Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
08/2005
08/25/2005US20050186176 Compounds and compositions for delivering active agents
08/25/2005CA2555884A1 Amino-substituted tricyclic derivatives and methods of use
08/25/2005CA2554465A1 Piperidine derivatives useful as ccr3 antagonists
08/25/2005CA2552565A1 Aryloxyalkylcarbamate-type derivatives, preparation method thereof and use of same in therapeutics
08/24/2005EP1565192A2 Method and compositions for temporarily incapaciting subjets
08/24/2005EP1565178A2 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
08/24/2005EP1334085B1 Sulfamides as gamma-secretase inhibitors
08/24/2005EP1299349B1 Compounds to treat alzheimer's disease
08/24/2005EP1218341B1 Sulfonyl carboxamide derivatives, method for their production and their use as medicaments
08/24/2005EP1158980B1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
08/24/2005EP1019075B1 Beta 2-adrenergic receptor agonists
08/24/2005CN1659157A Terphenyl derivatives, preparation thereof, compositions containing same
08/24/2005CN1659131A (2-((2-alkoxy) -phenyl) -cyclopent-1-enyl) aromatic carbo and heterocyclic acid and derivatives
08/24/2005CN1658855A O-substituted hydroxyaryl derivatives
08/24/2005CN1216056C Sulfamato hydroxamic acid metalloprotease inhibitor
08/24/2005CN1216055C Paroxetine hydrochloride anhydrous compound and its preparation method and use
08/24/2005CN1216054C 1,4-dihydro pyridine-3,5-carboxylic-acid derivatives and preparation method thereof
08/23/2005US6933358 Functionalized monomers for synthesis of rubbery polymers
08/23/2005CA2370888C Renin inhibitors
08/23/2005CA2176360C Pharmaceutical emulsion
08/23/2005CA2064373C Piperidine derivatives
08/18/2005WO2005075455A2 Methods for making 4-tetrazolyl-4-phenylpiperidine compounds
08/18/2005WO2005075424A1 New pyridin-2-one compounds useful as inhibitors of thrombin
08/18/2005WO2005075423A1 Extracts of marasmins androsaceus l.es, piperdinone derivatives and the use as antihypertensive agents
08/18/2005WO2005075420A2 Pyrrolidine derivatives acting as ccr3-receptor antagonists
08/18/2005WO2005075410A1 New compounds, methods for their preparation and use thereof
08/18/2005WO2005075384A1 Process for production of aromatic compounds
08/18/2005WO2005074933A1 Small molecule inhibitors of her2 expression
08/18/2005WO2005074919A1 Diurea derivatives
08/18/2005WO2005074513A2 N-benzyl-3,4-dihyroxypyridine-2-carboxamide and n-benzyl-2,3-dihydroxypyridine-4-carboxamide compounds useful as hiv integrase inhibitors
08/18/2005WO2005046601A3 4-phenyl piperdine sulfonyl glycine transporter inhibitors
08/18/2005WO2005037755A3 Bridged ring structures as pharmaceutical agents
08/18/2005WO2005030794A3 Hemiasterlin derivatives and uses thereof
08/18/2005US20050182260 Reacting substituted or unsubstituted aniline with maleic acid, succinic acid or glutaric acid in presence of polyphosporic acid; cyclization; imidation; chemical intermediates for drugs
08/18/2005US20050182096 Haloalkyl containing compounds as cysteine protease inhibitors
08/18/2005US20050182095 Piperdine derivatives useful as CCR3 antagonists
08/18/2005US20050182094 N-[[4-(2-Chloro-4-fluorophenoxy)[1,4'-bipiperidin]-1'-yl]carbonyl]-4-methyl benzenesulfonamide, used for prophylaxis of respiratory system disorders or as antiallergens
08/18/2005US20050182068 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
08/18/2005US20050182040 Benzamide derivatives
08/18/2005US20050181455 aryl sulfonates and sulfates used for inhibiting bioadhesion to surfaces
08/18/2005US20050181232 White light-emitting OLED device including spaced anode and cathode, and having blue light-emitting and yellow, orange, or red light-emitting layers, the blue light-emitting layer including a monoanthracene derivative, stability
08/18/2005CA2720312A1 Methods for making 4-tetrazolyl-4-phenylpiperidine compounds
08/18/2005CA2555453A1 Cross-coupling process for production of aromatic compounds from aliphatic organic compounds and aromatic organometallic reagents
08/18/2005CA2554120A1 N-benzyl-3,4-dihydroxypyridine-2-carboxamide and n-benzyl-2,3-dihydroxypyridine-4-carboxamide compounds useful as hiv integras inhibitors
08/18/2005CA2553604A1 New pyridin-2-one compounds useful as inhibitors of thrombin
08/18/2005CA2552942A1 New compounds, methods for their preparation and use thereof
08/18/2005CA2552928A1 Pyrrolidine derivatives acting as ccr3-receptor antagonists
08/18/2005CA2551566A1 Diurea derivatives
08/17/2005EP1563821A1 Dental composition with light stability
08/17/2005EP1562986A2 Compounds and methods for modulating functions of classical cadherins
08/17/2005EP1562937A2 N-substituted piperidine derivatives as serotonin receptor agents
08/17/2005EP1562932A1 4-tetrazolyl-4-phenylpiperidine derivatives for treating pain
08/17/2005EP1562928A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors
08/17/2005EP1562925A1 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
08/17/2005EP1562906A2 Heterocyclic selective androgen receptor modulators and methods of use thereof
