Patents
Patents for C07D 501 - Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula: , e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (7,574)
06/1997
06/05/1997WO1997013772A3 Cephalosporin antibiotics
06/04/1997CN1150950A Cephalosporin derivatives
06/03/1997US5635501 Alphalosporins and 1-carba-1-dethia cephalosporins
06/03/1997US5635500 Cephem compound and pharmaceutical composition containing the compound
05/1997
05/28/1997EP0775145A1 Process for making quinolonyl lactam antimicrobials and novel intermediate compounds
05/28/1997EP0775114A1 Process for making antimicrobial compounds
05/21/1997EP0774466A1 Novel cephem derivatives
05/21/1997EP0773928A1 2-(2-azetidinon-n-yl)-2- and 3-butenoic acids derivatives and their use in the cephalosporine synthesis
05/21/1997CN1150429A Cephalosporin compounds and processes for preparation thereof
05/21/1997CN1034940C Preparation process for new cephalosporin
05/20/1997US5631378 Protected aminothiazolylacetic acid derivatives
05/20/1997US5631367 E-rotamers of 3-hydroy cephem derivatives
05/20/1997US5631366 Process for making 3-formylcephem derivatives
05/20/1997US5631256 Antimicrobial quinolone thioureas
05/15/1997WO1997017352A1 De-esterification process
05/14/1997CN1149874A Cephalosporin antibiotics
05/13/1997US5629306 B-lactamase inhibitors
05/13/1997US5629171 Recombinant bioprocess for the preparation of 7-amino cephalosporanic acid (7-ACA)
05/07/1997EP0771803A1 Pyrazolo(1,5-a)pyrimidinium substituted cephem derivatives, their preparation and their use as antimicrobial agents
05/05/1997WO1997017353A1 Process for the preparation of 3-halogenocephem derivatives
04/1997
04/29/1997US5625058 Process for the preparation of cephalosporins
04/23/1997CN1148044A Prepn. and use of 7-[(2-carboalkoxy-1-methylethenyl) amino]-3-hydroxymethyl-3-cephem-4-cargoxylic acids
04/17/1997WO1997013772A2 Cephalosporin antibiotics
04/17/1997CA2234255A1 Cephalosporin antibiotics
04/16/1997EP0497978B1 Cephalosporin compounds and production thereof
04/16/1997CN1147516A Bioavailable crystalline form of cefuroxime axetil
04/16/1997CN1034571C A method for producing a pyrrolidire derivative
04/15/1997US5621095 Cephalosporins
04/15/1997US5621084 Process for removal of allyl group or allyloxycarbonyl group
04/15/1997US5620969 Bactericides
04/15/1997US5620968 7-substituted-amino-3-substituted-3-cephem-4-carboxylic acids
04/10/1997WO1997012890A1 New cephem compounds
04/09/1997CN1034504C Process for preparing thioalkylthio cephalosporin derivs.
04/02/1997CN1146770A Cephalosporin synthesis
04/01/1997US5616703 Separation of cephalosporin isomers
03/1997
03/26/1997EP0764648A1 Cephem derivatives and process for the preparation thereof
03/25/1997US5614623 Diastereomers of 1-(isopropoxycarbonyloxy)ethyl 3-cephem-4-carboxylate and processes for their preparation
03/25/1997CA1339021C Ó-crystals of cefazolin sodium
03/19/1997EP0763043A1 Process for the preparation of trihydrated cefixime
03/13/1997WO1997009052A1 Therapeutic azide compounds
03/13/1997CA2231442A1 Therapeutic azide compounds
03/13/1997CA2184971A1 Cephalosporin derivatives
03/12/1997EP0761673A1 Cephalosporin derivatives
03/12/1997EP0761672A1 Cephalosporin containing in position 7 a substituted benzyloxyimino radical, processes for their preparation and intermediates for their preparation, their use as medicaments
03/12/1997EP0761671A1 Cephem derivatives
03/12/1997EP0760820A1 Cephalosporin compounds and processes for the preparation thereof
03/06/1997WO1997008174A1 Interleukin converting enzyme and apoptosis
03/06/1997WO1997007805A1 Interleukin converting enzyme and apoptosis
03/05/1997EP0548186B1 Cephalosporin derivatives and their homologues
03/05/1997CN1144274A Improved enzymatic process for producing penicillins and cephalosporins
03/05/1997CN1144222A New cephem compounds
03/05/1997CN1034177C Process for preparing cefalexin
03/04/1997US5608055 Beta lactam production
