Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304) |
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12/17/2002 | US6495525 N-((4-(((2-methylphenylamino)carbonyl)amino)phenyl)acetyl)-l -prolyl-3-methyl)-beta-alanine; very late antigen-4 cell adhesion inhibitor; inflammation and immune reactions |
12/17/2002 | US6495496 Hydroxy aromatic mannich base condensation products and the use thereof as soot dispersants in lubricating oil compositions |
12/17/2002 | CA2064783C Cytoprotective fatty moiety compounds |
12/12/2002 | WO2002099077A2 Methods and compositions related to tagging of membrane surface proteins |
12/12/2002 | WO2002098854A2 Process for preparing chiral diol sulfones and dihydroxy acid hmg coa reductase inhibitors |
12/12/2002 | WO2002098850A2 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors |
12/12/2002 | WO2002098849A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer’s disease and similar diseases |
12/12/2002 | WO2002098839A1 Biphenylcarboxamides and process for preparation thereof |
12/12/2002 | WO2002098420A1 4-substituted-1-(arylmethylidene)thiosemicarbazide, 4-substituted-1-(arylcarbonyl)thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof |
12/12/2002 | WO2002098406A1 Novel compounds and compositions as cathepsin inhibitors |
12/12/2002 | US20020188137 Low shrinkage thermosetting resin compositions and methods of use thereof |
12/12/2002 | US20020188136 Pesticides and herbicides |
12/12/2002 | US20020188120 Such as 4-(4-methyoxy-benzenesulfonyl)-1-(3-phenyl-propyl)-piperidine-4-carboxylic acid hydroxyamide for treatment of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone diseases, diabetes, and HIV |
12/12/2002 | US20020187993 Bifunctional energy-reversible acyl-compositions |
12/12/2002 | US20020187992 Prodrugs via acylation with cinnamate |
12/12/2002 | DE10125882A1 Arzneimittel enthaltend einen Effektor des Glutathionmetabolismus zusammen mit alpha-Liponsäure im Rahmen der Behandlung des Diabetes mellitus Medicines containing an effector of the glutathione metabolism together with alpha-lipoic acid in the treatment of diabetes mellitus |
12/12/2002 | CA2449813A1 Process for preparing chiral diol sulfones and dihydroxy acid hmg coa reductase inhibitors |
12/12/2002 | CA2449021A1 Novel compounds and compositions as cathepsin inhibitors |
12/12/2002 | CA2448834A1 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases |
12/12/2002 | CA2448418A1 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors |
12/11/2002 | EP1264597A2 Methods and compositions for treating cancer |
12/11/2002 | EP1263849A1 Degradable cross-linking agents and cross-linked network polymers formed therewith |
12/11/2002 | EP1263773A1 Oligonucleotide analogues, methods of synthesis and methods of use |
12/11/2002 | EP1263760A1 Novel compounds |
12/11/2002 | EP1263743A1 Heterocycle substituted diphenyl leukotriene antagonists |
12/11/2002 | EP1263730A1 Amine derivatives for the treatment of apoptosis |
12/11/2002 | EP1263729A1 Azacyclic compounds for use in the treatment of serotonin related diseases |
12/11/2002 | EP1263727A1 2-oxo-1-pyrrolidine derivatives, process for preparing them and their uses |
12/11/2002 | EP1263726A1 N-acylpyrrolidin-2-ylalkylbenzamidine derivatives as inhibitors of factor xa |
12/11/2002 | EP1263725A1 Novel compounds |
12/11/2002 | EP1263724A1 Novel compounds |
12/11/2002 | EP1263723A1 Ningalin b analogs employable for reversing multidrug resistance |
12/11/2002 | EP1263712A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds |
12/11/2002 | EP1263711A1 Novel use of phenylheteroalkylamine derivatives |
12/11/2002 | EP1058678B1 Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes |
12/11/2002 | EP0721455B1 Tetrahydropyridine-(or 4-hydroxypiperidine)alkylazoles having an affinity for sigma and/or 5ht1a receptors |
12/11/2002 | EP0662958B1 1-(2-oxo-acetyl)-piperidine-2-carboxylic acid derivatives as multi-drug-resistent cancer cell sensitizers |
12/11/2002 | EP0624155B2 Carbamates and plant-protecting agents containing them |
12/11/2002 | CN1384830A Novel spiroheterocyclic compoundsus reversible inhibitors of cysteine proteases |
12/11/2002 | CN1384820A Process for production of N-methyl pyrrolidone using gamma butyrolactone and mixed methylamines as starting materials |
12/11/2002 | CN1384743A Remedies or preventives for diseases in association with chemokines |
12/11/2002 | CN1384100A Benzo-1,3-dioxole and benzofuran substituted pentazane derivative |
12/11/2002 | CN1095835C Tricyclo-substituted isohydroxyloxime acid derivative |
12/10/2002 | USRE37936 Pesticidal 1-polyarylpyrazoles |
12/10/2002 | US6492553 A method for preparing a n-((aliphatic or aromatic)carbonyl) )-2-aminoacetamide compound, and for preparing a cyclized compound therefrom, as well as novel resin bound intermediate compounds that are useful for preparing such compounds. |
12/10/2002 | US6492541 Process for the preparation of 3-amino-2-oxo-pyrrolidines, novel intermediates and their use |
12/10/2002 | US6492534 Process and intermediate compounds for the preparation of pyrrolidines |
12/10/2002 | US6492523 Subjecting a pyrrole derivative, methyl aminocrotonate and 2-chlorobenzaldehyde to a hantzsch reaction, and converting the pyrrole residue of the resulting product to an amine group by the action of hydroxylamine hydrochloride. |