08/17/2005EP1562902A1 2-pyridone derivatives as inhibitors of neutrophile elastase
08/17/2005EP1562901A1 17beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
08/17/2005EP1562897A1 Phenylcarboxamide beta-secretase inhibitors for the treatment of alzheimer s disease
08/17/2005EP1562895A1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
08/17/2005EP1343761B1 Piperidine mch antagonists and their use in the treatment of obesity
08/17/2005EP1256575B1 Phenoxyalkylamine derivatives useful as opioid delta receptor agonists
08/17/2005EP1161240B1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
08/17/2005EP1140841B1 3-phenyl-2,6-dioxopiperidin-3-yl propionamide derivatives and method for preparing same
08/17/2005EP0993447B1 A process for the preparation of amlodipine benzenesulphonate
08/17/2005EP0894085B1 Benzyl(idene)-lactam derivatives, their preparation and their use as selective (ant)agonists of 5-ht1a- and/or 5-ht1d receptors
08/17/2005CN1656107A Plasma carboxypeptidase B inhibitors
08/17/2005CN1656071A New piperidine derivative
08/17/2005CN1656070A Melanocortin receptor ligands
08/17/2005CN1655785A N-acyl piperidine derivatives for use as melanocortin receptor ligands in the treatment of feeding disorders
08/17/2005CN1655777A A non-hormonal approach to male contraception
08/17/2005CN1655773A Compounds useful in the treatment of anthrax and inhibiting lethal factor
08/17/2005CN1215055C Arylsulfonamido-substituted hydroxamic acid derivatives
08/16/2005US6930200 Mono-and di-substituted alpha-amino acid derivatives useful as raw materials for pharmaceutical and agro-chemical products
08/16/2005US6930197 Preparing 4-(cyclopropylcarbonyl)benzene acetic acid ester; making intermediates useful for the synthesis of fexofenadine and related compounds
08/16/2005US6930186 Process for the preparation of paroxetine substantially free of alkoxy impurities
08/16/2005US6930106 Inhibitors of HCV NS5B polymerase
08/16/2005CA2166059C Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives
08/11/2005WO2005073192A1 Novel piperidines as chemokine modulators (ccr)
08/11/2005WO2005072735A1 Piperidinyl prostaglandin e analogs
08/11/2005WO2005053663A3 Norepinephrine reuptake inhibitors useful for treatment of cognitive failure
08/11/2005WO2005036961A3 N-substituted azacycles
08/11/2005US20050176962 Aminating a -cyanophenylalanine derivative with hydroxylamine hydrochloride in the presence of sodium carbonate in alcoholic-aqueous solution at reflux temperature to a 3-amidino derivative; chemical intermediates as highly efficient urokinase inhibitors
08/11/2005US20050176821 Meta-substituted phenylene sulphonamide derivatives
08/11/2005US20050176781 Process for the preparation of [S(-) amlodipine - L (+)- hemitartarate
08/11/2005US20050176780 2,5-disubstituted 3-mercaptopentanoic acid
08/11/2005US20050176775 Substituted pyridinones
08/11/2005US20050176766 2,3-Oxidosqualene-lanosterol cyclase inhibitors
08/11/2005US20050176760 and tumors; imino-, thiocarbonyl- or hydroxyimino-substituted N-heterocyclic amide compounds such as 2-(3-aminomethylphenylamino)-N-[3-chloro-4-(2-hydroxyiminopyrrolidin-1-yl)phenyl]-2-phenylacetamide
08/11/2005US20050176758 2-(hydroxy or methoxymethoxy)-4-(carboxy or alkoxycarbonyl)-5-(fluoro or hydrogen)-7-oxabicyclo(4.1.0)hept-3-ene chemical intermediates to neuraminidase inhibitors
08/11/2005US20050176757 For example, 6-[4-(4-Amino-5-chloro-2-methoxy-benzoylamino)-3-methoxy-piperidin-1-yl]-hexanoic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester; for treatment of gastrointestinal disorders including gastroparesis, gastroesophageal reflux
08/11/2005US20050176752 Such as 2,2,4-trimethyl-1,3-dioxolo[4,5-c]piperidin-7-ol; reacting methanesulfonic acid 6-hydroxy-2,2,6-trimethyl-tetrahydro-furo[3,4-d][1,3]dioxol-4-ylmethyl ester with phthalimide; avoids the use of reagents such as corrosive triflic anhydride and toxic sodium azide; intermediates to antivirals
08/11/2005US20050176731 N-[5-({(2S)-3-[(4-{4-[(4-benzylpiperidin-1-yl)carbonyl]phenyl}cyclohexyl)amino]-2-hydroxypropyl}oxy)-2-hydroxyphenyl]methanesulfonamide; beta 3 receptors agonist; gastrointestinal diseases; antiobesity, antidiabetic, cicatrizing agents, tocolytics, dysmenorrhea, antiglaucomatous; amidation
08/11/2005US20050176727 Male erectile dysfunction; 1-(3-chlorophenyl)-3-(4-pyridin-2-yl-piperazin-1-yl)propan-1-one O-methyloxime
08/11/2005US20050176708 Piperidine derivatives useful as modulators of chemokine receptor activity
08/11/2005CA2553387A1 Piperidinyl prostaglandin e analogs
08/11/2005CA2553089A1 Novel piperidines as chemokine modulators (ccr)
08/10/2005EP1560825A1 Novel 2,3-dihydro-4(1h)-pyridinone derivatives, method for production thereof and pharmaceutical composition comprising the same
08/10/2005EP1560814A1 Process for making risperidone and intermediates therefor
08/10/2005EP1560813A1 Novel piperidine derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
08/10/2005EP1560810A1 Bifunctional phenyliso(thio)cyanates; method and intermediate products for the production thereof