| Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304) |
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| 09/12/2003 | WO2003074049A1 Antitumor agents |
| 09/12/2003 | WO2003073999A2 Pini-modulating compounds and methods of use thereof |
| 09/12/2003 | WO2003002522A3 Peptide deformylase inhibitors |
| 09/12/2003 | CA2477749A1 Artificial receptors, building blocks, and methods |
| 09/12/2003 | CA2477715A1 8-azaprostaglandin derivative compound and agent comprising the compound as active ingredient |
| 09/11/2003 | WO2003074500A2 N-aminoacetyl-pyrrolidine-2-carbonitriles and their use as ddp-iv inhibitors |
| 09/11/2003 | WO2003074482A1 Method for the simultaneous production of tetrahydrofurans and pyrrolidones |
| 09/11/2003 | US20030171599 An alpha-diazoacetamide is reacted under conditions promoting intramolecular C-H insertion, for example in the presence of a rhodium salt such as Rh2(OAc)4 |
| 09/11/2003 | US20030171578 Pyrrolidinone derivative compound |
| 09/11/2003 | US20030171404 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors |
| 09/11/2003 | US20030171377 Therapy for non-insulin dependent diabetes |
| 09/11/2003 | US20030171361 Treatment of impotence, sexual dysfunction in female, stable, unstable and variant angina, hypertension, pulmonary hypertension, congestive heart failure, atherosclerosis |
| 09/11/2003 | US20030171352 Sulfonylaminocarboxylic acid N-arylamides as guanylate cyclase activators |
| 09/11/2003 | US20030171309 Pharmaceutically active pyrrolidine derivatives as bax inhibitors |
| 09/11/2003 | US20030171301 Novel form of (S)-1-(N2-(1-carboxy-3-phenylpropyl)-L-lysyl)-L-proline known under the generic name lisinopril. Further, the present invention also relates to the use of the novel amorphous form of lisinopril |
| 09/11/2003 | US20030171219 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides |
| 09/11/2003 | US20030171218 Substituted 3-heteroaryl(amino- or oxy) pyrrolidin-2-ones of the formula (I), processes for preparing them, and their use as herbicides or as plant growth regulators. |
| 09/11/2003 | US20030170917 4-Hydroxyalkylphenethamines, used as an intermediate, hapten, or immunogen in the production of antibodies specific for ecstasy drugs; binding the antibody to the analyte and detecting the adduct formed; immunoassay |
| 09/11/2003 | US20030170381 Piezoelectric element and process for production thereof |
| 09/10/2003 | EP1342718A1 Method and reagents for n-alkylating ureides |
| 09/10/2003 | EP1341785A2 HYDROLYSIS OF R(R*,R*)]-2-(4-FLUOROPHENYL)-$g(b),$g(d) -DIHYDROXY-5-(1-METHYLETHYL)-3-PHENYL-4- (PHENYLAMINO)CARBONYL]-1H-PYRROLE-1-HEPTANOIC ACID ESTERS WITH CALCIUM HYDROXIDE |
| 09/10/2003 | EP1341780A2 Substituted heterocyclic phthalic acid diamide arthropodicides |
| 09/10/2003 | EP1341758A2 Coniosetin and derivatives thereof, method for producing the same and use thereof |
| 09/10/2003 | EP1341757A1 Pyrrolcarboxamides and pyrrolcarbothioamides and their agrochemical uses |
| 09/10/2003 | EP1341755A1 Carboxylic acid amide derivatives and their use in the treatment of thromboembolic diseases and tumours |
| 09/10/2003 | EP1127871B1 New esters derived from substituted phenyl-cyclohexyl compounds |
| 09/10/2003 | EP1082300B1 3-[(1'-n-methylamino)ethyl-n-benzyl]pyrrolidine monomethanesulfonate |
| 09/10/2003 | EP0991619B1 Inhibitors of alpha 4-beta 1 mediated cell adhesion |
| 09/10/2003 | EP0934264B1 Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists |
| 09/10/2003 | CN1441800A Beta 3 adrenergic agonists |
| 09/10/2003 | CN1441779A Proline derivatives and use thereof as drugs |
| 09/10/2003 | CN1441771A Method for producing 3,3-diarylpropylamines |
| 09/09/2003 | US6617480 Molecular weight-enlarged ligands for asymmetric, homogeneously soluble hydrogenation catalysts, process for the production thereof and use |
