Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
12/2004
12/23/2004US20040259804 (Substituted)Acyl dipeptidyl inhibitors of the ICE/ced-3 family of cysteine proteases
12/23/2004CA2528905A1 Neurocyte protective agent
12/23/2004CA2528652A1 Nk1 antagonist
12/23/2004CA2528644A1 Novel piperazinyl-aryloxy and piperazinyl-heteroaryloxy-n-aryl lactams
12/23/2004CA2527033A1 2-substitued 5,6-diaryl-pyrazine derivatives as cb1 modulators
12/23/2004CA2526209A1 Cyclic hydroxylamine as psychoactive compounds
12/23/2004CA2525207A1 Substituted piperidine carbamates for use as inhibitors of hormone sensitive lipase
12/22/2004EP1489106A1 Arene-ruthenium complexes immobilized on polymers, catalysts consisting of the complexes, and processes for organic syntheses with the same
12/22/2004EP1487817A1 Piperidine derivatives useful as modulators of chemokine receptor activity
12/22/2004EP1487811A1 N-sulfonylurea apoptosis promoters
12/22/2004EP1487807A2 New compounds
12/22/2004EP1487798A1 Substituted tetrahydroisoquinolines as c5a receptor modulators
12/22/2004EP1487793A1 Piperidine derivatives useful as modulators of chemokine receptor activity
12/22/2004EP1440067B1 N-formyl derivatives of paroxetine
12/22/2004CN1556805A Piperidine derivative as NMDA receptor antagonist
12/22/2004CN1556105A Synthesis method of N-benzyl-4-piperidyl formaldehgde
12/22/2004CN1181056C 4-acylamino piperidin-N-oxides
12/21/2004US6833458 Practical syntheses of chiral trans-3, 4-disubstituted piperidines and the intermediates
12/21/2004US6833457 Process for preparation of benzylpiperidine compounds
12/16/2004WO2004108674A1 Amino alcohol derivative, medicinal composition containing the same, and uses of these
12/16/2004WO2004108673A2 Inhibitors of papilloma virus
12/16/2004WO2004108636A2 Isotopically labeled chemically stable reagents and process for the synthesis thereof
12/16/2004WO2004108215A1 Piperidinyl prostaglandin e analogs
12/16/2004US20040254377 Novel processes for the preparation of peripheral opioid antagonist compounds and intermediates thereto
12/16/2004US20040254374 Alanyl-piperidine heterocyclic derivatives useful against cardiovascular diseases
12/16/2004US20040254344 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
12/16/2004US20040254327 Bisphenol a derivatives containing one biaryl group and a spacer; monomers for polycarbonates
12/16/2004US20040254280 Blends of waxes and polymer additives
12/16/2004US20040254219 Muscarinic receptors; chronic obstructive pulmonary disease; asthma
12/16/2004US20040254218 Substituted piperidine compounds and methods of their use
12/16/2004US20040254195 heterocyclic amines such as 1-{1-[1-(4-Choro-phenyl)-cyclopropylmethyl]-piperidin-3ylmethyl}-4-(2-methoxy-phenyl)-piperazine used as dopamine, serotonin or norepinephrine transporters
12/16/2004US20040254182 Enhanced propertied pharmaceuticals
12/16/2004CA2528179A1 Piperidinyl prostaglandin e analogs
12/16/2004CA2526506A1 Inhibitors of papilloma virus
12/15/2004EP1485370A1 Amino-derivatives as novel inhibitors of histone deacetylase
12/15/2004EP1485364A1 Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase
12/15/2004EP1485354A1 Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
12/15/2004EP1485353A1 New inhibitors of histone deacetylase
12/15/2004EP1485351A2 Process for the manufacture of optically active 3-substituted lactams by asymmetric hydrogenation of 3-alkylidenelactams
12/15/2004EP1485348A1 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
12/15/2004EP1485107A1 Phospholipids as caspase inhibitor prodrugs
12/15/2004EP1485099A1 Inhibitors of histone deacetylase
12/15/2004EP1263711B1 Novel use of phenylheteroalkylamine derivatives
12/15/2004EP1188742B1 Vinylated alkoxyamine, use thereof, and process for producing the same
12/15/2004EP0988263B1 Process for the production of radioiodinated neuroreceptor agents
12/15/2004CN1554768A Preparation of lactams from aliphatic alpha,omega dinitriles
12/15/2004CN1554746A Preparation of lactams from aliphatic alpha,omega dinitriles
12/15/2004CN1554649A Metabotropic glutamate receptor antagonists for treating central nervous system diseases
12/15/2004CN1554646A Preparation of lactams from aliphatic alpha,omega dinitriles
12/15/2004CN1554343A Compounds for treating fibromyalgia and chronic fatigue syndrome
12/15/2004CN1554341A Compounds for treating fibromyalgia and chronic fatigue syndrome
12/14/2004US6831199 Pyrimidine compounds and derivatives thereof
12/14/2004US6831176 Reacting a ketoaldonic acid methyl ester of the sugar with the protected hydroxyl groups with a an alkylamine or hydroxyalamine salt in an organic solvent with a tert-amine to react with acid generated to produce oxime methyl ester
12/14/2004US6831089 1,4-di-substituted piperidines, some of which have M2 selectivity even higher than that of 3-alpha-chloroimperialine for treating cognitive disorders such as Alzheimer's disease
12/10/2004WO2004108677A1 Antithrombotic ethers
