| Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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| 01/20/2005 | US20050014721 reacting oxabenzonorbornadiene with nucleophiles;in presence of rhodium complex catalyst forming 2-pyrrolidin-1-ol-1,2-dihydronaphthalen-1-ol; drug used as analgesics, Parkinson's disease, anticancer agents; aids |
| 01/20/2005 | US20050014700 Cbi analogues of cc-1065 and the duocarmycins |
| 01/20/2005 | CA2528626A1 Indoles useful in the treatment of inflammation |
| 01/20/2005 | CA2528336A1 Tetrahydrocarbazole derivatives and their pharmaceutical use |
| 01/19/2005 | EP1498411A1 Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient |
| 01/19/2005 | EP1498406A1 Novel hydronaphthalene compounds, prepared by a rhodium catalysed ring opening reaction in the presence of phosphine ligand |
| 01/19/2005 | EP1497282A2 Inhibitors of serine protease, particularly hepatitis c virus ns3-ns4 protease |
| 01/19/2005 | EP1497279A2 Substituted indoles and their use as 5ht-reuptake inhibitors and as 5ht ligands |
| 01/19/2005 | EP1497278A1 Heterocyclic amide derivatives as cytokine inhibitors |
| 01/19/2005 | EP1497274A2 Terphenyl derivatives, preparation thereof, compositions containing same |
| 01/19/2005 | EP1497268A2 Nitric oxide donors, compositions and methods of use |
| 01/19/2005 | EP1497240A1 Non-heating clay composites for building materials |
| 01/19/2005 | EP1496838A2 Substituted amides |
| 01/19/2005 | EP0958293B1 Nanomolar, non-peptide inhibitors of cathepsin d |
| 01/19/2005 | EP0831813B1 Methods of inhibiting pneumocystis carinii pneumonia and compounds useful therefor |
| 01/19/2005 | CN1568370A Treatment of CNS disorders using D-amino acid oxidase and D-aspartate oxidase antagonists |
| 01/19/2005 | CN1568311A 1h-indole derivatives as a highly selective cyclooxygenase-2 inhibitor |
| 01/19/2005 | CN1568310A Heterocyclic inhibitors of glycogen synthase kinase GSK-3 |
| 01/19/2005 | CN1566092A Indene ketone diindyl class compound, preparation method and medical use thereof |
| 01/19/2005 | CN1566091A Molindone derivatives and use for preparing antineoplastic medicine thereof |
| 01/19/2005 | CN1185234C Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives |
| 01/19/2005 | CN1185214C Novel indeno indolone compound, its preparation method and drug composition comprising the same |
| 01/18/2005 | US6844446 Catalysts containing per-ortho aryl substituted aryl or heteroaryl substituted nitrogen donors |
| 01/18/2005 | US6844445 Central nervous system disorders; psychological disorders |
| 01/18/2005 | US6844366 Such as N-hydroxy-2(R)-((3,4-methylenedioxybenzyl)-(4-methoxy-2,3,6-trimethylbenzene-sulfonyl) amino)-3-methylbutyramide for treatment of diseases treatable with pro-collagen C-proteinase inhibitors |
| 01/18/2005 | US6844362 Inflammatory, allergic and respiratory disorders; beta 2 adrenoceptors agonists; such as 5-(-2-((-2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethyl)amino)propyl) -N-(2-methoxybenzyl)-1H-indole-2-carboxamide |
| 01/18/2005 | US6844359 As inhibitors of tumor necrosis factor; for therapy of cachexia, arthritis, rheumatoid arthritis, osteoarthritis, reperfusion injury, congestive heart failure, Crohn's disease, ulcerative colitis, systemic lupus erythrematosis |
| 01/18/2005 | US6844342 Heterocyclic substituted 2-methyl-benzimidazole antiviral agents |
| 01/13/2005 | WO2005003153A1 Novel method of synthesising perindopril and the pharmaceutically-acceptable salts thereof |
| 01/13/2005 | WO2005003098A1 Heterocyclically substituted pentanol derivatives, method for the production thereof, and use thereof as anti-inflammatory agents |
