Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041) |
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07/10/2008 | US20080167475 Intermediates of 2-substituted carbapenem derivatives and process for production thereof |
07/10/2008 | CA2710046A1 N3-heteroaryl substituted triazoles and n5-heteroaryl substituted triazoles useful as axl inhibitors |
07/10/2008 | CA2673965A1 Pyrazolopyrimidine compound |
07/09/2008 | EP1940847A2 Pyrazolopyrimidines as protein kinase inhibitors |
07/09/2008 | EP1940835A1 Pyrazolo[3,4-b]pyridine compounds, and their use as pde4 inhibitors |
07/09/2008 | EP1940401A2 Acylated spiropiperidine derivatives as melanocortin-4 receptor modulators |
07/09/2008 | CN101214248A Triazolo[4,5-d] pyrimidine derivatives and their application as purinergic receptor antagonists |
07/09/2008 | CN100400540C Isoxazoline derivatives as anti-depressants |
07/09/2008 | CN100400042C Methods for making sustained release pharmaceutical compositions of ergot alkaloids having improved bioavailability and compositions thereof |
07/08/2008 | US7396926 Compound for use in the measurement of gene expression |
07/03/2008 | WO2008077811A1 Spiro-piperidine derivatives |
07/03/2008 | US20080161572 Preparation Method |
07/03/2008 | CA2674518A1 Spiro-piperidine derivatives |
07/02/2008 | EP1939202A1 Novel adenine compound |
07/02/2008 | EP1937691A1 Thieno-pyrimidine compounds having fungicidal activity |
07/02/2008 | EP1474425B9 Deazapurines and uses thereof |
07/02/2008 | CN100398545C Thienopyrazoles |
07/01/2008 | US7393957 Generation triple-targeting, chiral, broad-spectrum antimicrobial 7-substituted piperidino-quinolone carboxylic acid derivatives, their preparation, compositions and use as medicaments |
07/01/2008 | US7393859 Amide substituted imidazoquinolines |
07/01/2008 | US7393551 Denatured carob flour (DCF) with a low content of soluble tannins and sugars, meant for human consumption and process to obtain it |
06/26/2008 | WO2008075109A1 Substituted piperidines having protein kinase inhibiting activity |
06/26/2008 | WO2008047201A3 Solid dispersion comprising a poorly water soluble drug |
06/26/2008 | US20080153899 Fatty amine drug conjugates |
06/26/2008 | US20080153855 Chemical Compounds |
06/25/2008 | EP1670796B1 Imidazopyridine-derivatives as inducible no-synthase inhibitors |
06/25/2008 | EP1430147A4 Fluorescent quenching detection reagents and methods |
06/19/2008 | WO2008072655A1 Imidazothiazole derivatives |
06/19/2008 | WO2008072634A1 Fused heterocyclic compound |
06/19/2008 | WO2008071964A1 Naphthyridine bactericides |
06/19/2008 | WO2008071962A1 Pteridines and pyrimidinopyridines as antibacterial agents |
06/19/2008 | WO2008071937A1 Novel fluorescent kinase ligands and assays employing the same |
06/19/2008 | US20080146546 Bicyclic and Tricyclic Heteroaromatic Compounds |
06/19/2008 | CA2673097A1 Fused heterocyclic compound |
06/19/2008 | CA2672565A1 Imidazothiazole derivatives |
06/18/2008 | EP1931674A2 Deazapurines useful as inhibitors of janus kinases |
06/18/2008 | CN101203519A 2-amido-6-amino-8-oxopurine derivatives as ToII-like receptor modulators for the treatment of cancer and viral infections, such as hepatitis c |
06/18/2008 | CN101203516A Purine and imidazopyridine derivatives for immunosuppression |
06/18/2008 | CN101200457A Dihydro pteridinone, method for making the same and uses as pharmaceutical preparation thereof |
06/12/2008 | WO2008068392A1 Novel imidazo[1,2-a]pyridine-3-ylamine fluorophore derivatives and process for the preparation thereof |
06/12/2008 | WO2008068185A1 Spiro-piperidine derivatives as via receptor antagonists |
