Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
10/2003
10/16/2003CA2479522A1 New pharmaceutical compositions based on anticholinergics and p38 kinase inhibitors
10/16/2003CA2479520A1 P38 kinase inhibitors for treating mucus hypersecretion_
10/15/2003EP1352650A1 Inhibitors against the production and release of inflammatory cytokines
10/15/2003EP1351959A1 Novel pleuromutilin derivatives
10/15/2003EP1351956A1 Semicarbazides and their uses as cyclin dependent kinase inhibitors
10/15/2003EP1351943A1 Benzophenone uv-absorbers with heterocyclic substituents
10/15/2003EP1351939A1 Coupler/developer and coupler/coupler hybrid dyes and coupler/developer and coupler/coupler hybrid dye intermediates
10/15/2003EP1005332B1 Pharmaceutical composition for reducing production of mcp-1 protein
10/15/2003EP0973747B1 Pesticidal 1-arylpyrazoles
10/14/2003US6632840 Monoacyl-substituted guanidines, a process for their preparation, their use as a medicament or diagnostic aid, and pharmaceutical compositions containing them
10/14/2003US6632830 ACE-2 inhibiting compounds and methods of use thereof
10/14/2003US6632825 Picornaviral 3C protease enzyme inhibitors; amide ester or amide acid derivatives
10/14/2003US6632815 Show selectivity for factor Xa versus other proteases of coagulation or the fibrinolytic cascades
10/09/2003WO2003082861A2 Morpholinyl-urea derivatives for use of the treatment of inflammatory diseases
10/09/2003WO2003082826A1 Substituted biaryl amides as c5a receptor modulators
10/09/2003WO2003082280A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
10/09/2003WO2003082205A2 Compounds and methods
10/09/2003WO2003082013A1 Method of purifying a pesticide
10/09/2003US20030191175 Indole sPLA2 inhibitors
10/09/2003US20030191171 Insecticidal and acaricidal agent
10/09/2003US20030191156 Antidiabetic agents; dietetics
10/09/2003US20030191118 Inhibitors of alpha4 mediated cell adhesion
10/09/2003US20030190298 Use as skin lightening agents
10/09/2003CA2480241A1 Method of purifying a pesticide
10/09/2003CA2480106A1 Morpholinyl-urea derivatives for use of the treatment of inflammatory diseases
10/09/2003CA2479928A1 Substituted biaryl amides as c5a receptor modulators
10/08/2003EP1349839A1 Phenylethenyl or phenylethinyl derivatives as glutamate receptor antagonists
10/08/2003EP1349613A2 Thrombopoietin mimetics
10/08/2003EP1349548A2 Methods and compositions for treating periodontal disease
10/08/2003EP1214318B1 Imidazo[1,2-a]pyridine and pyrazolo[2,3-a]pyridine derivatives
10/08/2003CN1447798A Process for prepn. of pyrazole compounds
10/08/2003CN1447789A Compounds to treat alzheimer's disease
10/07/2003US6630499 Control of arthropods in animals
10/07/2003US6630468 Disubstituted pyrazolines and triazolines as factor Xa inhibitors
10/07/2003US6630463 Heterocycle-containing carboxylic acid derivative and drug containing the same
10/07/2003CA2287552C Pyrazolopyrimidinone cgmp pde5 inhibitors for the treatment of sexual dysfunction
10/07/2003CA2263957C Diarylmethyl piperazine derivatives as delta opioid agonists
10/07/2003CA2107105C Heterocyclic-cyclic amine derivatives
10/07/2003CA2094808C Oxysulfonyl urea acat inhibitors
10/02/2003WO2003080583A1 Medicine for prevention and/or therapy of cardiomyopathy
10/02/2003WO2003080577A2 Amidoacetonitrile compounds
10/02/2003WO2003080545A2 Substituted phenylacetic acids
10/02/2003WO2003080053A1 Combination treatments for chemokine-mediated diseases
10/02/2003WO2003079973A2 Mitotic kinesin inhibitors
10/02/2003WO2003053358A3 Fused heterocyclic compounds and analogs thereof: modulators of nuclear hormone receptor function
10/02/2003WO2003045912A8 Inhibitors of factor xa and other serine proteases involved in the coagulation cascade
10/02/2003WO2003039529A8 Selective antibacterial agents
10/02/2003US20030187302 Enzyme inhibitors, 1-(4-methanesulfonyl-benzylidene)-3,4-dihydro-1H-naphthalene-2 -one oxime
10/02/2003US20030187033 Potassium channel modulators; cardiovascular disorders; antiarrhythmia agents
10/02/2003CA2780743A1 Substituted tetracycline compounds
10/02/2003CA2479338A1 Substituted phenylacetic acids
10/01/2003CN1445615A Electric photographic organic photoreceptor with new charge transfer matter
10/01/2003CN1445218A 3-phenyl pyrazole-5-ramification of carboxylic acid derivative as well as its preparing method and medicine appliction
10/01/2003CN1122665C Herbicidal N-alkenyl heteroaryloxyacetamides
10/01/2003CN1122442C Fungicidal mixtures
09/2003
09/30/2003US6627758 Ligand including (i) at least two different types of heteroatoms selected from nitrogen, phosphorus, and sulfur, and (ii) at least one of imidazole, pyrazole, and pyridine; transition metal complex for carbonylation to aldehyde
09/30/2003US6627643 Sodium-hydrogen exchanger type 1 (NHE-1) inhibitors of formula I' are useful for the prevention and treatment of myocardial ischemic injury. Myocardial ischemic injury can occur in out-patient in perioperative settings and can lead to sudden
09/30/2003US6627626 Antiinflammation agents and antiarthritic agents colon cancer, and Alzheimer's disease in mammals, preferably humans, dogs, cats and livestock animals.
