Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
05/2003
05/01/2003US20030083490 Coupling of H-phosphonate with a nucleoside alcohol to form the diester; oxidation with sulfur transfer agent to form a phosphorothioate triester
05/01/2003US20030083364 3-Substituted-3-(substitutedsulfonyl or sulfanyl)pyrroldine-2,5-diones useful for inhibition of farnesyl-protein transferase
05/01/2003US20030083349 Antimalaria agents
05/01/2003US20030083348 Farnesyl transferase inhibitors
05/01/2003US20030083337 Optically active 3-[(2-piperazinylphenyl)methyl]-1-[4-(trifluoromethyl)phenyl]-2-pyrrolidinone compounds as 5-HT1D receptor selective antagonists
05/01/2003US20030083331 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
05/01/2003US20030083268 Isoquinoline compounds having antiinfective activity
05/01/2003US20030083228 Treatments for female sexual dysfunction and methods for identifying compounds useful for treating female sexual dysfunction
05/01/2003US20030082225 Sterile, breathable patch for treating wound pain
05/01/2003US20030080320 Combining a tertiary amide with a pentavalent phosphorous halide in a solvent to form an alpha - haloiminium salt and converting the alpha -haloiminium salt to the alpha -haloenamine with a base
05/01/2003CA2464254A1 Inhibitors of post-proline cleaving proteases
05/01/2003CA2463309A1 Sterile, breathable patch for treating wound pain
04/2003
04/30/2003CN1414950A Substituted pyrrole Mannich bases to treating paint and allergic reactions
04/30/2003CN1414849A Carboxylic acid amides, medicaments containing these compounds and the use and preparation thereof
04/30/2003CN1107067C Carbapenem compounds, use and intermediate compounds thereof
04/30/2003CN1107061C Chemotaxis cell factor receptor-3 receptor antagonists
04/29/2003US6555714 P-hydrophenylpyruvate dioxygenases (HPPD) from plants is incubated with test substrate and enzymatic activity of enzyme is determined in comparison with activity of uninhibited enzyme
04/29/2003US6555700 1,3-propane diol esters and ethers and methods for their use in drug delivery
04/29/2003US6555694 Method for production of pyrrolidinone derivatives
04/29/2003US6555692 Polylactams having imidazole or pyrrole rings specifically bind with subnanomolar affinity to a predetermined DNA sequence; use in molecular biology and diagnostic medicine; gene expression control; target the minor groove of B-form
04/29/2003US6555572 Benzylated PDE4 inhibitors
04/29/2003US6555556 N-(4-(1-acetimidoylpiperidin-4-yl)oxyphenyl)-N-((E)-3-(3 -amidinophenyl)-2-methyl-2-propenyl)sulfamoylacetic acid dihydrochloride for example; factor Xa inhibitors
04/29/2003US6555541 Substituted phenyl compounds with immunosuppressing activity and pharmaceutical compositions
04/29/2003CA2083980C Aminoalkylpyrrolidinylthiocarbapenem derivatives
04/24/2003WO2003033484A1 Substituted piperazine cyclohexane carboxilic acid amides and the use thereof
04/24/2003WO2003032981A1 4-(4-alkoxy-3-hydroxyphenyl)-2-pyrrolidone derivatives as pde-4 inhibitors for the treatment of neurological syndromes
04/24/2003WO2003032971A1 5’-acylamino-1,1’-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors
04/24/2003WO2003032910A2 Carbinols for the treatment of neuropathic dysfunction
04/24/2003WO2002098850A3 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
04/24/2003US20030078444 Fluorous triphase and ther multiphase systems for effecting reactions and/or separation
04/24/2003US20030078438 N-heterocyclicamide compounds; used as anticoagulant agent
04/24/2003US20030078420 New derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
04/24/2003US20030078339 Degradable cross-linking agents and cross-linked network polymers formed therewith
04/24/2003US20030078302 As carriers for delivering active agents such as peptides, drugs by administration, such as oral, subcutaneous, sublingual, and intranasal administration
04/24/2003US20030078286 For therapy of central nervous system disorders such as anxiety, depression, motor disorders
04/24/2003US20030078261 Prostaglandin agonists
04/24/2003US20030078253 Matrix metalloprotease inhibitors
04/24/2003US20030078249 VLA-4 inhibitor compounds
04/24/2003US20030078247 Enzyme inhibitor of a dipeptidyl peptidase for treating hyperglycaemia
04/24/2003US20030078241 Treating effects of excessive reactive oxygen species
04/24/2003CA2463518A1 Carbinols for the treatment of neuropathic dysfunction
04/24/2003CA2463469A1 4-(4-alkoxy-3-hydroxyphenyl)-2-pyrrolidone derivatives as pde-4 inhibitors for the treatment of neurological syndromes
04/24/2003CA2463426A1 Substituted piperazine cyclohexane carboxilic acid amides and the use thereof
04/23/2003EP1304327A2 Glutamine-thiazolidide and -pyrrolidide and their use as dipeptidylpeptidase IV inhibitors
