Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
01/2004
01/14/2004CN1134411C Bicyclic amino derivatives and PGD2 antagonist containing same
01/14/2004CN1134410C Amine derivative, process for producing same, and use thereof as antiarrhythmic medicine
01/14/2004CN1134264C Antithrombotic agents
01/13/2004US6677487 Combining a tertiary amide with a pentavalent phosphorous halide in a solvent to form an alpha - haloiminium salt and converting the alpha -haloiminium salt to the alpha -haloenamine with a base
01/13/2004US6677382 Halogenated oxyamines, used as enzyme inhibitors for prophylaxis of atherosclerosis and cardiovascular disorders, and as antilipemic agents
01/13/2004US6677380 Antilipemic agents such as 3(3-(4-chloro-3-ethyl-phenoxy)-phenyl)((3-(1,1,2,2 -tetrafluoroethoxy)phenyl)methyl))amino)-1,1,1-trifluro-2-propanthiol, used for prophlaxis of cardiovascular disorders and atherosclerosis
01/13/2004US6677379 Such as 3-((3-(3-trifluoromethoxyphenoxy)phenyl)((3-(1,1,2,2-tetrafluoroethoxy) -phenyl)methyl) amino)-1,1,1-trifluoro-2-propanol for treatment of coronary artery disease
01/13/2004US6677378 Monoamine reuptake inhibitors for treatment of CNS disorders
01/13/2004US6677375 Substituted N,N-bis-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
01/13/2004US6677360 Biphenyl and biphenyl-analogous compounds as integrin antagonists
01/13/2004US6677353 Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
01/08/2004WO2004002977A1 Inhibitors of hcv ns5b polymerase
01/08/2004WO2004002944A1 Inhibitors of hcv ns5b polymerase
01/08/2004WO2004002943A1 4-(3,3-dihalo-allyloxy)phenoxy alkyl derivatives
01/08/2004WO2004002940A1 Inhibitors of hcv ns5b polymerase
01/08/2004WO2004002491A1 Morpholine and tetrahydropyran drivatives and their use as cathepsin inhibitors
01/08/2004WO2003030899A3 Use of 2-oxo-1-pyrrolidine derivatives for the treatment of dyskinesia and movement disorders
01/08/2004US20040006236 Diaminopropionic acid derivatives
01/08/2004US20040006233 Synthetic multimerizing agents
01/08/2004US20040006231 Process for the synthesis of 1,3-diols
01/08/2004US20040006166 Compatible with a wide variety of adhesive formulations and which provide substantial adhesion enhancement relative to base formulations to which they are added
01/08/2004US20040006107 For prophylaxis of asthma and other allergic diseases
01/08/2004US20040006096 Substituted alkanohydroxamic acids and method of reducing TNFalpha levels
01/08/2004US20040006078 For therapy of autoimmune diseases, asthma, osteoporosis, atherosclerosis, Alzheimer's disease
01/08/2004US20040006049 For therapy of prostatitis, benign prostate hyperplasia or prostate cancer
01/08/2004US20040006023 Intravenous administration of a alpha -halogen- acryloyl distamycin derivative for therapy of tumors
01/08/2004CA2491156A1 Inhibitors of hcv ns5b polymerase
01/08/2004CA2490950A1 Inhibitors of hcv ns5b polymerase
01/08/2004CA2489433A1 Inhibitors of hcv ns5b polymerase
01/08/2004CA2488525A1 Morpholine and tetrahydropyran derivatives and their use as cathepsin inhibitors
01/07/2004EP1378230A1 Para-phenylenediamine derivatives comprising a pyrrolidinyl group substituted by a cyclic radical and their use in colouring keratinic fibres
01/07/2004EP1377543A1 Oxalic acid derivatives
01/07/2004EP1377295A2 Carboxamide derivatives as therapeutic agents
01/07/2004EP1377278A1 Treatment of type 2 diabetes with inhibitors of dipeptidyl peptidase iv
01/07/2004EP1056733B1 Histamine h3 receptor ligands
01/07/2004CN1466572A 吡咯衍生物 Azole derivatives
01/07/2004CN1466571A Method for producing delta 1-pyrrolines
01/06/2004US6673920 Method for the production of N-alkenyl-amides
01/06/2004US6673829 Treatment of diseases of the central nervous system, the peripheral nervous system, the cardiovascular system, the pulmonary system, the gastrointestinal system and the endocrinological system.
