhibitor, a tumor cell infiltration inhibitor or a tumor metastasis inhibitor; inflammatory diseases, osteoarthritis, rheumatoid arthritis
12/25/2002CN1387531A Pyrazolo [4,3-d] pyrimidine derivs.
12/25/2002CN1387518A Heterocyclic substd, diphenyl leukotriene antagonists
12/25/2002CN1097054C Tricyclic pyrazole derivs. and composition
12/25/2002CN1097049C Processes for preparing intermediate product used in method of diastereoselective synthesis of nucleosides
12/24/2002US6498275 Use of compounds for the elevation of pyruvate dehydrogenase activity
12/24/2002US6498172 Prostaglandin agonists and their use to treat bone disorders
12/19/2002WO2002100853A1 Pyrazole derivatives as hiv reverse transcriptase inhibitors
12/19/2002WO2002100846A1 Compounds and methods for the treatment or prevention of flavivirus infections
12/19/2002WO2002100845A1 Hv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
12/19/2002WO2002100844A2 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
12/19/2002WO2002100833A1 Rho KINASE INHIBITORS
12/19/2002WO2002100822A1 Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ii diabetes
12/19/2002WO2002100821A1 3,3-dialkoxy-2-hydroxyiminopropionitriles, process for preparation thereof and process of preparing 5-amino -4-nitrosopyrazoles or salts thereof by the use of the same
12/19/2002WO2002100403A1 Modulators of peroxisome proliferator activated receptors (ppar)
12/19/2002WO2002088091A3 Inhibitors of human rhinovirus 2a cysteine protease
12/19/2002WO2002083651A3 Pyrimidine compounds as anti-ictogenic and/or anti-epileptogenic agents
12/19/2002WO2002070541A3 Peptide deformylase inhibitors
12/19/2002WO2002059080A3 Trisubstituted carbocyclic cyclophilin binding compounds and their use
12/19/2002WO2002042248A3 Naphthalene derivatives
12/19/2002US20020193610 Indazoles
12/19/2002US20020193411 Pesticidal 1-polyarylpyrazoles
12/19/2002US20020193368 Use of potassium channel openers for the treatment of insulitis
12/19/2002DE10121003A1 Anthranilsäureamide, Verfahren zur Herstellung, ihrer Verwendung als Medikament sowie sie enthaltende pharmazeutische Zubereitungen Anthranilic acid amides, processes for preparing, their use as a medicament as well as pharmaceutical compositions containing them
12/19/2002CA2450269A1 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
12/19/2002CA2450265A1 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
12/19/2002CA2448552A1 Modulators of peroxisome proliferator activated receptors (ppar)
12/19/2002CA2445653A1 Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ii diabetes
12/18/2002EP1267369A2 Pyridine compound, its use as charge transfer material, and photoelectrochemical cell
12/18/2002EP1265850A2 Insecticidal anthranilamides
12/18/2002EP0934300B1 The preparation and use of ortho-sulfonamido heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
12/18/2002CN1096449C Process for producing substituted aryl pyrazoles
12/17/2002US6495699 Antiarthritic agents; osteoporosis
12/17/2002US6495492 Substituted 3-aryl-pyrazoles
12/12/2002WO2002098893A1 Glucopyranosyloxypyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate therefor
12/12/2002WO2002098862A1 Methods of making indazoles
12/12/2002WO2002098861A1 Methods of making 1-(2-aminopropyl)-6-hydroxyindazole
12/12/2002WO2002098860A1 Novel fused indazoles and indoles and their use for the treatment of glaucoma
12/12/2002WO2002098849A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer’s disease and similar diseases
12/12/2002WO2002098420A1 4-substituted-1-(arylmethylidene)thiosemicarbazide, 4-substituted-1-(arylcarbonyl)thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof
12/12/2002WO2002081398A3 Additives for building industry obtained from by-products and process for their production
12/12/2002WO2002004424A9 Pyrazole derivatives
12/12/2002US20020188136 Pesticides and herbicides
12/12/2002US20020188120 Such as 4-(4-methyoxy-benzenesulfonyl)-1-(3-phenyl-propyl)-piperidine-4-carboxylic acid hydroxyamide for treatment of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone diseases, diabetes, and HIV
12/12/2002US20020188017 Thienylazolylalkoxyethanamines, their preparation and their application as medicaments
12/12/2002US20020188007 Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
12/12/2002CA2448834A1 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases
12/12/2002CA2447482A1 Methods of making indazoles
12/12/2002CA2447156A1 Novel fused indazoles and indoles and their use for the treatment of glaucoma
12/11/2002EP1264823A1 Process for the preparation of 2,3-dicyanopropionates