04/23/2003EP1304323A1 Preventives or remedies for atopic dermatitis
04/23/2003EP1303509A1 Beta3 adrenergic agonists
04/23/2003EP1303503A2 Aniline derivatives
04/23/2003EP1303486A1 Pyrrolidine derivatives as metalloprotease inhibitors
04/23/2003EP1303485A1 Pyrrolidine derivatives as inhibitors of endothelin-converting enzyme
04/23/2003EP1303483A1 Novel thiourea derivatives and the pharmaceutical compositions containing the same
04/23/2003EP1303307A2 Combined therapy against tumors comprising substituted acryloyl distamycin derivatives and alkylating agents
04/23/2003EP1102739B1 Glucocorticoid and thyroid hormone receptor ligands for the treatment of metabolic disorders
04/23/2003EP1082314B1 New dipeptidyl peptidase iv effectors
04/23/2003EP1063230B1 Cyclic amino compounds
04/23/2003EP1035848B1 Substituted alkanohydroxamic acids and method of reducing tnf-alpha levels
04/23/2003EP1007032B1 4-cyano-4-deformylsordaricin derivatives
04/23/2003EP0993442B1 Hydrazine derivatives
04/23/2003EP0937041B1 Use of a pharmaceutically acceptable salt of (3R,2'R)-3-[(Cyclopently-hydroxyphenylacetyl)oxy]-1,1-dimethyl-pyrrolidinium for the preparation of a medicament
04/23/2003EP0915846B1 2- and 2,5-substituted phenylketoenols
04/23/2003EP0836615B1 New thrombin inhibitors, their preparation and use
04/23/2003CN1413217A Olefin polymerization cocatalysts derived from group-15 compounds and process using them
04/23/2003CN1413207A 5-membered ring heterocyclic compounds with nitrogen
04/23/2003CN1413193A Nitrile derivatives as cathepsin K inhibitors
04/23/2003CN1413191A Method for production of N-alkenyl amides
04/23/2003CN1413190A EP4 receptor selective agonists in treatment of osteoporosis
04/23/2003CN1413189A Benzamidine derivatives
04/23/2003CN1412181A Carboxylic acid derivative capable of inhibiting combination of integrin and its receptor
04/23/2003CN1106380C New synthetic catechol derivatives, method for production and use thereof
04/22/2003US6552225 Such as n-(2,3-dichloro-4-(methylaminosulphonyl)phenyl)-3,3,3-trifluoro-2-hydroxy-2 -methylpropanamide; diabetes, obesity, lactic acidaemia
04/22/2003US6552216 Molecular model for VLA-4 inhibitors
04/22/2003US6552090 Perfluoroalkyl haloalkyl ethers and compositions and applications thereof
04/22/2003US6552067 EP4 receptor selective agonists in the treatment of osteoporosis
04/22/2003US6552061 Amino acid derivatives and anti-inflammatory agents
04/22/2003US6552051 Useful as high energy oxidizing agents in explosive and propellant formulations, and drugs for vasodilation
04/22/2003US6552041 Cyclized amide derivatives useful for treating or preventing neuronal damage associated with neurological disease
04/22/2003US6552038 Anticoagulant agents
04/22/2003US6552022 Atherosclerosis in a mammal, pancreatitis, non-insulin dependent diabetes mellitus, coronary heart disease in a lowering serum lipid levels
04/17/2003WO2003031440A1 3,4-di-substituted maleimide compounds as cxc-chemokine receptor antagonists
04/17/2003WO2003031414A1 Novel heterocyclic compound and anti-inflammatory agent
04/17/2003WO2003030900A1 Remedies for attention-deficient/hyperreactivity disorder
04/17/2003WO2003030899A2 Use of 2-oxo-1-pyrrolidine derivatives for the treatment of dyskinesia and movement disorders
04/17/2003WO2003030897A1 Pyrrolidinone derivatives
04/17/2003WO2003030889A1 Para-amino benzoic acids as integrin antagonists
04/17/2003WO2003030886A2 Allylamides useful in the treatment of alzheimer's disease
04/17/2003WO2003013484A3 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents
04/17/2003WO2003006454A3 Heterocyclic carboxamides and their use as fungicides
04/17/2003WO2002036641A3 Improved productivity catalysts and microstructure control
04/17/2003WO2001053275A3 Substituted aryl ketones
04/17/2003WO2000037430A3 Use of androgen receptor suppressors
04/17/2003US20030073851 Arylphenyl-substituted cyclic ketoenols
04/17/2003US20030073845 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors
04/17/2003US20030073836 Heteroarylcarboxylic acid amides, the preparation thereof and their use as pharmaceutical compositions
04/17/2003US20030073832 Novel aminophenyl ketone derivatives
04/17/2003US20030073731 Alkylation therapy; anticancer agent
04/17/2003US20030073682 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors
04/17/2003US20030070241 Substituted 2-aminoalkyl-1,4-Diaminobenzene compounds and oxidation dye precursor compositions containing same
04/17/2003CA2463198A1 Pyrrolidinone derivatives
04/17/2003CA2462875A1 Allylamides useful in the treatment of alzheimer's disease
04/17/2003CA2462862A1 3,4-di-substituted maleimide compounds as cxc-chemokine receptor antagonists
04/17/2003CA2462301A1 Para-amino benzoic acids as integrin antagonists