Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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06/30/2005 | US20050142322 Optical recording media and dipyrrpomethene-metal chelate compounds |
06/30/2005 | DE10354629A1 2-Ethyl-4,6-dimethyl-phenyl substituierte spirocyclische Tetramsäure-Derivate 2-ethyl-4,6-dimethyl-phenyl substituted spirocyclic tetramic acid derivatives |
06/30/2005 | CA2550886A1 Polymorphic forms of tegaserod base and salts thereof |
06/30/2005 | CA2549825A1 N-(4-carbamimidoyl-benzyl) -2-alkoxy-2-heterocyclyl acetamides as inhibitors of the formation of coagulation factors xa, ixa and thrombin induced by factor viia |
06/30/2005 | CA2549660A1 Cyclopropane compounds and pharmaceutical use thereof |
06/30/2005 | CA2549598A1 N-substituted-n-sulfonylaminocyclopropane compounds and pharmaceutical use thereof |
06/30/2005 | CA2549167A1 Inhibitors of hepatitis c virus ns3/ns4a serine protease |
06/30/2005 | CA2549072A1 Tricyclic indole hydroxyethylamine derivatives and their use in the treatment of alzheimer's disease |
06/29/2005 | EP1547603A2 Compositions and methods for use in targeting vascular destruction |
06/29/2005 | EP1547590A1 Melanin extinguisher |
06/29/2005 | EP1546371A1 Substrates for o6-alkylguanine-dna alkyltransferase |
06/29/2005 | EP1546153A1 Broadspectrum substituted oxindole sulfonamide hiv protease inhibitors |
06/29/2005 | EP1546142A2 Indoles having anti-diabetic activity |
06/29/2005 | EP1546116A1 Vanilloid receptor ligands and their use in treatments |
06/29/2005 | EP1546108A1 1,4-substituted cyclohexane derivatives |
06/29/2005 | EP1546099A2 3,6-disubstituted azabicyclo 3.1.0 hexane derivatives useful as muscarinic receptor antagonists |
06/29/2005 | EP1546098A1 3,6-disubstituted azabicyclo [3.1.0]hexane derivatives useful as muscarinic receptor antagonists |
06/29/2005 | EP1546088A2 Compounds for use in the treatment of autoimmune diseases, immuno-allergical diseases and organ or tissue transplantation rejection |
06/29/2005 | EP1546087A1 3-amino-2-hrydroxyalkanoic acids and their prodrugs |
06/29/2005 | EP1545528A2 Indole-type derivatives as inhibitors of p38 kinase |
06/29/2005 | EP1545510A1 Substituted phenylindoles for the treatment of hiv |
06/29/2005 | EP1545508A1 3,6-disubstituted azabicyclo [3.1.0] hexane derivatives useful as muscarinic receptor antagonist |
06/29/2005 | EP1485352B1 Azaspiro compounds for the treatment of pain |
06/29/2005 | EP1373272B1 Tert. alkylphenoxy substituted polycyclic compounds |
06/29/2005 | EP1274701B1 [1,4']-bipiperidine compounds |
06/29/2005 | EP1242069B1 Albumin-binding compounds that prevent nonenzymatic glycation and that may be used for treatment of glycation-related pathologies |
06/29/2005 | EP0901459B1 Calcilytic compounds |
06/29/2005 | CN1633296A Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
06/29/2005 | CN1631880A Carbazole dithioformate RAFT reagent and preparation method and application thereof |
06/29/2005 | CN1631879A Substituted phenyl keto enols as pesticides and herbicides |
06/29/2005 | CN1631878A C2 phenyl-substituted cyclic keto-enols used as pesticides and herbicides |
06/29/2005 | CN1208333C Indole derivatives useful for the treatment of osteoporosis |
06/29/2005 | CN1208329C Aniline derivatives |
06/29/2005 | CN1208322C Dihydroindole and tetrahydroquinoline derivatives |
06/28/2005 | US6911468 Useful as a prophylactic or therapeutic agent for diabetes or the like |