12/11/2002EP1263743A1 Heterocycle substituted diphenyl leukotriene antagonists
12/11/2002EP1263734A1 3-thiomethylpyrazoles as pesticides
12/11/2002EP1263712A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
12/11/2002EP1100805B1 Medicine nitrate salts
12/11/2002EP0722446B1 Distamycin a analogues as antitumour or antiviral agents
12/11/2002EP0624155B2 Carbamates and plant-protecting agents containing them
12/11/2002CN1384829A Sodium-hydrogen exchanger type 1 inhibitor crystals
12/11/2002CN1384818A Novel compounds having cyano and insecticides and miticides
12/11/2002CN1384741A Selective COX-2 inhibitory novel esters from indolealkanols and novel amides from indolealkylamines
12/10/2002USRE37936 Pesticidal 1-polyarylpyrazoles
12/10/2002US6492529 Bis pyrazole-1H-pyrazole intermediates and their synthesis
12/10/2002US6492411 Substituted pyrazolyl benzenesulfonamides for the treatment of inflammation
12/10/2002US6492401 Sodium hydrogen exchanger type 1 inhibitors; reducing perioperative myocardial tissue damage
12/10/2002US6492396 Substituted thioacetamides
12/10/2002US6492393 Compounds useful as anti-inflammatory agents
12/10/2002US6492372 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4
12/10/2002US6492368 Benzamidine derivatives as factor XA inhibitors
12/10/2002CA2260412C Parasiticidal pyrazoles
12/10/2002CA2252344C Improved methods of preparing 4-cyano-4-(substituted indazole)cyclohexane-carboxylic acids useful as pde4 inhibitors
12/10/2002CA2208792C Substituted indazole derivatives
12/09/2002WO2002004403A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments
12/09/2002CA2412116A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments
12/05/2002WO2002096882A1 Substituted anilide derivatives, intermediates thereof, agricultural and horticultural chemicals, and their usage
12/05/2002WO2002096516A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
12/05/2002WO2002011707A3 Drugs for incontinence
12/05/2002US20020183519 Antithrombotic carboxylic acid amides
12/05/2002US20020183367 2,1-Oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase IV and method
12/05/2002US20020183362 2-Fluorobenzenesulfonyl compounds for the treatment of inflammation
12/05/2002US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm
12/05/2002US20020183334 For therapy of sleepiness, promotion of wakefulness, treatment of Parkinson's disease, cerebral ischemia, stroke, sleep apneas, eating disorders, stimulation of appetite and weight gain, treatment of attention deficit hyperactivity disorder
12/05/2002CA2447657A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
12/04/2002EP1261630A2 Bacterial genes and proteins that are essential for cell viability and their uses
12/04/2002EP1261587A1 Stilbene derivatives, their preparation and their use as antiviral agents
12/04/2002EP1261336A2 Il-8 receptor antagonists
12/04/2002EP1261321A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof
12/04/2002CN1383425A Uracil substituted phenyl sulfamoyl carboxamides
12/03/2002US6489452 An azo dye represented by the following general formula (1) and a process for making the azo dye is disclosed. the process comprises a step in which a diazonium salt is formed by the reaction between an aminopyrazole and aromatic coupling agent
12/03/2002US6489365 Ltb4-antagonistic compounds for treatment of inflammation, allergy or gastropathy induced by non-steroidal antiinflammatory agents in a warm-blooded animals
12/03/2002US6488734 Nitrification inhibitors, and the use of polyacids which contain a nitrification inhibitor for the treatment of inorganic fertilizers
12/03/2002CA2065644C Pyrazolopyridine compound and processes for preparation thereof
11/2002
11/28/2002WO2002094793A1 Acylated 4-aminopyrazoles
11/28/2002WO2002094792A1 Herbicidal substituted benzoylpyrazoles
11/28/2002WO2002094791A1 Diamide invertebrate pest control agents containing a non-aromatic heterocyclic ring
11/28/2002WO2002039997A3 Ace-2 modulating compounds and use thereof
11/28/2002WO2002009759A3 Aldosterone antagonist and cyclooxygenase-2 inhibitor combination therapy to prevent or treat inflammation-related cardiovascular disorders
11/28/2002US20020177600 Two or more ligand moieties covalently linked together by one or more linking groups enabling binding to multiple binding sites; increased efficacy, selectivity and duration; anti-proliferative and anticarcinogenic
11/28/2002US20020177594 Inhibitors of histone deacetylase
11/28/2002DE10138577A1 New 4-benzoyl-5-oxy-pyrazole derivatives, useful as herbicides, especially pre- and post-emergence selective herbicides