Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
03/2005
03/02/2005EP1077698B1 Metabolites of ecteinascidin 743
03/02/2005CN1589307A Phosphorescent compounds and devices comprising the same
03/02/2005CN1589262A Cyanoguanidine prodrugs
03/02/2005CN1589153A Preventives/remedies for urinary disturbance
03/01/2005US6861527 Nitration in a static micromixer
02/2005
02/24/2005WO2005016891A1 7-phenylsulfonyl-tetrahydro-3-benzazepine derivatives as antipsychotic agents
02/24/2005WO2005016890A1 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor
02/24/2005WO2005016889A1 Compounds having antiestrogenic and tissue selective estrogenic properties
02/24/2005WO2005016876A2 Cyclic amine bace-1 inhibitors having a benzamide substituent
02/24/2005WO2005016867A2 Anthranilic acid derivatives and their use as activators of the hm74a receptor
02/24/2005WO2005016862A1 Substituted arylalkanoic acid derivative and use thereof
02/24/2005WO2005016344A1 Piperazine derivatives for the treatment of hiv infections
02/24/2005WO2005016264A2 Diamine derivatives of quinone and uses thereof
02/24/2005US20050043552 Process for the synthesis of amine ethers from secondary amino oxides
02/24/2005US20050043358 Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
02/24/2005US20050043351 Fused compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor
02/24/2005US20050043340 Process for reacting alkaloids and use of the reaction products in the preparation of medicaments
02/24/2005US20050043304 Lower alkyl molecular weight amine as enzyme inhibitors for use in the treatment of tryptase enzyme inhibitors inhibitorsfor respiratory system disorders, antiinflammatory agents, inflammatory bowel disease, hyperprolific skin disorders, vascular edema and rheumatoid arthritis
02/24/2005US20050043300 Piperazine derivatives
02/24/2005US20050042407 containing a cyanovinylene group; can be written on or read by blue light, preferably laser light
02/24/2005CA2743534A1 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor
02/24/2005CA2535665A1 Substituted arylalkanoic acid derivative and use thereof
02/24/2005CA2534950A1 Cyclic amine bace-1 inhibitors having a benzamide substituent
02/24/2005CA2534866A1 Piperazine derivatives for the treatment of hiv infections
02/23/2005EP1507764A1 Novel enantiomers of tetrahydroisoquinoline derivatives and their pharmaceutically acceptable salts, their preparations and pharmaceutical compositions
02/23/2005EP1507763A1 Tetrahydroisoquinoline derivatives
02/23/2005EP1507504A1 Cycloalkyl inhibitors of potassium channel function
02/23/2005CN1583725A Preparation of liensinine, isoliensinine and methylliensinine extracted from lotus seed
02/23/2005CN1190427C Method for preparing pyrimidine derivative
02/22/2005US6858735 Preparation of quinapril hydrochloride
02/17/2005WO2005014576A1 Isoquinolinone derivative, process for producing the same and use thereof
02/17/2005WO2004094386A8 Isoquinoline-5-sulfonic acid amides as inhibitors of akt (protein kinase b)
02/17/2005WO2004092115A3 Hydroxamates as therapeutic agents
02/17/2005US20050038035 Heterocyclic amide compounds as apolipoprotein b inhibitors
02/17/2005US20050038027 Melanocortin-4 receptor agonists; obesity, type II diabetes; such as N-(2-(2-(2,4-dichlorophenyl)ethyl)-1-oxo-2,3-dihydro-1H-isoindol-5-yl) -3-methyl-N'-(2,6,6-trimethylbicyclo(3.1.1)hept-3yl)piperazine-1-carboximidamide
02/17/2005CA2531796A1 Aryl and heteroaryl compounds, compositions, and methods of use
02/16/2005EP1506188A1 Process for the preparation of a hydrate of an anthranilic acid derivative
02/16/2005EP1506166A1 Aminotetralin-derived urea modulators of vanilloid vr1 receptor
02/15/2005US6855715 Drugs such as 1-(3-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4-(4-fluoro-2 -methylsulphonylphenyl)piperazine, used as anticoagulants
02/15/2005US6855512 Phenylacetic or heteroarylacetic acid derivatives; retinoid like activity
02/10/2005WO2005011697A2 Sulfonamide derivatives with activity on protein kinase a and b
02/10/2005US20050032794 For example, 2-Dimethylamino-N-(3-dimethylamino-1,4-dioxo-1,4-dihydro-naphthalen-2-yl)-N-methyl-acetamide; ability to function as gene expression modulators for genes found in cancer cells, especially genes involved in misregulated signal transduction pathways typical of cancers of colon and breast
02/10/2005US20050032790 For example, 1-(2-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4,4'-bispiperidine; for treatment of thrombosis, emphysema, cirrhosis; antiarthritic agents, anticancer agents, antihistamines
02/10/2005US20050031903 Multilayer; charge generating compound, charge transfer compound; blue phosphorescence
02/09/2005EP1505062A1 Heterocyclic derivatives and their use as antithrombotic agents
02/09/2005EP1503989A1 Dopamine receptor modulators as antipsychotic agents
