Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
09/2004
09/30/2004US20040192744 Inhibition of Histone Deacetylase; antiproliferative; antitumor: cell differentiation; 3,5-Dimethyl-isoxazole-4-carboxylic acid (2-amino-4,5-dichloro-phenyl)-amide
09/30/2004US20040192735 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
09/30/2004US20040192681 N-acylsulfonamide apoptosis promoters
09/30/2004US20040192667 Novel pyrazole analogs acting on cannabinoid receptors
09/30/2004US20040192666 Nonnucleoside reverse transcriptase inhibitors
09/30/2004US20040192653 P38 inhibitors and methods of use thereof
09/30/2004US20040191660 Electrophotographic printing method, monoazo iron complex compound, charge controlling agent using the same and toner using the charge controlling agent
09/29/2004EP1461345A2 Copper deposition using copper formate complexes
09/29/2004EP1461334A2 Pyrazole derived kinase inhibitors
09/29/2004EP1461311A2 Urea derivatives as vr1-antagonists
09/29/2004EP0736016B1 Trisubstituted phenyl derivatives, processes for their preparation and their use as phosphodiesterase (type iv) inhibitor
09/29/2004CN1533380A N-pyrazolylcarboxanilides as fungicides
09/28/2004US6797731 Resorcinol derivatives
09/28/2004US6797723 Heterocycle substituted diphenyl leukotriene antagonists
09/23/2004WO2004080999A1 Pyrazole compounds useful in the treatment of inflammation
09/23/2004WO2004080984A1 Insecticidal phthalamide derivatives
09/23/2004WO2004080973A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors
09/23/2004WO2004080972A1 Pirazole modulators of atp-binding cassette transporters
09/23/2004WO2004080962A1 2,4,6-phenyl substituted cyclic ketoenols
09/23/2004WO2004080947A1 Imino ether derivative compounds and drugs containing the compounds as the active ingredient
09/23/2004WO2004080486A1 Tumorigenesis inhibitor
09/23/2004WO2004080376A2 Hydroxyethylamine compounds having asp2 inhibitory activity for the treatment of alzheimer’s disease
09/23/2004WO2004050613A3 2-substituted-3-propenamide derivatives and methods of using the same
09/23/2004WO2003105751A3 Novel curcumin derivatives
09/23/2004US20040186156 useful for solid tumors and leukemia; auto-immune diseases such as psoriasis, alopecia and multiple sclerosis; cardiovascular diseases such as stenoses, arterioscleroses and restenoses; infectious diseases caused by unicellular parasites; nephrological diseases, neurodegenerative diseases
09/23/2004US20040186154 treating or preventing a hypercholesterolemia-related or an inflammation-related condition ; apical sodium co-dependent bile acid transport inhibitor and an amount of a cyclooxygenase-2 (COX-2) selective inhibitor or its prodrug; kits
09/23/2004US20040186145 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
09/23/2004US20040186108 such as N-{2-[2-(4-1,2-Benzisothiazol-3-yl-piperazin-1-yl)-ethyl]-phenyl}-2-(2,5-dimethoxy-phenyl)-acetamide; antagonists of dopamine D2 receptors and of serotonin 2A (5HT2a) receptors; for treatment of depression and dementia/schizophrenia
09/23/2004US20040186060 [1-(3-cyano-benzyl)-1-([[(5-cyano-thiophen-2-ylmethyl)-carbamoyl]-methyl]-carbamoyl)-3-methanesulfonyl-propyl]-carbamic acid methyl ester; trypsin-like serine protease; for treatment of tumors and metastasis cancer
09/23/2004US20040185352 Photothermographic element comprising improved base precursors and methods for their use
09/23/2004US20040182279 Colorant or dye covalently bonded to benzophenone derivative; storage stability
09/23/2004DE10311300A1 New 2-alkoxy-4-halo-6-alkylphenyl-substituted (hetero)cyclic ketoenols, useful as total or selective herbicides and pesticides, e.g. insecticides, acaricides and nematocides for plant protection
09/23/2004CA2518986A1 Imino ether derivative compounds and drugs containing the compounds as the active ingredient
09/23/2004CA2517885A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors
09/22/2004EP1460077A1 Novel pyrazolopyrimidones and their use as PDE inhibitors
09/22/2004EP1458685A2 Substituted phenyl derivatives
09/22/2004EP1458670A1 Method for producing 2-halogenacyl-3-amino-acrylic acid derivatives
09/22/2004EP1458383A2 Heteroaryl substituted pyrazole modulators of metabotropic glutamate receptor-5
09/22/2004EP1458379A1 Hydroxyphenyl-pyrazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
09/22/2004EP1458375A2 Compositions for decreasing activity of hormone-sensitive lipase
09/22/2004EP1458374A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/22/2004EP1000062B1 Tricyclic vasopressin agonists
09/22/2004EP0805148B1 Benzamidoxime derivative, process for production thereof, and agrohorticultural bactericide
09/22/2004CN1531536A Process for preparation of pyrazolo[4,3-D] pyrimidine derivative
09/22/2004CN1167685C Released development inhibiting primary blue former
09/22/2004CN1167683C Aromatic pyrozole compound, its preparation, agricultural composition containnig it and use thereof
09/21/2004US6794512 Antiinflammatory agents; cyclooxygenase inhbitors; anticancer agents; autoimmune disease
