Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041) |
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01/19/2010 | CA2239904C Inhibitors of interleukin-1.beta. converting enzyme |
01/14/2010 | WO2010004837A1 Therapeutic agent for amyotrophic lateral sclerosis |
01/14/2010 | WO2010004394A1 9-substituted-b-carboxy-oxadiazino-quinolone derivatives, their preparation and their application as anti-bacterials |
01/14/2010 | CA2727820A1 9-substituted-5-carboxy-oxadiazino-quinolone derivatives, their preparation and their application as anti-bacterials |
01/14/2010 | CA2727282A1 Novel pyrrolidine derivatives as metap-2 inhibitors |
01/12/2010 | US7645763 dipeptidylpeptidase-IV inhibitors; antidiabetic agents, antiarthritic agents, obesity, allograft transplantation, and osteoporosis caused by calcitonin; 1,3-disubstituted-7-(2-butyn-1-yl)-8-(3-aminopiperidin-1-yl)-xanthine compounds |
01/12/2010 | US7645758 (4-Methyl-piperazin-1-yl)-(6H-thieno[2,3-b]pyrrol-5-yl)-methanone; (2,3-Dichloro-6H-thieno[2,3-b]pyrrol-5-yl)-(4-methyl-piperazin-1-yl)-methanone; histamine H4 receptor antagonist; treats allergic rhinitis |
01/12/2010 | CA2399818C Preventive and therapeutic medicament for gastroesophageal reflux disease |
01/07/2010 | US20100004463 Process for synthesizing carbapenem using raney nickel |
01/06/2010 | EP2139334A1 2-cyanophenyl fused heterocyclic compounds, and compositions and uses thereof |
01/06/2010 | EP1885364B1 Halogenated quindoline dimers for the treatment of cancer |
01/05/2010 | US7642362 Compounds as semaphorin inhibitors |
01/05/2010 | US7642229 Synergistic antineoplastic effect; side effect reduction |
01/05/2010 | CA2318192C .beta.2-adrenergic receptor agonists |
12/31/2009 | US20090326221 New oxabispidine compunds useful in the treatment of cardiac arrhythmias |
12/31/2009 | US20090326218 Azepinoindole and Pyridoindole Derivatives as Pharmaceutical Agents |
12/31/2009 | US20090324625 Heterocyclic Aromatic Compounds Useful As Growth Hormone Secretagogues |
12/30/2009 | WO2009158396A1 Diketopiperidine derivatives as hiv attachment inhibitors |
12/30/2009 | WO2009158394A1 Diketo azolopiperidines and azolopiperazines as anti-hiv agents |
12/30/2009 | WO2009156863A2 Substituted tricyclic derivatives |
12/30/2009 | EP2138498A1 Substituted tricyclic derivatives against neurodegenerative diseases |
12/30/2009 | EP2137196A1 Tricyclic nitrogen containing compounds as antibacterial agents |
12/30/2009 | EP1562949B1 Methods for the preparation of pyrrolotriazine compounds useful as kinase inhibitors |
12/30/2009 | CA2728728A1 Substituted tricyclic derivatives |
12/29/2009 | CA2563761C Inhibitors of the hiv integrase enzyme |
12/23/2009 | WO2009155017A2 Novel substituted azabenzoxazoles |
12/23/2009 | WO2009154132A1 Spirodiamine-diarylketoxime derivative |
12/23/2009 | WO2009153025A1 Process for the preparation of bisindole alkaloid derivatives |
12/23/2009 | WO2009152712A1 Vinflunine salts, preparation process and pharmaceutical composition thereof |
12/23/2009 | EP2135872A1 Process for the preparation of bisindole alkaloid derivatives |
12/23/2009 | EP2134343A2 Pyrrolo-pyridine kinase modulators |
12/23/2009 | EP2134342A2 Monocyclic anilide spirolactam cgrp receptor antagonists |
12/23/2009 | EP1879901B1 Pyrrolobenzodiazepines |
12/23/2009 | CN101611041A Fused heterocyclic compound |
12/23/2009 | CN101607968A Vinflunine salt, preparation method and pharmaceutical composition thereof |
