Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
04/2005
04/06/2005CN1604893A Cyclic amine compounds
04/06/2005CN1604890A 取代的环己烷衍生物 Substituted cyclohexane derivatives
04/06/2005CN1603291A Novel intermediates useful for the preparation of antihistaminic piperidine derivatives
04/06/2005CN1195762C Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same
04/06/2005CN1195741C Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
04/06/2005CN1195737C HIV proteinase inhibitor
04/06/2005CN1195736C Gatrokinetic monocyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
04/05/2005US6875888 Method for the production of esters of unsaturated carboxylic acids
04/05/2005US6875870 Discoloration inhibition, colorfastness for candle wax; polymers
04/05/2005US6875831 Mono and multifunctional alkoxyamines for the preparation of functionalized macromers
04/05/2005US6875780 Compounds that modulate PPAR activity and methods for their preparation
04/05/2005US6875777 Compounds
04/05/2005US6875776 Antihistamines; antiallergens; antiinflammatory agents; autoimmune diseases; rheumatic diseases
04/05/2005US6875775 Triphenylalkene derivatives and their use as selective estrogen receptor modulators
04/05/2005US6875760 Glucagon antagonists/inverse agonists
04/05/2005US6875759 Anticancer agents; analgesics
04/05/2005CA2339621C 2-substituted-1-piperidyl benzimidazole compounds as orl1-receptor agonists
04/05/2005CA2245686C In situ block copolymer formation during polymerization of a vinyl aromatic monomer
03/2005
03/31/2005WO2005028467A1 Antibacterial 3,5-diaminopiperidine-substitute aromatic and heteroaromatic compounds
03/31/2005WO2005028440A1 Novel gamma secretase inhibitors
03/31/2005WO2005028439A1 Cinnamoyl compound and use of the same
03/31/2005WO2005028438A1 Novel piperidine derivative
03/31/2005WO2005028436A2 Thalidomide analogs as tnf-alpha modulators
03/31/2005WO2005028429A2 Haloalkyl containing compounds as cysteine protease inhibitors
03/31/2005WO2005028426A1 Novel 4-phenylamino-benzaldoxime derivative and use thereof as mek inhibitor
03/31/2005WO2005028425A2 Amidines and derivatives thereof and pharmaceutical compositions containing them
03/31/2005WO2005005394A3 Thiophenylaminoimidazolines as prostaglandin i2 antagonists
03/31/2005WO2005005345A3 Use of functionalized onium salts as a soluble support for organic synthesis
03/31/2005US20050070582 For example,1-{[2-(3,5-dimethylphenoxy)-5-nitrophenyl]sulfonyl}-4-ethylpiperazine or 1-{[2-(3,5-dichlorophenoxy)-5-nitrophenyl]sulfonyl}piperazine; for the treatment of asthma, atopic dermatitis, allergic rhinitis and other inflammatory/immunological disorders
03/31/2005US20050070549 heterocylic amines such as 2-(5-{3-[4-(4-Chloro-2-methyl-phenyl)-piperazin-1-yl]-propylidene}-5,11-dihydro-10-oxa-1-aza-dibenzo[a,d]cyclohepten-7-yl)-propan-2-ol, used for treating diseases associated with aberrant leukocyte recruitment and/or activation
03/31/2005US20050070539 Such as 1-(4-{4-[2-(cyclopropylmethyl-amino)-5-nitro-benzoyl]-piperazin-1-yl}-3-fluoro- phenyl)-ethanone for treatment of psychoses, pain, neurodegenerative disfunction in memory and learning, schizophrenia, dementia, attention deficit disorders, or Alzheimer's disease
03/31/2005US20050070520 Aza-cyclic compounds as modulators of acetylcholine receptors
03/31/2005US20050069555 Vaccine adjuvants; hepatitis c virus; modulation immunology response
03/31/2005CA2808646A1 Thalidomide analogs
03/31/2005CA2551037A1 Novel piperidine derivative
03/31/2005CA2539842A1 Amidines and derivatives thereof and pharmaceutical compositions containing them
03/31/2005CA2538960A1 Cinnamoyl compound and use of the same
03/31/2005CA2538864A1 Thalidomide analogs as tnf-alpha modulators
03/31/2005CA2538590A1 Novel gamma secretase inhibitors
03/31/2005CA2521811A1 Haloalkyl containing compounds as cysteine protease inhibitors
03/30/2005EP1517894A1 N-benzyl-3-phenyl-3-heterocyclyl-propionamide compounds as tachykinin antagonists and/or serotonin reuptake inhibitors
03/30/2005EP1517882A1 Amide linker peroxisome proliferator activated receptor modulators
03/30/2005EP1360184B1 Piperidine derivatives as neurokinin 1 antagonists
03/30/2005EP1087765B1 Use of optically pure (-) norcisapride in the treatment of irritable bowel syndrome
03/30/2005EP1047674B1 Process for production of donepezil derivatives
03/30/2005CN1602191A Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
03/29/2005US6872832 Hydroxy substituted N-alkoxy hindered amines and compositions stabilized therewith
03/29/2005US6872741 Sodium channel modulators
03/29/2005US6872735 LFA-1 antagonist compounds
03/29/2005US6872716 Sexual diosrders; schizophrenia; drug abuse; eating disorders anxiolytic agents
03/24/2005WO2005026171A1 Substance which exhibits antiviral and antibacterial activity and is based on derivatives of 2,8-dithioxo-1h-pyrano[2,3d¸6,5-d']dipyrimidyne and 10-aza-analogue thereof