03/04/1997US5607927 Cephalosporin derivative
03/04/1997US5607926 Active against methicillin resistant bacteria
02/1997
02/27/1997WO1997007121A1 Purification process
02/27/1997WO1997007112A1 Amine acid salt compounds and process for the production thereof
02/26/1997EP0759437A1 Processes for the production of 2-isocephem derivatives
02/26/1997EP0759436A1 Processes for the preparation of beta-lactam derivative
02/25/1997US5605895 Cephalosporin antibiotics and processes for preparation thereof
02/18/1997US5604222 Reacting penicillin sulfoxide ester with n-chlorohalogenating agent in inert organic solvent in presence of phosphate acid scavenger
02/18/1997US5604218 Cephalosporin antibiotics
02/18/1997US5604217 7-acyl-3-(substituted carbamoyloxy) cephem compounds and process for their preparation
02/17/1997CA2183469A1 New cephalosporins containing a substituted benzyloxyimino radical in position 7; process and intermediates for preparing them and use thereof as therapeutic agents
02/12/1997EP0757991A1 Bioavailable crystalline form of cefuroxime axetil
02/12/1997EP0757691A1 Cephalosporin synthesis
02/11/1997US5602117 Cephalosporin compounds
02/06/1997WO1997003990A1 Isomer separation
02/05/1997CN1141923A Process for selective sulfoxide reduction of 3-hydroxy cephem and 3-methylene cepham sulfoxide compounds
02/05/1997CN1141922A Cephalosporin derivative
02/04/1997CA2179359A1 Bioavailable crystalline form of cefuroxime azetil
01/1997
01/28/1997US5597914 Process for the production of cephalosporins
01/28/1997US5597817 7-vinylidene cephalosporins and methods of using the same
01/23/1997WO1997002268A1 7,7-disubstituted cephem-4-ketones
01/23/1997WO1997002024A1 Use of stat 5 sh2 domain specific compounds to enhance erythropoiesis
01/23/1997CA2225666A1 Use of stat 5 sh2 domain specific compounds to enhance erythropoiesis
01/22/1997EP0754184A1 Cephalosporin antibiotics
01/22/1997CN1140714A Preparation of cephalosporin antibiotic using syn-isomer of thiazolyl intermediate
01/21/1997US5596096 Azetidinone derivatives and method for producing azetidinone and cephalosoporin derivatives
01/21/1997US5596095 Removal of neopentyl protecting groups and regeneration of parent drugs
01/21/1997US5595986 Stably storable and readily water soluble composition of cephalosporin for injections
01/15/1997CN1140175A 7-acyl-3-(substd. carbamoyloxy) cephem compounds and their preparation process
01/14/1997US5594133 Crystalline acid addition salts of diastereomerically pure 1-(2,2-dimethylpropinonyloxy)-ethyl-3-cephem-4-carboxylate
01/14/1997US5594132 7-acylamino-3-substituted cephalosporanic acid derivatives
01/14/1997US5594131 Process for preparing cephalosporin intermediates
01/14/1997US5594130 N-acylation of 7-amino-3-((1-methyl-1-pyrrolidinio)-methyl) ceph-3-em-4-carboxylate with syn-2-(2-aminothiazol-4-yl)-2-methoxyimino acetyl chloride hydrochloride
01/14/1997US5594129 Process for the preparation of a cephalosporin antibiotic
01/14/1997US5593986 Cephalosporin antibiotics
01/14/1997US5593985 Cephalosporin compounds
01/14/1997US5593984 Cephalosporin derivatives
01/14/1997CA1338842C Cephem compound and a process for preparation thereof
01/09/1997WO1996030540A3 Substrates for beta-lactamase and uses thereof
01/09/1997DE19626616A1 Verfahren zur Herstellung von 1,1-Dioxo-cephem-4-ketonen A process for the preparation of 1,1-dioxo-cephem-4-ketones
12/1996
12/31/1996US5589594 Process for the preparation of cephem prodrug esters
12/31/1996US5589593 Crystalline form of a cephalosporin antibiotic
12/31/1996US5589592 Process for preparing β-lactam derivative and synthetic intermediate
12/31/1996CA1338820C Intermediates useful for preparing cephem compounds and process for preparing same
12/24/1996US5587474 Method for removing the protecting group for carboxyl group
12/24/1996US5587473 Blocking; condensation; deblocking
12/24/1996US5587373 Elastase inhibitors
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