| Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041) |
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| 08/31/2010 | US7786135 Substituted pyrroline kinase inhibitors |
| 08/31/2010 | US7786107 Treating neurodegenerative diseases, psychological disorders, pain, glaucoma, dru eye, dry mouth, Sjogren's syndrome, asthma, bradycardia, wound healing, gastrointestinal disorders; amide- or urea-functional 1,2,3,4-tetrahydrospiro[benzo[b]azepine-5,4'-piperidine] rings; selective as to subtypes M1-M5 |
| 08/26/2010 | US20100216970 Methods, compositions, and apparatuses for forming macrocyclic compounds |
| 08/26/2010 | US20100216252 use of the complexes obtained as fluorescent markers, and as relaxation agents for NMR or for NMR imaging |
| 08/25/2010 | EP2221309A1 Novel naphthyridine derivative monohydrate and method for producing the same |
| 08/25/2010 | EP2220095A1 Inhibitors of human immunodeficiency virus replication |
| 08/25/2010 | EP2220083A2 Imidazo[1,2-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
| 08/25/2010 | EP1339402B1 Azaphenanthridone derivatives and their use as parp inhibitors |
| 08/25/2010 | CN101812079A Piprazine compound containing polysulfide bond and preparation method and application thereof |
| 08/24/2010 | US7781450 protein kinase C or glycogen synthase kinase-3-beta inhibitors such as 3-(2-chlorophenyl)-4-[1-(3-hydroxypropyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-1H-pyrrole-2,5-dione, used for treating cardiovascular, skin, nervous system disorders and immunological disorders, diabetes, inflammatory diseases and cancer |
| 08/24/2010 | US7781431 Thienopyrroles as antiviral agents |
| 08/24/2010 | CA2520897C Pyrrolo (2,1-c)(1,4) benzodiazepine dimers as antitumour agents and process thereof |
| 08/19/2010 | WO2010093341A1 C-7 isoxazolinyl quinolone/naphthyridine derivatives useful as antibacterial agents |
| 08/19/2010 | WO2009061453A8 Solubilized thiazolopyridines |
| 08/19/2010 | US20100210679 Preventive and therapeutic medicament for gastroesophageal reflux disease |
| 08/18/2010 | EP2218705A1 Method of separating isomers of chiral substances and apparatus therefor |
| 08/18/2010 | EP2217606A1 Solubilized thiazolopyridines |
| 08/18/2010 | CN1922182B Pyrrolotriazine compounds as kinase inhibitors |
| 08/18/2010 | CN101805699A Method for preparing gliocladicillin C and application thereof |
| 08/18/2010 | CN101805359A Method for preparing biapenem with high purity |
| 08/18/2010 | CN101440099B Industrial large scale extracting method for nimbin dry powder |
| 08/17/2010 | US7777058 A thrombolytic agent in combination with a compound such as2-methylthioisosorbide 5-mononitrate; cardiovascular diseases such as, atherosclerosis, cardiac allograft vasculopathy, and tissue damage due to ischemia and/or to ischemia-reperfusion |
| 08/17/2010 | US7776867 Furanopyrimidines |
| 08/12/2010 | WO2010090077A1 Organic electroluminescent element, and illumination device and display device each comprising the element |
| 08/12/2010 | WO2010011546A3 Pyrrolo [3, 2-b]pyridines and pyrazolo [4, 3 -b] pyridines having 5-ht6 receptor affinity |
| 08/12/2010 | US20100204267 Preventive and therapeutic medicament for gastroesophageal reflux disease |
| 08/11/2010 | EP2215095A1 Cyclopropyl fused indolobenzazepine derivatives for the treatment of hepatitis c |
| 08/11/2010 | EP2215093A1 Novel piperazino-dihydrothienopyrimidine derivatives |
| 08/11/2010 | EP2215092A1 Substituted piperidino-dihydrothienopyrimidines |
| 08/11/2010 | EP2215090A1 Purine derivatives useful as pi3 kinase inhibitors |
| 08/11/2010 | CN101801971A Deazapurines useful as inhibitors of janus kinases |
| 08/11/2010 | CN101801376A Pyrazolo (3, 4-b) pyridine derivatives as phosphodiesterase inhibitors |
| 08/10/2010 | US7772229 Oxabispidine compounds useful in the treatment of cardiac arrhythmias |
