Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
05/2005
05/25/2005EP1532105A1 Anthranyl derivatives having an anticholecystokinin activity (anti-cck-1), a process for their preparation, and pharmaceutical use thereof
05/25/2005EP1531807A1 Bazedoxifene treatment regimens
05/25/2005EP1442016A4 1h-indole derivatives as a highly selective cyclooxygenase-2 inhibitor
05/25/2005EP1259231B1 Naphthoquinone derivatives as cd45 inhibitors
05/25/2005EP1140814B1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
05/25/2005EP1039911B1 MORPHOLINO-N-ETHYL ESTER PRODRUGS OF INDOLE sPLA 2 INHIBITORS
05/25/2005DE10347383A1 New 1-amino-tetrahydronaphthalene derivatives, useful for treatment of e.g. inflammation, bind with high selectivity to glucocorticoid receptors
05/25/2005CN1620429A Derivatives of alpha-phenylthiocarboxylic and g(a)-phenyloxy-carboxylic acids useful for the treatment of diseases responding to PPAR alpha activation
05/25/2005CN1620313A Method of examining effect of angiogenesis inhibitors mediated by the inhibition of integrin expression
05/24/2005US6897276 Coordination polymerization catalyst for alpha-olefins
05/24/2005US6897240 Thio semicarbazone and semicarbazone inhibitors of cysteine proteases and methods of their use
05/24/2005US6897237 MMP-12 inhibitors
05/24/2005US6897207 Kinase inhibitors; angiogenesis inhibitors, anticancer agents, antiinflammatory agents and chronic obstructive pulmonary disease inhibitors
05/24/2005CA2174000C Process for the preparation of a substituted 2,5-diamino-3-hydroxyhexane
05/21/2005CA2486838A1 Organic amine salts of glutamic acid derivatives and their application
05/19/2005WO2005044923A1 Cyanine dye labelling reagents
05/19/2005WO2005044796A1 2-halogen-6-alkyl-phenyl substituted spirocyclic tetramic acid derivatives
05/19/2005WO2005044261A1 Melatonin analogue prodrugs
05/19/2005WO2005044260A1 Use of crth2 antagonist compounds in therapy
05/19/2005WO2005028436A3 Thalidomide analogs as tnf-alpha modulators
05/19/2005WO2005016868A3 Matrix metalloproteinase inhibitors
05/19/2005WO2004041780A3 N-(indole-2-carbonyl) amides as anti-diabetic agents
05/19/2005US20050107618 Processes for the preparation of N-substituted phthalimides
05/19/2005US20050107543 Fluoro linkers and their use as linkers for enzyme-activated drug conjugates
05/19/2005US20050107463 Novel prostamides for the treatment of glaucoma and related diseases
05/19/2005US20050107458 used as diagnostic kits, bioassay and/or drugs for preventing cancers, Alzheimer's disease, amyotrophic lateral sclerosis, Parkinson's disease, stroke, ischaemia, Huntington's disease, epilepsy, multiple sclerosis, neuropathy, or injuries of the brain or spinal chord, or as tyrosine kinase inhibitors
05/19/2005US20050107445 Active compounds with carbamic acid for diseases such as cancer, leukemia, atheriosclerosis, alzheimers disease or arthritis
05/19/2005US20050107362 Indolamid derivatives which possess glycogenphosphorylase inhibitory activity
05/19/2005US20050107321 FLK-1 is a receptor for vascular endothelial growth factor
05/19/2005US20050107258 Auxinic analogues of indole-3-acetic acid
05/19/2005US20050106709 First reactive functional group used to provide attachment to a surface of a substrate, second reactive functional group is a N-sulfonyldicarboximide group reacted with an amine-containing material, to form a connector group between the substrate and amine containing material (protein, peptide, dna rna)
05/19/2005US20050106106 In-vivo diagnostic method by near infrared radiation