06/28/2005 | US6911465 For treating inflammatory diseases including rheumatoid arthritis, glomerular nephritides, lung fibrosis, restenosis, alveolitis, asthma, psoriasis, inflammatory bowel disease, multiple sclerosis and brain trauma, stroke, ischemia |
06/28/2005 | US6911464 N-alkyl-hydroxamic acid-isoindolyl compounds and their pharmaceutical uses |
06/28/2005 | US6911463 Capable of increasing lipolysis and energy expenditure in cells and therefore is useful for treating Type 2 diabetes and/or obesity |
06/28/2005 | CA2159071C 4-arylisoindole analgesics |
06/28/2005 | CA2108621C Process for the preparation of mono- or diacetoxyindole |
06/23/2005 | WO2005056693A1 Polymeric dispersant |
06/23/2005 | WO2005056527A1 Substituted tetrahydrocarbazole and cyclopentanoindole derivatives |
06/23/2005 | WO2005056013A1 Dpp-iv inhibitors |
06/23/2005 | WO2005014584A9 3-(indol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones,3-(benzimidazol-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones, and 3-(indolin-1-yl)-4-(indol-3-yl)-pyrrole-2,5-diones; their preparation and use as modulators of apoptosis |
06/23/2005 | WO2005000406A3 Treatment of amyloid- and epileptogenesis-associated diseases |
06/23/2005 | WO2004055026A8 Tetracyclic 3-substituted indoles having serotonin receptor affinity |
06/23/2005 | WO2002068380A8 Synthetic excitatory amino acids |
06/23/2005 | US20050137405 Reacting o-chlorobenzaldehyde with an alkyl 4-(phthalimido)ethoxy)acetoacetate to yield alkyl 2-(o-chlorobenzylidene)-4-(2-phthalimidoethoxy)acetoacetate which upon reacting with an alkyl -3-aminocrotonate yields a phtahalimiamlodipine; good yields and purity; useful as reference standards or markers |
06/23/2005 | US20050137246 Organic amine salts of glutamic acid derivatives and their application |
06/23/2005 | US20050137230 Factor Xa-inhibitors; preventing thromboembolic illnesses and tumors; 2-amino-N-(2'-methylsulfonylbiphenyl-4-yl)-3-phenylpropionamide |
06/23/2005 | US20050137220 Beta-carboline compounds and analogues thereof as mitogen-activated protein kinase-activated protein kinase-2 inhibitors |
06/23/2005 | US20050137215 Antiarthritic and antiinflammatory agents; analgesics; the proline derivatives do not displace gabapentin from alpha-2-delta receptors |
06/23/2005 | US20050137190 Compositions useful as inhibitors of voltage-gated sodium channels |
06/23/2005 | US20050137168 inhibit the formation of coagulation factors Xa, IXa and thrombin induced by factor VIIa and tissue factor; for treatment and/or prevention of arterial and venous thrombosis, deep vein thrombosis, pulmonary embolism, unstable angina pectoris, cardiac infarction, stroke |
06/23/2005 | CA2548602A1 Substituted tetrahydrocarbazole and cyclopentanoindole derivatives |
06/22/2005 | EP1542973A1 2,4-substituted indoles and their use as 5-ht6 modulators |
06/22/2005 | EP1542692A1 Amino-pyridine, -pyridine and pyridazine derivatives for use as vanilloid receptor ligands for the treatment of pain |
06/22/2005 | EP1525265A4 Chiral indole intermediates and their fluorescent cyanine dyes containing functional groups |
06/22/2005 | EP1320523B1 Branched chain amino acid-dependent aminotransferase inhibitors and their use in the treatment of neurodegenerative diseases |
06/22/2005 | EP1154774B1 Quinazoline derivatives as angiogenesis inhibitors |
06/22/2005 | EP1082127B1 Succinamide inhibitors of interleukin-1beta converting enzyme |
06/22/2005 | EP1047672B1 Process for preparing sparingly soluble aromatic amines |
06/22/2005 | CN1630673A Indole resins epoxy resins and resin compositions containing the same |