| 08/10/2010 | US7772227 such as (R)-3-Cyclohexyl-2,3-dihydro-6-(4-ethylpiperazin-1-ylcarbonyl)pyrrolo[1,2,3-de]-1,4-benzoxazine hydrochloride salt, used as analgesics for the treatment of post-operative pain, chronic pain neuropathic pain, cancer pain and spasticity associated with multiple sclerosis |
| 08/10/2010 | CA2477967C Purine derivatives as kinase inhibitors |
| 08/10/2010 | CA2451605C Diamine derivatives |
| 08/10/2010 | CA2440714C Pyrazolopyrimidines as therapeutic agents |
| 08/05/2010 | WO2010086638A1 Dimeric pyrrolopyrimidinedione and its use in therapy of respiratory diseases |
| 08/05/2010 | US20100196387 Disulfide, Sulfide, Sulfoxide, and Sulfone Derivatives of Cyclic Sugars and Uses Thereof |
| 08/05/2010 | CA2751054A1 Dimeric pyrrolopyrimidinedione and its use in therapy of respiratory diseases |
| 08/04/2010 | EP2213673A1 Pyridone-substituted-dihydropyrazolopyrimidinone derivative |
| 08/04/2010 | EP2212333A1 Thienopyrimidine and pyrazolopyrimidine compounds and their use as mtor kinase and pi3 kinase inhibitors |
| 08/04/2010 | EP2212332A1 Substituted tricyclic compounds and methods of use thereof |
| 08/04/2010 | EP2212321A2 (1,4-diaza-bicyclo[3.2.2]non-6-en-4-yl)-heterocyclyl-methanone ligands for nicotinic acetylcholine receptors, useful for the treatment of disease |
| 08/04/2010 | CN101792457A Method for preparing 5,5',7,7'-tetramethyl-2,2'-linked-([1,2,4]-triazol [1,5-a]) pyrimidine |
| 08/03/2010 | US7767813 Eliminating excess bipiperidinyl-1'-carbonyl chloride after it has reacted with 7-ethyl-10-hydroxy camptothecin and crystallizing the pure irinotecan hydrochloride formed |
| 08/03/2010 | US7767808 Porphyrin-phthalocyanine dimer and tetramer having directly-bound π electron systems and production method thereof |
| 07/29/2010 | WO2010084425A1 New adenosine receptor ligands and uses thereof |
| 07/29/2010 | US20100190898 Weakly Basic Hindered Amines Compounds Having Carbonate Skeletons, Synthetic Resin Compositions And Coating Compositions |
| 07/29/2010 | CA2750449A1 New adenosine receptor ligands and uses thereof |
| 07/28/2010 | EP2210891A1 New adenosine receptor ligands and uses thereof |
| 07/28/2010 | EP2209375A1 Parp inhibitor compounds, compositions and methods of use |
| 07/28/2010 | CN101790533A cyclopropyl fused indolobenzazepine hcv inhibitors |
| 07/27/2010 | US7763727 electrophotographic photoconductor, an organic transistor, an organic electroluminescent device and an organic solar cell; naphthalene monoimide derivative, naphthalene monoimide monohydrazone derivative |
| 07/27/2010 | US7763641 such as [(1S,2R)-2-hydroxy-3-[N-[4-(2-methylaminothiazol-4-yl)phenylsulfonyl]-N-(2-methylpropyl)amino]-1-(phenylmethyl)propyl]carbamic acid, [(3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl]ester, used for treating human immunodeficiency virus infections |
| 07/27/2010 | CA2481241C Fused quinoxaline derivatives as inhibitors of akt activity |
| 07/22/2010 | US20100184754 Quinolinone derivatives |
| 07/21/2010 | CN101784552A 6-cycloamino-s-(pyridazin-4-yl)imidazo[1,2-b]-pyridazine and derivatives thereof preparation and therapeutic application thereof |
| 07/21/2010 | CN101784551A bicycloaniline derivative |
| 07/21/2010 | CN101781322A Process method for preparing vinorelbine |
| 07/21/2010 | CN101369633B Pyran derivative |
| 07/20/2010 | US7759361 treating a cancer, autoimmune diseases and cardiovscular disorders comprising administering drugs such as Isobutyric acid 2-isobutyryloxymethyl-3-oxo-1-aza-bicyclo[2.2.2]oct-ylmethyl ester; antiproliferative agents |
| 07/15/2010 | US20100179128 Xanthine derivatives as selective hm74a agonists |
| 07/14/2010 | EP2205610A1 Thienopyrimidiene derivatives as pi3k inhibitors |
| 07/14/2010 | EP2205603A1 Pyrimidine derivatives as protein kinase inhibitors |
| 07/14/2010 | EP1636224B1 Pyrrolopyridine-2-carboxylic acid amide inhibitors of glycogen phoshorylase |
| 07/14/2010 | CN101775028A Method for gathering and purifying agrimonine in agrimony |
