Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
09/2005
09/14/2005EP1572645A2 Derivatives of succinic and glutaric acids and analogs thereof useful as inhibitors of phex
09/14/2005EP1572197A1 4- 1- (sulfonyl) -1h-indol-2-yl)-4- (hydroxy) -cyclohexa-2,5-dienone compounds and analogs thereof as therapeutic agents
09/14/2005EP1283825B1 N-substituted peptidyl nitriles as cysteine cathepsin inhibitors
09/14/2005EP1071420B1 Indolyl-3-glyoxylic acid derivatives with antitumoral activity
09/14/2005CN1668721A Immunoadhesin comprising a glycoprotein VI domain
09/14/2005CN1668709A Polymerisable diketopyrrolopyrroles, use of such compounds in colour filters and polymers prepared from these compounds
09/14/2005CN1668703A Charge transport compositions on the basis of triarylmethanes and their use in electronic devices
09/14/2005CN1668622A 1-aza-dibenzoazulenes as inhibitors of tumor necrosis factor production and intermediates for the preparation thereof
09/14/2005CN1668616A Charge transport compositions comprising fluorizated quinazoline derivatives
09/14/2005CN1668611A 1-[(indol-3-yl)carbonyl] piperazine derivatives
09/14/2005CN1668595A Method of forming a carbon-carbon or carbon-heteroatom linkage
09/14/2005CN1668591A Phenol derivatives and method of use thereof
09/14/2005CN1668590A 1-heterocyclylalkyl-3-sulfonyl-indole or -indazole derivatives as 5-hydroxytryptamine-6 ligands
09/14/2005CN1668589A Indoline derivatives substituted in the 6 position, their preparation and their use as medicaments
09/14/2005CN1668588A Indole derivatives, method for preparing same and pharmaceutical compositions containing same
09/14/2005CN1668587A Indole derivatives and drugs containing the same
09/14/2005CN1668586A Method for preparing 13 5-triaminobenzene and hydrolyzing it into high-purity phloroglucinal
09/14/2005CN1668585A 3, 6-disubstituted azabicyclo [3.1.0]hexane derivatives useful as muscarinic receptor antagonists
09/14/2005CN1668298A Antitumor compound and therapeutic uses thereof
09/14/2005CN1668296A Methods and compositions using selective cytokine inhibitory drugs for treatment and management of cancers and other diseases
09/14/2005CN1668291A Substituted phenylsulfonamide inhibitors of beta amyloid production
09/14/2005CN1218936C Carboxamide-substituted phenylurea derivatives, process for their preparation and their use as medicaments
09/14/2005CN1218919C Fluorene derivatives and their application
09/13/2005US6943188 For manufacture of medicament for use in treating asthma, multiple sclerosis, inflammatory disease
09/13/2005US6943174 6,5-Fused bicyclic heterocycles
09/13/2005CA2179634C 4-arylisoindole analgesics
09/09/2005WO2005082882A1 Hydrazide type compounds and the use thereof in pharmaceutical compositions for the treatment of cardiovascular diseases
09/09/2005WO2005082851A2 Charge transport compounds and electronic devices made with such compounds
09/09/2005WO2005082850A1 Process for producing monatin
09/09/2005WO2005058884A3 Cyclopropane compounds and pharmaceutical use thereof
09/09/2005WO2005058819A8 Polymorphic forms of tegaserod base and salts thereof
09/09/2005WO2005014584A8 3-(indol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones,3-(benzimidazol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones, and 3-(indolin-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones; their preparation and use as modulators of apoptosis
09/09/2005CA2556830A1 Methods and compositions comprising non-peptide small molecules that solubilize beta amyloid peptide fiber
09/09/2005CA2554439A1 Hydrazide type compounds and the use thereof in pharmaceutical compositions for the treatment of cardiovascular diseases