06/22/2005 | CN1630642A Benzenesulfonamide derivatives |
06/22/2005 | CN1630636A Indoline derivatives and their use as 5-HT2 receptor ligands |
06/22/2005 | CN1630632A Aromatic amino acid derivates and medicinal compositions |
06/22/2005 | CN1630629A 酯化合物及其医药用途 Ester compounds and pharmaceutical use |
06/22/2005 | CN1630555A Hydroxylation of beta-dicarbonyls with zirconium catalysts |
06/22/2005 | CN1629140A 3-cyano-1-alkoxy indole derivatives, preparing process and application thereof |
06/22/2005 | CN1207281C Trifluoromethyl-substd. spirocyclic ketoenols |
06/21/2005 | US6909006 Invention provides cyclopropylindole compounds with structures that allow them to be joined to combinatorial chains, as well as combinatorial libraries containing cyclopropylindoles themselves |
06/21/2005 | US6908935 Calcium receptor modulating agents |
06/21/2005 | US6908929 Central nervous system disorders |
06/21/2005 | US6908927 Reduction physical cigarette smoking |
06/21/2005 | US6908922 Linear cyclic ureas |
06/21/2005 | CA2382387C Pharmaceutical formulations and use thereof in the prevention of stroke, diabetes and/or congestive heart failure |
06/16/2005 | WO2005054249A1 Novel compounds |
06/16/2005 | WO2005054195A1 Method for producing (3-oxo-2,3-dihydro-1h-isoindol-1-yl) acetylguanidine derivatives |
06/16/2005 | WO2005054194A1 A method for the preparation of (2s, 3ar, 7as)-octahydro-1h-indole-2-carboxylic acid as key intermediate in the preparation of trandolapril by reacting a cyclohexyl aziridine with a dialkyl malonate |
06/16/2005 | WO2005054193A1 1-alkyl-3-thio-substituted indole-2-alkynoic acids useful for the treatment for alzheimer's disease and related conditions |
06/16/2005 | WO2005054176A1 Peroxisome proliferator activated receptor modulators |
06/16/2005 | WO2005053686A1 Indolinone based protein kinase inhibitors |
06/16/2005 | WO2005053685A1 Nitrooxyderivatives of carvedilol and other beta blockers as antihypertensive drugs |
06/16/2005 | WO2005053614A2 Advanced indolinone based protein kinase inhibitors |
06/16/2005 | WO2005053610A2 Diamine and iminodiacetic acid hydroxamic acid derivatives |
06/16/2005 | WO2005040116A3 Indolinone derivatives and their use in treating disease-states such as cancer |
06/16/2005 | WO2005016326A3 Analogs of thalidomide as potential angiogenesis inhibitors |
06/16/2005 | WO2004046107A8 Indole derivatives as somatostatin agonists or antagonists |
06/16/2005 | US20050131237 Indole derivatives |
06/16/2005 | US20050131226 Rearranged pentanols, a process for their production and their use as anti-inflammatory agents |
06/16/2005 | US20050131167 Indole resins epoxy resins and resin compositions containing the same |
06/16/2005 | US20050131053 Indole derivatives substituted with long-chain alcolhols and medicaments containing them |
06/16/2005 | US20050131043 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles |
06/16/2005 | US20050131032 (Oxime)carbamoyl fatty acid amide hydrolase inhibitors |
06/16/2005 | US20050131018 Acetylene derivatives as inhibitors of histone deacetylase |
06/16/2005 | US20050130976 Bicyclic inhibitors of MEK and methods of use thereof |
06/16/2005 | US20050130965 Inhibitors of p38 kinase |
06/16/2005 | US20050130963 Indole-amid derivatives which possess glycogen phosphorylase inhibitory activity |
06/16/2005 | US20050130943 Bicyclic inhibitors of MEK and methods of use thereof |
06/16/2005 | US20050130221 Synthesis for the preparation of compounds for screening as potential tubulin binding agents |