| 09/09/2003 | US6617454 Process for the preparation of amine oxides |
| 09/09/2003 | US6617320 Protease inhibitor; anticoagulants |
| 09/09/2003 | US6617317 Boronic ester and acid compositions |
| 09/04/2003 | WO2003072556A1 Glutaminyl based dpiv inhibitors |
| 09/04/2003 | WO2003072546A1 Novel coupling agents, the active intermediates and the conjugates thereof and the use of said conjugates in diagnostic methods |
| 09/04/2003 | WO2003072545A1 Cyclic amine compound and ccr3 inhibitory drug containing the same as active ingredient |
| 09/04/2003 | WO2003072544A1 Crystalline anhydrous and monohydrate benzoate salts of (2's,3s)-3-hydroxy-n-{2{n-methyl-n-4-(n-propylamino-carbonyl)phenyl]amino-2-phenyl}-ethylpyrrolidine |
| 09/04/2003 | WO2003072535A2 Substituted hydroxyethylamines |
| 09/04/2003 | WO2003072532A1 Ester compound and medicinal use thereof |
| 09/04/2003 | WO2002074737A3 Process for the preparation of 2-hydroxymethyl-pyrolidine-3,4-diols |
| 09/04/2003 | WO2002032376A3 Bile-acid conjugates for providing sustained systemic concentrations of drugs |
| 09/04/2003 | US20030166947 Extraction, purification |
| 09/04/2003 | US20030166926 Pyrroloazepine derivatives |
| 09/04/2003 | US20030166717 Substituted amide compound containing hydroxy and amino groups; useful for treating Alzheimer's disease and other similar diseases |
| 09/04/2003 | US20030166707 Tetramic acid derivatives, useful in treating or preventing bacterial diseases, especially diseases caused by gram-positive pathogens resistant to other antibiotics |
| 09/04/2003 | US20030166693 Benzene derivatives and pharmaceutical use thereof |
| 09/04/2003 | US20030166690 Use of compounds for decreasing activity of hormone-sensitive |
| 09/04/2003 | US20030166685 Acid derivatives of benzene useful as anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and as metastasis inhibitors in treating cancer |
| 09/04/2003 | US20030166681 Aminopyrrolidine sulfonamides as serine protease inhibitors |
| 09/04/2003 | US20030166680 For treating serine protease or dual-serine protease mediated disorders |
| 09/04/2003 | US20030166674 1-Azabicyclo[2.2.2]octan-3-one derivatives and maleimide derivatives and their use for treating cancer tumors |
| 09/04/2003 | US20030166668 Substituted heteroarylalkanoic acids |
| 09/04/2003 | US20030166644 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase |
| 09/04/2003 | CA2479812A1 Glutaminyl based dpiv inhibitors |
| 09/04/2003 | CA2477634A1 Crystalline anhydrous and monohydrate benzoate salts of (2's,3s)-3-hydroxy-n-{2{n-methyl-n-4-(n-propylamino-carbonyl)phenyl]amino-2-phenyl}-ethylpyrrolidine |
| 09/04/2003 | CA2477607A1 Substituted hydroxyethylamines |
| 09/03/2003 | EP1340980A1 Derivatives of amphetamine, antibodies against said derivatives, reagent kits, methods of producing said antibodies, and methods of detecting said derivatives |
| 09/03/2003 | EP1340744A2 Hiv protease inhibitors |
| 09/03/2003 | EP1339685A2 Biphenylcarboxamides useful as lipid lowering agents |
| 09/03/2003 | EP1339684A1 Mch antagonists and their use in the treatment of obesity |
| 09/03/2003 | EP1339678A2 Ep4 receptor selective agonists in the treatment of osteoporosis |
| 09/03/2003 | EP1339677A1 Aminoalkylpyrrolidine serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their synthesis |
| 09/03/2003 | EP1339670A1 Substituted cyclohexane derivates and the use thereof in medicaments for treating cardiovascular diseases |
| 09/03/2003 | EP1339668A2 Bisubstituted carbocyclic cyclophilin binding compounds and theirus |
| 09/03/2003 | EP1060178B1 Heterocyclic compounds as inhibitors of rotamase enzymes |
| 09/03/2003 | EP0975588B1 Antipicornaviral compouds, compositions containing them, and methods for their use |
| 09/03/2003 | EP0775689B1 Novel amine derivative, process for producing the same, and use thereof as antiarrhythmic |
