Patents
Patents for C07D 203 - Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom (1,097)
07/2006
07/18/2006US7078418 e.g., 2,6-bis(1-aziridino-1-hydroxyiminomethyl)pyridine; treating colon, stomach, lung, breast and uterus cancer
07/05/2006EP1676635A2 Immobilisable ligands derived from ethylenediamine
06/2006
06/29/2006US20060142586 Synthesis of 2-alkyl amino acids
06/15/2006WO2006039383A3 Synthesis by chiral diamine-mediated asymmetric alkylation
06/14/2006EP1187798B1 PRODUCTION OF OPTICALLY ACTIVE $g(a)-HYDROXYACETALS
05/2006
05/16/2006CA2237752C Novel substituted aryl compounds useful as modulators of acetylcholine receptors
04/2006
04/12/2006CN1759093A Azide free process for preparing 1,2-diamino compounds
03/2006
03/30/2006US20060069078 long chain retinyl ketone; prevent retinotoxic accumulation; inhibits, antagonizes, or short-circuits the visual cycle at a step of the visual cycle that occurs outside a disc of a rod photoreceptor
03/28/2006US7019000 administering nitrogen-sulfur compounds, e.g. 4,4-dithiodimorpholine to inhibit binding of the E6 protein by human papilloma virus; treatment of cervical cancer
03/08/2006EP1451167B1 Phenylalkynes
03/07/2006US7008945 Amide derivatives
02/2006
02/22/2006EP1627868A2 Aspartic ester functional compounds
02/22/2006CN1738799A Methods for preparing phenylalkyne derivatives
02/09/2006US20060030718 Cobalt-based catalysts for the cyclization of alkenes
02/08/2006EP1318978B1 N-acylsulfonamide apoptosis promoters
02/02/2006US20060025596 Method for deuteration or tritiation of heterocyclic ring
02/01/2006CN1239451C Process for preparing chiral desubstituted carbinol with high selectivity
01/2006
01/19/2006US20060010609 Mixture with 1,4-diazabicyclo[2.2.2]octane and polar solvent; curing agents; leather treatment, coatings, textile printing; storage stability
01/12/2006US20060009449 Naphthaline derivatives as H3 inverse agonists
01/11/2006CN1720223A Stabilised compositions containing polyfunctional aziridine compounds as hardening constituents
12/2005
12/21/2005EP1606242A1 Azide free process for preparing 1,2-diamino compounds
12/20/2005US6977303 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same
12/15/2005WO2005117865A1 Naphthaline derivatives useful as histamine-3-receptor ligands
12/08/2005US20050272774 Substituted cyclohexane derivatives
11/2005
11/24/2005US20050261203 Azabicyclo-octane inhibitors of IAP
11/17/2005WO2005016264A3 Diamine derivatives of quinone and uses thereof
11/16/2005EP1330464B1 Phosphino-aminophosphines, catalyst complexes and enantioselective hydrogenation
11/08/2005US6962633 cyclic compounds with amine and azide functional groups suitable as hypergolic fuel components for rockets
11/03/2005US20050245551 Amide derivatives
10/2005
10/26/2005EP1589017A2 12,13-modified epothilone derivatives
10/13/2005WO2005094818A1 Azabicyclo-octane inhibitors of iap
10/13/2005CA2558615A1 Azabicyclo-octane inhibitors of iap
10/12/2005CN1680361A Preparation of cyclohexene carboxylate derivatives
10/11/2005US6953806 Cyclohexane derivatives containing amine or amine oxide, useful for treating hypercholesterolemia and hyperlipemia
10/06/2005US20050222081 Cross-linked hyaluronate compounds
10/05/2005EP1581496A2 2-substituted-3-propenamide derivatives and methods of using the same
09/2005
09/07/2005EP1569898A1 Stabilised compositions containing polyfunctional aziridine compounds as hardening constituents
09/06/2005US6939932 Initiator systems, polymerisable compositions, and uses thereof for bonding low surface energy substrates
09/01/2005US20050192317 Novel diamines having a casr modulating activity
08/2005
08/31/2005EP1567494A1 Methods for preparing phenylalkyne derivatives
08/25/2005US20050187392 Hydrolytic kinetic resolution of cyclic substrates
08/11/2005US20050176758 2-(hydroxy or methoxymethoxy)-4-(carboxy or alkoxycarbonyl)-5-(fluoro or hydrogen)-7-oxabicyclo(4.1.0)hept-3-ene chemical intermediates to neuraminidase inhibitors
08/04/2005US20050171082 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same
08/03/2005CN1649861A Kinetics resolution method
08/02/2005US6924378 Method for production of aziridines and N-vinylamides
07/2005
07/06/2005EP1549761A1 Methods and compositions for the modification of nucleic acids
06/2005
06/30/2005US20050143586 N-(di)nitrobenzenesulfonyl-protected-aziridine-2-carboxylic acid derivatives and intermediates; their preparation from haloalanine derivatives that may be N-(di)nitrobenzenesulfonyl-protected, preferably using metal 3,3-dimethyl-3-(optionally protected-amino)propynylides
06/16/2005WO2005054194A1 A method for the preparation of (2s, 3ar, 7as)-octahydro-1h-indole-2-carboxylic acid as key intermediate in the preparation of trandolapril by reacting a cyclohexyl aziridine with a dialkyl malonate
06/15/2005CN1206217C Method for synthesizing azirdine compound
