Patents
Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041)
03/2012
03/15/2012US20120064181 P2X3 Receptor Antagonists for Treatment of Pain
03/15/2012CA2810696A1 Pyrazoloquinoline compound
03/15/2012CA2810659A1 Quinoxaline compound
03/14/2012EP1474420B1 Quinazoline compounds
03/14/2012CN102372731A Preparation method for vinblastine
03/14/2012CN102372730A Bridged ring substituted phosphodiesterase inhibitor
03/14/2012CN102372717A Pyrrolopyrimidine compound and use thereof
03/14/2012CN102372712A Imidazodiazanaphthalene PI3K (phosphatidyl inositol 3 kinase) and mTOR (mammalian target of rapamycin) dual inhibitor
03/14/2012CN102372711A Imidazo quinoline PI3K and mTOR (mammalian target of rapamycin) dual inhibitor
03/13/2012US8133992 Azepinoindole and pyridoindole derivatives as pharmaceutical agents
03/08/2012WO2012028331A1 Substituted tetrahydropyrrolopyrazine derivatives
03/08/2012DE102010040233A1 Bicyclische Aza-Heterocyclen und ihre Verwendung Aza-bicyclic heterocycles and their use
03/08/2012CA2810071A1 Substituted tetrahydropyrrolopyrazine derivatives
03/06/2012US8129386 Fused azole-pyrimidine derivatives
03/01/2012WO2012025186A1 Triazolopyrazine derivatives
03/01/2012CA2809331A1 Triazolopyrazine derivatives
02/2012
02/29/2012EP1532153B1 Azepinoindole and pyridoindole derivatives as pharmaceutical agents
02/29/2012CN102365280A New adenosine receptor ligands and uses thereof
02/29/2012CN102363622A Compound and preparation method and use thereof
02/29/2012CN101723960B Benzopyran zofuran compound as well as preparation method and application thereof
02/29/2012CN101346380B Pyrimidine derivatives for the treatment of abnormal cell growth
02/28/2012US8124600 5-HT3 receptor modulators, methods of making, and use thereof
02/23/2012US20120046271 2,5-Methano- and 2,5-Ethano-Tetrahydrobenzazepine Derivatives And Use Thereof To Block Reuptake Of Norepinephrine, Dopamine, and Serotonin
02/22/2012EP2420502A1 Fused pyrrolopyridine derivative
02/22/2012EP1507778B1 Anti-tumour polycyclic carboxamides
02/21/2012US8119648 Arthritis, obesity, (non-insulin dependent) diabetes calcitonin-induced osteoporosis; administering allograft transplantation; dipeptidyl peptidase-IV (DPP-IV) inhibitors
02/21/2012US8119631 Inhibitors of interleukin-1β converting enzyme
02/16/2012WO2012021907A2 Vincristine immunoassay
02/16/2012WO2012020217A1 Amino- imidazolothiadiazoles for use as protein or lipid kinase inhibitors
02/16/2012WO2012020215A1 Amino- imidazolothiadiazoles for use as protein or lipid kinase inhibitors
02/16/2012WO2012019954A1 Pyrazolopyridine compounds as pde10a inhibitors
02/16/2012US20120040989 2-hydroxyethyl-1h-quinolin-2-one derivatives and their azaisosteric analogues with antibacterial activity
02/16/2012US20120040380 Optically-detectable enzyme substrates and their method of use
02/15/2012EP2417140A1 Inhibitors of hiv replication
02/15/2012EP2417138A1 Pyrazolo [1, 5-a] pyrimidine derivatives as mtor inhibitors
02/15/2012EP2124944B1 Pyrazolo[3,4-b]pyridine derivatives as phosphodiesterase inhibitors
02/15/2012CN101899059B 含有吡咯烷并环的头孢菌素衍生物 A cephalosporin derivative and the pyrrolidine ring contains
02/09/2012WO2012018909A1 Fused heterocyclic compounds
02/09/2012WO2012017869A1 Metal complex dye, photoelectric conversion element and photoelectrochemical cell
02/09/2012US20120035178 Quinuclidine Compounds as Alpha-7 Nicotinic Acetylcholine Receptor Ligands
02/09/2012US20120035158 Xanthine Derivatives, the Preparation Thereof and Their Use as Pharmaceutical Compositions
02/09/2012US20120032158 Charge transport compositions and electronic devices made with such compositions
02/08/2012EP1706403B1 Imidazo[4,5-c]pyridine compounds and methods of antiviral treatment
02/08/2012EP1235938B1 Fluorescent quenching detection reagents and methods
02/02/2012US20120028965 Compounds useful as protein kinase inhibitors
02/01/2012CN102341399A Quinoxaline compounds
02/01/2012CN102341398A Sulfonylated tetrahydroazolopyrazines and their use as medicinal products
02/01/2012CN102336772A Preparation method of cefozopran hydrochloride intermediate
02/01/2012CN102336712A Nitrogen-containing heterocyclic ring derivatives synthesized by transition metal salt induced intermolecular cyclization and preparation method thereof
01/2012
01/31/2012CA2508233C New substituted imidazo-pyridinones and imidazo-pyridazinones, the preparation thereof and their use as pharmaceutical compositions