05/19/2005DE10347386A1 New 1-amino-tetrahydronaphthalene derivatives, useful for treatment of e.g. inflammation, bind with high selectivity to glucocorticoid receptors
05/19/2005DE10346939A1 New arylalkanol derivatives used for treating e.g. respiratory diseases, joint diseases, vascular inflammations, skin disorders, kidney and liver diseases and neurological diseases
05/19/2005CA2544752A1 Bicyclic pyrazolyl and imidazolyl compounds and uses thereof
05/19/2005CA2544548A1 2-halogen-6-alkyl-phenyl-substituted tetramic acid derivatives
05/19/2005CA2544537A1 2-halogen-6-alkyl-phenyl substituted spirocyclic tetramic acid derivatives
05/19/2005CA2543199A1 Use of crth2 antagonist compounds in therapy
05/18/2005EP1530572A2 Analogs of indole-3-carbinol metabolites as chemotherapeutic and chemopreventive agents
05/18/2005EP1530564A2 Compounds derived from aryl carbamates, preparation thereof and uses of same
05/18/2005EP1317430B1 (2-azabicyclo [2.2.1]hept-7-yl)methanol derivatives as nicotinic acetylcholine receptor agonists
05/18/2005EP1263724B1 Novel compounds
05/18/2005EP1176139B1 Medicinal compositions with 2.2.1] and 3.1.1] bicycloskeleton antagonistic to both of pgd 2?/txa 2? receptors
05/18/2005EP0946173B1 Preparation of 3-fluoro oxindole derivatives
05/18/2005CN1617865A Phenylalkynes
05/18/2005CN1617860A [1.2]-oxazin-3, 5-diones
05/18/2005CN1617855A Inhibitors of cytosolic phospholipase A2
05/18/2005CN1617854A Pheny(alkyl)carboxylic acid derivatives and dionic phenylalkylheterocyclic derivatives and their use as medicines with serum glucose and/or serum lipid lowering activity
05/18/2005CN1617718A N-aryl-N'-arylcycloalkyl-urea derivatives as MCH antagonists for the treatment of obesity
05/18/2005CN1616455A Processes for producing 7-isoindoline-quinolonecarboxylic acid derivative and its intermediate
05/18/2005CN1616428A Acenaphthene heterocyclic compound and its cell fading inducing and anti-tumor use
05/18/2005CN1616427A New method for preparing medicine mitiglinide for treating diabetes
05/18/2005CN1616426A Indolyl styrene salt compound, high density recording medium including said compound and its preparing method
05/18/2005CN1616425A Noval benzoindoline compounds, their preparing method and pharmaceutical composition containing them
05/18/2005CN1616386A Intermediate for preparing isothiazole derivatives
05/18/2005CN1202093C Substituted heterocyclic compound
05/18/2005CN1202052C Enantioselective reduction of ketones with silane agent/metal compound/chiral ligand system
05/18/2005CN1201735C Mycobacterial inhibitors
05/17/2005US6894185 Substituted chiral allosteric hemoglobin modifiers
05/17/2005US6894174 Water-soluble polyimides and methods of making and using same
05/17/2005US6894072 Compounds as NS3-serine protease inhibitors of hepatitis C virus
05/17/2005US6894070 Herbicides
05/17/2005US6894005 Heterocyclic compound containing phenyl groups; postemergence herbicides
05/17/2005US6893650 Fungicides; locus infestation; such as N,N-dimethyl-N'-(4-(3-trifluoromethylbenzylthio)-2,5-xylyl)formamidine
05/17/2005CA2347757C Method for producing (+)-exo-6-phenyl-3-azabicyclo-[3.2.0]heptanes
05/17/2005CA2103845C 9-[(substituted glycyl)-amido]-6-demethyl-6-deoxytetracyclines
05/12/2005WO2005042513A1 Phenyl carboxamide and sulfonamide derivatives for use as 11-beta-hydroxysteroid dehydrogenase
05/12/2005WO2005042497A2 Benzimidazoles useful as modulators of ion channels
05/12/2005WO2005042469A1 Aromatic amino acid labeled with stable isotope, method for incorporating the same into target protein and method for analyzing protein structure using nmr
