Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
07/2005
07/28/2005DE10360745A1 Neue Amid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel New amide compounds with MCH-antagonistic activity and pharmaceutical compositions containing them
07/28/2005CA2554382A1 Compounds useful in therapy
07/28/2005CA2552965A1 Carboxamide derivative and use thereof
07/28/2005CA2552550A1 Piperidine derivatives as gcs inhibitors
07/27/2005EP1556351A1 Secondary amino anilinic piperidines as mch1 antagonists and uses thereof
07/27/2005EP1556350A1 Process for the preparation of stabilizers for polymers
07/27/2005EP1556349A1 1,4-disubstituted piperidine derivatives and their use as 11-betahsd1 inhibitors
07/27/2005EP1556330A2 Phenyl compounds
07/27/2005EP1556046A1 Phenylpiperidines and phenylpyrrolidines as histamine h3 receptor modulators
07/27/2005EP1556045A1 4-aminopiperidine derivatives, processes for their preparation and their use as medicaments
07/27/2005EP1556029A2 Thiomolybdate analogues and uses thereof
07/27/2005EP1309555B1 Process for making amlodipine maleate
07/27/2005EP1274411B1 Phenylethylamines and condensed rings variants as prodrugs of catecholamines, and their use
07/27/2005EP1133489B1 Isonipecotamides for the treatment of integrin-mediated disorders
07/27/2005CN1646509A Piperazinyl- or piperidinylamine-sulfamic acid amides as inhibitors of steroid sulfatase
07/27/2005CN1646491A Compounds used to prepare camptothecin derivatives
07/27/2005CN1644208A China fir extracts with lycopodine A and B composition and their preparing method
07/26/2005US6921758 Amino acid derivatives
07/26/2005CA2315481C Selective inhibition of aggrecanase in osteoarthritis treatment
07/26/2005CA2286914C Process for producing 1-chlorocarbonyl-4-piperidinopiperidine or hydrochloride thereof
07/26/2005CA2193388C Aryl and heteroaryl alkoxynaphthalene derivatives
07/26/2005CA2137623C Phenyl-substituted 1,4-dihydropyridines
07/21/2005WO2005066181A1 Process for the preparation of 1,3-dioxolo [4,5-c] piperidin-7-ols and related compounds
07/21/2005WO2005066159A1 Cathepsin cysteine protease inhibitors
07/21/2005WO2005066128A1 Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
07/21/2005WO2005066127A1 Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
07/21/2005US20050159622 Reacting a primary or secondary amine with of SO3 or a source in the presence of a tert-amine and reacting the sulfamate formed with a phosphorus halide; the product may be reacted with NH3 to form the sulfamide, the NH2 group of which may then be acylated with a N-heterocycl-N-ylbenzoyl derivative
07/21/2005US20050159455 1,4-dihydropyridine and pyridine compounds as calcium channel blockers
07/21/2005US20050159452 Nociceptin analogs
07/21/2005US20050159451 NMDA (N-methyl-D-aspartate) receptors; eg 6-(4-benzylpiperidin-1-carbonyl)-1,5-dihydro-oxazolo[4,5-f]indole-2-one
07/21/2005US20050159450 Derivative of n-[phenyl(piperidin-2-yl)methyl]benzamide, the preparation method thereof and application of same in therapeutics
07/21/2005US20050159427 N-acylsulfonamide apoptosis promoters
07/21/2005US20050159416 Substituted urea derivatives activate the cardiac sarcomere by potentiating cardiac myosin; systolic heart failure including congestive heart failure; 1-[3-(1-Acetyl-piperidin-3-yloxy)-5-fluoro-phenyl]-3-(6-methoxy-pyridin-3-yl)-urea
07/21/2005US20050159407 Carboxylic acid substituted heterocycles, derivatives thereof and methods of use
07/21/2005US20050159405 Substituted 10-aryl-11h-benzo[b]fluourenes and 7-aryl-5, 6-dihydro-benzo[a]anthracenes for selective effects on estrogen receptors
07/21/2005US20050159402 Polyarylcarboxamides useful as lipid lowering agents
07/21/2005US20050156753 Digital sound processing system for a vehicle
07/21/2005DE4120550B4 Verfahren zur Herstellung eines gereinigten N,N'-Bis-(2,2,6,6-tetramethyl-4-piperidyl) -alkandiamins A process for producing a purified N, N'-bis (2,2,6,6-tetramethyl-4-piperidyl) -alkandiamins
07/21/2005CA2552946A1 Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
07/21/2005CA2552850A1 Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
07/21/2005CA2552726A1 Cathepsin cysteine protease inhibitors
07/20/2005EP1554267A1 Dihydropyridine compounds having simultaneous ability to block l-type calcium channels and to inhibit phosphodiesterase type 3 activity
07/20/2005EP1554260A1 Aryloxyalkylamine derivatives as h3 receptor ligands
07/20/2005EP1554247A2 Process for the preparation of (s,s)-cis-2-phenyl-3-aminopiperidine
07/20/2005EP1554246A2 Dihydropyridinone derivatives as hne inhibitors
07/20/2005EP1554245A1 Piperidinetriol derivatives as inhibitors of glycosylceramidsynthase
07/20/2005EP1554242A1 Watersoluble prodrugs of propofol
07/20/2005EP1553937A2 Glycinenitrile-based inhibitors of dipeptidyl peptidase iv and methods
07/20/2005EP1175402B1 Piperidine derivatives useful as ccr5 antagonists
07/20/2005EP1175401B1 Piperazine derivatives useful as ccr5 antagonists
