Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865) |
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01/06/2005 | US20050004360 Compounds and methods for modulation of estrogen receptors |
01/06/2005 | US20050004230 Retroviral protease inhibitors |
01/06/2005 | US20050004167 Such as dibenzofuran-2-carboxylic acid 2-(phenylsulfonyl)hydrazide |
01/06/2005 | US20050004164 2-Cyanopropanoic acid amide and ester derivatives and methods of their use |
01/05/2005 | EP1492771A1 Quinoline and isoquinoline derivatives, method for the production thereof and use thereof as anti-inflammatory agents |
01/05/2005 | EP1274687B1 1,2,3,4- tetrahydroisoquinoline derivatives |
01/05/2005 | CN1183117C Intermediates for making HIV-protease inhibitors and method of making HIV-protease inhibitors |
01/05/2005 | CN1183116C Substituted isoquinoline derivatives and pharmaceutical composition containing them, its preparation method and use |
01/05/2005 | CN1183107C Alkynyl containing hydroxamic acid compounds as TACE inhibitors |
01/04/2005 | US6838465 N-acyltetrahydroisoquinoline derivatives |
12/30/2004 | US20040266817 3-Substituted 6,7-dihydroxytetrahydroisoquinoline derivatives for use as antibacterial agents |
12/29/2004 | WO2004113391A2 Improved pharmaceutical drug candidates and methods for preparation thereof |
12/29/2004 | WO2004113330A1 Immunosuppressant compounds and compositions |
12/29/2004 | WO2004113302A1 N-substituted 6,8-dialkoxy-1,2,3,4-tetrahydro-1h-isoquinoline as potassium channels modulators |
12/29/2004 | WO2004113301A1 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders |
12/29/2004 | WO2004113277A2 Methods and compositions for treating amyloid-related diseases |
12/29/2004 | WO2004113275A2 Methods and compositions for treating amyloid-related diseases |
12/29/2004 | WO2004112793A1 Guanidino-substituted quinazolinone compounds as mc4-r agonists |
12/29/2004 | EP1491532A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetyloholine receptors |
12/29/2004 | EP1490341A1 Novel adamantane derivatives |
12/29/2004 | EP1490340A1 Heteroaromatic urea derivatives as vr-1 receptor modulators for treating pain |
12/29/2004 | EP1490339A1 Novel chalcone derivatives and uses thereof |
12/29/2004 | EP1490062A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
12/29/2004 | CN1182121C Compound with activity for resisting platelet aggregation and its preparation method |
12/29/2004 | CA2529524A1 Substituted piperidine compounds and methods of their use |
12/29/2004 | CA2529257A1 Methods and compositions for treating amyloid-related diseases |
12/29/2004 | CA2529256A1 Methods and compositions for treating amyloid-related diseases |
12/29/2004 | CA2524700A1 N-substituted 6,8-dialkoxy-1,2,3,4-tetrahydro-1h-isoquinoline as potassium channels modulators |
12/29/2004 | CA2524027A1 Immunosuppressant compounds and compositions |
12/29/2004 | CA2523015A1 Guanidino-substituted quinazolinone compounds as mc4-r agonists |
12/28/2004 | US6835739 Benzamides and related inhibitors of factor Xa |
12/28/2004 | US6835725 Cyanine dye containing heterocylic rings; satisfies light stability, favorable signal/noise rato, damage free application to the substrate material, use in the information layer in a write-once optical data carrier |
12/28/2004 | US6835469 Phosphorescent compounds and devices comprising the same |
12/28/2004 | CA2126072C Tri-substituted phenyl derivatives and processes for their preparation |
12/23/2004 | WO2004111010A1 Isoquinoline -1,3,4-trione, the synthetic method and the use thereof |
12/23/2004 | WO2004111009A1 Fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor |
12/23/2004 | WO2004110986A1 Benzamide derivative or salt thereof |
12/23/2004 | WO2004099150A3 3-(1-naphthyl)-2-cyanopropanoic acid derivatives as estrogen receptor ligands |
12/23/2004 | US20040259912 N-(4-benzhydryloxy-3-isobutyrylphenyl)-N'-(3,4-dimethoxyphenyl)urea for example; vanilloid receptor agonists; use as analgesic and or for treating urinary frequency and/or urinary incontinence |
12/23/2004 | US20040259910 Glutamine fructose-y-phosphate amidotransferase (GFAT) inhibitors |
12/23/2004 | US20040259804 (Substituted)Acyl dipeptidyl inhibitors of the ICE/ced-3 family of cysteine proteases |
12/23/2004 | CA2756058A1 Fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor |
12/23/2004 | CA2526872A1 Fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor |
12/23/2004 | CA2526387A1 Benzamide derivative or salt thereof |
12/22/2004 | EP1489071A1 N-substituted, 3,4-dihydro-1H-isoquinoline as potassium channels modulators |
12/22/2004 | EP1487801A1 7-arylsulfonamido-2,3,4,5-tetrahydro-1h-benzo[d]azepine derivatives with 5-ht6 receptor affinity for the treatment of cns disorders |
12/22/2004 | EP1487798A1 Substituted tetrahydroisoquinolines as c5a receptor modulators |
12/22/2004 | EP1487795A2 Synthesis of enantiomerically pure amino-substituted fused bicyclic rings |
12/22/2004 | EP1487449A1 Tyrosyl derivatives and their use as p2x7 receptor modulators |
