Patents
Patents for C07D 203 - Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom (1,097)
07/2002
07/10/2002EP1220838A2 1-aziridino-1-hydroxyiminomethyl-derivatives, method for the production thereof and medicaments containing said compounds
07/09/2002US6417010 Methods and apparatus for synthesizing labeled combinatorial chemistry libraries
07/04/2002US20020086887 N-Acylsulfonamide apoptosis promoters
06/2002
06/11/2002US6403824 Process for the preparation for 4,5-diamino shikimic acid derivatives
06/04/2002US6399638 Anticarcinogenic agents; microtubule stabilizing effects
05/2002
05/30/2002US20020065417 Useful as ligands for metal catalysts for asymmetric reactions, in particular as rhodium complexes for asymmetric hydrogenation of enamide, itaconate, and alpha-ketoester compounds
05/22/2002CN1350530A 酰胺衍生物 Amide derivatives
05/16/2002US20020058823 Dehydrationg cyclohexylalcohol compound
05/09/2002US20020055642 Processes for the preparation of aziridine compounds and vapor-phase reaction processes
05/09/2002US20020055631 N-acylsulfonamide apoptosis promoters
05/08/2002EP1147082A4 Synthesis of ethyleneimine dimer
05/08/2002EP0915648B1 Methods and compositions for the selective modification of nucleic acids
05/08/2002DE10153414A1 Verfahren zur Herstellung von Aziridinverbindungen und Dampfphasen- Reaktionsverfahren Process for the preparation of aziridine compounds and vapor phase reaction method
05/08/2002CN1347693A Noval compound, its synthetizing process and therapeutic use
05/02/2002EP0765336B1 Synthesis of conduritol epoxides and aziridines and methods of using such to synthesize higher disaccharides
04/2002
04/30/2002US6380395 Anticancer agents
04/11/2002US20020042508 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same
04/11/2002US20020040725 Washing with acidity solution
04/11/2002DE10147370A1 Waschverfahren für Destillationssysteme von Stickstoff enthaltenden polymerisierbaren Monomeren Washing method for distillation systems of nitrogen-containing polymerizable monomers
04/04/2002WO2002026750A2 Phosphino-aminophosphines, catalyst complexes and enantioselective hydrogenation
04/04/2002WO2002026705A2 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and their preparation
03/2002
03/28/2002WO2002024636A2 N-acylsulfonamide apoptosis promoters
03/27/2002EP0920410B1 Preparation of cyclohexene carboxylate derivatives
03/21/2002US20020034724 Methods to selectively inactivate microorganisms in biological compositions
03/20/2002EP1187798A1 PRODUCTION OF OPTICALLY ACTIVE $g(a)-HYDROXYACETALS
03/14/2002US20020032338 Enantiomerically pure compounds by reacting water and carbocycle or heterocycle having an electrophilic center in the presence of an asymmetric tetradentate ligand complexed with a metal atom, which has a geometric shape
02/2002
02/26/2002CA2206776C N-sulfonylindoline derivatives carrying an amide functional group, their preparation and the pharmaceutical compositions in which they are present
02/14/2002WO2002012186A1 Optically active aziridine-2-carboxylate derivatives and a process for preparing them
02/14/2002WO2002012184A1 Process for preparing alpha-amino acids and their derivatives including phenylalanine and homophenylalanine and their intermediates
02/14/2002WO2002012181A1 Novel diamines having a casr modulating activity
02/13/2002EP1179530A1 Processes for preparing optically active amino acid derivatives
02/13/2002EP0975616B1 Substituted benzyl oximino compounds
01/2002
01/17/2002US20020006960 Neuraminidase inhibitors
01/03/2002WO2002000590A1 Synthesis of functionalized and unfunctionalized olefins via cross and ring-closing metathesis
12/2001
12/19/2001EP1163237A1 Amide derivatives
12/11/2001US6329359 Substituted benzyl oximino compounds
11/2001
11/27/2001US6323346 Process for producing aziridine compounds
10/2001
10/30/2001US6310246 Fluorovinloxyacetamides, process for preparing same and herbicidal composition comprising same
10/24/2001EP1147227A1 Lipophilic quenching of viral inactivating agents
10/24/2001EP1147082A1 Synthesis of ethyleneimine dimer
10/16/2001US6303659 Administering adamantane derivative for therapy of rheumatoid arthritis
10/11/2001WO2001021585A3 Bis(1-aziridino-1-hydroxyiminomethyl)-derivatives, method for the production thereof and use thereof as anti-tumoral agents
10/10/2001EP1140844A1 Process for the formation of intermediates useful for the preparation of pharmaceuticals
10/02/2001US6297230 N-carbamoyl-substituted
09/2001
09/26/2001CN1071744C 1,2,3-trisubstituted aziridine, preparing method and use
09/11/2001US6288224 Preparation of n-arylmethyl aziridine derivatives, 1,4,7,10-tetraazacyclododecane derivatives obtained therefrom and n-arylethyl-ethanolamine sulphonate esters as intermediates
09/05/2001EP1129728A1 Methods and compositions for the selective modification of nucleic acids
08/2001
08/29/2001EP1127872A1 Tamiflu via Diels-Alder
