Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
07/2005
07/13/2005EP1551804A1 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
07/13/2005EP1551798A1 Novel sulphones for inhibition of gamma secretase
07/13/2005EP1551797A1 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors
07/13/2005EP1551795A1 Inhibitors of histone deacetylase
07/13/2005EP1235802B1 Carbamate derivatives having muscarinic receptor antagonist activity
07/13/2005EP1161415B1 N-cyanomethylamides as protease inhibitors
07/13/2005CN1639159A N-aminoacetyl-pyrrolidine-2-carbonitriles and their use as DDP-IV inhibitors
07/13/2005CN1639147A Synthesis of 4, 5-dihydro-pyrazolo [3, 4-c] pyrid-2-ones
07/13/2005CN1639142A Method for producing 3-amidinophenylalanine derivatives
07/13/2005CN1639125A New inhibitors of histone deacetylase
07/13/2005CN1639124A Aminotetralin derivatives as muscarinic receptor antagonists
07/13/2005CN1639123A 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derativatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
07/13/2005CN1638757A 组织蛋白酶半胱氨酸蛋白酶抑制剂 Cathepsin cystatin
07/13/2005CN1636993A Process for producing novel form of paroxetine hydrochloride anhydrate
07/13/2005CN1636986A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636985A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636984A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636980A 二肽腈组织蛋白酶k抑制剂 Dipeptide nitrile cathepsin inhibitors k
07/13/2005CN1636979A Method for separating cis-3, 5-dimethylpiperidine from a mixture of its geometrical isomers
07/13/2005CN1636976A Mutilin derivatives and their use as antibacterials
07/13/2005CN1636565A Modified form of the r(-)-n-(4, 4-di(3-methylthien-2-yl)but-3-enyl)-nipecotic acid hydrochloride
07/13/2005CN1210274C Piperazine and piperidine derivatives
07/13/2005CN1210268C (Cyclo) alkyl substituted-gamma-aminobutyric acid derivatives (=GABA analogurs), their preparation and their use in the treatment of neurolog disorders
07/13/2005CN1210263C N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
07/13/2005CN1210262C Method for preparing methylsulfonate trihydrate of 1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperid-1-yl)-1-propanol
07/13/2005CN1210261C Arylpiperidine and aryl-1,2,5,6-tetrahydropyridine amide derivatives having 5HT1A receptor activity
07/12/2005US6916957 Antiinflammatory agents; antihistamines; antiallergens
07/12/2005US6916929 Via hydrolysis of 1-benzyl-4-cyano-4-phenylpiperidine in acidic medium; for tachykinin antagonist drugs
07/12/2005US6916850 Pyruvate derivatives
07/12/2005US6916833 Substituted piperidines
07/12/2005US6916830 Substituted tetrahydroisoquinolines as C5a receptor modulators
07/12/2005US6916829 Method for enhancing mutant enzyme activity in gaucher disease
07/12/2005US6916822 For preventive and/or therapeutic treatment of nerve system diseases including schizophrenia, depression, cerebral apoplexy, epilepsy, Alzheimer's disease, and Parkinson's disease
07/12/2005US6916817 Inhibitors of metalloproteinases
07/12/2005CA2137525C Isopropyl 2-methoxyethyl 4-(2-chloro-3-cyano-phenyl)-1,4-dihydro-2,6-dimethyl-pyridine-3,5-dicarboxylate
07/09/2005CA2455018A1 Process for the preparation of piperidine derivatives
07/07/2005WO2005061483A2 Modulators of peripheral 5-ht receptors
07/07/2005WO2005061470A1 1-akan-2-ol substituted piperazine and piperidine compounds
07/07/2005WO2005061457A1 Organic compounds
07/07/2005WO2005061453A1 Antharquinone compounds as anti cancer compounds
07/07/2005WO2005061442A1 Opioid receptor antagonists
07/07/2005WO2005060947A2 Agonist and antagonist ligands of the nociceptin receptor
07/07/2005WO2005060603A2 Nitric oxide releasing pyruvate compounds, compositions and methods of use
07/07/2005WO2005049593A3 N-acylsulfonamide apoptosis promoters
07/07/2005WO2005042521A3 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
07/07/2005WO2005037782A3 Derivatives of n-[phenyl(alkylpiperidine-2-yl)methyl]benzamide, preparation method thereof and application of same in therapeutics
07/07/2005US20050148637 Neurotrophic low molecular weight ketones and tioester compounds for treatment of nervous system disorders and neurodegenerative conditions
07/07/2005US20050148629 Hydroxyamidealkylsulfonamide compounds for anthrax treatment
07/07/2005US20050148613 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
07/07/2005US20050148595 heterocylcyclic amines used for treating or preventing conditions ameliorated by monoamine reuptake such as vasomotor symptoms, sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders
07/07/2005US20050148588 LFA-1 antagonist compounds
