Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
02/2004
02/18/2004EP1169301B1 A topical antiandrogen for hair loss and other hyperandrogenic conditions
02/18/2004CN1476434A Novel compounds
02/18/2004CN1476431A Process for preparing distamycin derivatives
02/18/2004CN1476430A Delta 1-pyrrolines used as pesticides
02/18/2004CN1476429A EP4 receptor selective agonists in treatment of osteoporosis
02/18/2004CN1476428A Delta 1-pyrrolines for use as pesticides
02/18/2004CN1138757C Prepn. of N-bromosuccinimide
02/17/2004US6693202 Multibinding ligands containing such as amine, amide, ester, hydroxyl, carbamate, urea and/or imino functionality
02/17/2004US6693199 Deprotecting carbamate group and amidating in presence of such as hydroxybenzotriazole hydrate promoter
02/17/2004US6693193 Coupling an n- and o-protected 2,3-dihydroxy-pyrrolidine to the 2-position and deprotecting
02/17/2004US6693123 (4-(3-pyridylaminomethylene)-2-phenylbenzoyl)-n -methylmethionine, methyl ester for example; restenosis, hyperplasia
02/17/2004US6693099 Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance
02/17/2004US6693092 Herbicides; pesticides
02/12/2004WO2004013282A2 Bis (amino acid) molecular scaffolds
02/12/2004WO2004013098A1 Novel gamma-lactams as beta-secretase inhibitors
02/12/2004WO2004013097A1 Process for the preparation of amino-pyrrolidine derivatives
02/12/2004WO2004013094A2 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/12/2004WO2004012732A2 Use of a proteasome inhibitor in the treatment of endothelial dysfunction and/or in a low-dose proteasome inhibitor therapy
02/12/2004WO2004012731A1 Pyrrolidine derivatives as tryptase inhibitors
02/12/2004WO2003103604A3 Gamma lactams as prostaglandin agonists and use thereof
02/12/2004WO2003088909A3 Methods for modulating phototoxicity
02/12/2004WO2003070665A3 Desolvating solvates of atorvastatin hemi-calcium
02/12/2004WO2002100344A3 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
02/12/2004US20040030155 One pot process; halogenation an acid; reacting with base
02/12/2004US20040030132 Anticancer agents; arterosclerosis; bone disorders; antiarthritic agents; vision defects
02/12/2004US20040030129 NF-kappaB inhibitor comprising phenylmethyl benzoquinone as an active ingredient
02/12/2004US20040030072 Using coordination catalyst
02/12/2004US20040029951 cyclooxygenase-2 (COX-2) inhibitors; Non-steroidal anti-inflammatory drugs (NSAIDs) with side effect reduction; N-propyl-3-(4-methylsulfonylphenyl)-4-(4-chlorophenyl)-2,5-dihydropyrrole-2-one for example; rheumatoid arthritis
02/12/2004US20040029933 Substituted phenylacetic acids
02/12/2004US20040029887 Cardiovascular disorders; antiinflammatory agents; central nervous system diosrders; psychological disorders
02/12/2004US20040029862 Alzheimer's disease
02/12/2004US20040029814 Cathepins inhibitor; antiinflammatory agents; antiarthritic agents
02/12/2004US20040029810 Process for preparing distamycin derivatives
02/12/2004US20040029735 Substituted herbicidal phenyluracils
02/12/2004CA2494404A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/12/2004CA2492830A1 Pyrrolidine derivatives as tryptase inhibitors
02/11/2004EP1387824A1 Method for purifying a raw melt of at least one monomer by crystallization
02/11/2004EP1387820A2 Method for the production of a purified melt of at least one monomer
02/11/2004EP1387679A1 Sulfonamides
02/11/2004EP1299356B1 Novel compounds
02/11/2004EP1098866B1 Method for producing ortho-alkylated benzoic acid derivatives
02/11/2004EP0936912B1 Inhibitors of cysteine protease
02/11/2004CN1474810A Substituted urea neuropeptide YY5 antagonists
02/11/2004CN1474809A Cyanopyrolidine derivatives
02/11/2004CN1473814A Intemediate for preparing alkyl-dihalogeno phenyl substituted keto-enol
02/10/2004US6689909 Substituted N-phenyl 2-hydroxy-2-methyl-3,3,3-trifluoropropanamide derivatives which elevate pyruvate dehydrogenase activity
02/10/2004US6689890 Efficient lactam synthesis
02/10/2004US6689771 Amide derivatives as inhibitors of matrix metalloproteinases, TNF-α, and aggrecanase
02/10/2004US6689174 N-benzyl-p-phenylenediamine-derivatives containing coloring agents for keratin fibres and novel n-benzyl-p-phenylenediamine-derivatives
02/05/2004WO2004011431A1 Pleuromutilin derivatives as antimicrobbials
02/05/2004WO2004011423A2 Structural carotenoid analogs for the inhibition and amelioration of disease
02/05/2004WO2004011418A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc-chemokine receptor ligands
02/05/2004WO2004010945A2 Cyclooxygenase- 2 selective inhibitors, compositions and methods of use
