Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
11/1995
11/21/1995US5468742 Antibacterial agents, feed additives
11/21/1995CA2149854A1 Substituted furoxanes
11/15/1995EP0682030A1 8-Amino-10(azabicycloalkyl)-pyrido[1,2,3-d,e] [1,3,4] benzoxadiazine derivatives, process for their preparation and antibacterial agents containing them
11/15/1995EP0682029A1 Process for producing bicozamycin benzoate
11/15/1995EP0682027A1 Pyrrolopyrimidine derivatives with antiproliferative action
11/15/1995EP0681584A1 Condensed heterocyclic glutamic acid derivatives as antiproliferative agents
11/15/1995CN1111632A Imidazodiazepine
11/14/1995US5466689 Morpholine derivatives and their use
11/12/1995CA2148866A1 8-amino-10-(azabicycloalkyl)-pyrido[1,2,3-d,e][1,3,4] benzoxadiazine derivatives
11/12/1995CA2148865A1 8-amino-pyrido(1,2,3-d,e)(1,3,4)benzoxadiazine derivatives
11/09/1995WO1995029894A1 Novel quinolone 5-(n-heterosubstituted amino) antimicrobials
11/09/1995CA2188918A1 Novel quinolone 5-(n-heterosubstituted amino) antimicrobials
11/08/1995EP0681005A1 Triphendioxazine reactive dyes
11/08/1995CN1111247A Protein kinase C inhibitors
11/07/1995US5464842 Azabicyclo oxime and amine cholinergic agents and methods of treatment
11/07/1995US5464841 Use of delta opioid receptor antagonists to treat immunoregulatory disorders
11/07/1995US5464796 7-isoindolinyl-quinolone-carboxylic acid derivatives
11/07/1995US5464617 1H-2,6a-diazacyclobut(cd)indene-6-carboxylic acid derivatives, antibiotics
11/07/1995CA1337523C Pyridonecarboxylic acids and antibacterial agents
11/04/1995CA2148324A1 Pyrrolopyrimidine derivatives having pharmacological activity
11/02/1995WO1995029169A2 Process for preparing 2-piperazine carboxylic acid derivatives
11/02/1995EP0679641A1 Sulfonamide and sulfonic ester derivatives each having tricyclic hetero ring
11/02/1995EP0679084A1 Hydantoin and succinimide-substituted derivatives of spiroindanylcamphorsulfonyl oxytocin antagonists
11/02/1995EP0599862B1 Moisture-scavenging iminoalcohol-oxazolidine mixtures
11/02/1995DE19515371A1 New spiro:oxazine photochromic cpds.
10/1995
10/31/1995US5463053 Optically active pyridobenzoxazine derivatives
10/31/1995US5463048 Rapamycin amidino carbamates
10/31/1995US5462938 Arthropodicidal oxadiazinyl, thiadiazinyl and triazinyl carboxanilides
10/26/1995WO1995028406A1 Rapamycin hydroxyesters, process for their preparation and pharmaceutical compositions containing them
10/26/1995WO1995028397A1 Alpha1c adrenergic receptor antagonists
10/26/1995WO1995028391A1 Cck or gastrin modulating 1,5 benzodiazepines derivatives
10/26/1995CA2187767A1 Alpha1c adrenergic receptor antagonists
10/26/1995CA2186872A1 Cck or gastrin modulating 1,5 benzodiazepines derivatives
10/25/1995EP0678506A2 Intermediates for the preparation of 1-(phenyl)-1-hydroxy-2-amino-3-fluoro propane derivatives
10/25/1995EP0358774B1 Novel spirooxazine compounds
10/25/1995CN1110685A Nitrogen-containing spirocycles
10/24/1995US5461146 Enzyme inhibitor protecting nerve cells from degeneration
10/24/1995US5461058 Methods of inhibiting transplant rejection in mammals using rapamycin and derivatives and prodrugs thereof
10/24/1995US5461048 Tricyclic compounds having cholecystokinin antagonist activity
10/24/1995CA1337419C (2-imidazolin-2-yl) fused heteropyridine compounds, intermediates for the preparation of and use of said compounds as herbicidal agents
10/19/1995WO1995027716A1 6,7-heteroannealed 2,2-diphenyl chromenes and use thereof in ophthalmic optics
10/18/1995EP0677519A1 Chroman derivative and medicinal use thereof
10/18/1995EP0677516A1 Cyclic amide derivatives
10/18/1995EP0677511A2 Intermediates for the preparation of 1-(phenyl)-1-hydroxy-2-amino-3-fluoro propane derivatives
10/18/1995EP0676961A1 Use of macrolides for the treatment of cerebral ischemia
10/17/1995US5459152 Platelet activating factor antagonists
10/17/1995US5459141 Compounds 31668P and 31668U, a process for their production and their use
10/17/1995CA2082809C Pure crystalline form of rifapentine
10/17/1995CA1337351C Spiro-isoquinoline-pyrrolidine tetrones and analogs thereof useful as aldose reductase inhibitors
10/12/1995WO1995026966A1 Cephalosporin antibiotics
10/12/1995CA2186894A1 Cephalosporin antibiotics
10/11/1995EP0676401A1 Annelated spirofluorene-2H-benzopyrans and their use in ophthalmic optics