01/06/2004US6673817 Anticoagulants
01/06/2004US6673803 Quinazoline derivatives and pharmaceutical compositions containing them
01/06/2004US6673772 Dipeptide compounds and their use as antiviral agents
01/06/2004US6673257 Blends employing at least two organic compounds having known melt temperatures, exhibit improved thermal properties and performance characteristics
01/02/2004EP1375482A1 Benzamidine derivative
01/02/2004EP1375481A1 Method of purifying n-(2-hydroxyethyl)-2-pyrrolidone
01/02/2004EP1375480A1 Para-phenylene-diamine derivatives comprising a silyl substituted pyrrolidine group and their use for the colouring of keratinic fibres
01/02/2004EP1375479A1 Pyrrolidine derivative and process for producing the same
01/02/2004EP1375465A1 Cyclooctanone derivative and cyclodecanone derivative, and use thereof
01/02/2004EP1373494A2 Succinimide and maleimide derivatives and their use as topoisomerase ii catalytic inhibitors
01/02/2004EP1373208A1 A process for the synthesis of an aliphatic cyclic amine
01/02/2004EP1373202A1 Preparation of non-crystalline atorvastatin calcium
01/02/2004EP1373191A1 Acylated indanyl amines and their use as pharmaceuticals
01/02/2004EP1372692A2 Asymmetric synthesis of (s, s, r)-(-)-actinonin and its analogs and uses therefor
01/02/2004EP1372655A2 Cathepsin cysteine protease inhibitors
01/02/2004EP1140819B1 Alfa-sulfenimino acid derivatives
01/02/2004EP1027339B1 Method and reagents for n-alkylating ureides
01/01/2004US20040002609 Antidiabetic agents; metabolism diseases; hypotensive agents; cardiovascular disorders
01/01/2004US20040002542 Succinoylamino hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors
01/01/2004US20040002539 Enzyme inhibitors; anticoagulants; blood collecting device
01/01/2004US20040002533 Culture product of Streptomyces; lanosterol synthase inhibitor; anticholesterol agents, fungicides
01/01/2004US20040002515 Antihistamines; antiallergens; antiinflammatory agents; autoimmune diseases; rheumatic diseases
01/01/2004US20040002491 Melatonergic receptors
01/01/2004US20040002490 Melatonergic receptors
01/01/2004US20040002485 Enzyme inhibitors; viricides
12/2003
12/31/2003WO2004000828A1 New compounds useful for the treatment of obesity, type ii diabetes and cns disorders
12/31/2003WO2004000806A1 Amides of cyclic amino acids used as pde 4 inhibitors
12/31/2003WO2004000802A2 Scaffolded maleimide clusters for multivalent peptide assembly
12/31/2003WO2004000797A1 Alpha-sulfonylamino-acetonitriles
12/31/2003WO2003073999A3 Pini-modulating compounds and methods of use thereof
12/31/2003WO2003069303A3 Antimalarial and antiproliferative pharmacophore models, novel tryptanthrin compounds having increased solubility, and methods of making and using thereof
12/31/2003WO2003063576A3 Arylsulfonamidobenzylic compounds
12/31/2003WO2003035058A3 Polymaleide compounds and their medical use
12/31/2003CN1464881A New dipeptidyl peptidase iv inhibitors and their uses as anti-cancer agents
12/31/2003CN1463967A Opioid receptor containing 3-pyrroline, process for preparing the same and use thereof
12/31/2003CN1132836C 各种片螺素化合物和类似物的合成及中间体 And various synthetic intermediates lamellarin compounds and the like
12/31/2003CA2490124A1 Scaffolded maleimide clusters for multivalent peptide assembly
12/31/2003CA2486989A1 New compounds useful for the treatment of obesity, type ii diabetes and cns disorders
12/30/2003US6670483 Catalytically hydrogenating n-methyl-succinimide to form n-methylpyrrolidone
12/30/2003US6670479 Amination process
12/30/2003US6670386 For therapy of nuclear hormone receptor-associated conditions, such as age related diseases, for example sarcopenia
12/30/2003US6670358 Substituted thioacetamides
12/30/2003US6670357 Antiinflammatory agents
12/30/2003CA2198637C Preparation of quaternized glycine nitriles
12/30/2003CA2052884C Angiotensin 11 antagonists in the treatment of hyperuricemia
12/30/2003CA2051399C Therapeutically useful 2-aminotetralin derivatives
12/25/2003US20030236438 Enantioselective 1,4-addition of aromatic nucleophiles to alpha,beta-unsaturated aldehydes using chiral organic catalysts
12/25/2003US20030236415 Etherifying mucochloric or mucobromic acid with an alcohol, alkylation, hydrogenation, dehydrochlorination or dehydrobromination, decyclization by reductive amination and carboxylation; 3-Aminomethyl-5-methyl-hexanoic acid
12/25/2003US20030236403 Certain substituted 1-aryl-3-piperazine-1'-yl propanones
12/25/2003US20030236401 Asymmetric synthesis of amino-pyrrolidinones
12/25/2003US20030236254 Novel heterocyclic compounds having hypolipidemic, hypocholesteremic activities process for their preparation and pharmaceutical compositions containing them and their use in medicine
12/25/2003US20030236250 Antidepressants, anxiolytic agents, analgesics, antiinflammatory agents, reduce concentration of tachykinins
12/25/2003US20030236248 Kappa agonist compounds and pharmaceutical formulations thereof
12/25/2003US20030236198 For treatment of infections by drug resistant bacteria
12/24/2003WO2003106456A2 New compounds
12/24/2003WO2003106445A1 Compounds and methods for controlling bacterial virulence
12/24/2003WO2003106417A1 Mitotic kinesin inhibitors
12/24/2003WO2003106405A1 Aspartyl protease inhibitors
12/24/2003WO2003106390A1 Polymerisation inhibitor
12/24/2003WO2003105855A1 Mitotic kinesin inhibitors
12/24/2003WO2003105756A2 Stereoselective synthesis of 1,2-disubstituted cycloalkyls