06/12/2008 | WO2007081597A3 Peri condensed tricyclic compounds useful as antibacterial agents |
06/12/2008 | US20080139812 Heterocyclical Chromophore Architectures |
06/12/2008 | CA2671990A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
06/12/2008 | CA2670674A1 Spiro-piperidine derivatives as via receptor antagonists |
06/11/2008 | EP1492803B1 New analogs of nitrobenzylthioinosine |
06/11/2008 | EP1255739B1 3-aminoquinazolin-2,4-dione antibacterial agents |
06/11/2008 | CN100393789C Composition stablized to heat, oxidation or optical degradation stablized mixture and its preparation process |
06/10/2008 | US7384952 1-(3-ethoxybenzyl)-4-[4-[4-[2-(dimethylamino)ethoxy]benzoyl]piperazin-1-yl]-1H-pyrazolo[3,4-d]pyrimidine; small conductance potassium channel (SK channel) blocking activity; gastrointestinal disorders |
06/10/2008 | US7384950 Respiratory system disorders; asthma; chronic obstructive pulmonary disease |
06/10/2008 | US7384946 M3 muscarinic acetylcholine receptor antagonists |
06/10/2008 | US7384931 Constrained compounds as CGRP-receptor antagonists |
06/10/2008 | US7384930 [9-(2,2-Dimethyl-propyl)-8-oxo-3,6,7,8,9,10-hexahydro-2,3,9-triaza-(S)-cyclohepta[e]inden-7-yl]-acetic acid methyl ester; calcitonin gene-related peptide receptor antagonist; analgesic, antiinflammatory agent; migraine, neurogenic vasodilation, circulatory shock, menopause, asthma |
06/10/2008 | US7384928 7-side chain is substituted with aminothiazole and 3-position with a cyclic-type quarternary ammoniummethyl group; antibacterial activities against cephem-resistant Pseudomonas aeruginosa which produce beta -lactamase; antibiotic resistance; pharmacokinetics; high water solubility; injection |
06/05/2008 | US20080132526 Purine Derivative |
06/05/2008 | DE60129697T2 Kondensierte azepinderivate und ihre verwendung als antidiuretisches mittel Condensed azepine derivatives and their use as antidiuretic agent |
06/04/2008 | CN101193899A Monomers, oligomers and polymers of thieno (3, 4-D) thiazole |
06/03/2008 | US7381723 Antiserotonine agents; stroke, brain disorders;trauma; Alzheimer's disease; neurodegenerative disease; schizophrenia; psychological disorders; anxiolytic agents; controlling stresses; eating disorders; sleep disorders; sexual disorders |
06/03/2008 | US7381720 Tumor suppression agents with reduced side effects; anticancer; antibacterial and antiviral |
06/03/2008 | CA2180829C Cephalosporin synthesis |
05/29/2008 | WO2008019356A3 Process for the preparation of substituted-1,2,3,4-tetrahydroisoquinoline derivates |
05/29/2008 | CA2636242A1 Heterobicyclic thiophene compounds and methods of use |
05/28/2008 | EP1925618A1 Imidazopyridine-based compounds and organic light emitting diode including organic layer comprising the imidazopyridine-based compounds |
05/28/2008 | EP1925614A1 Anxiolytic agents with reduced sedative and ataxic effects |
05/28/2008 | EP1660475B1 Pyrimidylpyrrole derivatives active as kinase inhibitors |
05/28/2008 | EP1501507B1 Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity |
05/28/2008 | CN101189227A New derivatives of pyrrolyltriazine together with methods for obtaining them and their use as protecting agents against uv radiation |
05/28/2008 | CN100390178C Polycycloalkylpurines as adenosine receptor antagonists |
05/27/2008 | US7378534 Anti-first-pass effect compounds |
05/27/2008 | US7378524 e.g., 6-chloro-2-methyl-4-(N-(2-(N-(p-methoxyphenylsulfonyl)-N-(2-(2,5-dimethoxy-4-nitroanilinocarbonyl)ethyl)amino)ethyl)amino)quinoline; used to treat inflammatory and immune diseases by binding to CXCR3 receptors. |