12/23/2009 | CN101607958A Quinazoline compounds |
12/23/2009 | CA2727914A1 Spirodiamine-diaryl ketoxime derivative technical field |
12/23/2009 | CA2725940A1 Novel substituted azabenzoxazoles |
12/23/2009 | CA2724449A1 5-ht3 receptor modulators, methods of making, and use thereof |
12/17/2009 | WO2009152200A1 Tricyclic indole derivatives and methods of use thereof |
12/17/2009 | WO2009152072A1 Pyrrolo [2, 3-c] pyridine derivatives as p38 kinase inhibiting agents |
12/17/2009 | WO2009150230A1 2,4'-bipyridinyl compounds as protein kinase d inhibitors useful for the treatment of ia heart failure and cancer |
12/17/2009 | US20090312334 Immunomodulating Heterocyclic Compounds |
12/17/2009 | CA2727680A1 2,4'-bipyridinyl compounds as protein kinase d inhibitors useful for the treatment of ia heart failure and cancer |
12/17/2009 | CA2727620A1 Tricyclic indole derivatives and methods of use thereof |
12/17/2009 | CA2727315A1 Pyrrolo [2, 3-c] pyridine derivatives as p38 kinase inhibiting agents |
12/16/2009 | CN100569772C Azaindoles useful as inhibitors of JAK and other protein kinases |
12/10/2009 | WO2009148062A1 Polycyclic compound and organic electroluminescent device using the same |
12/09/2009 | CN100567293C N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists |
12/08/2009 | US7629338 for treating migraine, headaches; N-[(4S)-3-Methyl-2,5-dioxo-1',3'-dihydrospiro[imidazolidine-4,2'-inden]-5'-yl]-2-((6+-)-2-oxo-6-phenylpiperidin-1-yl)acetamide |
12/08/2009 | CA2361525C Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands |
12/03/2009 | WO2009091856A3 Beta-lactamase inhibitors |
12/03/2009 | WO2009077741A3 3-substituted-4-0x0-3, 4-dihydro-imidazo- [5, 1-d] [1,2,3,5] -tetrazine-8-carboxylic acid amides as anticancer agents |
12/03/2009 | US20090299060 Compounds and methods for inhibiting mitotic progression |
12/02/2009 | EP2128163A1 Spiro-ring compound |
12/02/2009 | EP2124560A1 2-aminopyrimidine modulators of the histamine h4 receptor |
12/02/2009 | EP1633759B1 Cross-linked glycopeptide-cephalosporin antibiotics |
12/02/2009 | CN101595110A 7-substituted purine derivatives for immunosuppression |
12/02/2009 | CN101591348A Tetrahydrochysene carboline acyl aminoacid benzyl ester, preparation method and application thereof |
12/01/2009 | US7626032 4-Amino-3,3-dimethylpiperidine; reduced toxicity, and improved pharmacology and pharmacokinetics |
12/01/2009 | US7625901 for treating migraine, headaches; 2-[(8S)-8-(3,5-Difluorophenyl)-6-oxo-7-azaspiro[4.5]dec-7-yl]-N-(2'-oxo-1',2',5,7-tetrahydrospiro[cyclopenta[b]pyridine-6,3'-pyrrolo[2,3-b]pyridin]-2-yl)acetamide |
12/01/2009 | US7625892 Pharmaceutical compositions for the treatment of diseases related to neurotrophines |
11/26/2009 | WO2009141288A2 Switchable special effect substances |
11/26/2009 | CA2724842A1 Imidazo[1,2-a]pyridine compounds |
11/25/2009 | EP2123654A1 Pyrazolopyrimidine compound |
11/25/2009 | EP2120951A1 Inhibitors of akt activity |
11/25/2009 | EP2120929A1 Use of inhibitors of the degradation of p27, in particular argyrin and derivatives thereof, for the treatment of proliferative diseases |
11/24/2009 | US7622481 Gramnegative and Grampositive bacterial infections; substituted Piperidine derivatives specially optionally substituted pyrido [3,2, -b][1,4] thiazin-yl; 6-({(3R,4S)-3-Fluoro-1-[(R)-2-hydroxy-2-(2-methoxy-quinolin-8-yl)-ethyl]-piperidin-4-ylamino }-methyl)-4H-pyrido[3,2-b][1,4]thiazin-3-one; nontoxic |
