Patents
Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041)
08/2009
08/18/2009CA2585557C Pyrazolo[4,3-d] pyrimidine derivatives useful as pde-5 inhibitors
08/18/2009CA2219675C Pentacyclic compound
08/13/2009WO2009098369A1 Antimitotic compounds derived from vinca alkaloids, preparation thereof and therapeutic use thereof
08/13/2009CA2714419A1 Dual pharmacophores - pde4-muscarinic antagonistics
08/13/2009CA2714418A1 Dual pharmacophores - pde4 -muscarinic antagonistics
08/12/2009EP2086999A1 Inhibitors for disrupting the interaction of ubiquitination related enzymes and uses thereof
08/12/2009CN101506207A Compound having pyridoindole ring structure having substituted pyridyl group attached thereto, and organic electroluminescence element
08/11/2009US7572784 Inhibit Aurora kinase; cancer; 4-[9-Chloro-7-(2-fluoro-phenyl)-5H-benzo[c]pyrimido[4,5-e]azepin-2-ylamino]-N-(2-methylamino-ethyl)-benzamide; 9-Chloro-N-(4-{[3-(dimethylamino)azetidin-1-yl]carbonyl}phenyl)-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-amine
08/11/2009CA2359772C Cyclic substituted fused pyrrolocarbazoles and isoindolones
08/11/2009CA2222552C N-oxides as antibacterial agents
08/06/2009WO2009097446A1 Pyrazolopyrimidine pi3k inhibitor compounds and methods of use
08/06/2009WO2009096445A1 Nerve trunk cell propagation accelerator
08/06/2009WO2009096435A1 Condensed heterocyclic derivatives and uses thereof
08/06/2009WO2009095787A1 Substituted heteroarylamide oxazepinopyrimidone derivatives
08/06/2009WO2009095254A1 Pyrazolopyrimidines, a process for their preparation and their use as medicine
08/06/2009US20090198454 Standard sample for test and /or calibration of circular dichroism dispersion meter and uv-visible spectrophotometer
08/06/2009CA2713289A1 Substituted heteroarylamide diazepinopyrimidone derivatives
08/06/2009CA2713248A1 Substituted heteroarylamide oxazepinopyrimidone derivatives
08/06/2009CA2711759A1 Pyrazolopyrimidine pi3k inhibitor compounds and methods of use
08/06/2009CA2711575A1 Pyrazolopyrimidines, a process for their preparation and their use as medicine
08/05/2009EP2085400A1 Substituted heteroarylamide oxazepinopyrimidone derivatives
08/05/2009EP2085398A1 Pyrazolopyrimidines, a process for their preparation and their use as medicine
08/05/2009EP2084162A2 Bicyclic triazoles as protein kinase modulators
08/05/2009EP2083844A2 Hcv ns3 protease inhibitors
08/05/2009CN101501042A Pyrazolopyrimidines, a process for their preparation and their use as medicine
08/05/2009CN101501037A Organic electroluminescent device and material for organic electroluminescent device
08/05/2009CN101501036A Substituted pyrazolopyrimidines, a process for their preparation and their use as medicine
08/05/2009CN101500563A Cycloalkanopyrolocarbazole derivatives and the use thereof as PARP, VEGFR2 and MLK3 inhibitors
08/05/2009CN101497623A Compound containing imidazopyridine
08/05/2009CN101497622A Pyridine methyl sulfinyl imidazopyridine derivative
08/04/2009US7569569 Pyrrolo[2,3-d]pyrimidine compounds
07/2009
07/30/2009WO2009093008A1 Thieno-pyridine derivatives as mek inhibitors
07/30/2009WO2009050242A3 Heterocycle-substituted piperazino-dihydrothienopyrimidines
07/30/2009US20090192177 2-ARYL pyrrologpyrimidines for A1 and A3 receptors
07/30/2009CA2711487A1 Quinolizidinone m1 receptor positive allosteric modulators
07/29/2009EP2083014A2 Inhibitors of interleukin-1ß converting enzyme
07/29/2009EP2081937A2 Triazolopyridazine protein kinase modulators
07/29/2009EP1713809B1 Dimeric azacyclic compounds and their use