09/08/2005US20050197501 Reacting calcium hydroxide with an ester derivative or protected ester derivative of the statin; rosuvastatin, pitavastatin and atorvastatin, simvastatin and lovastatin
09/08/2005US20050197383 Quaternary ammonium compounds and their use as anti-tussive agents
09/08/2005US20050197382 Indolinone combinatorial libraries and related products and methods for the treatment of disease
09/08/2005US20050197380 Condensed indoline derivatives and their use as 5HT, in particular 5HT2C, receptor ligands
09/08/2005US20050197373 Substituted fused bicyclic amines as modulators of chemokine receptor activity
09/08/2005US20050197362 Preventives/remedies for urinary disturbance
09/08/2005US20050197343 N-[(4-phenyl-1-piperazinyl)alkyl]-substituted heteroarene carboxamide or 2-ferrocenyl compounds; psychiatric diseases: schizophrenia , unipolar depression, disturbances of consciousness, antidepressant; neurodegenerative diseases: Parkinson's disease, attention deficit hyperactivity syndrome; drug abuse
09/08/2005US20050197331 Novel anti-inflammatory and analgesic heterocyclic amidines that inhibit nitrogen oxide (NO) production
09/08/2005US20050197301 3,4-(cyclopentyl)-fused proline compounds as inhibitors of hepatitis C virus NS3 serine protease
09/08/2005US20050197299 Peptidomimetic protease inhibitors
09/08/2005DE102004006785A1 Verfahren zur CC-Bindungsknüpfung zwischen elektrophilen Substraten und TT-Verbindungen in neutralen bis basischen wässrigen oder alkoholischen Lösungsmitteln ohne den Einsatz einer Lewis- oder Protonensäure Process for carbon-carbon bond between electrophilic substrates and TT compounds in neutral to basic aqueous or alcoholic solvents without the use of a Lewis or protic acid
09/07/2005EP1571142A1 Novel anti-inflammatory and analgesic heterocyclic amidines that inhibit nitrogen oxide (NO) production
09/07/2005EP1569916A1 Substituted aralkyl derivatives
09/07/2005EP1569911A1 Indazole derivatives as crf antagonists
09/07/2005EP1569904A1 Substituted arylalcanoic acid derivatives as ppar pan agonists with potent antihyperglycemic and antihyperlipidemic activity
09/07/2005EP1569903A2 Methods of using and compositions comprising selective cytokine inhibitory drugs for the treatment and management of myeloproliferative diseases
09/07/2005EP1569902A1 Substituted indole oxo-acetyl amino acetic acid derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1)
09/07/2005EP1569901A2 ARYL, ARYLOXY, AND ALKYLOXY SUBSTITUTED i 1H /i -INDOL-3-YL GLYOXYLIC ACID DERIVATIVES AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR-1 (PAI-1)
09/07/2005EP1569900A2 Substituted 3-carbonyl-1-yl acetic acid derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1)
09/07/2005EP1569899A2 SUBSTITUTED 3-ALKYL AND 3-ARYLALKYL i 1H /i -INDOL-1-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR-1 (PAI-1)
09/07/2005EP1569639A2 Substituted dihydropyrano indole-3,4-dione derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1)
09/07/2005EP1569638A1 Aminoalkoxyindoles as 5-ht6-receptor ligands for the treatment of cns-disorders
09/07/2005EP1495023B1 Novel 1,2,3-substituted indolizine derivatives, inhibitors of fgfs, method for making same and pharmaceutical compositions containing same
09/07/2005EP1333824B1 Treatment of sexual dysfunction with bombesin receptor antagonists
09/07/2005EP1254133B9 Indol-3-yl derivatives and their use as integrin inhibitors
09/07/2005EP1192132B1 Serine protease inhibitors
09/07/2005EP1188747B1 Phenoxypropylamine compounds
09/07/2005EP1178794B1 Use of succinic acid derivatives to obtain a medicine for treating inflammation
09/07/2005CN1666577A Electronic devices made with electron transport and/or anti-quenching layers
