Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
04/1995
04/25/1995US5409921 Renin inhibitors
04/25/1995US5409919 Pharmaceutically acceptable salt of 7B-[2-(5-amino-1,2,4-thio-diazol-3-yl)-2(Z)-metho-xyiminoacetamido]-3-[(imidazo[1,2-b]pyridazinium-1-yl)methyl]-3-cephem-4-carboxylate and composition comprising same
04/25/1995US5409913 Oxazocinyl/thiazocinyl terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
04/25/1995CA1335377C Photochromic compound and photochromic composition
04/22/1995CA2133169A1 Cation-sensing composite structure and compounds for use therein
04/19/1995EP0648209A1 Contrast agents for mr diagnosis
04/19/1995CN1028235C Pyranobenzoxadiazole derivatives
04/18/1995US5407943 Azaspiro quinolone antibacterial agents
04/18/1995US5407938 Certain 1-methyl-piperidine-4-spiro-4'-(1'-3'-oxazolines) and corresponding -(1',3' thiazolines)
04/18/1995US5407932 Bactericides
04/15/1995CA2101623A1 A method for making 2-¬18f|fluoro-2-deoxy-d-glucose
04/13/1995WO1995009857A1 O-aryl, o-alkyl, o-alkenyl and o-alkynyl-macrolides having immunosuppressive activity
04/13/1995CA2172124A1 O-aryl, o-alkyl, o-alkenyl and o-alkynyl-macrolides having immunosuppressive activity
04/12/1995EP0647644A1 Antibacterial pyrido 1,2,3-d,e 1,3,4 benzoxacin derivatives
04/12/1995EP0647641A1 Substituted heterocyclylisoquinolinium salts and compositions and methods of usethereof
04/12/1995CN1028143C Fungicidal oxazolidinones
04/11/1995US5405958 Photochromic spiro(indoline)naphthoxazine compounds
04/11/1995US5405956 Cyclic oligomers for production of linear polyketones, polyphthalazines and polyisoquinolines
04/11/1995US5405829 Substituted pyrazolypyrazoles and their use as herbicides
04/06/1995WO1995009175A1 Ring-expanded nucleosides and nucleotides
04/06/1995DE4333697A1 Process for the preparation of 3-aminopyridines from 3-nitropyridines
04/05/1995EP0646583A1 Derivatives of Imidezol-4-yl piperidine, their preparation and use in therapy
04/05/1995EP0646115A1 Heterocyclic-cyclic amine derivatives
04/05/1995CN1101047A Intermediates useful in the preparation of pyranyl cyanoguanidine derivatives and methods of preparing same
04/05/1995CA2133491A1 Imidazol-4-ylpiperidine derivatives, their preparation and their application in therapeutics
04/04/1995US5403839 Pyrrolophenothiazine carboxamides
04/04/1995US5403833 Methods of inhibiting transplant rejecton in mammals using rapamycin and derivatives and prodrugs thereof
04/04/1995US5403572 Diagnosis/medical/
04/03/1995CA2133373A1 Method for preparing 3-aminopyridines from 3 nitropyridines
03/1995
03/31/1995CA2133180A1 Rapamycin formulation for iv injection
03/29/1995EP0645391A2 Aminobenzoic acid derivatives
03/29/1995EP0645378A1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors
03/29/1995EP0645377A1 Benzoxazepine derivatives useful as squalene synthetase inhibitors
03/29/1995EP0346427B1 Macrocyclic compounds
03/28/1995US5401741 Cream with ofloxacin for inflammation of ears
03/28/1995US5401737 Cholecystokinin antagonists
03/25/1995WO1999013871A2 Fused imidazole derivatives for improving oral bioavailability of pharmaceutical agents
03/25/1995CA2132794A1 Condensed 7-membered cyclic compounds and their use
03/25/1995CA2132792A1 Condensed cyclic compounds and their use
03/23/1995WO1995007918A2 Pyrimidine derivatives for labeled binding partners
03/23/1995WO1995007911A1 K-252a DERIVATIVES WHICH ENHANCE NEUROTROPHIN-INDUCED ACTIVITY
03/22/1995EP0643966A1 Sensitivity enhancer for antineoplasic agent
03/22/1995EP0643700A1 New substituted pyrazolylpyrazoles, processes for their preparation, as well as intermediates, and their use as herbicides.