01/26/2012WO2012010633A1 Herbicidal isoxazolo[5,4-b]pyridines
01/26/2012CA2805354A1 Herbicidal isoxazolo[5,4-b]pyridines
01/25/2012EP2410002A1 Compound and element using same
01/25/2012EP2408304A1 Cgrp receptor antagonists
01/25/2012EP2328890B1 6 substituted 2-heterocyclylamino pyrazine compounds as chk-1 inhibitors
01/25/2012EP2215092B1 Substituted piperidino-dihydrothienopyrimidines
01/25/2012CN102329334A 6H-indole[3, 2-b]quinoxaline derivative and organic light-emitting diode thereof
01/25/2012CN102329330A Method for extracting conodurine from Ervatamia officinalis Tsiang
01/19/2012WO2012008508A1 Heterocyclic ring compound
01/19/2012US20120012819 Organic semiconductor compounds
01/19/2012CA2804970A1 Spirocyclic compounds
01/18/2012EP2310395B1 9-substituted-b-carboxy-oxadiazino-quinolone derivatives, their preparation and their application as anti-bacterials
01/18/2012EP2300485B1 Pyrrolo-[2, 3-c]-pyridine derivatives as p38 kinase inhibiting agents
01/18/2012CN102326273A Organic electroluminescent element
01/18/2012CN102321092A Triprenyl phenol compound, process for production of triprenyl phenol compound, and thrombolysis enhancer
01/17/2012CA2484640C Vitamin-mitomycin conjugates
01/12/2012WO2012006203A1 N-cyclyl-3 - (cyclylcarbonylaminomethyl) benzamide derivatives as rho kinase inhibitors
01/12/2012WO2012005342A1 Novel organic compound and organic light-emitting device including the same
01/12/2012WO2012004259A1 Ring-fused 4 -aminopyrimidines and use thereof as stimulators of soluable guanylate cyclases
01/12/2012WO2012003576A1 Imidazopyridine, imidazopyrimidine and imidazopyrazine derivatives as melanocortin-4 receptor modulators
01/12/2012WO2010135524A8 Benzoxazepines based p13k/mt0r inhibitors against proliferative diseases
01/12/2012US20120010208 6-CYCLOAMINO-3-(1H-PYRROLO[2,3-b]PYRIDIN-4-YL)IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
01/12/2012US20120010192 Fused Heterocyclic Compounds as Ion Channel Modulators
01/12/2012US20120009141 Functionalized pyrrolidines and use thereof as iap inhibitors
01/12/2012CA2804471A1 Ring-fused 4 -aminopyrimidines and use thereof as stimulators of soluable guanylate cyclases
01/12/2012CA2803448A1 Imidazopyridine, imidazopyrimidine and imidazopyrazine derivatives as melanocortin-4 receptor modulators
01/11/2012EP2404922A1 Quinoxaline compounds
01/11/2012EP2403854A1 Sulfonylated tetrahydroazolopyrazines and their use as medicinal products
01/10/2012CA2505389C Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions
01/05/2012WO2012003498A1 2 -quinolinyl- acetic acid derivatives as hiv antiviral compounds
01/05/2012WO2012003262A1 Heterocyclic compounds and their use as inhibitors of pi3k activity
01/05/2012WO2012000595A1 2,4- diaryl - substituted [1,8] naphthyridines as kinase inhibitors for use against cancer
01/05/2012US20120004201 Phosphodiestarase inhibitors
01/05/2012CA2803665A1 2,4- diaryl - substituted [1,8] naphthyridines as kinase inhibitors for use against cancer
01/05/2012CA2803259A1 Heterocyclic compounds and their use as inhibitors of pi3k activity
01/05/2012CA2802492A1 2-quinolinyl-acetic acid derivatives as hiv antiviral compounds
01/04/2012EP2403028A1 Organic electroluminescent element
01/04/2012EP2402347A1 Pharmaceutical compounds
01/04/2012EP2402334A1 Inhibitors of E1 Activating Enzymes
01/04/2012EP2401275A1 Novel bronchodilating diazaheteroaryls
01/04/2012CN1926107B Weakly basic hindered amines having carbonate skeletons, synthetic resin compositions, and coating compositions
01/04/2012CN102304141A Calixarene constructed supramolecular polymer material and preparation method thereof
01/03/2012CA2551723C Single-layer organic electroluminescent device
01/03/2012CA2445835C 6h-oxazolo[4,5-e]indole derivatives as nicotinic acetylcholine receptor ligands and/or serotonergic ligands
01/03/2012CA2397661C 2,4-disubstituted thiazolyl derivatives
12/2011
12/29/2011WO2011163527A1 Pyrrolo- pyrazine derivatives useful as inhibitors of atr kinase
12/29/2011WO2011163195A1 Fused pyrrole derivatives as pi3k inhibitors
12/29/2011WO2011161262A1 Evaporable organically semiconductive material and use thereof in an optoelectronic component
12/29/2011CA2803802A1 Pyrrolo- pyrazine derivatives useful as inhibitors of atr kinase
12/28/2011CN102300865A 二聚的吡咯并嘧啶二酮和它在呼吸性疾病中的治疗用途 Dimeric pyrrolopyrimidine dione and its therapeutic use in respiratory diseases
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