Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
01/2005
01/05/2005EP1492568A1 Cancer treatment method comprising administration of an erb-family inhibitor and a raf and/or ras inhibitor
01/05/2005EP1492539A1 Statin therapy for enhancing cognitive maintenance
01/05/2005EP1492537A1 Morpholine derivatives with a substituted acetamide group in the 2-position for use as ccr-3 antagonists for the treatment of inflammatory diseases
01/05/2005EP1492534A1 Carbamic acid compounds comprising a piperazine linkage as hdac inhibitors
01/05/2005EP1492526A2 Improved prodrugs of cc-1065 analogs
01/05/2005EP0957914B1 Formulation of 5-ht agonists
01/05/2005CN1561393A Inhibitors of glycogen synthase kinase-3 (GSK-3) for treating glaucoma
01/05/2005CN1561341A Hydrolysis of [R(R*, R*)]-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino) carbonyl]-1H-pyrrole-1-heptanoic acid esters with calcium hydroxide
01/05/2005CN1561334A Indole derivatives as COXII inhibitors
01/05/2005CN1561327A Novel aminobenzoephenones
01/05/2005CN1561212A Benzimidazolidinone derivatives as muscarinic agents
01/05/2005CN1561211A Nociceptin analogs
01/05/2005CN1560035A 5-hydroxylic indole-3-carboxylic ester kind derivantion
01/05/2005CN1183111C Cycloalkano-indole and cycloalkane-azaindole derivatives, process for their preparation and pharmaceutical commposition containing the same
01/05/2005CN1183107C Alkynyl containing hydroxamic acid compounds as TACE inhibitors
01/04/2005US6838484 Androgen receptor targeting agents which demonstrate androgenic and anabolic activity of a nonsteroidal ligand for the androgen receptor
01/04/2005US6838483 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
01/04/2005US6838461 Psychological disorders; schizophrenia; Alzheimer's disease; Parkinson's disease; Huntington's disease; cardiovascular disorders; hypotensive agents; side effect reduction
01/04/2005US6838415 Substituted benzoylisoxazoles and the use thereof as herbicides
01/04/2005CA2293834C Substituted naphthopyrans
12/2004
12/30/2004US20040266861 Administering a therapeutically effective amount of a compound which is a cannabinoid receptor agonist, a pharmaceutically acceptable salt of the compound, an isomer of the compound, or a pharmaceutically acceptable salt of the isomer
12/30/2004US20040266855 Effective against Src family; cancer, osteoporosis
12/30/2004US20040266822 Secondary amines; tissue specificity; reduced side effects; cardiovascular diseases, diabetes, bronchial and urinary smooth muscle spasms, ischemia, anoxic nerve injury
12/30/2004US20040266789 Substituted amino carboxylic acids
12/30/2004US20040266788 treatment of diabetes and/or cancer; useful in the treatment of syndrome X; capable of inhibiting Protein tyrosine phosphatase
12/30/2004US20040266782 Cyclic amine derivatives-CCR-3 receptor antagonists
12/30/2004US20040266733 Substituted naphthyl indole derivatives as inhibitors of plasminogen activator inhibitor Type-1 (PAI-1)
12/30/2004US20040265985 Such as 1S,4R)-1-amino-4-(hydroxymethyl)-2-cyclopentene via N-acetylamino-alcohol hydrolase isolated from Rhodococcus, Gordona, Arthrobacter, Alcaligenes, Agrobacterium/Rhizobium, Bacillus, Pseudomonas or Alcaligenes/Bordetella
12/30/2004US20040262576 such as tris(2-phenylpyridine)iridium which luminesce when voltage is applied; improved electroluminescent efficiency
12/29/2004WO2004113453A1 Crystalline nonsolvated polymethine compound
12/29/2004WO2004113394A2 Living radical polymerization initiator comprising a functional group capable of reacting with polypeptides or the like, comb polymer obtained therewith, polypeptide conjugates and drugs obtained therefrom
