Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
02/2003
02/05/2003CN1395467A Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
02/05/2003CN1100778C Pyrrolopyriidines and processes for preapring thereof
02/05/2003CN1100535C Pharmaceutical agents for treatment of emesis
02/04/2003US6515179 Process for the removal of nitrobenzenesulfonyl
02/04/2003US6515167 Said process comprising reacting a carboxylic acid or salt thereof having formula (I) with dimethyl carbonate having formula (II) in the presence of a catalyst selected from the group consisting of 1,8 diazabicyclo(5.4.0)undec-7-ene;
02/04/2003US6515155 Group 4 metal complexes of the constrained geometry type, catalysts derived therefrom and polymerization processes using the same, characterized by a nitrogen containing aliphatic or cycloaliphatic moiety that is substituted with one or more
02/04/2003US6515143 Method for producing ortho-alkylated benzoic acid derivatives
02/04/2003US6515142 Intermediates of aromatic amidine derivatives which have anticoagulation action
02/04/2003US6515027 Substituted benzanilides as CCR5 receptors ligands, antiinflammatory agents and antiviral agents
02/04/2003US6515024 Succinoylamino hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors
02/04/2003US6515023 Thrombin receptor antagonists
02/04/2003US6515021 The compounds according to the invention have pronounced activity in the fields of cell differentiation and cell proliferation
02/04/2003US6515013 For diseases or conditions caused by or exacerbated by histamine-3 receptor activity
02/04/2003US6515012 Reacting 3-benzoylthio-2-methylpropionoic acid chloride with 4-phenylthio-L-proline; hypotnsive agents
02/04/2003US6515011 Anticoagulants
02/04/2003US6514992 Caspases and apoptosis
02/04/2003US6514970 Urotensin-II receptor antagonists
02/04/2003US6514925 O-substituted N,N-diacylhydroxylamine bleach activators and compositions employing the same
02/04/2003US6514664 Radiation sensitive compositions containing image quality and profile enhancement additives
01/2003
01/30/2003WO2003008410A2 Polypyrroles as agents for treating cancer, treating viral diseases and causing immunosuppression
01/30/2003WO2003008380A1 Carboxylic acid derivatives
01/30/2003WO2003008379A1 Azasugar compounds
01/30/2003WO2003008378A1 Dolastatin 10 derivatives
01/30/2003WO2003008377A1 Prostaglandin analogues_as ep4 receptor agonists
01/30/2003WO2003008371A1 Substituted 4-aminocyclohexanol derivatives
01/30/2003WO2003007954A2 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors
01/30/2003WO2003007941A1 2 pyrrolidone derivatives as prostanoid agonists
01/30/2003WO2003007930A2 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors
01/30/2003WO2003002522A8 Peptide deformylase inhibitors
01/30/2003US20030023123 Reduced production of unwanted byproducts; purity, efficiency
01/30/2003US20030023100 For therapy of inflammatory and allergic reactions, drug or alcohol abuse, diarrhoea, gastritis, ulcers, cardiovascular diseases, urinary incontinence, depressions, states of shock, migranes, narcolepsy, overweight, asthma, glaucoma, etc.
01/30/2003US20030023087 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
01/30/2003US20030023031 Acryloyl substituted distamycin derivatives, process for preparing them, and their use as antitumor and antiviral agents
01/30/2003US20030022891 Melanin-concentrating hormone (MCH); treating metabolic and eating disorders, such as hyperphagia, and diabetes; urea, thiourea and cyano-guanidine compounds of given formula
01/30/2003CA2453987A1 Dolastatin 10 derivatives
01/30/2003CA2453636A1 Polypyrroles as agents for treating cancer, treating viral diseases and causing immunosuppression
01/30/2003CA2453613A1 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors
01/30/2003CA2453602A1 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors
01/30/2003CA2451392A1 Prostaglandin analogues as ep4 receptor agonists
01/29/2003EP1278784A2 Catalysts containing n-pyrrolyl substituted nitrogen donors
01/29/2003EP1278743A1 Novel anti-infectives
01/29/2003EP1278733A1 Process for the preparation of sterically hindered aryloxyamines
01/29/2003EP1278728A1 Pyrrolidine and piperidine derivatives and their use for the treatment of neurodegenerative disorders
01/29/2003EP1278726A1 Method for producing cyclic lactams
01/29/2003EP1278723A2 P-(sulfonyl)-aryl and -heteroaryl amines
01/29/2003EP1192145A4 Process for preparing chiral cyclopropane carboxylic acids and acyl guanidines
01/29/2003EP0910573B1 New amino acid derivatives and their use as thrombin inhibitors
01/29/2003EP0835243B1 Dialkyl phenyl halide-substituted keto-enols for use as herbicides and pesticides
01/29/2003EP0832081B1 Bicyclic-aromatic compounds
01/29/2003EP0817772B1 Pyrrolidinyl hydroxamic acid compounds and their production process
01/29/2003EP0754175B1 Alkoxy-alkyl-substituted 1-h-3-aryl-pyrrolidine-2,4-diones used as herbicides and pesticides
01/28/2003US6512120 Functionalized pyrrolidine compounds through the use of intramolecular Diels Alder reactions. further in situ and resin-bound synthetic generation of chemical libraries.
