Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
03/2004
03/25/2004WO2003070696A3 Substituted aryl ketones
03/25/2004WO2003069350A3 Small molecule modulators of apoptosis
03/25/2004WO2003051846A3 Substituted phenyl derivatives
03/25/2004WO2003004480A3 Substituted piperazine and diazepanes as histamine h3 receptor agonists
03/25/2004US20040059128 Method of producing 1-alkyl-3-aryl-5-difluoromethoxy-ih-pyrazoles
03/25/2004US20040059116 Aryl aniline beta2 adrenergic receptor agonists
03/25/2004US20040058990 Thrombopoietin mimetics
03/25/2004US20040058937 Heterocyclic mutilin esters and their use as antibacterials
03/25/2004US20040058820 Central nervous system disorders; psychological disorders; antiinflammatory agents; multiple sclerosis
03/25/2004US20040058819 Process for the preparation of pesticidal compounds
03/25/2004CA2497550A1 Pyrazolo[3,4-b]pyridine compounds, and their use as phosphodiesterase inhibitors
03/25/2004CA2496315A1 4-(3,5-dicyanophenoxy) pyrazole derivatives for use as reverse transcriptase modulators in the treatment of i.a. hiv
03/24/2004EP1400529A1 Glucopyranosyloxypyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate therefor
03/24/2004EP1400516A1 Substituted anilide derivatives, intermediates thereof, agricultural and horticultural chemicals, and their usage
03/24/2004EP1400515A1 Cyclic diamine compound having five-membered cyclic group
03/24/2004EP1400508A1 Dithiocarbamic acid ester
03/24/2004EP1399497A1 Production of masked isocyanates, particularly masked polyisocyanates
03/24/2004EP1399159A1 4-substituted-1-(arylmethylidene)thiosemicarbazide, 4-substituted-1-(arylcarbonyl)thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof
03/24/2004EP1399156A2 Alkylidene pirazolidinedione derivatives and their use for treating diabetes and obesity
03/24/2004EP1131318B1 Process for making 5-substituted pyrazoles using dithietanes
03/24/2004EP1082110B1 Use of compounds for the elevation of pyruvate dehydrogenase activity
03/24/2004EP0904079B1 Antidiabetic agents
03/24/2004CN1484638A I-aryl-or-I-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-b ligands
03/24/2004CN1142917C N-cycloalkyl-3-alkenylbenzoyl-pyrazole derivs.
03/23/2004US6710069 1-aryl- or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
03/18/2004WO2004022544A1 Novel aminoindazole derivatives as medicines and pharmaceutical compositions containing same
03/18/2004WO2004022543A1 Preventive and/or therapeutic drugs for inflammatory intestinal diseases
03/18/2004WO2004022529A2 Diarylurea derivatives and their use as chloride channel blockers
03/18/2004WO2004022526A1 Cathepsin cysteine protease inhibitors
03/18/2004WO2004022523A2 1, 3-diamino-2-hydroxypropane prodrug derivatives
03/18/2004WO2004021984A2 Heterocyclic aromatic compounds useful as growth hormone secretagogues
03/18/2004WO2004011453A3 Method for preparing 3-halo-4,5-dihydro-1h-pyrazoles
03/18/2004US20040054186 Autoimmune diseases; anticancer agents; antiproliferative agents; skin disorders
03/18/2004US20040053985 Such as 1-(1-cyclooctyl-3-((nitrooxy)methyl)pyrazol-5-yl)-4-(methylsulfonyl)benzene; for synthesis of nitric oxide/ endothelium-derived relaxing factor; antiinflammatory agents; kits
03/18/2004US20040053971 A fluorinated compounds, microbiocides, synthesis with chemical intermediates, amidation, debromination, benzylation, oximination
03/18/2004US20040053970 Emzyme inhibitors, a 4-pyridinyl-3-pyrazoles derivatives, treating animal having cancer, restenosis, psoriasis, endometriosis, atherosclerosis, ischemia, myocardial ischemic; a plant having yeast infection and viral infection
03/18/2004US20040053953 Treatment of chemokine mediated diseases
03/18/2004US20040053945 Process for the preparation of a pyrazolo[4,3-d]pyrimidine derivative
03/18/2004US20040053935 Anticancer agents
03/18/2004US20040053934 Anticancer agents
03/18/2004US20040053890 Naphthalene derivatives
03/18/2004US20040053786 Insecticidal 1,8-naphthalenedicarboxamides
03/18/2004CA2497979A1 1, 3-diamino-2-hydroxypropane prodrug derivatives
03/18/2004CA2497955A1 Medicament for preventing and/or treating inflammatory bowel disease
03/18/2004CA2495939A1 Cathepsin cysteine protease inhibitors
03/18/2004CA2495284A1 Diarylurea derivatives and their use as chloride channel blockers
03/17/2004EP1398029A1 NR3B1 nuclear receptor binding 3-substituted pyrazole derivatives
03/17/2004EP1397341A1 6-(aryl-amido or aryl-amidomethyl)-naphthalen-2-yloxy-acidic derivatives as inhibitors of plasminogen activator inhibitor type-1 (pai-1)
03/17/2004EP1147102B1 Heteroaryl acetylenic sulfonamide and phosphinic acid amide hydroxamic acid tace inhibitors
03/17/2004EP1144365B1 Inhibitors of alpha-4 beta-1 mediated cell adhesion
03/17/2004EP1140802B1 Substituted aryl and heteroaryl derivatives, their production and their use as medicines
03/17/2004EP0971588B1 Novel cannabinoid receptor modulators
03/17/2004CN1482911A A method for treating allergies using substituted pyrazoles
03/17/2004CN1482119A Method for preparing 3.5-dimethylpyrazole
03/17/2004CN1142134C Processes for preparing pesticidal intermediates
03/16/2004US6706927 Intermediates in preparation of 1,5-diarylpyrazole antiinflammatory agents
03/16/2004US6706911 Reacting n-substituted 3-aminoacrylic esters with haloalkylcarboxylic anhydrides in presence of base; pyrazole-4-carboxylic acid chemical intermediates; haloacylation
03/16/2004US6706765 Aminoguanidines and alkoxyguanidines as protease inhibitors
03/16/2004US6706743 β3 adrenergic receptor agonists and uses thereof
03/16/2004US6706729 A method for dissociating a metal ion from a zinc finger-containing protein; inhibiting virus
03/16/2004US6706711 Substituted diaminopyrazoles; treating diseases, such as cancer, inflammatory disorders, restenosis, and cardiovascular disease. coatings for implantable medical devices, such as prostheses, artificial valves, etc.