02/09/2005EP1503761A1 Substituted piperazines as melanocortin receptor ligands
02/09/2005EP1487795A4 Synthesis of enantiomerically pure amino-substituted fused bicyclic rings
02/09/2005EP0983999B1 Process for producing amide derivatives and intermediates
02/09/2005CN1578663A Inhibitors of histone deacetylase
02/09/2005CN1188121C Therapeutic substituted guanidines
02/08/2005CA2096525C Retroviral protease inhibitors
02/08/2005CA2096409C Retroviral protease inhibitors
02/08/2005CA2096408C Retroviral protease inhibitors
02/03/2005WO2004072102A3 Benzene acetamide compounds useful as serine protease inhibitors
02/03/2005US20050027007 Allylamides useful in the treatment of alzheimer's disease
02/02/2005EP1501804A1 Isoquinoline derivatives mao-b inhibitors
02/02/2005EP1501803A2 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
02/02/2005EP0828754B1 Dipeptides which promote release of growth hormone
02/02/2005CN1187332C Tetrahydroisoquinoline hydroximic acid sulfamide compound, its synthesis method and its application
02/01/2005US6849733 Compounds containing amidated guanidine derivative type functional group of structure N-C(=N)-N-CO-N-C=N or N-C(=N)-N-CO-N
02/01/2005US6849632 Heteroaryl alkyl piperazine derivatives
01/2005
01/27/2005WO2005007838A1 Cell diffrentiation inhibitor, cell culture method using the same, liquid culture medium and cultured cell line
01/27/2005WO2005007621A2 Ubiquitin ligase inhibitors
01/27/2005US20050020684 Modulators of peroxisome proliferator activated receptors
01/27/2005US20050020623 5-Substituted isoquinoline derivatives
01/27/2005US20050020597 Attention deficit disorders; hyperactivity; post-trauma stress disorders; anxiolytic agents; obsessive compulsive disorders; analgesics; Parkinson's disease
01/27/2005US20050020584 Benzamide derivatives as antagonists of orexin receptors
01/26/2005EP1499898A2 Regulation of tnf-alpha
01/26/2005EP1499319A1 Bicyclo 4.4.0 antiviral derivatives
01/26/2005EP1499313A2 Heterocyclic derivatives as opioid receptor modulators
01/26/2005CN1186325C Tetrahydroisoquinoline derivative kind addition salt for treating cardiac and cerebral vascular diseases and its prepn
01/25/2005US6846825 Antibacterial agents
01/20/2005WO2005005392A1 Azacyclic compounds as inhibitors of sensory neurone specific channels
01/20/2005WO2005004868A1 Anti-coronavirus drug
01/20/2005US20050014946 Substituted amino ketone compounds
01/20/2005US20050014721 reacting oxabenzonorbornadiene with nucleophiles;in presence of rhodium complex catalyst forming 2-pyrrolidin-1-ol-1,2-dihydronaphthalen-1-ol; drug used as analgesics, Parkinson's disease, anticancer agents; aids
01/20/2005US20050014702 Inhibition of pdf enzyme as bactericidal agents for veterinary medicines
01/19/2005EP1498406A1 Novel hydronaphthalene compounds, prepared by a rhodium catalysed ring opening reaction in the presence of phosphine ligand
01/19/2005EP1497268A2 Nitric oxide donors, compositions and methods of use
01/19/2005CN1566099A Isoquinoline-1, 3, 4-trione compounds, preparation method and uses thereof
01/19/2005CN1566098A Isoquinoline compound, preparation method and application of salt thereof
01/19/2005CN1185234C Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
01/18/2005US6844367 Benzamides and related inhibitors of factor Xa
01/13/2005WO2004099129A3 Intermediates useful in the synthesis of hiv-protease inhibitors and methods for preparing the same
01/13/2005US20050009871 Ubiquitin ligase inhibitors
01/13/2005US20050009864 Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them
01/13/2005US20050009863 Used for treating renal disorders such as acute or chronic renal failure, biliary function disorders, respiratory disorders such as snoring or sleep apneas and strokes.
01/13/2005US20050009812 Remedies for stress diseases comprising mitochondrial benzodiazepine receptor antagonists
01/13/2005CA2531327A1 Compounds and therapeutical use thereof
01/12/2005EP1495009A2 Cyanamides useful as reversible inhibitors of cysteine proteases
01/12/2005EP1495004A2 Benzenesulfonamide derivatives and their use as dopamine d3 and d2 receptor ligands
01/12/2005EP1494997A1 Substituted aryl amides
01/12/2005EP1228043B1 Isoquinoline and quinazoline deivatives having a combined 5ht1a, 5ht1b and 5ht1d receptor activity
01/12/2005CN1562974A Method for synthesizing 1, 2, 3, 4 ramification of tetrahydro-isoquinoline
01/12/2005CN1184298C Color-safe bleach boosters, composns. and laundry methods employing same
01/11/2005US6841560 Substituted isoquinoline derivatives and their use as anticonvulsants
01/11/2005CA2104909C Decahydroisoquinolines as excitatory amino acid receptor antagonists
01/06/2005WO2004103967A3 Thiocarbamate inhibitors of alpha-4 integrins
01/06/2005WO2004101528A3 Isoquinoline derivatives and their use as gfat inhibitors
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