| 01/13/2005 | WO2005003091A1 Novel method of synthesising (2s, 3as, 7as)-perhydroindole-2-carboxylic acid, and use thereof for synthesis of perindopril |
| 01/13/2005 | WO2005002525A2 Cox-2 and faah inhibitors |
| 01/13/2005 | WO2005002523A2 Process for preparing highly pure and free-flowing solid of 7-ethyltryptophol |
| 01/13/2005 | WO2004099129A3 Intermediates useful in the synthesis of hiv-protease inhibitors and methods for preparing the same |
| 01/13/2005 | WO2004072047A8 Indoles, benzimidazoles or naphhimidazoles as histone deacetylase (hdac) inhibitors |
| 01/13/2005 | US20050010055 Methylation, benzylation of indole using 1,4-diazabicyclo(2.2.2)octane as basic catalyst under microwave irradiation |
| 01/13/2005 | US20050009920 Taxol enhancer compounds |
| 01/13/2005 | US20050009903 1-Methoxy-, 1-deoxy-11-hydroxy- and 11-hydroxy-1-methoxy- Delta 8-tetrahydrocannabinols and 1-alkyl-3(1-naphthoyl)indoles, useful for the treatment of pain (especially pain resulting from inflammation) and cancer (especially glioma tumors). |
| 01/13/2005 | US20050009898 New substituted indolinones, their manufacture and their use as medicaments |
| 01/13/2005 | US20050009897 Method of treatment |
| 01/13/2005 | US20050009871 Ubiquitin ligase inhibitors |
| 01/13/2005 | US20050009819 1-Aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands |
| 01/13/2005 | US20050009808 Azabicyclo compound matrix metalloprotease inibitor and skin preparation |
| 01/13/2005 | US20050009799 Cyclohexyl derivatives as selective estrogen receptor modulators |
| 01/13/2005 | US20050006246 Nitrogen atom transfer |
| 01/13/2005 | CA2531060A1 Heterocyclically-substitued pentanol derivatives, process for their production and their use as anti-inflammatory agents |
| 01/13/2005 | CA2530808A1 Cox-2 and faah inhibitors |
| 01/12/2005 | EP1496050A1 Novel chemiluminescent compounds and their use |
| 01/12/2005 | EP1496041A1 Novel aromatic compound and organic electroluminescnet element containing the same |
| 01/12/2005 | EP1495023A1 Novel 1,2,3-substituted indolizine derivatives, inhibitors of fgfs, method for making same and pharmaceutical compositions containing same |
| 01/12/2005 | EP1495016A2 Heterocyclic compounds and their use as modulators of p38 map kinase |
| 01/12/2005 | EP1495004A2 Benzenesulfonamide derivatives and their use as dopamine d3 and d2 receptor ligands |
| 01/12/2005 | EP1495000A1 Alpha, omega-dicarboximide derivatives as useful uro-selective a1a adrenoceptor blockers |
| 01/12/2005 | EP1494997A1 Substituted aryl amides |
| 01/12/2005 | EP1494989A2 Compounds that modulate ppar activity and methods for their preparation |
| 01/12/2005 | CN1564820A Heterocyclic compounds for use in the treatment of disorders of the urinary tract |
| 01/12/2005 | CN1562970A PPAR full activator of amino acids of aralkyl possessing excellent activity for lowering sugar and ester |
| 01/12/2005 | CN1184202C Method for preparing N-methyl carbazole |
| 01/11/2005 | US6841685 Methods for making bis-heterocyclic alkaloids |
| 01/11/2005 | US6841569 Treatment of central nervous system disorders; anticonvulsants, antiepileptics, neuroprotective agents and muscle relaxants |
| 01/11/2005 | US6841568 Inducing contraception, treat progesterone-related carcinomas and adenocarcinomas; hormone replacement therapy |
| 01/11/2005 | US6841552 3a,4,5,9b-tetrahydro-1H-benz[e]indol-2-yl amine-derived neuropeptide Y receptors ligands useful in the treatment of obesity and other disorders |
| 01/11/2005 | US6841504 Polymerization catalyst activator and its use in a polymerization process |
