Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
07/2003
07/24/2003WO2003059898A2 Eponemycin and epoxomicin analogs and uses thereof
07/24/2003WO2003059875A2 DERIVATIVES OF α-PHENYLTHIOCARBOXYLIC AND α-PHENYLOXY-CARBOXYLIC ACIDS USEFUL FOR THE TREATMENT OF DISEASES RESPONDING TO PPARα ACTIVATION
07/24/2003WO2003059865A1 Processes for the preparation of glutamic acid compounds and intermediates thereof and novel intermediates used in the processes
07/24/2003WO2003059864A2 Pheny(alkyl)carboxylic acid derivatives and dionic phenylalkylheterocyclic derivatives and their use as medicines with serum glucose and/or serum lipid lowering activity
07/24/2003WO2003059807A2 Crystalline solids of carvedilol and processes for their preparation
07/24/2003US20030139630 Organic compound in liquid or dissolved form is mixed with formylation reagent in liquid or dissolved form in microreactor; efficiency, simplification
07/24/2003US20030139628 Process for the preparation of optically active amines or salts thereof
07/24/2003US20030139609 Aziridinyl quinone antitumor agents based on indoles and cyclopent[b]indoles
07/24/2003US20030139605 Antiproliferative agents, treating or preventing osteoporosis, inflammation, and angiogenesis disorders, treating liver cancer
07/24/2003US20030139475 Novel tricyclic compounds and drug compositions containing same
07/24/2003US20030139464 Reduction of carbonyl compounds using the carbonyl reductase of kluyveromyces marxianus
07/24/2003US20030139453 Difluorobutyric acid metalloprotease inhibitors
07/24/2003US20030139449 Anxiolytic agents; psychological disorders; cognition activators
07/24/2003US20030139424 Dietetic therapy
07/24/2003US20030139404 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents
07/24/2003US20030139388 Antiinflammatory agents; osteoporosis
07/24/2003US20030139379 Autoimmune disease, osteoporosis, rheumatic diseases, skin disorders
07/24/2003US20030139348 Animal growth regulators
07/24/2003US20030138376 A compressed tablets comprising an embedded polymer matrix, insoluble and disintegrable in the solvents, removed by filtration, separation from a formed soluble product
07/24/2003CA2472419A1 Coumarin derivatives, process for their production and use thereof
07/24/2003CA2472377A1 Crystalline solids of carvedilol and processes for their preparation
07/24/2003CA2472223A1 Derivatives of alpha-phenylthiocarboxylic and alpha-phenyloxy-carboxylic acids useful for the treatment of diseases responding to pparalpha activation
07/24/2003CA2472209A1 Pheny(alkyl)carboxylic acid derivatives and dionic phenylalkylheterocyclic derivatives and their use as medicines with serum glucose and/or serum lipid lowering activity
07/23/2003EP1328550A2 Methods of selecting compounds for modulation of bladder function
07/23/2003EP1328525A2 2,3,4,5-tetrahydro-1h-[1,4]diazepino[1,7-a]indole compounds
07/23/2003EP1328515A1 Indoline derivatives and their use as 5-ht2 receptor ligands
07/23/2003EP1328514A1 Amide derivatives as nmda receptor antagonists
07/23/2003EP1328513A2 Diindolylmethane and c-substituted diindolylmethane compositions and methods for the treatment of multiple cancers
07/23/2003EP1328510A2 Carbamic acid compounds comprising a sulfonamide linkage as hdac inhibitors
07/23/2003EP0983274B1 Phthalocyanine and use of phthalocyanine as a marking agent
07/23/2003EP0888278B1 Antidiabetic agents
07/23/2003CN1431999A Indole derivatives with vascular damagine activity
07/23/2003CN1431998A Growth hormone secretagogues
07/23/2003CN1431997A 2-acyl indol derivatives and their use as anti-tumour agents
07/23/2003CN1431996A C2 phenyl-substituted cyclic keto-enols used as pesticides and herbicides
07/23/2003CN1431901A S-methyl-dihydro-zipprasidone for treatment of psychiatric and ocular disorders
07/23/2003CN1431197A Alanine class compound, its preparing method and use
07/23/2003CN1115343C Process for prepn. of (1S,4R)-or (1R,4S)-4-(2-amino-6-chloro-9H-purin-9-yl) -2-cyclopentene-1-methanol
07/23/2003CN1115330C N-(4-carbamimido-phenyl)-phenylglycinamid derivatives
07/22/2003USRE38200 Indole-2,3-dione-3-oxime derivatives
07/22/2003US6596877 Reaction with dimethyl carbonate using 4-(dimethylamino)pyridine, 1,4-diazabicyclo(2.2.2)octane, or 1,8-diazabicyclo(5.4.0)undec-7-ene basic catalyst
07/22/2003US6596873 2-and 2,5-substituted phenylketoenols
07/22/2003US6596772 Relates to trifluoromethyl sulfonyl and trifluoromethyl sulfonamido compounds and the physiologically acceptable salts and the prodrugs thereof. These compounds are expected to modulate the activity of protein tyrosine enzymes which are
07/22/2003US6596753 Compounds of the indolecarboxylic family and use thereof
07/22/2003US6596752 Inhibitors of α4β1 mediated cell adhesion
07/22/2003US6596732 1,3-dihydro-2h-indol-2-one, preparation method and pharmaceutical compositions containing same