12/09/2004WO2004106411A2 Biodegradable poly(beta-amino esters) and uses thereof
12/09/2004WO2004106303A1 Lactone-added hindered amine compound
12/09/2004WO2004106285A1 Benzamide nitrile derivatives
12/09/2004WO2004096761A8 Aromatic oxyphenyl and aromatic sulfanylphenyl derivatives
12/09/2004WO2004089901A3 Phospholipase c inhibitors for use in treating inflammatory disorders
12/09/2004WO2004069794A9 New arylpiperazinyl compounds
12/09/2004WO2001076599A8 Process of making racemic bupivacaine's enantiomers, levobupivacaine's pharmaceutical compositions, levobupivacaine's pharmaceutical compositions formulated on its free base form or its pharmaceutical acceptable salts and use of levobupivacaine's pharmaceutical compositions formulated on its free base form
12/09/2004US20040249160 Hydrogenation process
12/09/2004US20040249159 Novel piperidin-2,6-dione disulphate salts and their use for the treatment of stress related affective disorders
12/09/2004US20040249155 1-(omego-substituted-2-[(hetero)arylcarbonylamino]alkanoyl)-4-(1-methylpiperidin-4-yl)piperidine derivatives; e.g., 1-[N-(Indole-6-carbonyl)-D-serinyl]-4-(1-methylpiperidin-4-yl)piperidine Hydrochloride
12/09/2004US20040248981 Excellent inhibitory activity against factor Xa; anticoagulants; blood coagulation disorder, thrombotic disease, cerebral infarction, myocardial infarction, or peripheral circulation disorder
12/09/2004US20040248949 carbocyclic carboxy nitriles such as 4-chloro-N-[2-({[(1S)-1-cyano-2-thien-3-ylethyl]amino}carbonyl)cyclohexyl]benzamide, used as cathepsin inhibitors; antimetastatic and antitumor agents; prophylaxis of cardiovascular and bone disorders
12/09/2004US20040248938 Substituted piperidines
12/09/2004US20040248937 protein tyrosine phosphatase inhibitors such as N-[(4-{[4,6-bis(4-methoxyphenyl)pyrimidin-2-yl]amino}phenyl)sulfonyl]-N-methyl-L-phenylalanine, used for treatment of metabolic disorders related to insulin resistance or hyperglycemia
12/09/2004US20040248935 crystals, crystal structured, liquid crystals and/or amorphous forms of 4-[4[4-(hydroxy diphenyl methyl)-1-piperidenyl]-1-hydroxy butyl]- alpha , alpha -dimethylphenyl acetic acid, hydrochloride salts, used as antihistamines, antiallergens or bronchodilator agents
12/09/2004US20040248872 Safe for agricultural or gardening use; effective against insects and mammals
12/09/2004US20040248854 Piperidinyl prostaglandin E analogs
12/09/2004US20040248820 Administering 2-phthalimidoglutaric acid; vision defects; antitumor agents; anticancer agents
12/09/2004DE10322191A1 N-sulfonylierte Aminosäurederivate, Verfahren zu ihrer Herstellung und ihre Verwendung N-sulfonylated amino acid derivatives, processes for their preparation and their use
12/09/2004CA2527722A1 Biodegradable poly(beta-amino esters) and uses thereof
12/09/2004CA2527632A1 Benzamide nitrile derivatives
12/09/2004CA2527197A1 4-amino-2(5h)-furanones useful as cholecystokinin antagonists
12/08/2004EP1483241A2 Cyclic derivatives as modulators of chemokine receptor activity
12/08/2004EP1483236A1 Aminoalcohol derivatives as beta-3 adrenergic receptor agonists
12/08/2004EP1482940A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
12/08/2004EP1482926A2 Amino-methyl substituted tetracycline compounds
12/08/2004EP1482924A2 Cathepsin cysteine protease inhibitors
12/08/2004EP1363898A4 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
12/08/2004EP1061076B1 N-acyl cyclic amine derivatives
12/08/2004CN1553898A Method for producing 4-haloalkylnicotinic acid esters
12/08/2004CN1553797A Carboxylate-gated-nitroxide (CGN) compounds and compositions and methods of use thereof
12/08/2004CN1552758A Preparation of sterically hindered amine ethers
12/08/2004CN1178927C Histamine H3 receptor ligands
12/08/2004CN1178922C Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
12/08/2004CN1178915C Alkynyl containing hydroxamic acid derivatives and its preparation and its use as matrix metalloproteinase (MMP) inhibitors/TNF-alpha converting enzyme (TACE) inhibitors
12/08/2004CN1178914C 4-benzyl-1-[2-(4-hydroxy-phenoxy)-ethyl]-piperidine-3,4-diol
12/08/2004CN1178911C Pyrrolidine and piperidine derivatives and their use for treatment of neurodegenerative disorders
12/08/2004CN1178906C N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
12/08/2004CN1178905C Novel peptide derivative
12/07/2004US6828342 Nitrate salts of Salbutamol, Cetirizine, Loratadine, Terfenadine, Emedastine, Ketotifen, Nedocromil, Ambroxol, Dextromethorphan, Dextorphan, Isoniazide, Erythromycin, and Pyrazinamide; respiratory system pathology treatment
12/07/2004US6828339 Amlodipine salt forms and processes for preparing them
12/07/2004US6828319 Substituted indeno[1,2-c]isoquinoline derivatives and methods of use thereof
12/02/2004WO2004103991A1 2-substituted piperidines, focused library and a pharmaceutical compound
12/02/2004WO2004103972A1 Novel piperidine derivative
12/02/2004WO2004103971A1 Cyclic aminophenyl sulfamate derivative