07/07/2005US20050148584 N-(3-(2-(4-morpholino)ethyloxy)phenyl)-N-{(cis3-(benzylamino)cyclohexyl)methyl}-N'-phenylurea; useful for the treatment of gastrointestinal reflux disorders, eating disorders leading to obesity and irritable bowel syndrome
07/07/2005US20050148583 1-[2-[2-(4-Diethylcarbamoylbenzyl)phenoxy]ethyl]-4-(1,3-dihydro-2H-benzimidazol-2-on-1-yl)piperidine; agonist, antagonist, partial or inverse agonist; schizophrenia, depression, cerebral apoplexy, epilepsy, Alzheimer's disease, and Parkinson's disease; analgesic; pharmacokinetics
07/07/2005US20050146263 Liquid crystalline emitter and charge-transport materials for use in organic light emitting devices (OLED); photopolymerization; high luminous output; tetra-enes based on a fluorene ring skeleton and having at least one heterocyclic ring attached
07/07/2005DE10358539A1 Carbonsäureamidderivate Carboxamide
07/07/2005CA2550839A1 Antharquinone compounds as anti cancer compounds
07/07/2005CA2550257A1 1-akan-2-ol substituted piperazine and piperidine compounds
07/07/2005CA2549412A1 Nitric oxide releasing pyruvate compounds, compositions and methods of use
07/07/2005CA2549009A1 Opioid receptor antagonists
07/06/2005EP1549617A1 Organic acid salt of amlodipine
07/06/2005EP1549616A1 Organic acid salt of amlodipine
07/06/2005EP1549615A1 Naphthamide derivatives and their use
07/06/2005EP1549600A1 Ketones
07/06/2005EP0776327B1 New multimerizing agents
07/06/2005CN1634887A Process for chiral synthesis of (2S, 6R)-2, 6-dialkyl piperidine hydrochloride
07/06/2005CN1209351C N-(4-aryloxypiperidin-1-ylalkyl) cinnamic amides as CCR3 receptor antagonists
07/05/2005US6914142 Antiinflammatory agents; rheumatic diseases
07/05/2005US6914079 Antiproliferative agents; anticancer agents
07/05/2005US6913674 Process for fractionating water-containing crude amine mixtures from amine synthesis
07/05/2005CA2309485C New 4-arylpiperidine derivatives for the treatment of pruritus
07/05/2005CA2230082C Amide compounds and use thereof
07/05/2005CA2165446C Use of ropivacaine in the manufacture of a pharmaceutical with analgetic effect with minimal motor blockade
07/05/2005CA2119572C Oxygen substituted derivatives of nucleophile-nitric oxide adducts as nitric oxide donor prodrugs
07/05/2005CA2064382C Pharmaceutical compounds
06/2005
06/30/2005WO2005059037A1 Reagent for detecting an analyte
06/30/2005WO2005058972A1 Process for the oxidation of hydroxy compounds by means of nitroxy compounds
06/30/2005WO2005058885A2 Piperidine derivatives and their use as glycine transporter inhibitors
06/30/2005WO2005058884A2 Cyclopropane compounds and pharmaceutical use thereof
06/30/2005WO2005058826A1 New 5,6-dihydropyrin-2-one compounds useful as inhibitors of thrombin
06/30/2005WO2005058825A1 Amlodipine gentisate and a method of its preparation
06/30/2005WO2005058824A2 N-aryl piperidine substituted biphenylcarboxamides as inhibitors of apolipoprote in b
06/30/2005WO2005058822A1 Substituted amino-cycloalkanes
06/30/2005WO2005058818A1 Process for the recovery of nitroxy compounds from organic solutions and oxidation process
06/30/2005WO2005058808A1 N-substituted-n-sulfonylaminocyclopropane compounds and pharmaceutical use thereof
06/30/2005WO2004100960A8 Anti-inflammatory phosphonate compounds
06/30/2005WO2004096236A3 Immunomodulator phosphonate conjugates
06/30/2005WO2004089926A3 Genipin derivatives and uses thereof
06/30/2005WO2004055006A8 Novel compounds having selective inhibiting effect at gsk3
06/30/2005US20050143579 for the prevention and treatment of conditions ameliorated by monoamine reuptake including, inter alia, vasomotor symptoms (VMS), sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders
06/30/2005US20050143539 Polymerizable composition with free radicals and by controlling polymerization
06/30/2005US20050143456 Carboxamide-substituted phenylurea derivatives, process for their preparation and their use as medicaments
06/30/2005US20050143426 Osteoporosis, bone disorders, or diseases associated with excessive secretion of PTH, such as hyperparathyroidism; reduce or inhibit parathyroid hormone (PTH) secretion
06/30/2005US20050143419 Guanidine and amidine derivatives as factor Xa inhibitors
06/30/2005US20050143372 Compounds, pharmaceutical compositions and methods of use therefor
06/30/2005CA2550012A1 Urea derivative, process for producing the same and use
06/30/2005CA2549741A1 Reagent for detecting an analyte
06/30/2005CA2549660A1 Cyclopropane compounds and pharmaceutical use thereof
06/30/2005CA2549598A1 N-substituted-n-sulfonylaminocyclopropane compounds and pharmaceutical use thereof
06/30/2005CA2548793A1 5- or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication
06/30/2005CA2547064A1 New 5,6-dihydropyrin-2-one compounds useful as inhibitors of thrombin