Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
04/2004
04/01/2004US20040063643 Bombesin antagonists
04/01/2004US20040060127 E.g., p-(3-(3-trimethylsilanylpropoxy)-1-pyrrolidyl)-phenylamine
04/01/2004DE10243666A1 Dithiocarbaminsäureester Dithiocarbaminsäureester
04/01/2004CA2768674A1 Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-iv (dpp-iv)
04/01/2004CA2499701A1 Pyrrole derivatives as antimycobacterial compounds
04/01/2004CA2499490A1 Amide and sulfonamide ligands for the estrogen receptor
04/01/2004CA2499426A1 Process for preparing n-hydroxylamine compounds
04/01/2004CA2498335A1 4-pyrrolidino-phenyl-benzyl ether derivatives
03/2004
03/31/2004EP1401918A2 Biodegradable poly(beta-amino esters) and uses thereof
03/31/2004EP1401828A1 N-formyl hydroxylamine compounds as inhibitors of pdf
03/31/2004EP1401824A2 Aromatic hydroxamic acid derivatives useful as hdac inhibitors
03/31/2004EP1401821A1 Novel phenylalkyl diamine and amide analogs
03/31/2004EP1401817A1 Isoquinoline compounds having antiinfective activity
03/31/2004EP1401811A1 Method for producing pyrrolidones
03/31/2004EP1401810A1 Compounds having prolyl oligopeptidase inhibitory activity, methods for their preparation and their use
03/31/2004EP1401809A1 Tryptase inhibitors
03/31/2004EP1370258A4 Peptide deformylase inhibitors
03/31/2004EP1363623A4 Peptide deformylase inhibitors
03/31/2004CN1486172A Primary intermediates for oxidative coloration of hair
03/31/2004CN1143675C Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics
03/30/2004US6713635 As chemical intermediates used for the preparation of s-alpha-ethyl-2-oxo-1-pyrrolidine acetamide
03/30/2004US6713634 Pyrroloazepine derivatives
03/30/2004US6713603 Adjusted nucleotide sequences for use as antisense tools in genetic engineering
03/30/2004US6713504 Antifungal molecule 2-(3,4-dimethyl-2,5-dihydro-1H-pyrrol-2-yl)-1-methylethyl pentanoate
03/30/2004US6713503 1-(2,4-dimethyl-phenyl)-2,4-dihydroxy-3-(4-methyl-benzoyl)-5-oxo-2,5 -dihydro-1h-pyrrole-2-carboxylic acid methyl ester
03/30/2004US6713502 Anti-infectives
03/30/2004US6713492 N-acyloxylated cycloalkyl compounds, composition containing the same and methods of use therefor
03/30/2004US6713467 Anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and metastasis inhibitors in treating cancer
03/30/2004US6713059 Antibodies raised against immunogenic conjugates of gram-negative bacterial autoinducer molecules
03/30/2004CA2278687C 5-aroylnaphthalene derivatives
03/25/2004WO2004024991A1 Organic salts and their use as reagents in electrochemical reactions
03/25/2004WO2004024939A2 Ligands for the peroxisome proliferator-activated receptor, and methods of use thereof
03/25/2004WO2004024702A1 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof
03/25/2004WO2004024686A1 Biological low-molecular weight derivatives
03/25/2004WO2004024685A1 Novel dipeptide compound and medical use tehreof
03/25/2004WO2004024681A2 Novel compounds comprising a thiocarbonyl-sulfanyl group, which can be used for the radical synthesis of alpha-perfluoroalkylamines
03/25/2004WO2004024679A1 Inhibitors of factor xa and other serine proteases involved in the coagulation cascade
03/25/2004WO2004024143A1 Medicinal composition
03/25/2004WO2004024139A1 Melanin extinguisher
03/25/2004WO2003084941A3 Hydroxamic acid derivatives
03/25/2004WO2003082260A3 Tuberculosis treatment using pleuromutilin derivatives
03/25/2004WO2003048106A3 1,3-diarylprop-2-en-1-ones, compositions containing same and use thereof
03/25/2004WO2002096871A8 Allylmercaptocaptopril compounds and uses thereof
03/25/2004US20040059149 Method for the synthesis of compounds of formula 1 and derivatives thereof
03/25/2004US20040059129 2,5-bisphenyl-delta1-pyrroline derivative are chromatographed on a stationary chiral silica gel phase in presence of an eluent or mixture as liquid phase
03/25/2004US20040058968 Antiinflammatory agents; autoimmune diseases; antiarthritic agents
03/25/2004US20040058960 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
03/25/2004US20040058932 Novel piperazine derivatives
03/25/2004US20040058820 Central nervous system disorders; psychological disorders; antiinflammatory agents; multiple sclerosis
03/25/2004DE10243201A1 New N-acyl-aminoacid N-(succinimidyl-carbonyl-alkyl)-amide compounds, are broad-spectrum antibacterial agents useful in human or veterinary medicine
03/25/2004CA2499606A1 Biological low-molecular-weight derivatives
03/25/2004CA2497003A1 Inhibitors of factor xa and other serine proteases involved in the coagulation cascade
03/25/2004CA2496563A1 New carboxamide compounds having mch-antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture
03/24/2004EP1400516A1 Substituted anilide derivatives, intermediates thereof, agricultural and horticultural chemicals, and their usage
03/24/2004EP1400508A1 Dithiocarbamic acid ester
03/24/2004EP1399433A2 Fluoropyrrolidines as dipeptidyl peptidase inhibitors
03/24/2004EP1399431A2 Novel nitriles useful as reversible inhibitors of cysteine proteases
03/24/2004EP1399421A1 Substituted imidates as pesticidal agents
03/24/2004EP1399420A2 Pyrrolidines as dipeptidyl peptidase inhibitors
03/24/2004EP1399163A2 Compounds, methods and compositions useful for the treatment of bovine viral diarrhea virus (bvdv) infection and hepatitis c virus (hcv) infection
03/24/2004EP1399159A1 4-substituted-1-(arylmethylidene)thiosemicarbazide, 4-substituted-1-(arylcarbonyl)thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof
03/24/2004EP1399154A1 3-fluoro-pyrrolidines as antidiabetic agents
03/24/2004EP1399146A1 Novel compounds and compositions as cathepsin inhibitors
03/24/2004EP1214296B1 Substituted n-phenyl 2-hydroxy-2-methyl-3,3,3-trifluoropropanamide derivatives which elevate pyruvate dehydrogenase activity
03/24/2004EP1161232B1 Hydroxy diphenyl urea sulfonamides as il-8 receptor antagonists
03/24/2004EP1082110B1 Use of compounds for the elevation of pyruvate dehydrogenase activity
03/24/2004CN1484637A Pyrrolcarboxamides and pyrrolcarbothioamides and their agrochemical uses
03/24/2004CN1484527A Medicines for treatment and prevention of neurogenic pain
03/24/2004CN1142920C Quinazoline derivatives and pharmaceutical compositions containing them and preparation process and use
03/24/2004CN1142911C Compounds with growth hormone releasing properties
03/24/2004CN1142793C Epoxy-steroidal aldosterone antagonist and angiotensin 2 antagonist combination therapy for treatment of congestive heart failure
03/23/2004US6710186 Conformationally-restricted; analogous to poly(proline) ii helical structure
03/23/2004US6710179 Compounds with analgesic effect
03/23/2004US6710089 Substituted N-fused-phenyl-N-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
03/23/2004US6710061 Selective serine protease or dual-serine protease inhibitors of factor xa and tryptase
03/23/2004US6710040 Fluorinated cyclic amides as dipeptidyl peptidase IV inhibitors
03/23/2004CA2263319C Quinazoline derivatives and pharmaceutical compositions containing them
03/18/2004WO2004022536A1 New heterocyclic amide compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
03/18/2004WO2004022533A1 Novel vinyl carboxylic acid derivatives and their therapeutical use
03/18/2004WO2004022529A2 Diarylurea derivatives and their use as chloride channel blockers
03/18/2004WO2004022525A1 Amide derivatives and their use as chloride channel blockers
03/18/2004WO2004022523A2 1, 3-diamino-2-hydroxypropane prodrug derivatives
03/18/2004WO2004022053A1 Atorvastatin calcium form vi or hydrates thereof
03/18/2004WO2003099266A3 Acetamides and benzamides that are useful in treating sexual dysfunction
03/18/2004WO2003087094A3 Pyrrolidinium derivatives as antagonists of m3 muscarinic receptors
03/18/2004WO2003086563A3 Diabetes imaging probes
03/18/2004WO2003079975A3 Process for the manufacture of optically active 3-substituted lactams by asymmetric hydrogenation of 3-alkylidenelactams
03/18/2004WO2003035615A3 Tyrosine kinase inhibitors
03/18/2004WO2003035614A3 Tyrosine kinase inhibitors
03/18/2004WO2003018535A3 Novel aminobenzoephenones
03/18/2004US20040054194 Cyclization, deacylation nding amide in presence of diluent; insecticide for agriculture
03/18/2004US20040054193 Crystalline forms of [R-(R*,R*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1)
03/18/2004US20040054184 Preservative for organs, synthetic blood
03/18/2004US20040054009 Useful for potentiating glutamate receptor function in a mammal and therefore useful for treating wide variety of conditions such as psychiatric and neurological disorders
03/18/2004US20040053987 Bis-heterocyclic compounds with antitumour and chemosensitising activity
03/18/2004US20040053983 1, 2, 4-tribsubstituted benzenes as inhibitors of 15-lipoxygenase
03/18/2004US20040053981 Such as 2-(5(6)-nitro-2-benzimidazoyl)-5-(4-nitrophenyl)furan; fluorescent quantitative analysis; for treatment/prevention of cancer
03/18/2004US20040053953 Treatment of chemokine mediated diseases
03/18/2004US20040053933 Ligands of melanocortin receptors and compositions and methods related thereto
03/18/2004US20040053917 Reacting cyanophenyl-4-sulfonylchloride with a piperidine-4-oxo in presence of ethylene glycol to form an intermediate, reducing cyano group, followed by amidation, then reacting with an amine to form sulfonamide end