| 09/03/2003 | EP0612318B1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics |
| 09/03/2003 | CN1440405A Sulfonyl-pyrrolidine derivatives useful for treatment of neurological disorders |
| 09/03/2003 | CN1440390A Substituted diamide derivatives useful as motilin antagonists |
| 09/03/2003 | CN1440385A Pyrrole derivatives for treating AIDS |
| 09/03/2003 | CN1440383A PPARγ调制剂 PPARγ modulators |
| 09/03/2003 | CN1440381A Process for preparation of substituted octanoyl amides |
| 09/03/2003 | CN1439634A Preparation of 2-aryl-5-(trifluoride) pyrrole-3-nitrile and its use and preparation of its intermediate thereof |
| 09/03/2003 | CN1439633A Deodorant N-vinyl-2-pyrrolidone production |
| 09/03/2003 | CN1120167C Tetrahydropyridine-(or 4-hydroxypiperidine) alkylazoles having an affinity for alpha and/or 5HTIA receptors |
| 09/03/2003 | CN1120153C Novel 2,2'-Bi-1H-pyrrole derivatives with immunosuppressant activity |
| 09/03/2003 | CN1120152C Beta-halogamma-hydroxypyrrolidone and its synthesis process |
| 09/02/2003 | US6613920 25-(5-propylimidazol-2-yl)-26,27-cyclo-9, 10-secocholesta-5,7,10(19),22-tetraene-1,3,24-triol; antagonizes the action of calcitriol in HL 60 cells; hyperprolifierative diseases of the skin, tumor diseases and precancerous stages |
| 09/02/2003 | US6613916 Process for the preparation of amorphous atorvastatin |
| 09/02/2003 | US6613915 Polymerization of olefins |
| 09/02/2003 | US6613795 Respiratory system disorders; muscle relaxants |
| 09/02/2003 | US6613793 Anticancer activity of imino acid conjugates or methylglyoxal |
| 09/02/2003 | US6613791 N-substituted azaheterocyclic carboxylic acids and their use |
| 09/02/2003 | US6613787 Compounds that exhibit specific molecular recognition of mixed nucleic acid sequences and bind in the DNA minor groove as a dimer |
| 09/02/2003 | US6613764 Aspartic protease inhibitors |
| 08/28/2003 | WO2003070755A2 Compounds, compositions and method for transporting cyclosporin molecules through the blood brain barrier |
| 08/28/2003 | WO2003070702A1 Novel crystal forms of atorvastatin hemi-calcium and processes for their preparation, as well as novel processes for preparing atorvastatin hemi-calcium forms i, viii and ix |
| 08/28/2003 | WO2003070665A2 Desolvating solvates of atorvastatin hemi-calcium |
| 08/28/2003 | WO2003057131A3 Novel process for the preparation of trans-3- ethyl-2,5- dihydro-4- methyl-n-[2-[ 4-[[[[(4-methyl cyclohexyl) amino]carbonyl] amino]sulfonyl] phenyl]ethyl] -2-oxo-1h-pyrrole -1-carboxamide |
| 08/28/2003 | US20030162966 Reacting an amino alcohol derivative with a sulfonyl halide in a mixed solvent composed of an aprotic organic solvent and water in the presence of a non- water-prohibiting inorganic base to produce sulfonic acid ester derivative |
| 08/28/2003 | US20030162960 Compounds containing pyrroles as the key recognition element and a quinoxaline backbone as part of the compound for use in system with a built-in optical probe for selective sensing |
| 08/28/2003 | US20030162851 Methods of making intermediates from polyhydroxyalkanoates |
| 08/28/2003 | US20030162826 Degradation fragments |
| 08/28/2003 | US20030162820 Heterocyclic amides used as dipeptidyl aminopeptidase (DPIV) inhibitors, for prophylaxis of arthritis, obesity, allograft surgery, cancer, autoimmune, nervous system and skin disorders |
| 08/28/2003 | US20030162811 Heterocyclic amines such as 4-(3'-Thienyl)-alpha, alpha, 1-trimethyl-4-piperidinemethanol and/or prodrugs, used as analgesics for prophylaxis of neuropathic pain |
| 08/28/2003 | US20030162789 4-alkylpiperazine substituted phenol derivative or 4-alkylamide substituted phenols for treating neurodegerative diseases such as aging, cancer, diabetes, ischemic stroke, Parkinson's disease, dementia and Huntinton's disease |