Patents
Patents for C07D 203 - Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom (1,097)
05/2004
05/25/2004CA2048172C Substituted sulfonamids, preparation processes and drugs containing same
05/19/2004EP1229022B1 Process for the preparation of 7-azabicyclo (4.1.0)-hept-3-ene-3-carboxylic acid esters
05/06/2004EP1163237B1 Amide derivatives
05/05/2004CN1148348C 1-substituted-N-sulfinyl-2-aziridine methylenimine and its preparation and use
04/2004
04/21/2004EP1409453A1 Novel diamines having a casr modulating activity
04/13/2004US6720449 N-protecting an optically active 3-haloalanine derivative followed by cyclization for aziridine-2-carboxylic acid derivatives
04/13/2004US6720338 Bcl-x1 inhibiting compositions and methods of promoting apoptosis in a mammal
03/2004
03/24/2004CN1142923C 12,13-modified epothilone derivatives
03/18/2004US20040053316 Contacting composition with an aziridine derivative inactivating agent; killed virus-containing vaccines
03/18/2004US20040053208 Methods to selectively inactivate parasites in biological compositions
03/11/2004WO2004020429A1 Kinetic resolution method
03/11/2004US20040048235 Methods and compositions for the selective modification of nucleic acids
03/11/2004CA2495448A1 Kinetic resolution method
03/04/2004US20040044233 Nucleophilic kinetic resolution of cyclic substrates using silyl azides
02/2004
02/12/2004US20040030133 Amination of 2,3-dibromopropanoate menthol ester; crystallization
02/03/2004US6686477 Multistep chemical synthesis, including asymmetric hydrogenation of a lactam-enamide to produce an intermediate that can be used to make unspecified pharmaceuticals
01/2004
01/15/2004US20040010099 Initiator systems, polymerisable compositions, and uses thereof for bonding low surface energy substrates
01/01/2004US20040002604 Phenylalkynes
12/2003
12/24/2003WO2003066806A3 Therapeutic use of aziridino compounds
12/16/2003CA2268165C Preparation of caprolactam
12/09/2003US6660890 Production of optically active α-hydroxyacetals
11/2003
11/13/2003WO2003093512A1 Methods and compositions for the modification of nucleic acids
11/13/2003CA2484940A1 Methods and compositions for the modification of nucleic acids
11/05/2003CN1453268A Process for producing aziridine compound and N-vinyl amide
10/2003
10/30/2003WO2003089476A1 Cross-linked hyaluronate compounds
10/30/2003US20030204098 Producing the aziridines and the N-vinyl amides industrially advantageously by preventing a solid substance from forming and depositing in the decompressing system which is connected to the purifying step (vacuum distillation)
10/28/2003US6639087 Reacting a nucleophile and a chiral or prochiral cyclic substrate in the presence of a chiral, nonracemic catalyst; changing the oxidation state of catalyst residue to prevent degradation of product mixture; stereospecific
10/23/2003US20030199550 Cyclohexane derivatives containing amine or amine oxide, useful for treating hypercholesterolemia and hyperlipemia
10/22/2003EP1027041B1 Novel cyanoaziridines for treating cancer
09/2003
09/10/2003EP0983236B1 Process for the preparation of an oxirane, aziridine or cyclopropane
09/09/2003US6617157 Using inactivating agent of given formula to inactivate any virus contained in donor blood, blood products, or other biological compositions; can also use in vaccines
09/09/2003US6617101 Lipophilic quenching of viral inactivating agents
08/2003
08/27/2003EP0874809B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials
08/21/2003WO2003045906A3 Synthesis of 2-cyanoziridine-1-carboxamide
08/14/2003WO2003066806A2 Therapeutic use of aziridino compounds
08/14/2003US20030153771 Large scale synthesis of optically pure aziridines
08/14/2003CA2466251A1 Therapeutic use of aziridino compounds
07/2003
07/31/2003US20030144323 Phenylalkynes
07/30/2003EP1330464A2 Phosphino-aminophosphines, catalyst complexes and enantioselective hydrogenation
07/30/2003CN1116280C Prepn. of caprolactam
07/24/2003US20030139614 Catalyzing the decyclization of racemic and diastereomeric epoxides mixtures in the presence of a non-racemic, chiral catalyst; pharmaceutical synthesis
07/16/2003CN1429806A Preparation of cyclohexene carboxylic acid deravitive
07/16/2003CN1114637C Method of reactive amine catalysts for use in polyurethane formation
07/08/2003US6590115 Useful as ligands for metal catalysts for asymmetric reactions, in particular as rhodium complexes for asymmetric hydrogenation of enamide, itaconate, and alpha-ketoester compounds
07/03/2003WO2003053919A1 Substituted cyclohexane derivatives