| 01/11/2005 | US6841502 For catalytic polymerization of ethylene/olefin copolymers |
| 01/06/2005 | WO2005002293A2 Cox-2-targeted imaging agents |
| 01/06/2005 | WO2005001105A1 Method for producing monatin |
| 01/06/2005 | WO2005000814A1 Polymethine ethers |
| 01/06/2005 | WO2005000812A1 Process for producing indole compound |
| 01/06/2005 | WO2005000804A2 Substituted indoles and a process for preparing substituted indoles |
| 01/06/2005 | WO2005000803A2 Asymmetric urea compound and process for producing asymmetric compound by asymmetric conjugate addition reaction with the same as catalyst |
| 01/06/2005 | WO2005000775A2 Cyclohexyl derivatives as selective estrogen receptor modulators |
| 01/06/2005 | WO2005000406A2 Treatment of amyloid- and epileptogenesis-associated diseases |
| 01/06/2005 | WO2004099193A3 1-aryl-3-(indol-5-yl)-prop-2-en-1-ones, compositions comprising the same and use thereof |
| 01/06/2005 | WO1999044608A8 New use |
| 01/06/2005 | US20050004394 Processes of producing glutamic acid compounds and production intermediates therefore and novel intermediate for the processes |
| 01/06/2005 | US20050004369 Phenyl substituted carboxylic acids |
| 01/06/2005 | US20050004360 Compounds and methods for modulation of estrogen receptors |
| 01/06/2005 | US20050004207 Substituted isoindoles and the use thereof |
| 01/06/2005 | US20050004204 2-Iminopyrrolidine derivatives |
| 01/06/2005 | US20050004197 Thrombin receptors antagonists; oral efficacy |
| 01/06/2005 | US20050004167 Such as dibenzofuran-2-carboxylic acid 2-(phenylsulfonyl)hydrazide |
| 01/06/2005 | US20050004166 Imino acid derivatives as inhibitors of matrix metalloproteinases |
| 01/06/2005 | US20050004164 2-Cyanopropanoic acid amide and ester derivatives and methods of their use |
| 01/06/2005 | US20050004118 Prodrugs of non-steroidal anti-inflammatory and carboxylic acid containing compounds |
| 01/06/2005 | US20050004104 Methods for the protection of memory and cognition |
| 01/06/2005 | US20050004101 Therapy for schizophrenia, obsessive complusive disorders; antidepressants; anxiolytic agents; panic disorders; antiepileptic agents; analgesics; headaches; sleep disorders; eating disorders |
| 01/06/2005 | US20050004097 Indole derivatives |
| 01/06/2005 | US20050004096 Indole derivatives, process for producing the same and drugs containing the same as the active ingredient |
| 01/06/2005 | US20050003230 cyclized; organic light-emitting diodes (OLED); eliminate drawbacks of Alq3 as emitter and a host material for dopants; narrower emission bands; broad spectral range; low driver voltages; high photometric efficiency (low power consumption); high luminance (emission intensity); high thermal stability |
| 01/06/2005 | US20050002859 COX-2-targeted imaging agents |
| 01/06/2005 | CA2556706A1 Treatment of amyloid- and epileptogenesis-associated diseases |
| 01/06/2005 | CA2530408A1 Cox-2-targeted imaging agents |
| 01/06/2005 | CA2527659A1 Cyclohexyl derivatives as selective estrogen receptor modulators |
| 01/06/2005 | CA2526988A1 Substituted indoles and a process for preparing substituted indoles |
| 01/05/2005 | EP1493743A1 Substituted bipiperidine intermediates and derivatives thereof |
| 01/05/2005 | EP1492792A2 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino 4,5-b]indole-1-acetamide derivatives, preparation and use thereof in medicaments |
| 01/05/2005 | EP1492788A1 Indole-amid derivatives which possess glycogen phosphorylase inhibitory activity |
| 01/05/2005 | EP1492785A1 New compounds |
| 01/05/2005 | EP1492766A1 Improved cc-1065 analog synthesis |
| 01/05/2005 | EP1492756A1 Novel thyroid receptor ligands |