Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
08/2003
08/28/2003US20030162787 Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade
08/28/2003US20030162778 Carbocyclic side chain containing metalloprotease inhibitors
08/28/2003US20030162776 Substituted 5-membered polycyclic compounds useful for selective inhibition of the coagulation cascade
08/28/2003US20030162772 For example, N-(2-(3-((1-(3,4-dichlorobenzylpiperidinyl) aminohydroxypropoxy)phenyl)acetamide; use as modulators of chemokine receptor activity, and may be used in treatment of autoimmune, inflammatory, proliferative diseases
08/28/2003US20030162198 Medical diagnosis; complexing to Dna; calibration
08/28/2003CA2475864A1 Novel crystal forms of atorvastatin hemi-calcium and processes for their preparation, as well as novel processes for preparing atorvastatin hemi-calcium forms i, viii and ix
08/28/2003CA2475123A1 Desolvating solvates of atorvastatin hemi-calcium
08/27/2003EP1338588A1 Method of resolving optical isomers of amino acid derivative
08/27/2003EP1338336A1 Catalysts comprising n-substituted cyclic imides and processes for preparing organic compounds with the catalysts
08/27/2003EP1337532A2 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit
08/27/2003EP1337511A1 Bis-heterocyclic compounds with antitumour and chemosensitising activity
08/27/2003EP1257360A4 Chiral ferrocene phosphines and their use in asymmetric catalytic reactions
08/27/2003EP1165547B1 Substituted benzoylpyrazoles as herbicides
08/27/2003EP1073672B1 Antipicornaviral compounds, their preparation and use
08/27/2003EP0874809B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials
08/27/2003EP0862552B1 Succinimide and maleimide cytokine inhibitors
08/27/2003EP0802182B1 PROCESS FOR PRODUCING N-(D-alpha-METHYL-beta-MERCAPTOPROPIONYL)-L-PROLINE AND INTERMEDIATES THEREOF
08/27/2003CN1439010A Pyrrolo [2,3-d] pyrimidine compounds as immunosuppressive agents
08/27/2003CN1439006A Novel compounds possessing antibacterial, antifungal or antitumor activity
08/27/2003CN1439005A Pyrrole substituted 2-indolinone protein kinase inhibitors
08/27/2003CN1438999A Serine protease inhibitors
08/27/2003CN1438991A Cyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase
08/27/2003CN1119346C Benzothiadiaxoles and derivatives
08/27/2003CN1119340C Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4
08/27/2003CN1119147C Kappa-opiate agonists for inflammatory bowel disorders
08/26/2003US6610889 Using organometallic complex catalyst
08/26/2003US6610850 Contrast media for angiography
08/26/2003US6610731 Antiinflammatory
08/26/2003US6610730 Viricides; protease inbhibitor
08/26/2003US6610719 Use of prostaglandin (PGE2) receptor a (EP4) selective agonists for the treatment of acute and chronic renal failure
08/26/2003US6610710 Inflammatory bowel diseases, diabetes, tumor proliferation and tumor metastasis.
08/26/2003US6610708 Cyclic amino compounds
08/26/2003US6610707 Heterocyclic compounds as inhibitors of rotomase enzymes
08/26/2003US6610705 Process for the preparation of diaryl naphthyl methanes
08/26/2003US6610702 Ammonium salts of inositol hexaphosphate, and uses thereof
08/26/2003US6610660 O2-arylated or O2-glycosylated 1-substituted diazen-1-ium-1,2-diolates and O2-substituted 1-[(2-carboxylato) pyrrolidin-1-yl] diazen-1-ium-1,2-diolates
08/26/2003US6610284 Preparation for prevention and healing of inflammation affections
08/21/2003WO2003069303A2 Antimalarial and antiproliferative pharmacophore models, novel tryptanthrin compounds having increased solubility, and methods of making and using thereof
08/21/2003WO2003068740A1 Pyrrolylalkylidene-hydrazinecarboximidamide derivatives as 5-hydroxytryptamine-6 ligands
08/21/2003WO2003068739A1 Method of manufacturing an amorphous form of the hemi-calcium salt of (3r, 5r) 7- 3-phenyl-4-phenylcarbamoyl-2-(4-fluorophenyl)-5-isopropyl-pyrrol-1-yl!-3, 5-dihydroxyheptanoic acid (atorvastatin)
08/21/2003WO2003068738A1 Pyrrole derivatives as ligands of melanocortin receptors
08/21/2003WO2003068212A1 Use of sodium/hydrogen exchange inhibitors from the treatment of thrombotic and inflammatory diseases
08/21/2003WO2003067986A1 Δ1 pyrrolines and the use thereof in pest control
08/21/2003WO2003018549A3 Bicyclic compounds as inhibitors of chemokine binding to us28
08/21/2003WO2003007930A3 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors
08/21/2003WO2002062755A3 Polyamide analogs as dna minor groove binders
08/21/2003WO2002046158A3 Piperidine/piperazine-type inhibitors of p38 kinase
08/21/2003WO2002002512A3 Compounds to treat alzheimer's disease
08/21/2003US20030158441 Methods of making intermediates from polyhydroxyalkanoates
08/21/2003US20030158274 Hydrogenolyzing a polylactone to form a diol.
