Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
09/2004
09/08/2004CN1165536C Substituted pyrazole derivatives condensed with six-membered heterocyclic rings
09/02/2004WO2004074257A1 Non-nucleoside reverse transcriptase inhibitors
09/02/2004WO2004074256A1 Tetrahydroisoquinolinyl sulfamic acids
09/02/2004WO2004074243A2 Heterocyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands
09/02/2004WO2004074238A1 Phenethylamino sulfamic acids
09/02/2004WO2004073709A1 Antimicrobial agents
09/02/2004WO2004073642A2 2-aminoethyl substituted pyrimidin-2-ones, cyclopropanes, pyrazolines, pyrimidines and benzothiazepines and their use as urotensin ii and somatostatin 5 receptor ligands
09/02/2004WO2004073606A2 Sulfonamide derivatives as ppar modulators
09/02/2004WO2004049797A3 Pesticidal sulphonylaminopyrazoles
09/02/2004WO2003084539A3 New pharmaceutical compositions based on anticholinergics and p38 kinase inhibitors
09/02/2004US20040171881 N,N'-substituted-1,3-diamino-2-hydroxypropane derivatives
09/02/2004US20040171842 VIRICIDES; uSING A SECONDARY AMIDE COMPOUNDAIDS
09/02/2004US20040171781 From a sulfonate compound containing unsaturated ester group; membrane
09/02/2004US20040171670 Neurological diseases and disorders; such as 3-fluoro-10,11-dihydro-5-(2-aminoethyl)-5H-dibenzo[a,d]cycloheptene
09/02/2004US20040171649 Intermediates for anthranilic amide insecticides and blood coagulation factor Xa inhibitors
09/02/2004US20040171075 Modulation of protein functionalities
09/02/2004CA2515706A1 2-aminoethyl substituted pyrimidin-2-ones, cyclopropanes, pyrazolines, pyrimidines and benzothiazepines and their use as urotensin ii and somatostatin 5 receptor ligands
09/02/2004CA2515570A1 Heterocyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands
09/02/2004CA2512883A1 Sulfonamide derivatives as ppar modulators
09/01/2004EP1451175A1 Thrombin inhibitors
09/01/2004EP1451162A1 Substituted diphenyl heterocycles useful for treating hcv infection
09/01/2004EP1451160A2 Pyrazole-amides and-sulfonamides
09/01/2004EP1450901A2 (1-phenyl-2-heteroaryl)ethyl-guanidine compounds as inhibitors of mitochondrial f1f0 atp hydrolase
09/01/2004EP1450791A1 Hydrazonopyrazole derivatives and their use as therapeutics
09/01/2004EP0923530B1 Inhibition of matrix metalloproteases by substituted biaryl oxobutyric acids
09/01/2004CN1525957A Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
09/01/2004CN1525856A Stable high-concentration injection containing pyrazolone derivative
09/01/2004CN1164638C Dimethyl pyrazole-blocked isocyanate mixtures
08/2004
08/31/2004US6784195 Extracellular signal regulated kinase (erk); anticancer agents and protein kinase inhibitors
08/26/2004WO2004072101A2 Phenylglycine derivatives useful as serine protease inhibitors
08/26/2004WO2004047744A3 3-heterocyclic benzylamide derivatives as potassium channel openers
08/26/2004WO2004043355A3 Alpha, alpha-disubstituted benzylglycine derivatives as hiv protease inhibitors
08/26/2004WO2004043354A3 Ophthalmic compositions for treating ocular hypertension
08/26/2004WO2004013094A3 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
08/26/2004US20040167183 Protein tyrosine phosphatase inhibitor; antidiabetic agents; hypotensive agents; cardiovascular disorders; inflammatory bowel disorders; antiulcer agents; wound healing agents; anticancer agents
08/26/2004US20040167160 Skin disorders; controlling cell differentiation; antidiabetic agents; cardiovascular disorders; anticancer agents; central nervous system disorders
08/26/2004US20040167158 Heterocyclic compounds for the treatment of migraine
08/26/2004US20040167128 Aminopeptidase inhibitor; vision defects; administering to eye
08/26/2004US20040167127 atherosclerosis; antiarthritic agents; antidiabetic agents; cardiovascular disorders; autoimmune diseases; multiple sclerosis; chronic obstructive pulmonary disease
08/26/2004US20040167126 Such as (2RS,3R)-3-amino-4-cyclohexyl-2-hydroxy-N-phenoxybutanamide; methionine aminopeptidase type 2 inhibitors
08/26/2004US20040167122 Central nervous system disorders; anxiolytic agents; neurodegenerative disorders; obsessive compulsive disorders; schizophrenia; antidepressants; alzheimer's disease; neuropathic pain; stroke
08/26/2004US20040167116 Viricides
08/26/2004US20040167031 Arylphenyl-substituted cyclic ketoenols
08/26/2004DE10307329A1 New 4-amino-3(5)-phenyl-1(2)H-pyrazole derivatives, useful as pharmaceuticals, agrochemicals or their precursors, e.g. as antipyretic or antirheumatic agents
08/26/2004DE10306503A1 New 1-benzoyl-3-(heterocyclyl-phenyl)-urea derivatives, are glycogen phosphorylase a inhibitors useful e.g. for treating type II diabetes, dyslipidemia or arteriosclerosis
08/26/2004DE10305089A1 Neue heteroarylsubstituierte Acetonderivate als Hemmstoffe der Phospholiphase A2 New heteroaryl substituted acetone derivatives as inhibitors of phospholipase A2
