Patents
Patents for C07D 501 - Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula: , e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (7,574)
07/1996
07/02/1996US5532354 Antibiotics
07/02/1996US5532353 Antibiotics and bactericides
06/1996
06/25/1996US5530116 Antimicrobial quinolonyl lactams
06/20/1996WO1996018609A1 Formation and utility of sulfonic acid protecting groups
06/19/1996EP0716852A1 Pharmaceutical formulations of cefaclor
06/19/1996CN1124737A Method for production of t-butyl 3-oxobutyrates and their use
06/18/1996US5527906 Acylation in solution of sodium bicarbonate in aqueous acetone with 2-/2-aminothiazol-4-yl/-2-syn-methoxyimino acetic acid-2-benzothiazolyl thioester
06/18/1996US5527792 7-substituted-amino-3-substituted-3-cephem-4-carboxylic acids
06/18/1996US5527697 An esterase prepared by cultivation of microorganism of streptomyces, amycolatopsis or nocardia
06/14/1996CA2158511A1 Pharmaceutical formulations of cefaclor
06/13/1996WO1996017850A1 Cephem compounds and pharmaceutical use thereof
06/13/1996WO1996017849A1 7-alkylidene cephalosporanic acid derivatives and methods of using the same
06/13/1996WO1996017848A1 7-vinylidene cephalosporins and methods of using the same
06/13/1996WO1996017847A1 Process for the preparation of cephalosporins and analogues
06/13/1996WO1996017846A1 Process for the preparation of intermediates useful in the synthesis of cephalosporins
06/13/1996CA2206226A1 Process for the preparation of intermediates useful in the synthesis of cephalosporins
06/11/1996US5525599 7-substituted-amino-3-substituted-3-cephem-4-carboxylic acids
06/11/1996US5525483 By enzymatic reaction with parent amino beta-lactam
06/04/1996US5523400 3-(pyrrolidin-3-ylidene=ch-),7-((2-aminothiazol-4-yl)hydrox -iminoacetylamino-)-3-cephem derivatives; broad spectrum antibiotics
05/1996
05/30/1996WO1996016067A1 Silylation process
05/29/1996EP0233255B1 Conversion of cephalosporin hydrohalide salt to alkali metal salt
05/29/1996CN1123549A Crystalline benzathine salt of cefonicid and its preparation
05/29/1996CN1123274A Process for producing N-allyl-2,5-dimethyl-piperidinol-4-benzoyl ester
05/28/1996US5521308 Process for the preparation of crystalline TACA
05/15/1996EP0711774A1 Crystalline cephem-addition salts and process for their preparation
05/14/1996US5516902 Process for preparing cephalosporin compounds
05/07/1996US5514561 Fluorogenic and chromogenic β-lactamase substrates
05/07/1996US5514383 Process for the preparation of tablets of derivatives of cephalosporanic acid by direct compression
05/02/1996WO1996012712A1 Reactive phosphate derivatives of thiazolylacetic acid and process for preparing cephalosporin antibiotics using the same
05/01/1996EP0708779A1 Use of cephem derivatives as anti-metastatic agents
04/1996
04/23/1996US5510538 Process for the oxidation of primary and secondary alcohols to aldehydes and ketones and for the oxidation of 1,2-diols to α-ketols and α-diketones
04/17/1996CN1031571C Deprotection of allylic esters and ethers
04/11/1996DE4435478A1 New quinoline and naphthyridone carboxylic acid derivs.
04/10/1996EP0682669A4 Improved process for isolation of cefaclor after enzymatic acylation.