10/11/1995EP0575425B1 USE OF OXAZOLO- 2,3-a]ISOINDOLE AND IMIDAZO 2,1-a]ISOINDOLE DERIVATIVES AS ANTIVIRAL DRUGS, AND NEW OXAZOLO 2,3-a]ISOINDOLE DERIVATIVES
10/11/1995CN1109877A One-pot process for the preparation of 3-quinolone carboxylic acid derivatives
10/11/1995CN1109748A Rapamycin formulation for IV injection
10/10/1995US5457194 Substituted aliphatic amine-containing macrocyclic immunomodulators
10/10/1995US5457185 Rare earth cryptates, processes for their preparation, synthesis intermediates and application as fluorescent tracers
10/10/1995US5457184 Rare earth macrocyclic complexes and use thereof for reduction of disturbances in an assay using fluorescence
10/10/1995US5457111 Macrocyclic immunomodulators
10/10/1995US5457104 Quinolone- and naphthyridonecarboxylic acid derivatives
10/04/1995EP0675126A1 Amyloid beta-protein agglutination and/or deposition inhibitor
10/04/1995EP0674644A1 Herbicidal imidazolones and a process for their manufacture
10/04/1995CN1109471A Derivative of imidazol-4yl-piperidine, preparation of same and application of same in treatment
10/03/1995US5455249 Phosphorylcarbamates of rapamycin and oxime derivatives thereof
10/03/1995US5455241 Staurosporin derivatives as enzyme inhibitors for protein kinase C and platelet-derived growth factor kinase; antitumor agents, bactericides, antigrowth agents
10/03/1995CA1337200C .beta.-carbolines, their bio-isosteric benzofuran and benzothiophene analogues having cytostatic properties
09/1995
09/27/1995EP0673374A1 Pharmaceutical composition containing bicyclic type compounds
09/27/1995CN1109058A New extractive process for the recovery of naturally occurring macrolides
09/27/1995CN1108931A Rapamycin formulations for oral administration
09/26/1995US5453422 Animal growth promoters
09/21/1995WO1995025106A1 Oxazolidinone derivatives and pharmaceutical compositions containing them
09/20/1995EP0672670A1 Process for the preparation of clavulanic acid
09/20/1995EP0672669A1 Process for the preparation of clavulanic acid
09/20/1995EP0672668A1 Indolocarbazole derivatives and their use in the treatment of thrombocytopenia
09/20/1995EP0672666A2 Imidazodiazepins
09/20/1995EP0672043A1 Novel 4-(3-benzofuranyl)piperidinyl and 4-(3-benzothienyl)piperidinyl derivatives and pharmaceutical compositions containing them
09/20/1995EP0672034A1 Benzimidazole compounds which inhibit platelet aggregation
09/20/1995EP0672031A1 Catechol diethers as selective pde iv? inhibitors
09/19/1995US5451594 Nematocides, insecticides, miticides and fungicides
09/19/1995US5451585 GABA=gamma-aminobutyric acid
09/19/1995US5451343 Fluorone and pyronin y derivatives
09/19/1995CA2144941A1 Indolocarbazole derivatives
09/14/1995WO1995024408A1 Benzothiophene, benzofuran and indolethiazepinones, oxazepinones and diazepinones as inhibitors of cell adhesion and as inhibitors of hiv
09/14/1995WO1995024395A1 Quinoline derivatives as immunomodulators
09/14/1995CA2214521A1 Quinoline derivatives as immunomodulators
09/14/1995CA2181354A1 Benzothiophene, benzofuran and indole-thiazepinones, oxazepinones and diazepinones as inhibitors of cell adhesion and as inhibitors of hiv
09/13/1995EP0671401A1 Beta lactames
09/13/1995EP0671172A1 Amino acid derivative
09/12/1995CA2143519A1 Beta-lactams
09/12/1995CA1336976C Benzoxazepinone process
09/08/1995WO1995023870A1 Novel process for the isolation of clavulanic acid and of pharmaceutically acceptable salts thereof from the fermentation broth of streptomyces sp. p 6621 ferm p 2804
09/08/1995CA2184619A1 Novel process for the isolation of clavulanic acid and of pharmaceutically acceptable salts thereof from the fermentation broth of streptomyces sp. p 6621 ferm p 2804
09/06/1995EP0670321A1 Oxazopyrroloquinoline deivatives and use thereof
09/06/1995EP0669978A1 Flk-1 is a receptor for vascular endothelial growth factor
09/06/1995EP0669936A1 Novel mercaptoacetylamide bicyclic lactam derivatives useful as inhibitors of enkephalinase and ace
09/06/1995CN1108029A Diamine salts of clavulanic acid
09/05/1995CA1336905C Pyrido [3,2,1,ij]-1,3,4-benzoxadiazine derivatives
08/1995
08/31/1995WO1995022972A1 Rapamycin derivatives
08/30/1995EP0669339A1 Asymmetric epoxidation process using optically active manganese complexes
08/30/1995EP0669127A1 Prolonged-action pharmaceutical preparation