07/03/2003WO2003053918A2 Method for producing perfluoroalkane sulfonic acid esters and the salts thereof
07/03/2003CA2471038A1 Process for the preparation of perfluoroalkanesulfonic acid esters and salts thereof
07/02/2003EP1322609A2 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and their preparation
07/02/2003CN1113053C Preparation of cyclohexene carboxylate derivatives
06/2003
06/25/2003CN1112354C Stereo specific prepn. of chiral 1-aryl-and 1-heteroaryl-2-substituted ethyl-2-amines
06/19/2003WO2003050099A1 Phenylalkynes
06/19/2003CA2469893A1 Phenylalkynes
06/18/2003EP1318978A2 N-acylsulfonamide apoptosis promoters
06/05/2003WO2003045906A2 Synthesis of 2-cyanoziridine-1-carboxamide
06/03/2003US6573388 Synthetic intermediates for the synthesis of HIV protease inhibitors and oligopeptide mimetics
06/03/2003US6573387 Synthesis of α,β-substituted amino amides, esters, and acids
05/2003
05/28/2003CN1420866A Process for preparation of 7-azabicyclo ÒÇö4.1.0ÒÇò-hept-3-ene-3-carboxylic acid esters
05/22/2003WO2002026705A8 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and their preparation
05/21/2003EP1071656B1 Fluorovinyloxyacetamides, process for preparing same and herbicidal composition comprising same
05/20/2003US6566534 Processes for the preparation of aziridine compounds and vapor-phase reaction processes
05/14/2003EP1309550A1 Optically active aziridine-2-carboxylate derivatives and a process for preparing them
05/08/2003WO2002026750A8 Phosphino-aminophosphines, catalyst complexes and enantioselective hydrogenation
05/08/2003US20030088114 Kinetic resolution method
05/08/2003US20030087945 Sulfonylaminocarboxylic acids
05/06/2003US6559323 Degradation of hydrazone compound to diazo compound; catalysis with transition metal; reaction with sulfide
05/06/2003US6559321 Synthesis of ethyleneimine dimer
04/2003
04/23/2003CN1412179A Method for synthesizing aziridine compound
04/22/2003US6550485 Washing with acidity solution
04/16/2003EP1301458A1 Synthesis of functionalized and unfunctionalized olefins via cross and ring-closing metathesis
04/16/2003EP1040095B1 Cyclohexene carboxylates as neuraminidase inhibitors
03/2003
03/27/2003WO2003025017A1 Cytokine receptor
03/27/2003CA2460151A1 Cytokine receptor
03/19/2003EP1023264B1 New marker, production process and use thereof
03/12/2003EP0724569B1 Process for the preparation of an oxirane, aziridine or cyclopropane
02/2003
02/13/2003US20030032814 Process for preparing optically active amino acid derivatives
02/11/2003US6518438 Preparation of cyclohexene carboxylate derivatives
02/11/2003US6517836 Aziridin-1-yl nitrobenzamides as prodrugs in conjunction with nitroreductase enzymes
01/2003
01/02/2003EP1073648A4 12,13-modified epothilone derivatives
01/02/2003EP1073647A4 12,13-cyclopropane epothilone derivatives
01/01/2003CN1388119A Stereoselective preparation for chirality 1-aryl-and 1-heteroaryl-2-substituted-ethyl-2-amine
12/2002
12/11/2002EP0937039B1 Preparation of caprolactam
12/03/2002US6489515 Gas-phase dehydration reaction process
11/2002
11/26/2002US6486168 Formulations and methods for treatment of mucosal associated conditions with an immune response modifier
11/13/2002CN1094124C Method for purifying lactams
11/05/2002US6476236 Synthesis of 2-cyanoaziridine-1-carboxamide
10/2002
10/30/2002CN1376659A Process for preparing chiral desubstituted carbinol with high selectivity
10/24/2002US20020156300 Reacting chemical intermediate with reducing agent; neuraminidase inhibitor
10/16/2002EP0934316B1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
09/2002
09/26/2002WO2002024636A3 N-acylsulfonamide apoptosis promoters
09/26/2002US20020137978 Using as catalyst ruthenium or osmium carbene complexes containing an imidazolidine ligand
09/25/2002EP0922027B1 Method for purifying lactams
09/18/2002EP1036059B1 Adamantane derivatives
09/17/2002US6451824 Sulfonylaminocarboxylic acids
09/17/2002CA2261832C Method for purifying lactams
09/17/2002CA2122036C Bacterial nitroreductase for the reduction of cb 1954 and analogues thereof to a cytotoxic form
09/10/2002US6448414 Hydrolytic kinetic resolution of cyclic substrates
08/2002
08/13/2002US6433172 Cardiovascular disorders; hypotensive agents; anticholesterol agents
08/07/2002EP1229022A1 Process for the preparation of 7-azabicyclo 4.1.0]-hept-3-ene-3-carboxylic acid esters
07/2002
07/11/2002WO2002026750A3 Phosphino-aminophosphines, catalyst complexes and enantioselective hydrogenation
07/11/2002WO2002026705A3 Highly enantiomerically pure lactam-substituted propanoic acid derivatives and their preparation
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