07/22/2003US6596522 Compositions and optical methods for determining transmembrane potentials across plasma membrane of biological cells
07/22/2003US6596130 Using ionic liquids as solvents resulted in high yields with dramatically reduced reaction times
07/22/2003CA2245250C Benzofuran-acrylic acid derivatives and their use as modulators of rxrs or rars receptors
07/17/2003WO2003059014A1 Bis- and tris-(di)benzocarbazole-based materials as hole transport materials for organic light emitting devices
07/17/2003WO2003057697A1 Derivatives of 5-(pyridin-3-yl)-1-azabicyclo[3.2.1]octane, the preparation thereof and the application of same in therapeutics
07/17/2003WO2003057670A2 Indoles as naaladase inhibitors
07/17/2003WO2003057666A2 Inhibitors of dipeptidyl peptidase iv
07/17/2003WO2003057254A1 Preventives/remedies for urinary disturbance
07/17/2003WO2003057212A1 Polyamide derivatives possessing antibacterial, antifungal or antitumor activity
07/17/2003WO2003057169A2 4-dedimethylamino tetracycline compounds
07/17/2003WO2003057144A2 Change inhibitors of dipeptidyl peptidase iv
07/17/2003WO2002006280A3 INHIBITORS OF FACTOR Xa
07/17/2003US20030135051 Intermediates for making HIV-protease inhibitors and methods for making HIV-protease inhibitors
07/17/2003US20030135049 Preparing camptothecin intermediates
07/17/2003US20030134876 Inhibiting TNF alpha
07/17/2003US20030134863 Preventives/remedies for alzheimer's disease
07/17/2003US20030134827 Lactams or pharmaceutically acceptable salt forms thereof, wherein rings ring B is a 4-8 membered cyclic amide containing from 0-3 additional heteroatoms selected from N, O, and S, which are useful as metalloprotease inhibitors.
07/17/2003US20030131425 Colorants
07/17/2003CA2471760A1 Preventives/remedies for urinary disturbance
07/17/2003CA2471204A1 Inhibitors of dipeptidyl peptidase iv
07/16/2003EP1327636A2 Heterocyclic metallocenes and polymerisation catalysts
07/16/2003EP1326993A2 PRODUCTION OF g(a)-HYDROXY-CARBOXYLIC ACIDS USING A COUPLED ENZYME SYSTEM
07/16/2003EP1326867A2 Bridged piperazine derivatives
07/16/2003EP1326842A1 Arylpiperazine derivatives and their use as psychotropic agents
07/16/2003EP1326831A1 Substituted fused pyrroleimines and pyrazoleimines
07/16/2003EP1326830A1 2-, 3-, 4-, or 5-substituted-n1-(benzensulfonyl)indoles and their use in therapy
07/16/2003EP1326651A2 Dynamic organ function monitoring agents
07/16/2003EP1326650A2 Hydrophilic light absorbing compositions for determination of physiological function in critically ill patients
07/16/2003EP1326649A1 Tissue-specific exogenous optical agents
07/16/2003EP1326648A1 Novel dyes for organ function monitoring
07/16/2003EP1326623A1 Saururus chinensis extract for prevention and treatment of neurodegenerative disease
07/16/2003EP1326602A1 Indole compounds as minimally physiologial function monitioring agents
07/16/2003EP1326597A2 Methods for modulating bladder function
07/16/2003EP1076558B1 2-phenyl-1-[-(2-aminoethoxy)-benzyl -indole in combination with estrogens
07/16/2003CN1430607A Benzophenones as inhibitors of IL-1 beta and TNF-alpha
07/16/2003CN1430605A Process for synthesis of amine ethers from secondary amino oxides
07/16/2003CN1430604A Process for preparation of indole derivatives and intermediates of the process
07/16/2003CN1430603A Novel bicyclic compounds
07/16/2003CN1114608C Novel camptothecine analogues, prepn. method therefor, use thereof, and pharmaceutical compositions contg. same
07/15/2003US6593474 Adrenergic blocking agents
07/15/2003US6593347 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use
07/15/2003US6593327 Compounds and compositions as protease inhibitors
07/15/2003US6593322 Compounds and methods for modulation of estrogen receptors
07/15/2003US6593312 Cyclic α-amino-γ-hydroxyamide compounds
07/15/2003US6593148 Cyanine dye compounds and labeling methods
07/15/2003US6592894 Hydrogel-isolated cochleate formulations, process of preparation and their use for the delivery of biologically relevant molecules
07/10/2003WO2003055884A1 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino[4,5-b]indole-1-carboxamide derivatives, their preparation and therapeutic use
07/10/2003WO2003055848A2 Urea derivatives as vr1- antagonists
07/10/2003WO2003055847A1 Carboxylic acid derivative
07/10/2003WO2003055492A1 Use of oxindole derivatives in the treatment of dementia related diseases, alzheimer's disease and conditions associated with glycogen synthase kinase-3
07/10/2003WO2003055484A1 Urea derivatives
07/10/2003WO2003055478A1 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders
07/10/2003WO2003032908A3 Novel prodrugs of n-h bond-containing compounds and methods of making thereof
07/10/2003WO2003010140A3 Hepatitis c virus polymerase inhibitors with heterobicyclic structure