08/29/2001CN1310170A Process for producing 4,5-diamino shikimic acid derivative
08/23/2001WO2001060795A1 Processes for preparing optically active amino acid derivatives
08/23/2001CA2369678A1 Process for producing optically active amino acid derivatives
08/16/2001US20010014760 Gas-phase dehydration reaction process
08/16/2001US20010014744 Synthesis of ethyleneimine dimer
08/15/2001CN1308062A 1-substituted-N-sulfinyl-2-aziridine methylenimine and its preparation and use
08/08/2001EP1122228A1 Gas-phase dehydration reaction process
07/2001
07/25/2001CN1305453A Fluorovinyloxyacetamides, process for preparing the same and herbicidal composition comprising the same
07/17/2001US6262278 Reacting water and mixture of stereoisomers of chiral cyclic substrate in the presence of non-racemic chiral catalyst to produce by kinetic resolution stereoisomerically enriched cyclic substrate or stereoisomerically enriched hydrolyzate
07/10/2001US6258960 Catalytic asymmetric synthesis of chiral aziridines
07/10/2001US6258838 Compounds
07/04/2001EP1112250A1 Therapeutic compounds and methods
06/2001
06/27/2001EP1109550A2 Novel nitrophenylaziridine compounds and their use as prodrugs
06/07/2001US20010003121 Adamantane derivatives such as 2,4-dichloro-N-(tricyclo(3.3.1.13,7)dec-1-methyl)-benzamide; administering to treat rheumatoid arthritis; immunosuppressant
06/06/2001EP1104395A1 Stereoselective ring opening reactions
06/06/2001CN1298398A 12,13-modified epothilone derivatives
05/2001
05/29/2001US6239175 Carbamoyloxy derivatives of mutiline and their use as antibacterials
05/10/2001WO2001032617A1 Process for the preparation of 7-azabicyclo[4.1.0]-hept-3-ene-3-carboxylic acid esters
05/01/2001US6225341 For inhibiting neuraminidase; for therapy and prophylaxis of virus infection
04/2001
04/10/2001US6215003 Synthesis of ethyleneimine dimer
04/05/2001DE19947440A1 1-Aziridino-1-hydroxyiminomethyl-Derivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel 1-Aziridino-1-hydroxyiminomethyl derivatives, processes for their preparation and medicaments containing these compounds
03/2001
03/29/2001WO2001021585A2 Bis(1-aziridino-1-hydroxyiminomethyl)-derivatives, method for the production thereof and use thereof as anti-tumoral agents
03/20/2001US6204398 Useful as intermediates that are themselves useful in the synthesis of neuraminidase inhibitors
03/20/2001US6204379 Reacting pentenoic acid with carbon monoxide, hydrogen and ammonia in presence of a catalyst
03/13/2001US6201024 Effective p2x7 receptor antagonists for use in the treatment of inflammatory, immune or cardiovascular disorders
02/2001
02/22/2001WO2001012599A1 New ethylaziridine derivatives and their preparation methods
02/14/2001CN1284057A Adamantane derivatives
02/07/2001EP1073648A1 12,13-Modified epothilone derivatives
02/07/2001EP1073647A1 12,13-cyclopropane epothilone derivatives
01/2001
01/31/2001EP1071656A1 Fluorovinyloxyacetamides, process for preparing same and herbicidal composition comprising same
01/04/2001WO2001000545A1 PRODUCTION OF OPTICALLY ACTIVE α-HYDROXYACETALS
12/2000
12/12/2000US6159973 Aromatic amides, their preparation process, the compositions containing them and their use as pesticides
12/05/2000US6156744 Water solubility; diaphorase inhibitor
11/2000
11/21/2000US6150109 Lipophilic quenching of viral inactivating agents
11/01/2000CN1272105A Compound containing six-membered rings, processes for their preparation, and their use as medicaments
10/2000
10/24/2000US6136586 Methods for the selective modification of viral nucleic acids
10/04/2000EP1040095A1 Cyclohexene carboxylates as neuraminidase inhibitors
10/03/2000US6127550 By reacting a 2-amino-2-substituted ethyl alcohol having position 2 chirality(2-*) with a halide in the presence of a base to form a 2-substituted, 2-* aziridine, reacting with a lithium compound to form a salt, treating with strong acid
09/2000
09/28/2000WO2000056708A1 Catalytic asymmetric synthesis of chiral aziridines
09/27/2000EP1038866A1 Process for producing aziridine compound
09/21/2000WO2000055153A1 Amide derivatives
09/20/2000EP1036059A1 Adamantane derivatives
09/19/2000US6121281 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
09/05/2000US6114108 Methods and compositions for the selective modification of viral nucleic acids
08/2000
08/29/2000US6111132 Compounds and methods for synthesis and therapy
08/23/2000EP0805795B1 Novel aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
08/16/2000EP1027041A1 Novel cyanoaziridines for treating cancer
08/08/2000US6100396 Method for purifying lactams
08/03/2000WO2000044720A1 Synthesis of ethyleneimine dimer
08/02/2000EP1023264A1 New marker, production process and use thereof
08/02/2000CN1261873A Methods and compositions for selective modification of nucleic acids
07/2000
07/27/2000WO2000043549A1 Lipophilic quenching of viral inactivating agents
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