01/28/2003US6512101 Branched hydrazone linkers
01/28/2003US6512001 D-proline derivatives
01/28/2003US6511980 For therapy of gastrointestinal reflux disorders, eating disorders leading to obesity and irritable bowel disorder
01/28/2003US6511942 Animal husbandry, veterinary medicine
01/28/2003US6511663 Tri- and tetra-valent monospecific antigen-binding proteins
01/28/2003CA2083534C Indolopyrrolocarbazole derivatives
01/24/2003WO2002016308A1 Phenyl- and phenylalkyl-substituted ethanolamines and ethylenediamines
01/23/2003WO2003006454A2 Heterocyclic carboxamides and their use as fungicides
01/23/2003WO2003006423A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003WO2003005824A2 Substituted 3-heteroaryl (amino-or-oxy)-pyrrolidin-2-ones, method for the production thereof and use thereof as herbicides or as plant growth regulators
01/23/2003WO2002055491A3 1,2-DISUBSTITUTED CYCLIC INHIBITORS OF MATRIX METALLORPROTEASES AND TNF-$g(a)
01/23/2003US20030018202 Production method of pyrrolidone carboxylic acid and salt thereof
01/23/2003US20030018199 Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors
01/23/2003US20030018080 N-methoxymethyl-5,5-diphenylbarbituric acid
01/23/2003US20030018070 Bisaryl compound and medicament for cancer treatment comprising the same
01/23/2003US20030017964 Administration of agents via the PEPT-2 transporter
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/22/2003WO2002010131A1 Pyrrole derivatives
01/22/2003EP1277751A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277749A1 2- and 2,5-substituted phenylketo enols
01/22/2003EP1277735A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277734A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277733A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277729A1 Ppar (gamma) modulators
01/22/2003EP1277728A1 Novel TTDA derivatives and their use as gadolinium chelators for MRI imaging
01/22/2003EP1276732A1 Amides of r-2-(aminoaryl)-propionic acids for use in theprevention of leucocyte activation"
01/22/2003EP0898562B1 Hydroxamic acid derivatives for use with the treatment of diseases related to connective tissue degradation
01/22/2003EP0844241B1 Inhibitor for narcotic analgetic dependence/resistance acquisition
01/22/2003CN1392137A New cyclic alpha-amino-gamma hydroxy amide compound, its preparing method and medicinal composition containing said compound
01/22/2003CN1099425C 新的肽衍生物 New peptide derivatives
01/22/2003CA2416946A1 Pyrrole derivatives
01/21/2003US6509477 Small molecule inhibitors of rotamase enzyme activity
01/21/2003US6509474 Method of lithiating five membered heterocycles
01/21/2003US6509359 Pyrrolidin-2-one compounds and their use as neuraminidase inhibitors
01/21/2003US6509356 1-(4-(Substituted alkoxy)benzyl)naphthalene compounds having estrogen inhibitory activity
01/21/2003US6509309 Cleaning composition comprising alkoxy substituted perfluoro compounds
01/21/2003US6508957 Fluorescent maleimides and uses thereof
01/17/2003WO2002006269A1 Cyclic amino acid derivatives
01/17/2003CA2415964A1 Cyclic amino acid derivatives
01/16/2003WO2003004472A1 Arylamines for the treatment of conditions associated with gsk-3
01/16/2003WO2003004470A1 Crystalline forms of 'r-(r*,r*)!-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-'phenylamino)carbonyl!-1h-pyrrole-1-heptanoic acid calcium salt (2:1) (atorvastatin)
01/16/2003WO2003004469A1 Anticancer activity of imino acid conjugates of methylglyoxal
01/16/2003WO2003004468A1 Compounds having prolyl oligopeptidase inhibitory activity, methods for their preparation and their use
01/16/2003WO2003004457A2 Preparation process for atorvastatin and intermediates
01/16/2003WO2003004456A1 Process for the preparation of 7-amino syn 3,5-dihydroxy heptanoic acid derivatives via 6-cyano syn 3,5-dihydroxy hexanoic acid derivatives
01/16/2003WO2003004455A2 Process for the preparation of 7-amino syn 3,5-dihydroxy heptanoic acid derivatives, intermediates thereof and methods for their preparation
01/16/2003WO2003004450A1 Process for the preparation of intermediates useful in the synthesis of statin derivatives especially 7-amino 3,5-dihydroxy heptanoic acid derivatives, and intermediates thereof
01/16/2003WO2003004020A1 Heteroaryl carboxylic acid amides, the production thereof and the use of the same as inhibitors of the microsomal triglyceride transfer protein (mtp)