03/16/2004US6706707 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles
03/11/2004WO2004020445A2 4-(3,3-dihalo-allyloxy) phenol derivatives having pesticidal properties
03/11/2004WO2004020393A1 Dibenzylamine compound and medicinal use thereof
03/11/2004WO2003091264A3 Non nucleoside reverse transcriptase inhibitors
03/11/2004WO2003082861A3 Morpholinyl-urea derivatives for use of the treatment of inflammatory diseases
03/11/2004WO2003065789A3 N-biphenylmethyl aminocycloalkanecarboxamide derivatives
03/11/2004US20040049052 Benzophenone uv-absorbers with heterocyclic substituents
03/11/2004US20040048866 3-substituted with an oxy-, thio- or amino- group; increasing cGMP levels
03/11/2004US20040048864 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/11/2004US20040048858 Chalcone derivatives and their use to treat diseases
03/11/2004US20040048844 Acylsemicarbazides as cyclin dependent kinase inhibitors useful as anti-cancer and anti-proliferative agents
03/10/2004EP1396493A1 Heterocyclic compounds
03/10/2004EP1395571A1 Compounds and methods for the treatment or prevention of flavivirus infections
03/10/2004EP1395565A1 Herbicidal substituted benzoylpyrazoles
03/10/2004EP1395551A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases
03/10/2004EP1285014B1 Dimethylpyrazole-blocked isocyanate mixtures
03/10/2004CN1480454A Antagon of endostadin receptor pyrazole carboxylic acids
03/09/2004US6703426 Treatment of breast cancer
03/04/2004WO2004018476A1 Novel polymorph of n-methyl-n-(3-{3-[2-thienylcarbonyl]-pyrazol-[1,5-alpha]-pyrimidin-7-yl}phenyl)acetamide and compositions and methods related thereto
03/04/2004WO2004018428A1 Antibacterial benzoic acid derivatives
03/04/2004WO2004018414A2 Antibacterial agents
03/04/2004WO2004018410A1 Substituted benzanilide compound and pest control agent
03/04/2004WO2004017961A2 Derivatives of 3-hydroxy-4-(cyclyl-alkylaminoalkyl)-5-phenyl-1h-pyrazole as antagonists of the gonadotropin releasing hormone (gnrh) for use in the treatment of sex hormone related conditions, such as prostatic of uterine cancer
03/04/2004US20040044081 Hypotensive agents; cardiovascular disorders; anticholesterol agents; antiarrhythmia agents
03/04/2004US20040044062 Method of treatment of viral infection including HIV using water soluble fullerenes - III
03/04/2004US20040044049 Compounds for inhibiting insulin secretion and methods related thereto
03/04/2004US20040044008 Dietetics; antilipemic agents; non-insulin dependent diabetes; cardiovascular disorders
03/04/2004US20040043988 Cycloalkyl alkanoic acids as intergrin receptor antagonists
03/04/2004US20040043904 N-(4-pyrazolyl) amide derivatives, chemicals for agricultural and horticultural use, and usage of the same
03/04/2004US20040043388 Compositions and methods for isolating ligand binding polypeptides for a user-specified ligand, and for isolating small molecule ligands for a user-specified target polypeptide using an improved class of hybrid ligand compounds
03/04/2004US20040043247 Organic electroluminescence devices using pyrazolo [3,4B] quinoxaline derivatives
03/03/2004EP1392661A1 Diarylurea derivatives useful as anti-inflammatory agents
03/03/2004EP1392659A1 Methods of making indazoles
03/03/2004EP1392658A1 Novel fused indazoles and indoles and their use for the treatment of glaucoma
03/03/2004EP1392280A2 Arylsulfonamide ethers, and methods of use thereof
03/03/2004EP0986386B1 Use of nitrogen heterocyclic aromatic derivatives in the topical treatment of the epithelial tissues diseases
03/02/2004US6699994 Biaryl compounds as serine protease inhibitors
03/02/2004US6699991 Process for the preparation of pyrazoles
03/02/2004US6699990 Colorfastness; waterproofing; oxidative color hair dyes