Patents
Patents for C07D 203 - Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom (1,097)
12/2011
12/27/2011US8084452 Substituted enaminocarbonyl compounds used as insecticides
12/22/2011US20110311582 Novel lipids and compositions for the delivery of therapeutics
12/21/2011CN102292317A 氮丙啶官能化光活性交联化合物 Aziridine functionalized photoactive crosslinking compound
12/14/2011EP2394989A1 Method for producing a N-substituted aziridine
11/2011
11/15/2011USRE42930 Aziridinyl-epothilone compounds
11/09/2011EP2384319A1 Aziridine-functional photoactive crosslinking compounds
09/2011
09/15/2011US20110224431 Triazolium Carbene Catalysts and Stereoselective Bond Forming Reactions Thereof
07/2011
07/28/2011WO2011035064A3 Triazole catalysts and methods of making and using the same
07/27/2011CN101475520B Preparation of water-soluble fullerene
07/21/2011WO2011087664A1 (meth)acryloyl-aziridine crosslinking agents and adhesive polymers
07/06/2011CN102119151A Processes for the preparation of 4-oxo-octahydro-indole-1-carbocylic acid methyl ester and derivatives thereof
06/2011
06/29/2011CN102108133A (Methyl) acrylyl-aziridine crosslinking agent and adhesive polymer
06/23/2011US20110152445 (meth)acryloyl-aziridine crosslinking agents and adhesive polymers
06/21/2011CA2427046C A process for making polyaziridines
06/16/2011WO2011070459A1 Process for enantiomerically pure 8-aryloctanoic acids as aliskiren
06/09/2011US20110137047 Process for enantiomerically pure 8-Aryloctanoic acids as Aliskiren
05/2011
05/12/2011US20110112310 Aziridine synthesis
05/12/2011US20110112288 Metal Porphyrin Catalyzed Olefin Aziridination with Sulfonyl Azides
05/12/2011US20110112254 Polymeric compositions and method of making and articles thereof
05/05/2011US20110105458 Fatty acid inhibitors
05/04/2011EP2315748A1 Processes for the preparation of 4-oxo-octahydro-indole-1-carbocylic acid methyl ester and derivatives thereof
04/2011
04/28/2011WO2011021223A3 Novel salts of ethyl (3r, 4s, 5r)-4,5-imino-3-(l-ethylpropoxy)-1- cvclohexene-1-carboxylate and its use
04/21/2011US20110091508 Oligofluorinated cross-linked polymers and uses thereof
04/19/2011CA2517458C Azide free process for preparing neuraminidase inhibitors r6
04/06/2011CN102001985A Fullerene multi-nitrogen heterocyclic water-soluble derivatives as well as preparation method and application thereof
03/2011
03/24/2011WO2011035064A2 Triazole catalysts and methods of making and using the same
03/03/2011US20110054115 Acrylic pressure-sensitive adhesives with acylaziridine crosslinking agents
02/2011
02/22/2011CA2329181C 12,13-modified epothilone derivatives
02/16/2011CN1960727B Naphthalene derivatives useful as histamine-3-receptor ligands
01/2011
01/20/2011WO2010114291A3 Improved method for preparing dipeptidyl peptidase-iv inhibitor and intermediate
01/19/2011EP2275408A1 Method for synthesizing a n-substituted aziridine
01/18/2011US7872145 Aziridinyl-epothilone compounds
01/06/2011WO2010099206A3 Alkene aziridination
12/2010
12/22/2010EP2264030A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
12/16/2010US20100317832 Aziridine aldehydes, aziridine-conjugated amino derivatives, aziridine-conjugated biomolecules and processes for their preparation
12/07/2010CA2468542C Synthesis of 2-cyanoaziridine-1-carboxamide
11/2010
11/03/2010EP1220838B1 1-aziridino-1-hydroxyiminomethyl-derivatives, method for the production thereof and medicaments containing said compounds
10/2010
10/28/2010US20100273762 Method of combating infection
10/13/2010CN101284244B Catalyst for synthesizing the aziridine type compound
10/07/2010WO2010114291A2 Improved method for preparing dipeptidyl peptidase-iv inhibitor and intermediate
10/07/2010CA2800245A1 Improved method for preparing dipeptidyl peptidase-iv inhibitor and intermediate
10/05/2010CA2369595C Conjugate having a cleavable linkage for use in a liposome
09/2010
09/21/2010US7799934 Intermediates (synthons) in the synthesis of pharmaceuticals such as oseltamivir and other products; treating the arizidine with the nucleophile in the presence of a biaryl phosphoric acid catalyst
09/16/2010WO2010104645A1 Aziridine crosslinking agents for acrylic adhesives
09/09/2010US20100227969 Aziridine crosslinking agents for acrylic adhesives
09/02/2010WO2010099206A2 Alkene aziridination
08/2010
08/26/2010US20100215574 Process for producing an injectable medicament preparation
08/24/2010CA2423103C N-acylsulfonamide apoptosis promoters
08/10/2010CA2237099C Sulfonylaminocarboxylic acids
08/05/2010US20100197688 Epha4 rtk inhibitors for treatment of neurological and neurodegenerative disorders and cancer
08/04/2010EP2213653A2 Method for the stereoselective preparation of amino acid derivatives
07/2010
07/29/2010US20100191000 Method for synthesizing an n-unsubstituted or n-substituted aziridine
07/21/2010CN101781272A Method for preparing repaglinide amine and intermediate thereof
07/13/2010US7754899 Method for producing optically active aziridine compounds and amine compounds as well as complexes and their intermediates used in this method
07/13/2010US7754886 N-acylsulfonamide apoptosis promoters
07/01/2010US20100166871 Vermin poison
06/2010
06/10/2010WO2010065355A1 Aziridine-functional photoactive crosslinking compounds
06/09/2010CN1902159B Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents
06/03/2010US20100137469 Aziridine-functional photoactive crosslinking compounds
05/2010
05/27/2010WO2009129387A3 Cationic lipids and uses thereof
05/20/2010WO2010055887A1 Novel sulfonium salt, method for producing same and use of same
04/2010
04/29/2010US20100105647 Amide compound and use thereof for controlling plant diseases
04/29/2010US20100104515 Use of alpha-hydroxy carbonyl compounds as reducing agents
04/15/2010WO2010041748A1 Fluorene compound and use thereof for medical purposes
04/01/2010US20100081759 Heating an acrylic copolymer with an ester-, amide-, urea- or urethane-functional aziridine crosslinking agent to cure; adhesive tapes with exceptional load bearing capabilities at elevated temperatures; avoids use of VOCs
03/2010
03/24/2010CN101679234A Method for synthesizing an n-unsubstituted or n-substituted aziridine
03/18/2010WO2009146032A3 Metal porphyrin catalyzed olefin aziridination with sulfonyl azides
03/10/2010EP2160379A1 Method for synthesizing an n-unsubstituted or n-substituted aziridine
03/04/2010US20100056806 C-H Bond Amination and Olefin Aziridination with Beta-Diketiminato Copper Catalysts
02/2010
02/24/2010EP1461316B1 Synthesis of 2-cyanoziridine-1-carboxamide
02/23/2010US7666905 Compositions comprising hepoxilin analogs and their use in the treatment of cancer
02/18/2010WO2010018154A1 Processes for the preparation of 4-oxo-octahydro-indole-1-carbocylic acid methyl ester and derivatives thereof
02/18/2010CA2732095A1 Processes for the preparation of 4-oxo-octahydro-indole-1-carbocylic acid methyl ester and derivatives thereof
02/16/2010US7662969 Efficient aziridination of olefins catalyzed by dirhodium catalysts
01/2010
01/19/2010CA2368097C Amide derivatives of 3,4-dihydroquinazolinone compounds useful as cytokine inhibitors
01/14/2010US20100010094 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents
12/2009
12/31/2009DE10147370B4 Waschverfahren für Destillationssysteme von Alkyleniminen Washing method for distillation systems alkyleneimines
12/08/2009US7629332 Antitumor agents such as 2-[(2-Bromoethyl)-2,4-dinitro-6-[[[2-(phosphonooxy)ethyl]amino]-carbonyl]anilino]ethyl methanesulfonate; killing hypoxic cells in a tumor
12/03/2009WO2009146032A2 Metal porphyrin catalyzed olefin aziridination with sulfonyl azides
11/2009
11/11/2009CN101578262A Radiolabelling via fluorination of aziridines
10/2009
10/27/2009US7608617 N,N-alkylene-6-(piperidin-1-ylalkoxy)naphthalene-2-carboxamide derivatives, e.g., piperidin-1-yl-[6-(3-piperidin-1-yl-propoxy)-naphthalen-2-yl]-methanone and 3,4-dihydro-1H-isoquinolin-2-yl)-[6-(3-piperidin-1-yl-propoxy)-naphthalen-2-yl]-methanone; especially for treating obesity
10/01/2009US20090246390 Aziridine crosslinking agents having water solubilizing groups are more environmentally friendly, do not require VOCs, lower cost
09/2009
09/30/2009CN100545145C Azide free process for preparing 1,2-diamino compounds
09/16/2009EP2099749A2 C--h bond amination and olefin aziridination with beta-diketiminato copper catalysts
09/16/2009EP2099747A1 Radiolabelling via fluorination of aziridines
09/09/2009CN100537533C Stabilised compositions containing polyfunctional aziridine compounds as hardening constituents
09/02/2009EP1794129A4 Synthesis by chiral diamine-mediated asymmetric alkylation
08/2009
08/20/2009US20090208740 Improved balance of adhesive and cohesive characteristics, and load bearing capabilities at elevated temperatures; emulsions; environmentally friendly
08/12/2009CN101506140A Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors
08/11/2009CA2546660C Selective inhibitors of viral or bacterial neuraminidase
08/06/2009WO2009096907A1 Aziridine synthesis
07/2009
07/29/2009EP1461315B1 Catalytic carbonylation of three and four membered heterocycles
07/08/2009EP1073647B1 12,13-cyclopropane epothilone derivatives
07/08/2009CN101475520A Preparation of water-soluble fullerene
06/2009
06/25/2009WO2009078813A1 Method of forming oseltamivir and derivatives thereof
06/24/2009CN100503560C Substituted cyclohexane derivatives
05/2009
05/28/2009US20090137585 N-acylsulfonamide apoptosis promoters
05/27/2009EP1740173A4 Azabicyclo-octane inhibitors of iap
05/20/2009EP2059499A1 Processes of preparing asymmetric dinitrobenzamide mustard compounds, intermediate compounds useful therein and products obtained therefrom
05/19/2009CA2468879C Substituted cyclohexane derivatives
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