03/21/1995US5399687 For coating plastic lenses, less migration, better adhesion
03/21/1995CA1334850C Ureylene-2,4,6-pyrimidine-3-oxide derivatives, their preparation and use in cosmetics and dermopharmacy
03/21/1995CA1334847C Oxadiazolopyrimidones, their preparation and application in cosmetics and dermopharmacy
03/16/1995WO1995007269A1 Polar-substituted hydrocarbons
03/16/1995CA2171471A1 Polar-substituted hydrocarbons
03/15/1995EP0642516A1 Macrocyclic immunomodulators
03/15/1995CN1100095A Preparation of a sprio compound
03/15/1995CA2131967A1 Substituted heterocyclylisoquinolinium salts and compositions and method of use thereof
03/14/1995US5397791 Fibrinogen receptor antagonists
03/14/1995CA1334751C Ureylene-2,4,6-pyrimidine-3-oxide derivatives, their preparation and use in cosmetics and dermopharmacy
03/09/1995WO1995006649A1 Macrolides as antagonists of macrophilin binding immunosuppressants
03/08/1995EP0641343A1 4-mercaptoacetylamino- 2] benzazepinone(3) derivatives, and use as enkephalinase inhibitors
03/08/1995EP0641339A1 Azaspiro quinolone antibacterial agents
03/08/1995EP0641331A1 Chiral intermediates for the preparation of antidiabetics thiazoles
03/08/1995CN1099756A Tetrahydropyran derivatives
03/07/1995US5395834 New benzopyran compounds
03/02/1995WO1995003303A3 Aza spiro compounds acting on the cholinergic system with muscarinic agonist activity
03/01/1995EP0640592A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists
03/01/1995EP0640087A1 Use of tricyclic pyrimidine derivatives as anti-viral medicaments
03/01/1995CN1099392A Compounds containing a fused bicyclic ring and processes therefor
03/01/1995CN1099390A Process for the preparation of intermediates useful in the preparation of pyranyl cyanoguandine derivatives
02/1995
02/28/1995US5393775 Benzopyran compounds
02/28/1995US5393758 Substituted azetidinylpyridone naphthyridine carboxylic acid derivatives and their application as medical products
02/28/1995US5393752 Psycholigical disorders
02/23/1995WO1995005385A1 Spiro(indolino) oxazine photochromic compounds
02/23/1995CA2168475A1 Spiro(indolino) oxazine photochromic compounds
02/22/1995EP0639575A1 Bicyclic heterocycles, medicaments comprising these compounds and processes for their production
02/22/1995EP0639237A1 Dyes, their preparation and use in the coloration of substrates.
02/21/1995US5391763 3-aza-bicyclo[3.1.0]hexanes which are intermediates for anti-bacterial azabicyclo quinolone carboxylic acids
02/21/1995US5391730 Phosphorylcarbamates of rapamycin and oxime derivatives thereof
02/16/1995WO1995004741A1 Aza-5,5-fused heterocyclic acids as leukotriene antagonists
02/16/1995WO1995004738A1 C-22 ring stabilized rapamycin derivatives
02/16/1995WO1995004737A1 Condensed indole derivatives as 5-ht4-receptor antagonists
02/16/1995WO1995004735A1 Matrix metalloprotease inhibitors
02/16/1995WO1995004734A1 Hydroisoquinoline derivatives
02/16/1995WO1995004531A1 Fibrinogen receptor antagonists
02/16/1995CA2169277A1 C-22 ring stabilized rapamycin derivatives
02/16/1995CA2168853A1 Hydroisoquinoline derivatives
02/16/1995CA2168791A1 Matrix metalloprotease inhibitors
02/16/1995CA2168750A1 Condensed indole derivatives as 5-ht4-receptor antagonists
02/16/1995CA2168668A1 Aza-5,5-fused heterocyclic acids as leukotriene antagonists
02/16/1995CA2168581A1 Fibrinogen receptor antagonists
02/15/1995EP0638597A1 Polymeric adults of hindered amine-epoxydes as stabilizers
02/15/1995EP0638560A1 Remedy for osteoporosis and diazepine compound
02/15/1995EP0638082A1 Macrocyclic immunomodulators
02/14/1995US5389660 Substituted imidazo-fused 5-membered ring heterocycles as angiotensin II antagonists
02/14/1995US5389653 Inhibitors of the enzyme catechol-O-methyltransferase; useful as co-medication in treatment of Parkinson's disease
02/14/1995US5389639 Amino alkanoic esters of rapamycin
02/14/1995US5388815 Embossed card package production system with modular inserters for multiple forms
02/14/1995CA1334413C Amino-substituted bridged azabicyclic quinolone carboxylic acids and esters
02/14/1995CA1334392C Immunosuppressant agent
02/14/1995CA1334391C Immunosuppressant compound
02/09/1995WO1995004062A1 Synthesis of 4,10-dinitro-2,6,8,12-tetraoxa-4,10-diazatetracyclo[5.5.0.0?5,903,11¿]dodecane
02/09/1995WO1995004061A1 Activated macrolactams having immunomodulatory activities
02/09/1995WO1995004060A1 Rapamycin derivative with antimicrobial, anticancer and immunomodulation activity
02/09/1995WO1995004057A1 TRICYCLIC INHIBITORS OF THE GPIIbIIIa RECEPTOR
02/09/1995CA2166892A1 Activated macrolactams having immunomodulatory activities