05/12/2005WO2005041954A1 Indirubin-type compounds, compositions, and methods for their use
05/12/2005WO2005019169A3 Indoline derivatives as ppar-delta modulators
05/12/2005WO2005018531A3 Pharmaceutical compositions, azo-heterocyclic compounds and method for the production and use thereof
05/12/2005WO2005000803A8 Asymmetric urea compound and process for producing asymmetric compound by asymmetric conjugate addition reaction with the same as catalyst
05/12/2005WO2004096802A3 ANTIBIOTIC TETRAHYDRO-β-CARBOLINE DERIVATIVES
05/12/2005WO2004072087A3 Metal complexes as light-absorbing compounds in the information layer of optical data carriers
05/12/2005US20050101788 Method for manufacture of sertindole
05/12/2005US20050101786 N-alkylation of indole derivatives
05/12/2005US20050101781 Eponemycin and epoxomicin analogs and uses thereof
05/12/2005US20050101763 For use as building blocks in photolithographic solid-phase peptide synthesis; microarrays
05/12/2005US20050101661 Cyclooxygenase inhibitors; musculoskeletal and cardiovascular disorders; antiinflammatory agents
05/12/2005US20050101654 Process for the preparation of N-amino substituted heterocyclic compounds
05/12/2005US20050101623 Beta-carboline compounds and analogues thereof as mitogen-activated protein kinase-activated protein kinase-2 inhibitors
05/12/2005US20050101596 Such as N,N-dimethyl-3-(phenylsulfonyl)-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-amine; for treatment of central nervous system disorders related to or affected by serotonin receptor antagonists such as neurodegenerative disorders, attention deficit disorder, obsessive compulsive disorder, and drug abuse
05/12/2005US20050101584 Selective estrogen receptor-beta ligands
05/12/2005US20050101004 Screening for a compound to inhibit the urge for urinary incontinence by detecting activation of KCNQ protein in the host cell; measuring the membrane potential of the host cell and selecting the compound whose presence causes hyperpolarization in themembrane potential of the host cell
05/12/2005US20050100902 5-cyano-1h-indole derivatives as antagonist of the inerleukine-8 receptors
05/12/2005CA2543942A1 Indirubin-type compounds, compositions, and methods for their use
05/12/2005CA2543918A1 Benzimidazoles useful as modulators of ion channels
05/12/2005CA2540843A1 Phenyl carboxamide and sulfonamide derivatives for use as 11-beta-hydroxysteroid dehydrogenase
05/11/2005EP1530097A2 Organophotoreceptor with charge transport material having a vinyl ether group
05/11/2005EP1530096A2 Organophotoreceptor with a hydrazone polymer charge transport material
05/11/2005EP1530094A2 Organophotoreceptor with charge transport material having three arylamino groups
05/11/2005EP1529776A2 Amino acid derivatives and sweetening agent
05/11/2005EP1529034A1 Benzoylpyrazolones substituted by 3-aminocarbonyl
05/11/2005EP1529031A1 Acylated arylcycloalkylamines and their use as pharmaceuticals
05/11/2005EP1528923A1 N-((3-oxo-2,3-dihydro-1h-isoindol-1-yl)acetyl)guanidine derivatives as nhe1-inhibitors for the treatment of infarction and angina pectoris
05/11/2005EP1528919A2 Therapeutic use of aryl amino acid derivatives
05/11/2005EP1421064B1 Process for the preparation of 3-spiro'cyclohexam-1,3'-'3h!indolin-2'-one! derivatives
05/11/2005CN1615311A 3-biphenyl-substituted-3-substituted-4-ketolactam and ketolactone and their utilization as pesticide
05/11/2005CN1615305A Coumarin derivatives, process for their production and use thereof