02/05/2004WO2004010943A2 Substituted benzanilides as modulators of the ccr5 receptor
02/05/2004WO2003075857A3 Amino-methyl substituted tetracycline compounds
02/05/2004WO2002100886A8 Pyrrolidin-2-one derivatives as inhibitors of factor xa
02/05/2004WO2002041834A8 Atorvastatin hemi-calcium form vii
02/05/2004US20040024226 Reacting atorvastatin lactone, methanol, and methyl tert-butyl ether with sodium sodium hydroxide to form ring-opened salt; drying isolated product in vacuum pan dryer with continuously rotating agitator
02/05/2004US20040024215 Such as 4'-trifluoromethyl-biphenyl-2-carboxylic acid(4-(4-(alpha-methyl-benzyl)-piperazin-1-yl)-phenyl)-amide; apoprotein B-100 (apoB-100) and microsomal triglyceride transfer protein (MTP)
02/05/2004US20040024210 New compounds
02/05/2004US20040024132 A free radical polymerization in presence of a sulfur based chain transfer agents, controlling during the synthesis of polystyrene, polymethyl acrylate, polymethyl methacrylate
02/05/2004US20040024059 Novel pleuromutilin derivatives
02/05/2004US20040024046 By precipitating the atorvastatin using a solvent of a second type from a solution of atorvastatin which is provided with a solvent of a first type
02/05/2004US20040023945 Cyclic amp-specific phosphodiesterase inhibitors
02/05/2004US20040023806 Agrochemicals in agriculture for controlling acarids and insects and for preventing the infestation of crop plants by phytopathogenic fungi.
02/05/2004US20040023290 Novel therapeutic agents that modulate enzymatic processes
02/05/2004DE10022829B4 p-Aminophenol-Derivate und diese Verbindungen enthaltende Haarfärbemittel p-aminophenol derivatives and compositions containing these compounds Hair dyes
02/05/2004CA2495167A1 Structural carotenoid analogs for the inhibition and amelioration of disease
02/05/2004CA2493156A1 Cyclooxygenase-2 selective inhibitors, compositions and methods of use
02/04/2004EP1386913A1 Pyrrole derivative
02/04/2004EP1386912A1 Cyclic amidine derivative
02/04/2004EP1385841A1 Sulfonamides
02/04/2004EP1385840A1 Sulfonamides
02/04/2004EP1385822A1 Aminopyrrolidine sulfonamides as serine protease inhibitors
02/04/2004EP1385820A1 Anthranilic acid amides, method for the production thereof, their use as antiarrhythmia agents, and pharmaceutical preparations thereof
02/04/2004EP1385510A1 Prodigiosin composition for the treatment of rheumatic arthritis
02/04/2004EP1385508A1 Dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
02/04/2004EP1385507A1 Sulfonamides
02/04/2004EP1203585A4 Anti-ischemic agent
02/04/2004EP1115697B1 Unsaturated hydroximic acid derivatives as parp inhibitors
02/04/2004CN1473150A Bis-heterocyclic compounds with antitumour and chemosensitising activity
02/04/2004CN1473145A Method of resolving optical isomers of amino acid derivative
02/04/2004CN1473034A Photo-labile pro-fragrance conjugates
02/04/2004CN1137095C Preparation of i(N)-substituted-hydroxycycloalkylamine derivatives
02/03/2004US6686477 Multistep chemical synthesis, including asymmetric hydrogenation of a lactam-enamide to produce an intermediate that can be used to make unspecified pharmaceuticals
02/03/2004US6686390 Compounds having antiinflamatory activity: process for their preparation and pharmaceutical compositions containing them
02/03/2004US6686386 Combating photoinduced or chronological ageing of skin with retenoic acid receptor agonist
02/03/2004US6686353 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
02/03/2004US6686350 Cell adhesion inhibitors
02/03/2004US6685617 4-(((-1-carboxy-2-(4-((2,6-dichlorobenzoyl)amine)phenyl)ethyl) amino)carbonyl)-3-oxo-3-thiazolidinebutanoic acid, used as antagonists for cellular adhesion molecules, and administered as antiinflammatory agents
01/2004
01/29/2004WO2004009544A1 2-cyano-4-fluoropyrrolidine derivative or its salt
01/29/2004WO2004009533A1 Acetylamino benzoic acid compounds and their use for nonsense suppression and the treatment of disease
01/29/2004WO2004009531A1 Acetylenic compounds useful in treating inflammatory disorders
01/29/2004WO2004009527A1 Materials and methods for treating hypercholesterolemia
01/29/2004WO2004009017A2 Modulators of the glucocorticoid receptor and method
01/29/2004WO2003066035A3 Compounds for inhibiting insulin secretion and methods related thereto
01/29/2004WO2003053923A3 Pyrrolidine derivatives as prostaglandin modulators
01/29/2004WO2003000180A3 Dipeptidyl peptidase inhibitors for the treatment of diabetes
01/29/2004US20040019239 Catalytic compositions and methods for asymmetric aldol reactions
01/29/2004US20040019224 Low shrinkage thermosetting resin compositions and methods of use therefor