12/16/2004 | WO2004108682A2 Tetrahydroisoquinolines as antagonists of the 5ht1b receptor |
12/16/2004 | WO2004108681A1 Nitrogen-containing heteroaryl compounds and their use in increasing endogenous erythropoietin |
12/16/2004 | WO2004108663A1 N-alkynyl-2- (substituted aryloxy) alkylthioamide derivatives as fungicides |
12/16/2004 | WO2004108645A1 Method for the treatment or prevention of lower urinary tract symptoms |
12/16/2004 | WO2003063797A8 Cycloalkyl inhibitors of potassium channel function |
12/16/2004 | US20040254216 Inhibitors of p38 |
12/16/2004 | US20040254215 Novel nitrogen-containing heteroaryl compounds and methods of use thereof |
12/16/2004 | US20040254214 7-Amido-isoindolyl compounds and their pharmaceutical uses |
12/16/2004 | US20040254193 Novel tetrahydroquinolines |
12/16/2004 | US20040254188 such as N-(5-tert-butyl-2,3-dihydro-1H-inden-1-yl)-N'-5-isoquinolinylurea; for treating pain, inflammatory thermal hyperalgesia, urinary incontinence, or bladder overactivity |
12/16/2004 | CA2528756A1 Tetrahydroisoquinolines as antagonists of the 5ht1b receptor |
12/16/2004 | CA2527313A1 N-alkynyl-2-(substituted aryloxy) alkylthioamide derivatives as fungicides |
12/15/2004 | EP1485370A1 Amino-derivatives as novel inhibitors of histone deacetylase |
12/15/2004 | EP1485364A1 Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase |
12/15/2004 | EP1485357A1 Process for asymmetric hydrogenation of hexahydroquinoline salts |
12/15/2004 | EP1485356A1 NON-PEPTIDE GnRH ANTAGONISTS |
12/15/2004 | EP1485353A1 New inhibitors of histone deacetylase |
12/15/2004 | EP1485348A1 Carbonylamino-derivatives as novel inhibitors of histone deacetylase |
12/15/2004 | EP1485099A1 Inhibitors of histone deacetylase |
12/15/2004 | EP1226137B8 Phenyl- and pyridyl-tetrahydro-pyridines having tnf inhibiting activity |
12/15/2004 | CN1554649A Metabotropic glutamate receptor antagonists for treating central nervous system diseases |
12/15/2004 | CN1179948C HIV protease inhibitors |
12/14/2004 | US6831080 Cinnamide derivatives as KCNQ potassium channel modulators |
12/09/2004 | WO2004106305A1 New p2x7 receptor antagonists and their use |
12/09/2004 | US20040248989 Method for the treatment or prevention of lower urinary tract symptoms |
12/09/2004 | US20040248933 tertiary carbocyclic amines such as 4,7-diphenyl-2-methyl-1,2,3,4-tetrahydroisoquinoline, having preferential binding norepinephrine transporter protein (NET) over the other neurotransmitter transporters; side effect reduction |
12/09/2004 | US20040248932 Use of aryl- and heteroaryl-substituted tetrahydroisoquinolines in the treatment of chronic and neuropathic pain, migraine headaches, and urge, stress and mixed urinary incontinence |
12/09/2004 | US20040248895 Novel guanidino compounds |
12/09/2004 | US20040248872 Safe for agricultural or gardening use; effective against insects and mammals |
12/08/2004 | EP1484320A1 Jnk inhibitor |
12/08/2004 | EP1483244A1 Cyclic n-substituted alpha iminocarboxylic acids for selectively inhibiting collagenase |
12/08/2004 | EP1483233A2 Substituted tetrahydroisoquinoline compounds, methods of making, and their use |
12/02/2004 | WO2004103967A2 Thiocarbamate inhibitors of alpha-4 integrins |
12/02/2004 | WO2004103961A2 Sulfated bis-cyclic agents |
12/02/2004 | US20040242572 New carboxamide compounds having melanin concentrating hormone antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture |
12/02/2004 | CA2525934A1 Thiocarbamate inhibitors of alpha-4 integrins |
12/01/2004 | EP1481968A2 Cell adhesion-inhibiting anti-inflammatory and immune-suppressive compounds |
12/01/2004 | EP1480999A2 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases |
12/01/2004 | EP1480971A1 Isoquinoline derivatives |
12/01/2004 | EP1480954A1 Vanilloid receptor modulators |
12/01/2004 | EP1480941A2 Urea derivatives as hiv aspartyl protease inhibitors |
12/01/2004 | EP0886637B1 Inhibitors of microsomal triglyceride transfer protein and method |
12/01/2004 | CN1550496A Acetylenic alpha-amino acid-based sulfamide hydroxamic acid TACE inhibitors |
11/30/2004 | US6826033 Beta 3 adrenergic receptor agonists; treatment of pollakiuria, urinary incontinence, obesity or diabetes |
11/30/2004 | US6825354 Osteoporosis; rheumatic diseases |
11/30/2004 | US6825351 Selective hydrogenation of amino-substituted fused bicyclic aromatic ring system, preparation of racemic amino substituted fused bicyclic ring system via nitrosation, enzymatic resolution of racemic mixture to produce (r)- and (s)-forms |
11/30/2004 | US6825228 To treat infections by gram-positive bacteria, in particular drug- resistant strains |
11/30/2004 | US6825213 β3-adrenoreceptor agonists, agonist compositions and methods of using |
11/30/2004 | US6825189 Treating withdrawal symptoms caused by smoking cessation |
11/30/2004 | US6825184 For use as anti-inflammatory agents |
11/30/2004 | US6825181 Orally administrated to exhibit a strong anticoagulant effect by inhibiting activated blood- coagulation factor x |