05/27/2008 | US7378411 Substituted thienopyrimidinones as a mitotic kinesin inhibitor |
05/22/2008 | WO2008060301A1 7-substituted purine derivatives for immunosuppression |
05/22/2008 | CA2669886A1 Compounds useful as protein kinase inhibitors |
05/22/2008 | CA2669686A1 7-substituted purine derivatives for immunosuppression |
05/21/2008 | EP1456206B1 Azaindolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands |
05/15/2008 | WO2008057054A1 Dna complexing agents |
05/15/2008 | WO2008056187A1 Imidazolopyrimidines and imidazolotriazine derivatives as inhibitors of poly(adp-ribose) polymerase (parp) |
05/15/2008 | US20080114023 Azaindolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands |
05/15/2008 | US20080113972 Enzyme inhibitors of cGMP-metabolizing phosphodiesterases, for TREATMENT OF CARDIOVASCULAR DIORDERS, CEREBROVASCULAR DISORDERS, UROGENITAL DISORDERS AND ERECTILE DYSFUNCTION; chemical synthesis |
05/15/2008 | US20080113971 improved potency; reduced undesirable side effects; pain, inflammation, arthritis etc; ethyl 1-(2-aminoethyl)-3-pyridin-4-yl-1H-pyrazole-5-carboxylate dihydrochloride |
05/15/2008 | US20080113941 4-O esters of podophyllotoxin and 4'-demethylepipodophyllotoxin 4'-phosphonic acid or phosphonate derivatives; anticancer agents; type II DNA topoisomerase (topoisomerase II) inhibitors |
05/15/2008 | US20080109989 Stacking wall panel system and methods of installation and use |
05/15/2008 | CA2669432A1 Imidazolopyrimidines and imidazolotriazine derivatives as inhibitors of poly(adp-ribose) polymerase (parp) |
05/14/2008 | EP1919475A1 Tetrahydro- beta-carbolin-sulfonamide derivatives as 5-ht6 ligands |
05/13/2008 | US7371470 Pyran derivative |
05/08/2008 | WO2008055013A2 5-oxo-5,8 - dihydro - pyrido - pyrimidines as inhibitors of c-fms kinase |
05/08/2008 | WO2008052441A1 Inhibitors for disrupting the interaction of ubiquitination related enzymes and uses thereof |
05/08/2008 | US20080108644 alkaloids; anticarcinogenic, antiproliferative agent; inhibitor of cellular mitosis and cell proliferation; binding to tubulin leads to cell cycle arrest in M phase and subsequently to apoptosis; antiallergen, antiinflammatory, antidiabetic, autoimmune diseases; asthma, arthritis, Alzheimer' disease |
05/08/2008 | US20080108605 Anxiolytic agents with reduced sedative and ataxic effects |
05/08/2008 | US20080108141 2,3-diaminonaphthalene reacts with nitric oxide to give fluorescent naphthalenetriazole |
05/07/2008 | EP1383774B1 Dihydroimidazo¬4,5-e indole and 7h-pyrrolo¬3,2-f quinoxaline derivatives as nicotinic acetylcholine receptor ligands and/or serotonergic ligands |
05/07/2008 | CN101172981A 2,3-dihydroimidazo[2,1-b]oxazole compound |
05/07/2008 | CN100386329C Substituted 3-amino-thieno(2,3-b)pyridine-2-carboxylic acid amide compounds and processes for preparing and their uses |
05/06/2008 | US7368459 Heterocyclic compounds |
05/06/2008 | US7368438 Non-nucleotide compositions and method for inhibiting platelet aggregation |
05/06/2008 | US7368437 Bicyclic heterocycles, processes for their preparation and their use as herbicides and pharmaceutical agents |
05/06/2008 | CA2327468C Semi-synthetic ecteinascidins |
05/02/2008 | WO2008051552A2 Organic semiconductor materials and methods of preparing and use thereof |
05/02/2008 | WO2008050871A1 Crystalline carbapenem compounds |
05/02/2008 | WO2008049994A1 New fluorene derivatives, compositions containing the same and use thereof as inhibitors of the protein chaperone hsp 90 |
05/02/2008 | CA2667453A1 Triazolo-pyridazine protein kinase modulators |