12/10/2002 | US6492428 Macrophage migration inhibitory factor (mif); substituted iminoquinone or orthoquinone ring systems |
12/10/2002 | US6492424 Glucocorticoid and thyroid hormone receptor ligands for the treatment of metabolic disorders |
12/10/2002 | US6492423 Hepatitis c and b viricides |
12/10/2002 | US6492412 Prevention of loss and restoration of bone mass by certain prostaglandin agonists |
12/10/2002 | US6492400 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity |
12/10/2002 | US6492396 Substituted thioacetamides |
12/10/2002 | US6492393 Compounds useful as anti-inflammatory agents |
12/10/2002 | US6492367 Sulfamato hydroxamic acid metalloprotease inhibitor |
12/10/2002 | US6492355 Adamantane derivatives |
12/10/2002 | US6492351 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
12/10/2002 | US6492347 Treatment and/or prophylaxis of infection caused by protozoan parasite by administering compound to inhibit purine nucleoside hydrolase, purine nucleoside phosphorylase, and/or purine phosphoribosyl transferase |
12/10/2002 | CA2036360C Reagents and methods for stereospecific fluoromethylation |
12/09/2002 | WO2002004403A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments |
12/09/2002 | CA2412116A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments |
12/05/2002 | WO2002096882A1 Substituted anilide derivatives, intermediates thereof, agricultural and horticultural chemicals, and their usage |
12/05/2002 | WO2002096876A1 Carbamate and oxamide compounds as inhibitors of cytokine production |
12/05/2002 | WO2002096872A1 Substituted imidates as pesticidal agents |
12/05/2002 | WO2002096871A1 Allylmercaptocaptopril compounds and uses thereof |
12/05/2002 | WO2002096420A2 Method for treating nerve injury caused by surgery |
12/05/2002 | WO2002096398A2 Medicament containing an effector of the glutathione metabolism together with $g(a)-lipoic acid for treating diabetes mellitus |
12/05/2002 | US20020183535 Metal catalysts and methods for making and using same |
12/05/2002 | US20020183527 Process for the preparation of amorphous atorvastatin |
12/05/2002 | US20020183523 Cis-substituted aminocyclopropane derivative |
12/05/2002 | US20020183517 Reacting dihydric alcohol characterized by four to six carbons, preferably 1,5-pentanediol, with excess ammonia in presence of ZSM-5 catalyst modified with nickel, copper or cobalt |
12/05/2002 | US20020183512 Compounds for use in treatment of cancer |
12/05/2002 | US20020183397 Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity |
12/05/2002 | US20020183378 Novel crystal forms of atorvastatin hemi-calcium and processes for their preparation as well as novel processes for preparing other forms |
12/05/2002 | US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm |
12/05/2002 | US20020183334 For therapy of sleepiness, promotion of wakefulness, treatment of Parkinson's disease, cerebral ischemia, stroke, sleep apneas, eating disorders, stimulation of appetite and weight gain, treatment of attention deficit hyperactivity disorder |
12/05/2002 | US20020183303 Activity as selective serotonin re- uptake inhibitors (SSRIs); for therapy and prophylaxis of depression, attention deficit hyperactivity disorder, obsessive- compulsive disorder, post-traumatic stress disorder, sexual dysfunction |
12/05/2002 | DE10125963A1 Substituierte Imidate Substituted Imidates |
12/05/2002 | CA2449019A1 Method for treating nerve injury caused by surgery |
12/05/2002 | CA2448626A1 Carbamate and oxamide compounds as inhibitors of cytokine production |
12/04/2002 | EP1261584A1 Crystalline forms of antibiotic side chain intermediates |
12/04/2002 | EP1261329A2 Il-8 receptor antagonists |
12/04/2002 | EP1261321A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof |
12/04/2002 | EP1001930B1 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases |
12/04/2002 | EP0858262B1 Thrombin inhibitors |
12/04/2002 | CN1095463C Prepn. method of high purity N-formyl pyrrolidine and its homolog |
12/03/2002 | US6489515 Gas-phase dehydration reaction process |
12/03/2002 | US6489491 Synthesis of compounds useful in the manufacture of ketorolac |
12/03/2002 | US6489490 Pesticides |
12/03/2002 | US6489481 Compounds used for treatment and/or prevention of neuronal apoptosis and/or excitotoxicity related neurological disorders |
12/03/2002 | US6489480 Coordination polymerization catalyst for alpha-olefins |
12/03/2002 | US6489473 Pyrroloazepine derivatives |
12/03/2002 | CA2074933C Thiazole derivatives as active superoxide radical inhibitors |
11/28/2002 | WO2002094820A1 Crystalline salts of 2-(4-{2-[2-hydroxy-3-(2-thiophen-2-yl-phenoxy)-propylamino]-2-methyl-propyl}-phenoxy)-nicotinonitrile |
11/28/2002 | WO2002094767A2 Trisubstituted-n-[(1s)-1,2,3,4-tetrahydro-1-naphthalenyl] benzamides which inhibit p2x3 and p2x2/3 containing receptors |
11/28/2002 | WO2002094748A1 Impurity inhibition in olefin metathesis reactions |
11/28/2002 | WO2002094311A1 Use of proteasome inhibitors to treat dry eye disorders |
11/28/2002 | WO2002094261A1 Cxcr4-antagonistic drugs comprising nitrogen-containing compound |
11/28/2002 | WO2002094220A1 Liquid pharmaceutical composition |