04/10/1996CN1120045A New cephalosporins containing in position 7 a substituted benzyloxyimino radical, their preparation process, their use as medicaments
04/03/1996CN1119531A A stably storable and readily water soluble composition of cephalosporin for injections
04/02/1996US5504076 Antibiotics
03/1996
03/27/1996CN1119439A Improved process for isolation of cefaclor after enzymatic acylation
03/20/1996CN1119016A Crystalline ceftiofur free acid
03/14/1996WO1996007659A1 Novel crystal of cephalosporin compound
03/14/1996CA2199253A1 Novel crystal of cephalosporin compound
03/13/1996EP0700916A1 Cephem compound, process for producing the same, and antibacterial containing the compound
03/13/1996CN1118349A Oxime derivatives of cephalosporanic structure and compounds for their preparation
03/12/1996US5498787 Esterification of cephalosporin salts, quaternary ammonium or phosphonium catalyst
03/12/1996US5498777 3-thioheteroaryl cephalosporin compounds, compositions and methods of use
03/06/1996EP0699681A1 Cephalosporin derivatives
03/03/1996CA2155705A1 Cephalosporin derivatives
02/1996
02/28/1996CN1117383A Cefixime composition
02/22/1996WO1996005205A1 Novel cephem derivative
02/22/1996DE19530124A1 Verfahren zur Herstellung von N-Allyl-2,5-dimethyl-piperidinol-4- benzoylester A process for the preparation of N-allyl-2,5-dimethyl-4-benzoyl-piperidinol
02/15/1996WO1996004286A1 Process for making quinolonyl lactam antimicrobials and novel intermediate compounds
02/15/1996WO1996004247A1 Process for making antimicrobial compounds
02/08/1996WO1996003373A1 2-(2-azetidinon-n-yl)-2- and 3-butenoic acids derivatives and their use in the cephalosporine synthesis
02/07/1996EP0695548A1 A stably storable and readily water soluble composition of cephalosporin for injections
02/07/1996CN1116425A New cephem compounds
02/04/1996CA2155170A1 Stably storable and readily water soluble composition of cephalosporin for injections
02/01/1996WO1996002548A1 3-thioheteroaryl cephalosporin compounds, compositions and methods of use
02/01/1996WO1995035020A3 Glutaryl 7-aca derivatives and processes for obtaining them
01/1996
01/25/1996DE19526187A1 7-Diazo-beta-lactamderivate und Verfahren zu deren Herstellung 7-diazo-beta-lactam derivatives and process for their preparation
01/24/1996EP0693496A1 Novel cephalosporins having a substituted benzyloxyimino radical in position 7, process for their preparation and their use as medicaments
01/20/1996CA2154227A1 Cephalosporins with a substituted benzyloxyimino radical in position 7, process for their preparation and their application as medecines
01/16/1996US5484928 2-(2-aminothiazol-4-yl)-2-oxoacetic acid derivatives
01/10/1996EP0691343A1 Cephalosporin derivative
01/10/1996EP0690865A1 Crystalline benzathine salt of cefonicid and its preparation
01/10/1996EP0690864A1 Crystalline ceftiofur free acid
01/10/1996CN1030657C Method for preparing autibacterial compounds
01/03/1996CN1114507A Novel Cephem Derivative
01/03/1996CN1114315A Protected aminothiazolylacetic acid derivatives
01/02/1996US5480879 Quinolonecarboxylic acids
01/02/1996US5480720 Adhesive composition
12/1995
12/28/1995WO1995035020A2 Glutaryl 7-aca derivatives and processes for obtaining them
12/21/1995WO1995034567A1 Cyclohexanocephalosporins and their preparation procedure
12/20/1995EP0687676A1 Purification of a cephalosporin salt
12/14/1995WO1995033753A1 Process for the preparation of trihydrated cefixime
12/13/1995CN1113233A A method for producing a pyrrolidire derivative
12/06/1995EP0685232A2 Cefixim formulation
12/01/1995CA2150442A1 Cefixime composition
11/1995
11/30/1995WO1995032210A1 Cephalosporin compounds and processes for the preparation thereof
11/30/1995CA2190245A1 Cephalosporin compounds and processes for the preparation thereof
11/28/1995US5470972 Antibiotics
11/28/1995US5470717 Method for the preparation of certain β-lactam antibiotics
11/22/1995EP0682669A1 Improved process for isolation of cefaclor after enzymatic acylation
11/15/1995CN1111633A Process for preparing cephalosporin compounds from reactive organic acid derivatives
11/08/1995CN1111246A Novel cephalopsporin antibiotics and processes for the preparation thereof
11/07/1995US5464829 Cephalosporin derivatives
11/07/1995CA1337522C Syn-isomer of 3,7-disubstituted-3-cephem-4-carboxylic acid compounds and processes for the preparation thereof
11/02/1995WO1995029182A1 Cephalosporin synthesis
11/02/1995CA2533837A1 Cephalosporin synthesis
10/1995
10/31/1995US5462935 Antibiotic
10/25/1995EP0678520A1 Process for producing 3-substituted cephem compound
10/24/1995US5461044 Cephalosporin derivatives
10/24/1995US5461043 Diastereomers of 1-(isopropoxycarbonyloxy)ethyl 3-cephem-4-carboxylate
10/18/1995EP0677523A1 3-(substituted)-1-carba(dethia)-3-cephems and cephalosporins and a process for production therefor
10/12/1995WO1995026966A1 Cephalosporin antibiotics
10/12/1995CA2186894A1 Cephalosporin antibiotics
10/11/1995EP0676236A1 Process for removal of allyl group or allyloxycarbonyl group
10/11/1995CN1110057A Tricyclic defem sulphones as elastase inhibitors
10/11/1995CN1029965C Process and intermediates for beta-lactams having aminothiazole (iminoxyacetic acid) acetic acid sidechains
10/04/1995EP0675116A1 Protected aminothiazolylacetic acid derivatives
10/03/1995US5455239 3-aryl of heteroaryl-7-heteroaralkylamido cephalosporin compounds, compositions and methods of use
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