08/21/2003US20030158252 Especially trypsin-like serine proteases, such as chymotrypsin, trypsin, thrombin, plasmin and factor Xa.
08/21/2003US20030158225 Novel compounds
08/21/2003US20030158186 Compositions and methods for treating heart failure
08/21/2003US20030158185 Novel use of phenylheteroakylamine derivatives
08/21/2003US20030158173 NK 1 antagonists
08/21/2003CA2476446A1 Use of sodium/hydrogen exchange inhibitors from the treatment of thrombotic and inflammatory diseases
08/20/2003EP1335988A2 Synthesis of chiral intermediates useful in preparing pharmacologically active compounds
08/20/2003EP1335901A1 Pharmaceutically active sulfanilide derivatives
08/20/2003EP1335898A1 Carbamic acid compounds comprising an amide linkage as hdac inhibitors
08/20/2003EP1150944B1 N2-phenylamidine derivatives
08/20/2003EP0831829B1 Heterocyclic ring-fused pyrimidine derivatives
08/20/2003CN1437583A Trifluoromethylpyrrole carboxamides and trifluoromethylpyrrolethioamides as fungicides
08/20/2003CN1437578A (P-amino-hyaroxyphenyl)-acrylamide derivatives and dyes containing said compounds
08/20/2003CN1437485A Combined therapy against tumors comprising substituted acryloyl distamycin derivatives and alkylating agents
08/20/2003CN1437484A New formulation comprising a beta-blocker and optionally a cholesterol-lowering agent
08/20/2003CN1437473A Combined therapy against tumors comprising substituted acryloyl distamycin derivatives, taxanes and/or antimetabolites
08/20/2003CN1118467C 1,3,8-triaza-spiro [4,5] decan-4-on derivatives
08/19/2003US6608227 Benzylcycloalkyl amines as modulators of chemokine receptor activity
08/19/2003US6608196 Structurally diverse; parallel approach
08/19/2003US6608095 Sulfonylbenzene and sulfonamidobenzene compounds which inhibit COX-2; treatment of a medical condition in which prostaglandins are implicated as pathogens
08/19/2003US6608093 Polyarylpyrazole or polyarylpyrole or polyaryltriazole compounds or intermediates for pesticides
08/19/2003US6608061 Bisaryl compound and medicament for cancer treatment comprising the same
08/19/2003US6608019 Alkoxy-substituted perfluorocompounds
08/14/2003WO2003066889A2 Assay for acytyltransferase or deacetylase activity
08/14/2003WO2003066579A2 Novel bicyclic hydroxamates as inhibitors of histone deacetylase
08/14/2003WO2003066574A1 Aromatic amino acid derivatives and medicinal compositions
08/14/2003WO2003066035A2 Compounds for inhibiting insulin secretion and methods related thereto
08/14/2003US20030153788 Oxidizing an amino alcohol (obtained by ring opening the epoxy, aziding, reducing and reacting it with a carboxylic acid); stereoselectivity; protease inhibitors: antiallergens; anticarcinogenic and hypotensive agents
08/14/2003US20030153611 Antitumor agents promoting the detachment of endothelial cells forming tumor, inhibiting tubulin polymerization
08/14/2003US20030153596 Novel thiourea derivatives and the pharmaceutical compositions containing the same
08/14/2003US20030153577 Cyclic amine derivatives-CCR-3 receptor antagonists
08/14/2003US20030153559 Treatment of an oxygen and/or energy deficit; a poly(adenosine diphosphate ribose)-polymerase inhibitor; treating autoimmune, neurodegenerative and diseases caused by a toxic effect; viricides
08/14/2003US20030153555 Novel compounds
08/14/2003US20030153507 HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
08/14/2003US20030153465 Substituted aryl ketones
08/14/2003CA2473505A1 Novel bicyclic hydroxamates as inhibitors of histone deacetylase
08/13/2003EP1335250A1 Electrophotographic organophotoreceptors with novel charge transport materials
08/13/2003EP1334961A1 Process for the preparation of glycine-N,N-diacetic acid derivatives
08/13/2003EP1334097A2 Process for the preparation of ligands for olefin polymerization catalysts
08/13/2003EP1334085A1 Sulfamides as gamma-secretase inhibitors
08/13/2003EP1334084A2 Phosgene-free process for preparing carbamates
08/13/2003EP1334083A2 1,4-disubstituted benzenes as insecticides
08/13/2003EP1222166B1 Novel p-aminophenols and colorants containing said compounds
08/13/2003EP1019411A4 Process for synthesizing carbapenem side chain intermediates
08/13/2003EP0470128B2 Active carbonates of polyalkylene oxides for modification of polypeptides
08/12/2003US6605729 Crystalline forms of [R-(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1)
08/12/2003US6605728 Starting from atorvastatin lactone, where continuous agitation at a very low speed provides optimum drying conditions for avoiding clod formation and particle attrition
08/12/2003US6605677 Olefin polymerization processes using supported catalysts
08/12/2003US6605636 Atorvastatin hemi-calcium form VII
08/12/2003US6605632 Affinity for melatonin receptors