12/29/2004WO2004113301A1 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders
12/29/2004WO2004113296A1 A process for preparation of 1-[9h-carbazol-4-yloxy]- 3-[{2-(2-(-(methoxy)phenoxy)-ethyl}-amino]-propan-2-ol
12/29/2004WO2004113295A1 Process and intermediates for the preparation of (1r,2s,5s)-6,6-dimethyl-3-azabicyclo[3,1,0]hexane-2-carboxylates or salts thereof
12/29/2004WO2004113293A1 Novel crystalline forms of perindopril erbumine
12/29/2004WO2004113292A2 Fluvastatin sodium crystal forms, processes for preparing them, compositions containing them and methods of using them
12/29/2004WO2004113291A2 Fluvastatin sodium crystal forms xiv, lxxiii,lxxix, lxxx and lxxxvii, processes for preparing them, compositions containing them and methods of using them
12/29/2004WO2004113270A2 Propionic acid derivatives useful in the treatment of lipid disorders
12/29/2004WO2004112718A2 Compounds, compositions and methods for treatment and prevention of orthopoxvirus infections and associated diseases
12/29/2004WO2004085396A8 Preventive or therapeutic agent for ischemia/reperfusion injury, organ preservative, and screening method
12/29/2004WO2004002940A8 Inhibitors of hcv ns5b polymerase
12/29/2004WO2003045392A8 Use of n-(indolcarbonyl-)piperazine derivatives
12/29/2004EP1491524A2 Selective androgen receptor modulators and methods of use thereof
12/29/2004EP1491353A1 Optical recording media and dipyrromethene-metal chelate compounds
12/29/2004EP1491206A1 Induction method for cell differentiation
12/29/2004EP1490353A1 Method for manufacture of sertindole
12/29/2004EP1490334A1 Phthalimido derivatives as inhibitors of monoamine oxidase b
12/29/2004EP1490062A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
12/29/2004EP1425577A4 Apparatuses and methods for creating and testing pre-formulations and systems for same
12/29/2004EP1226138B1 Fab i inhibitors
12/29/2004EP1225882A4 Selective cox-2 inhibitory novel esters from indolealkanols and novel amides from indolealkylamines
12/29/2004EP1206442A4 Substituted chiral allosteric hemoglobin modifiers
12/29/2004EP1135123B1 Use of isatin derivatives as ion channel activating agents
12/29/2004EP1032560B1 Position-4 substituted 2-pyrrolidinone derivatives to reduce the level of extracellular glutamate
12/29/2004EP0869958B1 Novel indole-2,3-dione-3-oxime derivatives
12/29/2004CN1558900A Pseudopolymorphic forms of carvedilol
12/29/2004CN1558899A Spirocyclic 3-phenyl-3-substituted 4-ketolactams and 4-ketolactones
12/29/2004CN1558897A Antidiabetic agents
12/29/2004CN1558759A 病毒聚合酶抑制剂 Viral polymerase inhibitors
12/29/2004CN1182116C Mutilin derivatives and their use as antibacterials
12/29/2004CN1182103C Novel ethylamine derivatives
12/29/2004CA2613021A1 Fluvastatin sodium crystal form lxxx, processes for preparing, compositions and methods of using
12/29/2004CA2613013A1 Fluvastatin sodium crystal form lxxiii, processes for preparing, compositions and methods of using
12/29/2004CA2610635A1 Fluvastatin sodium crystal form lxxxvii, processes for preparing, compositions and methods of using
12/29/2004CA2610633A1 Fluvastatin sodium crystal form lxxix, processes for preparing, compositions and methods of using
12/29/2004CA2529859A1 Fluvastatin sodium crystal forms xiv, lxxiii ,lxxix, lxxx and lxxxvii, processes for preparing them, compositions containing them and methods of using them
12/29/2004CA2529820A1 Fluvastatin sodium crystal forms, processes for preparing them, compositions containing them and methods of using them
12/29/2004CA2529761A1 Compounds, compositions and methods for treatment and prevention of orthopoxvirus infections and associated diseases