09/07/2005CN1666357A Polymeric charge transport compositions and electronic devices made with such compositions
09/07/2005CN1665850A Heterocyclic nitrogen-containing activators and catalyst systems for olefin polymerization
09/07/2005CN1665849A Halogen substituted catalyst system for olefin polymerization
09/07/2005CN1665823A Process for preparing 1, 2, 3, 9-tetrahydro-9-methyl-3-[2-methyl-1h-imidazol-1-yl)methyl]-4h-carbazol-4-one
09/07/2005CN1665815A Novel tetracyclo-aryl-carbonyl indoles used as therapeutical agents with 5-hydroxy-tryptamine receptor affinity, their preparation process and pharmaceutical compounds containing same
09/07/2005CN1665809A Azaindoles
09/07/2005CN1665802A Bisarylsulfonamide compounds and their use in cancer therapy
09/07/2005CN1665780A Tricyclic steroid hormone nuclear receptor modulators
09/07/2005CN1665503A Utilization of heteroarene carboxamide as dopamine-D3 ligands for the treatment of cns diseases
09/07/2005CN1217933C Dihalopropene compound, insecticide/miticide containing the same and intermediate for producing the same
09/07/2005CN1217932C Antibacterial agents
09/07/2005CN1217931C Spirocyclic phenyl keto-enols as pesticides and herbicides
09/07/2005CN1217930C Process for preparation of indole derivatives and intermediates of the process
09/07/2005CN1217922C 2-amino-2-alkyl-4-hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors
09/06/2005US6939895 Renalosteodystrophy comprising a compound, or a pharmaceutically acceptable salt or hydrate thereof, having the formula: Ar5-(CHR16)t-W-(CH2)u-CHR17)-NH-CH(R18)-Ar6 wherein: Ar5 is phenyl, indole, carbazole, pyridine,
09/06/2005US6939890 Antiinflammatory agents; sepsis shock; rheumatic disorders
09/06/2005US6939889 Quarternary ammonium compounds
09/06/2005US6939888 Heterocyclic amides such as 3-(2-chloro-6-methoxyphenyl)-5-isopropyl-5-methyl-4-acetoxy-3-pyrrolidine-2 -one, used as insecticides or miticides
09/06/2005US6939886 Substituted naphthyl indole derivatives as inhibitors of plasminogen activator inhibitor Type-1 (PAI-1)
09/06/2005US6939875 Carbocyclic oxy sulfides such as [4-(Biphenyl-4-ylmethylsulfanyl)-5-methoxy-2-methyl-phenoxy]-acetic acid, used to control peroxisome proliferator activated receptors (PPAR), for prophylaxis of metabolic disorders
09/06/2005US6939869 Pyrrolo[2,1-c][1,4] benzodiazepine-indole derivatives, their preparation process, and uses of the same
09/06/2005US6939867 Phenyl sulfamide derivatives as dietetics, antidiabetics, and hypotensive agents
09/06/2005US6939515 Apparatuses and methods for creating and testing pre-formulations and systems for same
09/01/2005WO2005080361A1 Histamine-3 receptor modulators
09/01/2005WO2005080337A1 Oxime ester compound, photopolymerizable composition and color filter utilizing the same
09/01/2005WO2005080336A1 Novel benzofurans and indols
09/01/2005WO2005080335A1 3-3-di-substituted-oxindoles as inhibitors of translation initiation
09/01/2005WO2005080333A1 Process for purification of ropinirole
09/01/2005WO2005080332A1 Novel form of fluvastatin sodium
09/01/2005WO2005080331A1 Fluorescent probe
09/01/2005WO2005080330A1 Heteroarylphenylurea derivative
09/01/2005WO2005080329A2 Process for manufacture of racemic carvedilol
09/01/2005WO2005080322A1 Fluorene derivative
09/01/2005WO2005080317A2 Therapeutic amide derivatives
09/01/2005WO2005079497A2 Substituted fused bicyclic amines as modulators of chemokine receptor activity
09/01/2005WO2005079496A2 Substituted bicycloalkylamine derivatives as modulators of chemokine receptor activity
09/01/2005WO2003101941A3 Alpha acyloxyacetamides for kallikrein and urokinase inhibition