09/25/2003WO2003078408A1 Crystalline parecoxib sodium
09/25/2003WO2003078403A2 Derives d’aminoindazoles comme inhibiteurs de proteine-kinase
09/25/2003WO2003078402A1 Indazoles substituted with an anti-cancerous activity
09/25/2003WO2003078401A1 Preventive and/or therapeutic agent for hypoxic ischemic brain disorder
09/25/2003WO2003078400A1 Neurotensin active 2,3-diaryl-pyrazolidine derivatives
09/25/2003WO2003077847A2 Substituted amides
09/25/2003WO2003077828A2 Novel florfenicol-type antibiotics
09/25/2003WO2002024690A3 Efficient process for the preparation of a factor xa inhibitor
09/25/2003US20030181728 Fused heterocyclic compounds and analogs thereof, modulators of nuclear hormone receptor function
09/25/2003US20030181718 Process for synthesis of heteroaryl-substituted urea compounds useful as antiinflammatory agents
09/25/2003US20030181504 Administering 2-(benzo(g)indazol-1-yl)-ethylamines and 1-(4H-indeno(1,2-c)pyrazol-1-yl)-1-methylethylamines compounds for therapy of glaucoma
09/25/2003US20030181503 Administering 2-(benzo(g)indazol-1-yl)-ethylamines and 1-(4H-indeno(1,2-c)pyrazol-1-yl)-1-methylethylamines compounds for therapy of glaucoma
09/25/2003US20030181502 Methods of treating sepsis
09/25/2003US20030181496 Having Transforming Growth Factor- beta inhibitory activity and being useful as fibrosis inhibitors for organs or tissues
09/25/2003US20030181334 Herbicidal method
09/25/2003CA2478540A1 Indazoles substituted with an anti-cancerous activity
09/25/2003CA2478500A1 Crystalline parecoxib sodium
09/25/2003CA2478048A1 Novel florfenicol-type antibiotics
09/24/2003EP1345909A1 Phenylacetamido-pyrazole derivatives and their use as antitumor agents
09/24/2003EP1345902A1 Substituted heterocyclo-norbornylamine derivatives, method for producing the same, their use as medicament or diagnostic agent and medicament containing the same
09/24/2003EP1024137B1 Resolution of amines
09/24/2003CN1444573A Carboxamide compounds and their use as antagonists of human 11CBY receptor
09/24/2003CN1444564A Biphenyl carboxamides
09/24/2003CN1444477A Thrombopoietin mimetics
09/24/2003CN1122025C Method for preparing 1-phenylpyrrazolin-3-carboxylic acid derivatives
09/23/2003US6624309 Administering 4-heterocyclicbenzamide derivative
09/23/2003CA2127110C Carbamates and crop protection agents containing them
09/18/2003WO2003076410A1 Process for asymmetric intramolecular [3+2] cyclo- addition of hydrazones
09/18/2003WO2003076409A1 Derivatives of 1-phenyl-3-phenylpyrazole as herbicides
09/18/2003WO2003076408A2 Indazole derivatives that are activators of soluble guanylate cyclase
09/18/2003WO2003075917A1 Combination therapy for treating, preventing or managing proliferative disorders and cancers
09/18/2003WO2003075857A2 Amino-methyl substituted tetracycline compounds
09/18/2003WO2003075853A2 Cyclic derivatives as modulators of chemokine receptor activity
09/18/2003WO2003075836A2 Cathepsin cysteine protease inhibitors
09/18/2003WO2003053368A3 Chalcone derivatives and their use to treat diseases
09/18/2003WO2002076925A3 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
09/18/2003WO2002062750A9 Cannabinoid receptor ligands
09/18/2003US20030176708 Thiophene substituted hydroxamic acid derivatives as cyclooxygenase-2 and 5-lipoxygenase inhibitors
09/18/2003US20030176696 Preparing pyrazolopyrimidinone derivatives for the treatment of impotence
09/18/2003US20030176668 C-nitroso compounds and use thereof
09/18/2003US20030176478 For selectively modulating the activation, repression, agonism and antagonism effects of the glucocorticoid receptor in a patient; for therapy and prophylaxis of obesity, diabetes, depression, neurodegeneration or an inflammatory disease
09/18/2003US20030176466 For controlling parasites in or on an animal