Patents
Patents for C07D 501 - Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula: , e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (7,574)
10/1995
10/03/1995US5455238 Cephalosporins
10/01/1995CA2145012A1 Protected aminothiazolylacetic acid derivatives
09/1995
09/26/1995US5453504 Bicyclic β-lactams intermediates having a new amino protecting group
09/21/1995WO1995025109A1 Cephem compound, process for producing the same, and antibacterial containing the compound
09/21/1995WO1995019974A3 Calixarene-based compounds having antibacterial, antifungal, anticancer-hiv activity
09/20/1995EP0672738A2 Adhesive composition
09/19/1995US5451675 By-product inhibition
09/12/1995CA1336977C Azetidinone intermediates to carbacephalosporins and process
09/06/1995CN1107850A Separation of cephalosporin isomers
09/06/1995CN1107839A Carbox amide
09/02/1995CA2143170A1 Adhesive composition
08/1995
08/31/1995WO1995023153A1 Quinolonylcarboxamidocephalosporin derivatives and pharmaceutical compositions containing them
08/30/1995EP0669336A1 Novel cephem derivative
08/29/1995US5446037 2-[(substituted) methylene]cephalosporin sulfones as antiinflammatory, antidegenerative and antithrombin agents
08/23/1995EP0667868A1 New cephem compounds
08/23/1995EP0110955B1 Brain-specific drug delivery
08/15/1995US5442058 Using an oxidizer and an acid anhydride
08/15/1995US5441874 Method for the acylation of the 7-amino group of the cephalosporanic ring
08/09/1995EP0665847A1 Cephem compounds, and their pharmaceutical compositions
08/09/1995CN1106411A Novel cephalosporin antibiotics and processes for preparation thereof
08/09/1995CN1106410A Bicyclic beta-lactam/paraben complexes
08/09/1995CN1106409A Process for the preparation of cephalosporins
08/08/1995US5439904 2-spiro(2'-spirocycloalkyl)cyclopropyl cephalosporin sulfones as antiinflammatory and antigenerative agents
08/01/1995US5438053 Cephem compounds compositions and method
08/01/1995US5438052 Cephalosporin derivatives
07/1995
07/27/1995WO1995019974A2 Calixarene-based compounds having antibacterial, antifungal, anticancer-hiv activity
07/19/1995EP0662973A1 Novel cephalosporin derivatives and processes for the preparation thereof
07/19/1995CN1105365A Cephalosporin derivatives
07/18/1995US5434259 Process for isolation of cefaclor after enzymatic acylation
07/05/1995EP0661286A1 Novel cephalosporin antibiotics and processes for the reparation thereof
06/1995
06/28/1995EP0659742A1 An improved method for the preparation of 2-chloro sulfinyl azetidin-4-one
06/21/1995EP0658558A1 Separation of cephalosporin isomers
06/21/1995EP0658533A1 Process for the oxidation of primary and secondary alcohols to aldehydes and ketones and for the oxidation of 1,2-diols to alpha-ketols and alpha-diketones
06/15/1995WO1995015966A1 2-spiro(2'-spirocycloalkyl)cyclopropyl cephalosporin sulfones as antiinflammatory and antidegenerative agents
06/15/1995CA2178492A1 2-spiro(2'-spirocycloalkyl)cyclopropyl cephalosporin sulfones as antiinflammatory and antidegenerative agents
06/13/1995US5424203 Method for selectively deactivating catalase while retaining D-amino acid oxidase activity with a solution having a pH of about 11 to 12
06/13/1995US5424196 Enzymatic process for preparing 7-aminocephalosporanic acid and derivatives
06/07/1995CN1103403A Process for preparing cefalexin
05/1995
05/30/1995US5420269 3-fluorosulfonyloxyceph-3-em compounds
05/18/1995WO1995013281A1 Process for producing 3-substituted cephem compound
05/16/1995US5416081 Cephalosporin compounds
05/16/1995US5416080 Cephalosporins
05/10/1995EP0652220A1 Cephalosporin derivative
05/10/1995EP0651756A1 Tricyclic defem sulphones as elastase inhibitors
05/10/1995EP0651755A1 Cephalosporins and 1-carba-1-dethia cephalosporins
05/09/1995US5414081 Treating a 1-aza-3-thiabicycloalkane with base and phosphine or phosphite desulfurizing agent, and reacting the product with an active esterifying agent
05/02/1995US5412094 Bicyclic beta-lactam/paraben complexes
05/02/1995US5412093 3-heterocyclic thiomethyl cephalosporins
04/1995
04/26/1995EP0649849A1 Process for the preparation of cephalosporins
04/26/1995EP0204781B1 Process for the production of bissilylated 3-iodomethylcephalosporine derivatives