12/29/2004CA2528234A1 Propionic acid derivatives useful in the treatment of lipid disorders
12/28/2004US6835843 Amidation, deprotected by catalytic hydrogenation, salt formation with tributylamine
12/28/2004US6835752 Carboxylic acid derivatives, processes for the preparation thereof and pharmaceutical agents comprising the same as active ingredient
12/28/2004US6835744 3,3-substituted indoline derivatives
12/28/2004US6835729 2-phenyl-1-[4(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
12/28/2004US6835727 Bone disorders; osteoporosis; rheumatic diseases
12/28/2004US6835725 Cyanine dye containing heterocylic rings; satisfies light stability, favorable signal/noise rato, damage free application to the substrate material, use in the information layer in a write-once optical data carrier
12/28/2004US6835712 Compounds
12/28/2004US6835513 An organophotoreceptor comprising: (a) a charge transport compound having the formula carbazole compound dispersion of colorant particles in an organic liquid and charge transport compound having the formula of carbazole compound
12/28/2004CA2281426C Substituted indole compounds as anti-inflammatory and analgesic agents
12/28/2004CA2105923C 7-isoindolinyl-quinolone derivatives and 7-isoindolinyl-naphthyridone derivatives
12/23/2004WO2004111193A2 Prodrugs of mitotic kinesin inhibitors
12/23/2004WO2004111039A1 2,3-substituted 5,6-diaryl-pyrazine derivatives as cb1 modulators
12/23/2004WO2004110999A1 Tetrahydrocarbazole derivatives and their pharmaceutical use
12/23/2004WO2004110989A1 N-hydroxy-7-(arylamino)heptanamide derivatives useful for treating hyper-proliferative disorders
12/23/2004WO2004110986A1 Benzamide derivative or salt thereof
12/23/2004WO2004110983A2 New benzamides as pparϒ modulators
12/23/2004WO2004110436A1 Fused indoles as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
12/23/2004WO2004110149A1 Use of isoindolinone derivatives as insecticides
12/23/2004WO2004099150A3 3-(1-naphthyl)-2-cyanopropanoic acid derivatives as estrogen receptor ligands
12/23/2004WO2004099138A3 Process for the preparation of perindopril
12/23/2004WO2004091482A3 M3 muscarinic acetylcholine receptor antagonists
12/23/2004WO2004087048A3 Benzamide modulators of metabotropic glutamate receptors
12/23/2004WO2004085392A8 Melatonin derivatives and their use for treating neurological dysfunctions
12/23/2004WO2004064771A3 Geminally di-substituted nsaid derivatives as abeta 42 lowering agents
12/23/2004WO2003091689A3 Bis-transition-metal-chelate-probes
12/23/2004US20040259939 Dissolving and precipitation a solution of citalopram in acid with solvent, adding base to liberate free base.
12/23/2004US20040259919 for the treatment of diabetes, hyperglycemia, hypoglycemia, syndrome X, hyperinsulinemia, obesity, atherosclerosis, eating disorders, and nervous system disorders
12/23/2004US20040259917 Heteroaryl substituted imidazole modulators of metabotropic glutamate receptor-5
12/23/2004US20040259912 N-(4-benzhydryloxy-3-isobutyrylphenyl)-N'-(3,4-dimethoxyphenyl)urea for example; vanilloid receptor agonists; use as analgesic and or for treating urinary frequency and/or urinary incontinence
12/23/2004US20040259908 Integrin VLA-4 ( alpha 4 beta 1) and/or integrin LPAM-1 ( alpha 4 beta 7) antagonists, cell adhesion inhibitor; bioavailability, oral administration;treating inflammatory diseases; e.g. 3-[2-(2,6-dichlorobenzoylamino)pyrid-5-yl]-2-{3-[(2,2-dimethylpropionyl)isobutylamino]-4-methoxyphenyl}propionic acid
12/23/2004US20040259890 trans-3'-oxo-N-(trans-4-phenylcyclohexyl)-spiro[cyclohexane-1,1'(3'H)-isobenzofuran]-4-carboxamide e.g.; neuropeptide Y receptor antagonists for treatment of bulimia, obesity or diabetes for example