09/21/2004US6794400 4-substituted-1-(arylmethylidene)thiosemicarbazide, 4-substituted-1-(arylcarbonyl)thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof
09/21/2004CA2114017C Amide tetrazole acat inhibitors
09/16/2004WO2004078732A1 N-aryl heteroaromatic products, compositions containing same and use thereof
09/16/2004WO2004078116A2 P38 inhibitors and methods of use thereof
09/16/2004WO2004032975A3 Biphenyls and fluorenes as imaging agents in alzheimer's disease
09/16/2004WO2003028729A3 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
09/16/2004US20040181075 Process of making chalcone derivatives
09/16/2004US20040180964 anti-obestic activity; Neuropeptide Y antagonist
09/16/2004US20040180947 Sulfonamide compounds and pharmaceutical use thereof
09/16/2004US20040180944 Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3',5'-monophosphate phosphodiesterase (cGMP-PDE5) for the treatment of sexual dysfunction
09/16/2004US20040180906 Anti-inflammatory medicaments
09/16/2004US20040180896 P38 inhibitors and methods of use thereof
09/16/2004US20040180891 Pyrazole derivatives useful in the treatment of hyper-proliferative disorders
09/16/2004US20040180882 Small molecule modulators of hepatocyte growth factor (scatter factor) activity
09/16/2004US20040180871 Anti-inflammatory compositions and methods
09/16/2004CA2512243A1 N-aryl heteroaromatic products, compositions containing same and use thereof
09/15/2004EP1457490A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity
09/15/2004EP1457199A1 Coupling agents having a 2,3,5-triaminopyridine structure and their use for dyeing keratinic fibres
09/15/2004EP1456424A1 4-(alpha branched)acyl- (3h)-pyrazol-3-ones for use in the extraction of metals, especially copper, from solution
09/15/2004EP1456181A1 Methods for preparing sodium-hydrogen exchanger type-1 inhibitors
09/15/2004EP1456180A1 3,4-diarylpyrazoles and their use in the therapy of cancer
09/15/2004EP1456179A1 Deuterated substituted pyrazolylbenzylsulfonamides and medicaments comprising said compounds
09/15/2004EP1456151A1 Method for forming a carbon-carbon or carbon-heteroatom linkage
09/15/2004EP0986384A4 Inhibitors of protein isoprenyl transferases
09/15/2004CN1529595A 4,5-hydro-1H-pyrazole derivative having protent CB1-antagonistic
09/15/2004CN1166652C Preparation method of carbonyl aplpha-substitution nitrogenous compound
09/15/2004CN1166633C New alpha-amino acid sulfuryl compounds, its preparing method and medicinal composition containing them
09/14/2004US6790979 Use as antitumor agents, particularly for the treatment of cancers such as colon, skin and prostate cancer and to induce androgen receptor antagonist activity in subject with androgen-related affliction
09/10/2004WO2004076420A1 Heteroarylcarbamoylbenzene derivative
09/10/2004WO2004076414A2 Novel compounds
09/10/2004WO2004075840A2 Selective non-steroidal glucocorticoid receptor modulators
09/10/2004WO2004056727A8 Process of making chalcone derivatives
09/10/2004WO2004052847A3 Tricyclic steroid hormone nuclear receptor modulators
09/10/2004WO2004022523A3 1, 3-diamino-2-hydroxypropane prodrug derivatives
09/10/2004WO2004014352A3 Methods for treating carbonic anhydrase mediated disorders
09/10/2004CA2516684A1 Selective non-steroidal glucocorticoid receptor modulators
09/10/2004CA2516407A1 Heteroarylcarbamoylbenzene derivatives
09/09/2004US20040176595 Glucocorticoid receptor modulators
09/09/2004US20040176462 NPY Y5 antagonist
09/09/2004US20040176434 Pyrazoloanthrone derivatives as Jun N-terminal kinase inhibitors; diabetes; obesity
09/09/2004US20040176363 N-Acylpiperazine derivatives; cardiovascular disorders; anticoagulants
09/09/2004US20040176356 4-(Hydroxyalkyl-)-piperazinyl(thio)acetamide derivatives for treatment of cardiovascular disorders; antiarrhythmia agents; intermittent claudication, angina, congestive heart failure and myocardial infarction
09/09/2004US20040176325 P38 MAP kinase inhibitors comprising indazole derivatives; antiinflammatory and antiproliferative agents; autoimmune, bone, and neurodegenerative disorders; viricides, infections
09/09/2004US20040176308 Sodium dependent glucose transporter 1 inhibitors; blocking small intestine absorption of glucose; diabetes
09/09/2004US20040176253 Herbicides; broad active spectrum; on soil and above ground plant parts use
09/08/2004EP1454902A1 N- (substituted five-membered di-or triaza diunsaturated ring)carbonyl guanidine derivateives for the treatment of ischemia
09/08/2004EP1453801A1 Substituted 2-amino-cycloalkanecarboxamides and their use as cysteine protease inhibitors
09/08/2004EP1453789A2 N,n'-substituted-1,3-diamino-2-hydroxypropane derivatives
09/08/2004EP1289972B1 Serine protease inhibitors
09/08/2004EP0944581A4 Process of preparing substituted acrylamides
09/08/2004CN1527829A Pyrazole derivatives as HIV reverse transcriptase inhibitors
09/08/2004CN1527709A Therapeutic combinations for cardiovascular and inflammatory indications
09/08/2004CN1165546C New derivative of erythromycin, its preparation method and medicinal application