04/26/1995CN1101912A New cephem compounds
04/25/1995US5410044 Process for preparing Z and E-rotamers of 3-hydroxy cephem derivatives
04/25/1995US5410042 Acidification with trifluoroacetic acid, methanesulfonic acid and trifluoromethanesulfonic acid
04/25/1995US5409919 Pharmaceutically acceptable salt of 7B-[2-(5-amino-1,2,4-thio-diazol-3-yl)-2(Z)-metho-xyiminoacetamido]-3-[(imidazo[1,2-b]pyridazinium-1-yl)methyl]-3-cephem-4-carboxylate and composition comprising same
04/25/1995US5409918 Crystalline cephem acid addition salts and process for their preparation
04/19/1995CN1028236C Process for preparing acyl derivatives
04/18/1995US5407930 Cephalosporin derivatives
04/18/1995US5407929 Triazolylthiomethylthio cephalosporin hydrochhloride, its crystalline hydrate and the production of the same
04/12/1995EP0647230A1 Cephalosporins and 1-carba-1-dethia cephalosporins
04/11/1995US5405955 Chlorinating thiazolidine derivative in organic solvent, reacting product with arylsulfinic acid in solvent and acid, adding azetidinone product to solvent containing base
04/06/1995WO1995009171A1 Novel cephalosporin derivative
04/04/1995US5403929 Treating zinc salt of cephalosporin c with metal halide, ion exchanging
04/04/1995US5403835 Excellent antibacterial spectrum against sensitive or tolerant Gram-positive and Gram-negative bacteria, particularly glucose non-fermentative Gram-negative rods containing Pseudomonas aeruginosa
03/1995
03/28/1995US5401842 Antibiotics
03/28/1995US5401841 3-vinyl-substituted
03/28/1995US5401734 Cephem compounds
03/28/1995CA1334934C Antibacterial composition for oral administration
03/23/1995WO1995007912A1 Novel cephem derivative
03/16/1995WO1995007283A1 New cephem compounds
03/16/1995CA2157669A1 New cephem compounds
03/15/1995EP0643061A1 Novel cephalosporin antibiotics and processes for preparation thereof
03/14/1995US5397779 Cephalosporins
03/09/1995WO1995002603A3 Use of cephem derivatives as anti-metastatic agents
03/08/1995EP0641797A1 Cephem derivatives and antimicrobial agents containing the same
03/08/1995EP0641779A1 Novel 1-amidinopiperdines and 4-amidinomorpholines as aggregation inhibitions
03/08/1995CA2130864A1 Carboxamides
03/01/1995EP0640608A1 Intermediates in the synthesis of cephalosporins
02/1995
02/28/1995US5393882 Bicyclic β-lactam antibiotics
02/22/1995EP0639195A1 2-acyloxycephem derivatives as elastase inhibitors
02/21/1995USRE34865 Antibiotics
02/21/1995US5391729 Crystalline dihydrate of a cephalosporin salt
02/21/1995US5391728 Bicyclic B-lactams intermediates having a new amino protecting group
02/21/1995CA2006144C Microbial process for the production of immunosuppressive antibiotics
02/16/1995WO1995004740A1 7α-AMINO-1,1-DIOXOCEFEM L-VALYLAMIDES
02/16/1995WO1995004739A1 3-aryl or heteroaryl-7-heteroaralkylamido cephalosporin compounds, compositions and methods of use
02/15/1995EP0638574A1 Oxime derivatives of cephalosporanic structure and compounds for their preparation
02/15/1995EP0638573A1 Crystalline hydrates of cephalosporin and process for preparation thereof
02/14/1995US5389627 Cephem compounds
02/14/1995US5389626 3-aryloxmethyl-cephalosporin derivatives, and their medical use
02/14/1995US5389625 Sweet taste; oral administering
02/14/1995CA1334407C Method for the preparation of novel alcoyloxime derivatives of 7-amino-thiazolyl-acetamido-cephalosporanic acid
02/10/1995CA2128557A1 Oxime derivatives of cephalosporanic structure and compounds for their preparation
02/08/1995EP0637587A1 Bicyclic beta-lactam/paraben complexes
02/07/1995US5387748 Antimicrobial dithiocarbamoyl quinolones
02/07/1995US5387679 Process for the preparation of cephalosporins intermediates
02/01/1995EP0636627A1 Cephem compounds and antimicrobial agents
01/1995
01/26/1995WO1995002603A2 Use of cephem derivatives as anti-metastatic agents
01/26/1995CA2167194A1 Use of cephem derivatives as anti-metastatic agents
01/25/1995EP0635509A2 Novel cephalosporin antibiotics and processes for preparation thereof
01/18/1995EP0634415A2 Cephem compound, its production and its use for producing cephem antibiotics
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