| 07/13/2010 | US7754732 such as 4-Oxo-2-phenyl-1,3,8-triaza-spiro[4,5]dec-1-ene-8-carboxylic acid{1-7-methyl-1H-indazol-5-yl methyl)-2-[1,4]bipiperidinyl-1'-yl-2-oxo-ethyl}-amide, used as antagonists of calcitonin gene-related peptide receptors; used in the therapy of headaches and respiratory system disorders |
| 07/08/2010 | WO2010015518A3 4-dimethylamino-phenyl-substituted naphthyridines, and use thereof as medicaments |
| 07/08/2010 | US20100174058 Fluorescent quenching detecting reagents and methods |
| 07/08/2010 | US20100173895 Imidazolopyrimidines and imidazolotriazine derivatives as inhibitors of poly(adp-ribose)polymerase(parp) |
| 07/07/2010 | CN101772498A Heteroaryl amide analogues as p2x7 antagonists |
| 07/07/2010 | CN101768174A Method for preparing biapenem |
| 07/07/2010 | CN101768173A Norcantharidin dimer derivate as well as synthetic method and application thereof |
| 07/07/2010 | CN101298454B Cephalosporin derivate containing pyrazolo triazinium |
| 07/06/2010 | US7750152 Preparing 1-methyl,2-oxo,3-ethyl,4-cyclopentyl,6-chloro-1,2,3,4-tetrahydropteridine by reacting ethyl 2-N-cyclopentylaminobutyrate hydrochloride with 2,4-dichloro-5-aminopyrimidine; reducing, cyclizing and methylating by electrolytic substitution; antiproliferative, -carcinogenic and -tumor agents |
| 07/06/2010 | US7750148 chemical intermediates for making an oral antibiotics Sulbactam |
| 07/01/2010 | WO2010072399A1 7-azaindirubins, 7'azaindirubins, 7,7'-diazaindirubins and the corresponding 3'-oxime ether derivatives thereof, their production and use as a medicament |
| 07/01/2010 | WO2010046445A3 Urea derivatives of substituted nortropanes, medicaments containing such compounds and their use |
| 07/01/2010 | US20100168157 Preventive and therapeutic medicament for gastroesophageal reflux disease |
| 06/30/2010 | EP2202293A2 New mutactimycin and aldgamycin active compounds and the use thereof in therapy |
| 06/30/2010 | CN101765602A 6-cycloamino-3-(pyridin-4-yl)imidazo[1,2-b]pyridazine derivatives, preparation thereof and therapeutic use thereof |
| 06/30/2010 | CN101765599A Tropane derivatives useful as pesticides |
| 06/29/2010 | US7745619 alkaloids; anticarcinogenic, antiproliferative agent; inhibitor of cellular mitosis and cell proliferation; binding to tubulin leads to cell cycle arrest in M phase and subsequently to apoptosis; antiallergen, antiinflammatory, antidiabetic, autoimmune diseases; asthma, arthritis, Alzheimer' disease |
| 06/24/2010 | WO2010070452A1 Fused imidazole carboxamides as trpv3 modulators |
| 06/24/2010 | CA2746077A1 Fused imidazole carboxamides as trpv3 modulators |
| 06/23/2010 | EP2199292A1 7-azaindirubins, 7'-azaindirubins, 7-7'-diazaindirubin and the corresponding 3'-oxime ether derivates: production thereof, their production and use as a medicament |
| 06/23/2010 | CN101747352A Preparation method for biapenem condensation compound and crystalline solid thereof |
| 06/23/2010 | CN101747351A Synthetic method of Xyloketals compounds |
| 06/23/2010 | CN101007815B Pyrrolehexa-heterocyclic compound and pharmaceutical use thereof |
| 06/22/2010 | US7741343 6H-oxazolo[4,5 e]indole derivatives as nicotinic acetylcholine receptor ligands and/or serotonergic ligands |
| 06/22/2010 | US7741339 Fab I inhibitors |
| 06/22/2010 | US7741319 11-hydroxy-5h-pyrrolo[2,1-c][1,4] benzodiazepin-5-one derivatives as key intermediates for the preparation of c2 substituted pyrrolobenzodiazepines |
| 06/22/2010 | CA2540834C Imidazopyridine substituted tropane derivatives with ccr5 receptor antagonist activity for the treatment of hiv and inflammation |
| 06/22/2010 | CA2398988C Anti acid-fast bacterial agent containing pyridonecarboxylic acids as active ingredient |
| 06/17/2010 | WO2010067886A1 Dihydropyrimidopyrimidine derivative |
| 06/17/2010 | WO2010067332A1 5-amino-2-(1-hydroxy-ethyl)-tetrahydropyran derivatives |
| 06/17/2010 | CA2745970A1 Dihydropyrimidopyrimidine derivative |
| 06/17/2010 | CA2744456A1 5-amino-2-(1-hydroxy-ethyl)-tetrahydropyran derivatives |
| 06/16/2010 | CN1982308B Substituted pyrazoles |