08/25/2004EP1449894A2 Ink jet dye design
08/25/2004EP1448557A2 Heteroindanes: a new class of potent cannabimimetic ligands
08/25/2004EP1448554A1 Propylcarbamate derivatives as inhibitors of serine and cysteine proteases
08/25/2004EP1448539A1 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
08/25/2004EP1448534A1 6-membered unsaturated heterocyclic compounds useful for selective inhibition ofthe coagulation cascade
08/25/2004EP1278728B1 Pyrrolidine and piperidine derivatives and their use for the treatment of neurodegenerative disorders
08/25/2004EP0934302B1 Aminophenol derivates
08/25/2004CN1524075A Substitued arylketones
08/25/2004CN1163488C Process for preparing insecticide
08/25/2004CN1163486C Guanidinylamino heterocycle compounds useful as alpha-2 adrenoceptor agonists
08/24/2004US6780862 Such as amino-indazoles for treatment of central nervous system disorders
08/24/2004CA2285733C Process for preparation of pyrazolo[4,3-d]pyrimidin-7-ones and intermediates thereof
08/19/2004WO2004069837A1 Pyrazolo`1,5-a!`1,3,5!triazine derivatives as cannabinoid receptor ligands
08/19/2004WO2004069824A1 Pyrazole derivative
08/19/2004WO2004069805A1 Bis(hetero)aryl carboxamide derivatives for use as pgi2 antagonists
08/19/2004WO2004069797A1 Novel heteroaryl-substituted acetone derivatives as inhibitors of phospholipase a2
08/19/2004WO2004069394A2 Synthetic method for direct arylation of heterocyclic arenes
08/19/2004WO2004069158A2 Substituted pyrazoles, compositions containing such compounds and methods of use
08/19/2004WO2004046090A3 Aryl ureido derivatives and their medical use
08/19/2004WO2004002409A3 Cyclooxygenase-2 selective inhibitors, compositions and methods of use
08/19/2004WO2003049702A8 Vanilloid receptor ligands and their use in treatments
08/19/2004US20040162330 Stable high-concentration injection containing pyrazolone derivative
08/19/2004US20040162324 Thienylazolylalkoxyethanamines, their preparation and their application as medicaments
08/19/2004US20040162321 For therapy of disease characterized by inflammatory, allergic, or proliferative processes
08/19/2004US20040162282 Substituted piperazines
08/19/2004US20040162281 Pyridine ring containing biaryl compound useful to treat and/or prevent clotting disorders, and as antiinflammatory and anticoagulant agents
08/19/2004US20040162276 Indazole or indole derivatives, and use thereof in human medicine and more particularly in oncology
08/19/2004CA2515235A1 Bis(hetero)aryl carboxamide derivatives for use as pgi2 antagonists
08/19/2004CA2515147A1 Novel heteroaryl-substituted acetone derivatives as inhibitors of phospholipase a2
08/19/2004CA2515119A1 Pyrazole derivative
08/19/2004CA2513409A1 Pyrazolo`1,5-a!`1,3,5!triazine derivatives as cannabinoid receptor ligands
08/18/2004EP1447400A1 Bicyclic compound
08/18/2004EP1446405A2 Inhibitors of cyclin-dependent kinases, compositions and uses related thereto
08/18/2004EP1446384A1 Polymorphous form of rimonabant, preparation method and pharmaceutical compositions containing same
08/18/2004EP1446379A1 Aryl aniline beta-2 adrenergic receptor agonists
08/18/2004EP1446375A1 Dihalogenpropene compounds, method for the production thereof, agents containing said compounds and the use thereof as pest control agents
08/18/2004EP1268436B1 Novel diaminopyrazole derivatives and dyes containing said compounds
08/18/2004EP1222173B1 Process for preparing 4-trifluoromethylsulphinylpyrazole derivative
08/18/2004CN1522251A Azole compounds, process for preparation of the same and use thereof
08/18/2004CN1522250A Cyclic diamine compound having five-membered cyclic group
08/18/2004CN1522245A Substituted sulfonamide compounds, process for their use as medicament for the treatment of CNS disorders, obestity and type II diabetes
08/18/2004CN1522244A Anthranilic acid amides, method for the production thereof, their use as antiarrhythmia agents, and pharmaceutical preparations thereof
08/18/2004CN1162405C Substd. benzoyl ketones, methods for producing them and their use as herbicides
08/18/2004CN1162079C Poison baits containing N-phenyl or N-pyridyl pyrazoles for controlling insect pests
08/17/2004US6777437 Antidepressants, anxiolytic agents. sexual disorders
08/17/2004US6777419 Pyrazolo [4,3-d]pyrimidines
08/17/2004US6777418 For treating or preventing emphysema, cancer and dermatological disorders
08/12/2004WO2004067703A2 5ht7 antagonists and inverse agonists
08/12/2004WO2004067515A1 Pyrazolyl carboxanilides for controlling unwanted microorganisms
08/12/2004US20040158076 Tyrosine derivatives
08/12/2004US20040157904 Anilinopyrazole derivatives useful for the treatment of diabetes
08/12/2004US20040157892 Insecticides; miticides
08/12/2004US20040157849 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor
08/12/2004US20040157839 substituted pyrazolo[1,5-a][1,3,5]triazine compounds; in particular CB1 receptor antagonists