06/01/2005EP1534699A1 Kinetic resolution method
05/2005
05/24/2005US6897323 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same
05/18/2005CN1617865A Phenylalkynes
05/12/2005WO2005042471A1 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents
05/12/2005CA2544335A1 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents
05/11/2005CN1200924C Preparation of cyclohexene carboxylic acid derivative
05/04/2005CN1612887A Phosphino-aminophosphines
04/2005
04/28/2005CA2541509A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
04/27/2005EP1461316A4 Synthesis of 2-cyanoziridine-1-carboxamide
04/27/2005CN1610660A Method for producing perfluoroalkane sulfonic acid esters and the salts thereof
04/26/2005US6884803 Phenylalkynes
04/21/2005US20050085655 Method for producing perfluoroalkane sulfonic acid esters and the salts thereof
04/06/2005CN1604890A 取代的环己烷衍生物 Substituted cyclohexane derivatives
03/2005
03/17/2005WO2005002570A8 Use of an aziridino compound to selectively inactivate parasites in biological compositions
02/2005
02/24/2005WO2005016264A2 Diamine derivatives of quinone and uses thereof
02/10/2005US20050032794 For example, 2-Dimethylamino-N-(3-dimethylamino-1,4-dioxo-1,4-dihydro-naphthalen-2-yl)-N-methyl-acetamide; ability to function as gene expression modulators for genes found in cancer cells, especially genes involved in misregulated signal transduction pathways typical of cancers of colon and breast
01/2005
01/19/2005CN1185223C Novel Compounds and methods for synthesis and therapy
01/13/2005WO2005002570A1 Use of an aziridino compound to selectively inactivate parasites in biological compositions
01/11/2005US6841667 Nucleophilic kinetic resolution of cyclic substrates using silyl azides
01/04/2005CA2133091C Process for the manufacture of (s)-3-amino-1-substituted-pyrrolidines
12/2004
12/08/2004CN1178932C Amide derivatives
11/2004
11/24/2004EP1109550B1 Novel nitrophenylaziridine compounds and their use as prodrugs
11/04/2004US20040220413 Subjecting a specified olefin to an asymmetric aziridination or amination with a specified arylsulfonyl azide compound using using a specified ruthenium (salen) carbonyl complex as a catalyst
11/03/2004EP1472217A2 Method for producing perfluoroalkane sulfonic acid esters and the salts thereof
10/2004
10/27/2004EP1122228B1 Gas-phase dehydration reaction process
10/20/2004CN1171852C Method for inactivating virus in bio-composition
10/05/2004US6800766 Catalyzing the decyclization of racemic and diastereomeric epoxides mixtures in the presence of a non-racemic, chiral catalyst; pharmaceutical synthesis
10/05/2004CA2103837C Novel method of producing 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
09/2004
09/30/2004US20040192681 N-acylsulfonamide apoptosis promoters
09/29/2004EP1461316A2 Synthesis of 2-cyanoziridine-1-carboxamide
09/23/2004WO2004080944A1 Azide free process for preparing 1,2-diamino compounds
09/23/2004WO2004050613A3 2-substituted-3-propenamide derivatives and methods of using the same
09/22/2004CN1167673C Fluorovinyloxyacetamides, process for preparing the same and herbicidal composition comprising the same
09/21/2004US6794534 Synthesis of functionalized and unfunctionalized olefins via cross and ring-closing metathesis
09/16/2004US20040180933 multi-step process for preparing 2-aminoalcohols from 1,2-epoxides; useful as inhibitors of viral or bacterial neuraminidases; intermediates
09/15/2004EP1456171A1 Substituted cyclohexane derivatives
09/14/2004US6790964 Process for the preparation of 7-azabicyclo[4.1.0]hept-3-ene-3-carboxylic acid esters
09/01/2004EP1451308A2 Therapeutic use of aziridino compounds
09/01/2004EP1451167A1 Phenylalkynes
08/2004
08/25/2004EP1449831A1 Method of producing optically active aziridine compounds and amine compounds
08/19/2004WO2003053918A3 Method for producing perfluoroalkane sulfonic acid esters and the salts thereof
08/04/2004EP0942900A4 Stereospecific preparation of chiral 1-aryl- and 1-heteroaryl-2-substituted ethyl-2-amines
07/2004
07/07/2004EP1309550A4 Optically active aziridine-2-carboxylate derivatives and a process for preparing them
06/2004
06/30/2004EP1432734A1 Cytokine receptor
06/24/2004DE10256494A1 Stabilisierte Zusammensetzungen, enthaltend polyfunktionelle Aziridinverbindungen Stabilized compositions containing polyfunctional aziridine
06/17/2004WO2004050623A1 Methods for preparing phenylalkyne derivatives
06/17/2004WO2004050617A1 Stabilised compositions containing polyfunctional aziridine compounds as hardening constituents
06/17/2004WO2004050613A2 2-substituted-3-propenamide derivatives and methods of using the same
06/17/2004CA2507875A1 Methods for preparing phenylalkyne derivatives
06/03/2004US20040106788 asymmetric hydrogenation of a lactam-enamide; multi-step synthesis
06/03/2004US20040106593 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same
1 2 3 4 5 6 7 8 9 10 11