07/29/2009CN101492465A 7,7'-diaza indirubin compounds for antineoplastic medicament
07/29/2009CN101492464A Sulfhydryl imidazopyridine derivative containing dioxepane-pyridine
07/29/2009CN101492463A Imidazopyridine derivative containing dioxane-pyridine
07/29/2009CN100519560C Porphyrin/phthalocyanine dimer and tetramer directly bonded at pi system and processes for producing the same
07/28/2009US7566727 2-(1-aza-bicyclo[2.2.2]oct-3-yl)-2,3-dihydro-isoindole-1-one/5,6-dihydro-furo[2,3-c] pyrrol-4-one derivative ligands for alpha 7 nicotinic acetylcholine receptor
07/28/2009US7566725 2-(4-methylphenyl),3-(thien-2-yl-carbonyl),6-(methyl)imidazo(1,2-a)pyridine; GABA receptor inhibitors; anxiiolytic agents; sleep disorders (insomnia); psychological disorders; anticonvulsants; aggressiveness; antispasmodic agents; antidepressants/ bipolar disorders;cognition activators; analgesics
07/28/2009US7566707 For example, 2-[3-(Tert-butyloxycarbonylamino)-piperidin-1-yl]-3-(2-butyn-1-yl)-5-[(dibenzo[b,f][1,4]-oxazepin-11-yl)methyl]-3,5-dihydro-imidazo[4,5-d]pyridazin-4-one; inhibiting effect on activity of the enzyme dipeptidylpeptidase-IV; use in treatment of diabetes mellitus, arthritis, obesity
07/28/2009CA2462453C Azabicyclic-substituted fused-heteroaryl compounds for the treatment of disease
07/23/2009WO2008060597A8 Compounds useful as protein kinase inhibitors
07/23/2009US20090186889 Spiro-substituted pyrrolopyrimidines
07/23/2009CA2712783A1 Beta-lactamase inhibitors
07/22/2009EP2080762A1 Compound for organic electroluminescent device and organic electroluminescent device
07/22/2009EP2079750A1 Dna complexing agents
07/22/2009CN100516069C Process for preparing 6-alkylidene penem derivatives
07/21/2009US7563901 potent antimicrobial activity and a wide antimicrobial spectrum in a safe and cost effective reaction
07/21/2009US7563791 6-(Methoxymethyl)-5-(4-nitrophenyl)pyrrolo[2,1-f][1,2,4]triazin-4-amine; antiproliferative agents; angiogenesis inhibition; anticarcinogenic agents; breast cancer; colon cancer; antitumor agents
07/21/2009CA2478393C 1-allyl ergot alkaloid derivatives, methods for their production and their use for migraine prevention and treatment
07/21/2009CA2367921C Bicyclic heterocycles, processes for their preparation and their use as herbicides and pharmaceutical agents
07/16/2009WO2009087364A1 Electroluminescent materials
07/16/2009US20090181982 Substituted pyrroline kinase inhibitors
07/15/2009EP2078721A2 Thieno-pyrimidime compounds having fungicidal activity
07/15/2009EP2078010A2 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
07/15/2009EP2078009A1 New fluorene derivatives, compositions containing the same and use thereof as inhibitors of the protein chaperone hsp 90
07/15/2009EP1458726B1 Mitotic kinesin inhibitors
07/14/2009US7560454 1-(4-(10,11-dihydro-5H-pyrrolo[2,1-c](1,4)benzodiazepine-10-ylcarbonyl)-2-methyl-benzylcarbamoyl)-4methoxy-L-proline-N,N-dimethylamide; vasopressin agonists particularly useful in the treatment of urogenital disorders central diabetes insipidus, nocturnal enuresis and nocturia; blood disorders
07/10/2009WO2008083367A2 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
07/10/2009CA2710234A1 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
07/09/2009US20090176806 protein kinase C or glycogen synthase kinase-3-beta inhibitors such as 3-(2-chlorophenyl)-4-[1-(3-hydroxypropyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-1H-pyrrole-2,5-dione, used for treating cardiovascular, skin, nervous system disorders and immunological disorders, diabetes, inflammatory diseases and cancer