03/24/2005WO2005025568A1 Ophthalmic compositions for treating ocular hypertension
03/24/2005WO2005012220A3 Cycloalkylidene compounds as modulators of estrogen receptor
03/24/2005WO2004089922A3 Calcium channel inhibitors comprising benzhydril spaced from piperazine
03/24/2005WO2004087074A3 Process for making substituted pyrazoles
03/24/2005WO2004080583A3 PROCESS FOR THE PREPARATION OF threo-METHYLPHENIDATE HYDROCHLORIDE
03/24/2005WO2004064730A3 Compounds, compositions and methods
03/24/2005WO2004041161A3 Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity
03/24/2005US20050065346 anticoagulants; thrombosis; factor x inhibitor
03/24/2005US20050065345 pipecolic acid or an acid salt reacted with an amine (i,e 2,6-dimethylaniline) in an inert solvent in presence of a condensing agent such as dicyclohexylcarbodiimide, 1-ethyl-2-(2-dimethylaminopropyl)carbodiimide, methanesulfonyl chloride or phosphoryl chloride to form pipecolic acid-2,6-xylidide
03/24/2005US20050065339 Amino-alkyl derivatives
03/24/2005US20050065211 Ester derivatives
03/24/2005US20050065162 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
03/24/2005US20050065161 Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds, compositions and their uses
03/24/2005US20050065144 Dipeptidyl peptidase inhibitors
03/24/2005US20050065142 Antidiabetic agents; therapy for insulin resistance
03/24/2005US20050065140 Antidepressant; side effect reduction
03/24/2005US20050065139 Antidiabetic agents; controlling carbohydrate metabolism
03/24/2005US20050065095 Antibacterial agents
03/24/2005US20050065093 Inhibitors of the ICE/ced-3 family of cysteine proteases
03/24/2005CA2788502A1 Non-peptide agonists and antagonists of adrenomedullin and gastric releasing peptide
03/24/2005CA2539049A1 Quinazoline derivatives
03/24/2005CA2538410A1 2-pyridone derivatives as netrophil elastase inhibitors and their use
03/24/2005CA2537430A1 Ophthalmic compositions for treating ocular hypertension
03/23/2005EP1516872A1 Novel azasugar derivative and drug containing the same as the active ingredient
03/23/2005EP1515969A1 Spiroindolinepiperidine derivatives
03/23/2005EP1515951A1 Arylsulfonylhydroxamic acid and amide derivatives and their use as protease inhibitors
03/23/2005EP1515950A1 Cationic alkoxyamines and their use in producing nano particles from natural or synthetic clays
03/23/2005EP1515945A2 Method for making aryl hydrazines and substituted indoles
03/23/2005EP1280528B1 R-eliprodil for treating glaucoma
03/23/2005CN1599733A N-ureido-piperidines as antagonists viii for CCR-3 receptor
03/23/2005CN1599722A 4-piperidinyl alkylamine derivatives as muscarinic receptor antagonists
03/23/2005CN1599721A CCR-3 receptor antagonists VII
03/23/2005CN1599607A Carbinols for the treatment of neuropathic dysfunction
03/23/2005CN1597680A New method of synthesizing thalidomide and its derivative
03/23/2005CN1193788C Beta 2-adrenergic receptor agonist
03/22/2005US6869953 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents
03/17/2005WO2005023794A2 Compound libraries of 4-carboxamidopiperidine derivatives
03/17/2005WO2005023769A1 Process for the preparation of amlodipine salts
03/17/2005WO2005023768A1 An improved process for the preparation of pure nisoldipine
03/17/2005WO2005023767A2 Diastereomers of 4-aryloxy-3-hydroxypiperidines
03/17/2005WO2005023260A1 1- (2-amino-benzol) -piperazine derivatives as glycine uptake inhibitors for the treatment of psychoses
03/17/2005WO2005023183A2 Nitrosated ad nitrosylated diuretic compouds, compositions and methods of use
03/17/2005WO2005023182A2 Nitrosated and nitrosylated cardiovascular compounds, compositions and methods of use
03/17/2005WO2004056809A8 Novel piperidine derivatives as modulators of chemokine receptor ccr5
03/17/2005WO2004056808A8 Novel piperidine derivatives as modulators of chemokine receptor ccr5
03/17/2005WO2003045918A8 Piperidine-based mch antagonists for treatment of obesity and cns disorders
03/17/2005US20050059825 Reacting esters of 2,5-bis(2,2,2-trifluoroethoxy)-benzoic acid with primary amino group of 2-(aminomethyl)piperidine; high yield and purity; starting material has low toxicity; arrhythmia
03/17/2005US20050059712 Immunosuppressants for treating skin disorders, acne, alopecia, estrogen- or androgen-dependent tumors, rheumatoid arthritis, type I and II diabetes, lupus erythematosus, multiple sclerosis, ulcerative colitis, Crohn's disease, psoriasis, contact dermatitis, graft versus host disease, eczema, asthma
03/17/2005US20050059700 Reacting compunds such as 6-methyl-12-oxa-tricyclo[8.2.1.0]trideca-2,4,6-trien-11-ol with compounds such as 4-(2,6-dichloro-phenyl)-piperidine to produce (+-)-cis-1-methyl-7-[[4-(2,6-dichloro-phenyl)piperidin-1-yl)]methyl]-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ol