07/20/2005CN1642948A Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642915A Benzamide derivatives useful as histone deacetylase inhibitors
07/20/2005CN1642914A Certain 1-(D-cyclopropylglycinyl)-4-(piperidin-4-yl)piperazine compounds as inhibitors of the serine protease factor XA
07/20/2005CN1642913A Piperidine or 8-aza-bicyclo[3.2.1]oct-3-yl derivatives useful as modulators of chemokine receptor activity (especially CCR5)
07/20/2005CN1642912A Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642907A Carbonylamino-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642906A Novel arylamidine derivative or salt thereof
07/20/2005CN1642551A Inhibitors of histone deacetylase
07/20/2005CN1642535A Tuberculosis treatment using pleuromutilin derivatives
07/20/2005CN1211366C Methyl sulfonate trihydrate of 1-(4-hydroxy phenyl)-2-(4-hydroxy-4-phenyl piperid-1-yl)-1-propanol and its intermidiate preparing process
07/20/2005CN1211353C Unsaturated hydroximic acid derivatives as PARP inhibitors
07/19/2005US6919482 A 1,4-bis(N-(2-(4-hydroxy-3-hydroxymethylphenyl) -2-hydroxyethyl)amino)-cyclohexane or alkyl-cyclohexane or -pyrazine derivatives; treating respiratory diseases disorders, asthma, bronchitis, nervous system injury
07/19/2005US6919481 Alkoxyamines containing a vinyl group, their applications and methods of their production
07/19/2005US6919458 Preparation of terfenadine carboxylic acid metabolite and carebastine using a 1-(2-substituted isopropyl)-4-(cyclopropylcarbonyl)-benzene compound intermediate
07/19/2005US6919451 Synthesis of 4,5-dihydro-pyrazolo [3,4-c] pyrid-2-ones
07/19/2005US6919368 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
07/19/2005US6919367 Substituted thioacetamides
07/19/2005US6919356 Antihistamines, antiallergens, autoimmune disease, antiinflammatory agents
07/19/2005US6919355 Amide derivatives as NMDA receptor antagonists
07/19/2005US6919336 Hallogenated aminobenzophenones and aminobenzoylpyridines as inhibitors of IL-1 and TNF
07/14/2005WO2005064336A1 Pyrenyloxysulfonic acid fluorescent agents
07/14/2005WO2005063714A1 Analogs of benzoquinone-containing ansamycins for the treatment of cancer
07/14/2005WO2005063707A1 Enantiospecific process for the preparation of paroxetine intermediate
07/14/2005WO2005063706A1 Synthesis of nojirimycins
07/14/2005WO2005063705A1 Benzene compounds disubstituted with cyclic groups at the 1- and 2-positions
07/14/2005WO2005063704A1 Azetidine ring compounds and drugs comprising the same
07/14/2005WO2005063697A2 Substituted n-aryl amidines as selective d1 dopamine receptor antagonists for the treatment of obesity and cns disorders
07/14/2005WO2005063680A1 Process for the preparation of arylamines
07/14/2005WO2005063678A1 Process for producing phenylacetic acid derivative
07/14/2005WO2005063239A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders
07/14/2005WO2005063222A1 Hsp90 FAMILY PROTEIN INHIBITOR
07/14/2005WO2005046612A3 Hydroxy piperidine derivatives to treat gaucher disease
07/14/2005US20050154206 Adjusting pH of solution to generate nitrosonium ion and protonated hydroxylamine, removing solvent, then neutralizing
07/14/2005US20050154022 Selective antagonists for melanin concentrating hormone-1 (MCH1) receptors; antidepressants, anxiolytic agents; bipolar, eating, psychological, urogenital, and obsessive-compulsive disorders; phobias, post-traumatic stress disorder
07/14/2005US20050154021 N-and O-substituted 4-[2-(diphenylmethoxy)-ethyl]-1-[(phenyl)methyl]piperidine analogs and methods of treating CNS disorders therewith
07/14/2005US20050154020 4-Aryl piperidines
07/14/2005US20050154019 Substituted cyclic amine metalloprotease inhibitors
07/14/2005US20050154017 Novel azasugar derivative and drug containing the same as the active ingredient
07/14/2005US20050154011 such as S)-3-Methylcarbamoyl-7-sulfoamino-3,4-dihydro-1H-isoquinoline-2-carboxylic acid tert-butyl ester, used in the treatment of protein tyrosine phosphatase (PTPase) mediated disorder such as diabetes
07/14/2005US20050153996 Compounds that modulate ppar activity and methods for their preparation
07/14/2005US20050153963 exhibit a particular activity as specific inhibitors of the glycine transporters glyt1 and/or glyt2
07/14/2005US20050153456 Analysis of mass spectral data in the quiet zones
07/14/2005CA2550679A1 Substituted n-aryl amidines as selective d1 dopamine receptor antagonists for the treatment of obesity and cns disorders
07/14/2005CA2550649A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders
07/13/2005EP1553085A1 Cyclic amine derivatives and their use as drugs
07/13/2005EP1553084A1 Piperidine derivative, process for producing the same, and use
07/13/2005EP1553074A1 Fused benzene derivative and use
07/13/2005EP1552834A1 Neurotrophic factor production promoter
07/13/2005EP1551827A1 Piperidine derivatives as ccr5 inhibitors
07/13/2005EP1551805A1 Substituted gamma-phenyl-delta-lactams and uses related thereto