07/09/2009US20090176763 Azaindoles useful as inhibitors of JAK and other protein kinases
07/09/2009US20090173916 Fluorescent diketopyrrolopyrroles
07/08/2009EP2077268A1 Process for preparing inhibitors of nucleoside metabolism
07/08/2009EP1495022B1 Diazabicyclo alkane derivatives with nk1 antagonistic activity
07/08/2009CN100509811C Azaindoles
07/07/2009US7557099 Pyrrolobenzodiazepines as key intermediates in the synthesis of dimeric cytotoxic pyrrolobenzodiazepines
07/02/2009WO2009081197A1 Bicyclic derivatives for use in the treatment of androgen receptor associated conditions
07/02/2009WO2009080682A1 Pyrrolo[2,3-d]pyrimidine derivatives as cgrp receptor antagonists
07/02/2009WO2009079765A1 Compounds with activity at the 5-ht2c receptor
07/02/2009US20090169560 Disulfide, sulfide, sulfoxide, and sulfone derivatives of cyclic sugars and uses thereof
07/02/2009US20090169508 Opioid and opioid-like compounds and uses thereof
07/02/2009CA2709514A1 Bicyclic derivatives for use in the treatment of androgen receptor associated conditions
07/01/2009EP2074115A1 N3-heteroaryl substituted triazoles and n5-heteroaryl substituted triazoles useful as axl inhibitors
07/01/2009CN100506825C Heterotricyclyl 6-alkylidene-penems as beta epsilontaualpha-lactamase inhibitors
07/01/2009CN100506824C Preparation of 2,2'-di(3,4-ethylenedioxy-thiophene)
06/2009
06/30/2009US7553975 2-(((2-amino-1-oxo-3-mercapto-propyl)-amino)-methyl)-5-phenyl-thiazole-4-carbonyl-methionine; useful for treating restenosis or tissue proliferative diseases
06/25/2009WO2009077741A2 3-substituted-4-0x0-3, 4-dihydro-imidazo- [5, 1-d] [1,2,3,5] -tetrazine-8-carboxylic acid amides as anticancer agents
06/25/2009CA2709749A1 3-substituted-4-oxo-3,4-dihydro-imidazo[5,1-d][1,2,3,5]-tetrazine-8-carboxylic acid amides and their use
06/24/2009CN100503608C Deazapurines and uses thereof
06/23/2009US7550494 Small molecules useful in the treatment of inflammatory disease
06/23/2009US7550455 8-(piperazin-1yl)- and 8-([1,4]diazepan-1yl)-xanthines, the preparation thereof and their use as pharmaceutical composition
06/18/2009WO2009075359A1 Method of separating isomers of chiral substances and apparatus therefor
06/18/2009WO2009037394A3 6-cycloamino-s-(pyridazin-4-yl)imidazo[1,2-b]-pyridazine and derivatives thereof preparation and therapeutic application thereof
06/18/2009US20090156821 Quinazoline compounds
06/18/2009US20090156630 Anti-tumour polycyclic carboxamides
06/18/2009CA2707857A1 Organic compounds
06/17/2009EP2070930A1 Polycycloalkylpurines as adenosine receptor antagonists
06/11/2009US20090149468 Substituted heterocyclic compounds and methods of use
06/10/2009EP2066324A2 Cycloalkanopyrolocarbazole derivatives and the use thereof as parp, vegfr2 and mlk3 inhibitors
06/10/2009CN100497349C Improved Biapenem preparation method
06/09/2009US7544693 Spirofuropyridine aryl derivatives
06/09/2009US7544677 Cancer; 2-(methylthio)-6-phenyl-7-(4-{[4-(5-pyridin-2-yl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenyl)pyrido[2,3-d]pyrimidine;serine/threonine kinase (Akt) suppression; increased cellular potency or solubility, greater selectivity, enhanced pharmacokinetic properties, lack of off target activity
06/09/2009US7544312 Charge transport compositions and electronic devices made with such compositions
06/04/2009WO2009069589A1 Novel naphthyridine derivative monohydrate and method for producing the same
1 ... 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 ... 111