11/24/2009 | US7622476 1-allyl-( 5R,8S,10R)-terguride; antagonistic properties to 5-HT2 receptors for the prevention of migraine-related headache, Parkinson's disease, disorders of the thrombocyte function |
11/19/2009 | WO2009140101A2 Imidazopyridine compounds useful as mmp-13 inhibitors |
11/19/2009 | CA2722056A1 Hcv protease inhibitors |
11/18/2009 | EP2119720A1 Novel vinblastine derivatives, their preparation, use and pharmaceutical compositions comprising the said derivatives |
11/18/2009 | EP2118110A1 Cyclopropyl fused indolobenzazepine hcv inhibitors |
11/18/2009 | CN101583622A Inhibitors for disrupting the interaction of ubiquitination related enzymes and uses thereof |
11/18/2009 | CN101580535A Hcv protease inhibitors |
11/18/2009 | CN100560585C New benzimidazole derivative |
11/17/2009 | US7618959 6-({2-[4-(6-Methoxy-[1,5]naphthyridin-4-yl)phenyl]ethylamino}methyl)-4H-pyrido[3,2-b][1,4]thiazin-3-one;bacterial infections; antibiotic resistance; Staphylococcus aureus, Streptococcus pneumoniae and pyogenes, Enterococcus; Haemophilus influenzae, Moraxella catarrhalis, E-coli |
11/17/2009 | CA2521950C Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |
11/17/2009 | CA2407094C Diazabicyclic central nervous system active agents |
11/17/2009 | CA2393809C Heterocyclic dihydropyrimidines as potassium channel inhibitors |
11/12/2009 | WO2009136596A1 Organic electroluminescent element |
11/12/2009 | WO2009135927A1 Substituted n-phenyl-2,3-dihydroimidazo[2,1-b]thiazole-5-sulfonamide derivatives as 5-ht6 ligands |
11/12/2009 | WO2009135925A1 Substituted n-imidazo[2,1-b]thiazole-5-sulfonamide derivatives as 5-ht6 ligands |
11/12/2009 | WO2009135885A1 Fused pyrazine compounds useful for the treatment of degenerative and inflammatory diseases |
11/12/2009 | US20090280192 Method for treating or preventing alzheimer's disease |
11/12/2009 | CA2723745A1 Fused pyrazine compounds useful for the treatment of degenerative and inflammatory diseases |
11/11/2009 | EP2116547A1 Substituted N-imidazo(2, 1-b) thiazole-5-sulfonamide derivatives as 5-TH6 ligands |
11/11/2009 | EP2116546A1 Substituted N-phenyl-2,3-dihydroimidazo[2,1-b]thiazole-5-sulfonamide derivatives as 5-HT6 ligands |
11/11/2009 | EP2116538A1 Condensed tetrahydroquinoline derivative and use thereof for medical purposes |
11/11/2009 | EP1313734B1 Aza heterocyclic derivatives and their therapeutic use |
11/11/2009 | CN100558728C Calcitonin gene related peptide receptor antagonists |
11/10/2009 | US7615639 8-Methoxy-5-methyl-1-(6-methyl-pyridin-3-yl)-2-oxo-2,5-dihydro-1H-pyrido[3,2-b]indole-3-carbonitrile, for treating HIV, viral infection; effective treating mutant HIV viruses which has drug resistance against currently available reverse transcriptase inhibitors |
11/10/2009 | CA2481482C Tropane derivatives as ccr5 modulators |
11/05/2009 | WO2009134726A1 Substituted pyrimidine derivatives as histamine h4 receptor ligands |
11/05/2009 | WO2009104147A3 Azatricyclic antibiotic compounds |
11/04/2009 | EP1481077B1 Mitotic kinesin inhibitors |
11/04/2009 | EP1432700B1 Spiro-hydantoin compounds useful as anti-inflammatory agents |
11/04/2009 | CN101573365A Compounds useful as protein kinase inhibitors |
11/03/2009 | US7612094 Tri-substituted heteroaryls and methods of making and using the same |
11/03/2009 | US7612075 Anticaogulants; cardiovascular disorders |