| Patents for C07D 203 - Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom (1,097) |
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| 05/06/2009 | EP2054368A2 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors |
| 04/15/2009 | CN101407485A Method for preparing ethylene polyamine by ammonolyzing dichloroethane with alcohol as medium |
| 03/17/2009 | US7504512 BCL-X1 protein inhibitors; anticarcinogenic agents |
| 02/24/2009 | US7494988 Inhibitors of serine proteases, particularly hepatitis C virus NS3 protease |
| 01/27/2009 | US7482364 Histamine H3 antagonists; do not contain imidazolyl moiety; such as 1-[4-(4-piperidin-1-ylmethyl-phenyl)-but-3-ynyl]-piperidine |
| 01/22/2009 | US20090022664 Radiolabelling via fluorination of aziridines |
| 12/30/2008 | CA2294243C Novel cyanoaziridines for treating cancer |
| 12/24/2008 | WO2008155355A1 Method for synthesizing an n-unsubstituted or n-substituted aziridine |
| 12/11/2008 | WO2008024892A3 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors |
| 11/18/2008 | CA2361565C Synthesis of ethyleneimine dimer |
| 11/04/2008 | US7446104 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia |
| 10/28/2008 | US7442704 Amide derivatives |
| 10/23/2008 | DE102008001262A1 Kontinuierliches Verfahren zur Herstellung von Alkyleniminen A continuous process for the production of alkyleneimines |
| 10/16/2008 | WO2008073781A3 C--h bond amination and olefin aziridination with beta-diketiminato copper catalysts |
| 10/15/2008 | CN101284244A Catalyst for synthesizing the aziridine type compound |
| 10/08/2008 | EP1976848A2 Phenoxypiperidines and analogs thereof useful as histamine h3 antagonists |
| 09/04/2008 | US20080214838 Oligo-Tetracenes, Production and Use Thereof |
| 08/13/2008 | CN100409844C Noval compound, its synthetizing process and therapeutic use |
| 07/22/2008 | US7402670 Synthesis by chiral diamine-mediated asymmetric alkylation |
| 07/22/2008 | CA2313638C Cyclohexene carboxylates as neuraminidase inhibitors |
| 07/17/2008 | WO2008083729A1 Radiolabelling via fluorination of aziridines |
| 07/17/2008 | CA2674408A1 Radiolabelling via fluorination of aziridines |
| 07/16/2008 | EP1944288A1 Radiolabelling via fluorination of aziridines |
| 07/10/2008 | WO2008046232A8 Aziridine aldehydes, aziridine-conjugated amino derivatives, aziridine-conjugated biomolecules and processes for their preparation |
| 06/19/2008 | US20080146808 Antiapoptosis; cancers; inhibiting the caspases; |
| 06/19/2008 | CA2671783A1 C--h bond amination and olefin aziridination with beta-diketiminato copper catalysts |
| 05/01/2008 | US20080103135 Histamine H3 antagonists; do not contain imidazolyl moiety; such as 1-[4-(4-piperidin-1-ylmethyl-phenyl)-but-3-ynyl]-piperidine |
| 04/24/2008 | WO2008046232A1 Aziridine aldehydes, aziridine-conjugated amino derivatives, aziridine-conjugated biomolecules and processes for their preparation |
| 04/24/2008 | US20080096876 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia |
| 04/24/2008 | CA2702605A1 Unprotected amino aldehydes and applications for same |
| 04/16/2008 | EP1911350A1 Amidine compound and herbicide |
| 04/15/2008 | CA2337452C Process for the preparation of 4,5-diamino shikimic acid derivatives |
| 04/03/2008 | US20080081916 Method for Producing Optically Active Aziridine Compounds and Amine Compounds as Well as Complexes and their Intermadiates Used in this Method |
| 03/18/2008 | US7345081 Azabicyclo-octane inhibitors of IAP |
| 02/28/2008 | WO2008024892A2 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors |
| 02/28/2008 | CA2661401A1 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors |
| 02/19/2008 | US7332483 3-(5-benzamido-2-chlorophenyl)-7-methoxy-3,4-dihydroquinazolin-4-one;cytokines (tumor necrosis factor and interleukins) inhibitor; antiinflammatory agent, rheumatoid arthritis, osteoarthritis, psoriasis, chronic obstructive pulmonary disease |
| 01/16/2008 | EP1755593B1 Naphthalene derivatives useful as histamine-3-receptor ligands |
| 01/10/2008 | US20080009639 Preparation of oseltamivir phosphate (Tamiflu) and intermediates starting from D-glucose or D-xylose |
| 12/26/2007 | EP1868990A2 Novel heterocyclic derivatives |
| 12/20/2007 | US20070293465 Compounds for enzyme inhibition |
| 12/05/2007 | CN100352814C Preparation of cyclohexene carboxylate derivatives |
| 12/04/2007 | CA2193097C Synthesis of conduritol epoxides and aziridines and methods of using such to synthesize higher disaccharides |
| 11/28/2007 | CN101077345A Application of Tagalsin C and its homologous compound in preparing anti-tumor medicine |
| 11/15/2007 | US20070265254 Naphthaline derivatives as H3 inverse agonists |
| 11/08/2007 | DE10318326B4 Verfahren zur Herstellung von Aziridinen und N-Vinylamiden A process for the production of aziridines and N-vinylamides |
| 11/01/2007 | WO2006109146A3 Novel heterocyclic derivatives |
| 10/30/2007 | US7288540 Phenylalkynes |
| 10/04/2007 | US20070232581 Alzheimer's disease; compounds inhibit the production of A beta -peptide; improved pharmacokinetics; N-((4-amino-3,5-dichlorobenzylamino)(amino)methylene)-3-(isobutoxyimino)-3-(4-methoxyphenyl)propanamide |
| 09/27/2007 | US20070225505 Method for the Preparation of (2S, 3AR, 7AS)-Octahydro-III-Indole-2-Carboxylic Acid as Key Intermediate in the Preparation of Trandolapril by Reacting a Cyclohexyl Aziridine with a Dialkyl Malonate |
| 09/18/2007 | US7271130 N-alkynyl-2-(substituted phenoxy) alkylamides and their use as fungicides |
| 09/13/2007 | US20070213538 Ionic Liquids Having Fluoroalkyltrifluoroborate Anions |
| 09/11/2007 | US7268228 Optically active aziridine-2-carboxylate derivatives and a process for preparing them |
| 08/30/2007 | US20070203111 Cycloalkylamines as monoamine reuptake inhibitors |
| 08/21/2007 | US7259158 Naphthaline derivatives as H3 inverse agonists |
| 07/31/2007 | CA2263136C Preparation of cyclohexene carboxylate derivatives |
| 07/24/2007 | US7247740 Reacting perfluoroalkanesulfonic acid directly with dialkyl carbonate to give alkyl perfluoroalkanesulfonate optionally in the presence of a water or alcohol consuming reagent, and preparing an alkyl perfluoroalkanesulfonate with an alkylamine or alkylphosphine to prepare perfluoroalkanesulfonic acid |
| 07/11/2007 | CN1325486C Kinetics resolution method |
| 06/19/2007 | US7232914 Useful for more effective resolution of the mechanism of sphingomyelinase |
| 06/13/2007 | EP1794129A2 Synthesis by chiral diamine-mediated asymmetric alkylation |
| 05/22/2007 | US7220870 Resolution of epi(chloro or bromo)hydrin using transition metal catalyst |
| 05/09/2007 | CN1960727A Naphthalene derivatives useful as histamine-3-receptor ligands |
| 05/08/2007 | US7214803 Amidation of an alpha-pyrrolidinonylalkanoate by reaction with ammonium hydroxide |
| 05/01/2007 | USRE39606 Synthetic libraries of random oligomers, each member comprising an oligomer linked to a microchip encoded with information identifying structure of oligomer, for drug screening |
| 03/29/2007 | US20070072837 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia |
| 03/28/2007 | EP1767524A1 Process for production of optically active aziridines and amines, complexes used in the process, and intermediates thereof |
| 03/14/2007 | EP1606242B1 Azide free process for preparing 1,2-diamino compounds |
| 02/28/2007 | EP1755593A1 Naphthaline derivatives useful as histamine-3-receptor ligands |
| 02/27/2007 | US7182789 Stabilised compositions containing polyfunctional aziridine compounds as hardening constituents |
| 02/08/2007 | US20070032640 Cytokine receptor |
| 02/08/2007 | US20070032455 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents |
| 01/31/2007 | CN1297535C Method for producing perfluoroalkane sulfonic acid esters and the salts thereof |
| 01/24/2007 | EP1472217B1 Method for producing perfluoroalkane sulfonic acid esters and the salts thereof |
| 01/24/2007 | CN1902159A Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents |
| 01/18/2007 | WO2007007828A1 Ethylenediamine derivative and method for producing same |
| 01/10/2007 | EP1740173A1 Azabicyclo-octane inhibitors of iap |
| 01/10/2007 | EP1534699A4 Kinetic resolution method |
| 01/09/2007 | US7160903 Sulfonylaminocarboxylic acids |
| 01/02/2007 | US7157498 Diamines having a CaSR modulating activity |
| 12/28/2006 | US20060293518 Proccess for the preparation of phenylcarbamates |
| 12/27/2006 | EP0638123B1 Bacterial nitroreductase for the reduction of cb 1954 and analogues thereof to a cytotoxic form |
| 12/26/2006 | US7153979 For therapy of hepatic disorders |
| 12/20/2006 | EP1456171B1 Substituted cyclohexane derivatives |
| 12/14/2006 | US20060281734 3-[5-(3-acetamidobenzamido)-2-methylphenyl]-6-(4-methylpiperazin-1-yl)-3,4-dihydroquinazolin-4-one for example; treating rheumatoid arthritis, osteoarthritis, psoriasis, chronic obstructive pulmonary disease; inhibitor of cytokine-mediated disease |
| 12/12/2006 | US7148251 D-t-3',4'-ethylenedioxy-p4 derivatives; glucosyl ceramide inhibitors lower glycosphingolipid levels; anticarcinogenic, antitumor agents; angiogenesis inhibitors; tumor antigens |
| 11/16/2006 | US20060258859 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia |
| 11/02/2006 | EP1301458A4 Synthesis of functionalized and unfunctionalized olefins via cross and ring-closing metathesis |
| 10/25/2006 | EP1187798B8 Production of optically active alpha-hydroxyacetals |
| 10/19/2006 | WO2006109146A2 Novel heterocyclic derivatives |
| 10/18/2006 | CN1280267C Sulfonylaminocarboxylic acids |
| 10/18/2006 | CN1280258C Process for producing 4,5-diamino shikimic acid derivative |
| 10/17/2006 | US7122684 multi-step process for preparing 2-aminoalcohols from 1,2-epoxides; useful as inhibitors of viral or bacterial neuraminidases; intermediates |
| 09/21/2006 | US20060211870 cyclization; reacting 4-methylstyrene with p-toluenesulfonamide (TsNH2), N bromosuccinimide (NBS) in presence of dirhodium(II,II) carboxamidates compounds; stereospecific control |
| 09/20/2006 | EP1073648B1 12,13-modified epothilone derivatives |
| 09/20/2006 | CN1275941C Process for producing aziridine compound and N-vinyl amide |
| 09/19/2006 | US7109352 Process for producing optically active amino acid derivatives |
| 08/30/2006 | EP1694281A2 Biphenyl compounds and methods |
| 08/09/2006 | EP1687271A1 A method for the preparation of (2s, 3ar, 7as)-octahydro-1h-indole-2-carboxylic acid as key intermediate in the preparation of trandolapril by reacting a cyclohexyl aziridine with a dialkyl malonate |
| 08/08/2006 | CA2188835C Novel compounds and methods for synthesis and therapy |
| 07/19/2006 | EP1680394A1 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents |