Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
06/1996
06/25/1996US5529649 Containing 4,10-dinitro-2,6,8,12-tetraoxa-4,10-diazatetracyclo(5.5.0.0(5 ,9)0(3,11))-dodecane
06/20/1996DE4444244A1 Spiro:indoline cpd. useful for photochromic methacrylic] polymers
06/19/1996EP0717045A1 Process for producing indolocarbazole derivative
06/19/1996EP0716857A1 Use of rapamycin for treating anemia
06/19/1996CN1124925A Lotion
06/18/1996US5527907 Macrolide immunomodulators
06/18/1996CA2084840C Process for preparation of streptovaricin by fermentation
06/14/1996CA2164921A1 Method of treating anemia
06/13/1996WO1996017845A1 Rapamycin 42-oximes and hydroxylamines
06/13/1996CA2206965A1 Rapamycin 42-oximes and hydroxylamines
06/12/1996EP0594715B1 Preparation of diaminic compounds and intermediates
06/12/1996CN1124489A Tetracyclic compounds as dopamine agonists
06/12/1996CN1124247A Preparation of polyalkyl-1-*-bi-nitrogen-hetero-helidecane compound
06/11/1996US5525722 Process for producing biocozamycin benzoate
06/11/1996US5525610 Immunosuppressants, antiarthritic agents
06/06/1996WO1996016967A1 Hindered n-oxide esters of rapamycin and their use as medicaments
06/06/1996WO1996016957A1 3,4-dihydro-2,5,7,8-tetramethyl-benzopyran-6-ol derivatives for use as drugs
06/06/1996CA2205577A1 Hindered n-oxide esters of rapamycin and their use as medicaments
06/05/1996EP0714299A1 Benzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonists
06/05/1996EP0714295A1 Fibrinogen receptor antagonists
05/1996
05/30/1996WO1996016057A1 Certain 1-substituted aminomethyl imidazole and pyrrole derivatives; novel dopamine receptor subtype specific ligands
05/29/1996EP0713491A1 Spiro(indolino) oxazine photochromic compounds
05/29/1996CN1123545A Guanidine derivatives as inhibitors of Na+/H+ exchange in cells
05/28/1996US5521310 Process to obtain benzoxazines to be used for the synthesis of ofloxazine, levofloxazine and derivatives
05/28/1996US5521194 Antiproliferative agent for restenosis treatment
05/28/1996US5521182 1,2,3,4 tetrahydropteridinone cyclic amide derivatives
05/28/1996US5521181 Bicyclic substituted hexahydrobenz[e]isoindole α-1 adrenergic antagonists
05/23/1996WO1996015131A1 Macrocyclic lactone compounds and their production process
05/23/1996WO1996015121A1 Use of dioxomorpholines to combat endoparasites, novel dioxomorpholines and process for their production
05/23/1996WO1996015096A1 Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitiors
05/22/1996EP0712406A1 Condensed indole derivatives as 5-ht 4-receptor antagonists
05/22/1996EP0712402A1 Hydroisoquinoline derivatives
05/21/1996US5519131 Synthesis of pyridooxazinyl-indoles
05/21/1996US5519031 Carbamates of rapamycin
05/21/1996US5519016 Aryl group- or aromatic heterocyclic group-substituted aminoquinolone derivatives and anti-HIV agent
05/21/1996US5518588 Method for preparing 3-aminopyridines from 3-nitropyridines
05/17/1996WO1996014326A1 Antifungal sordaridin derivatives
05/17/1996WO1996014321A1 Substituted tetracyclic oxazepine and thiazepine derivatives with 5-ht2 receptor affinity
05/17/1996WO1996014320A1 Substituted tetracyclic azepine derivatives which have affinity for 5-ht2 receptors
05/17/1996CA2203664A1 Substituted tetracyclic oxazepine and thiazepine derivatives with 5-ht2 receptor affinity
05/17/1996CA2203661A1 Substituted tetracyclic azepine derivatives which have affinity for 5-ht2 receptors
05/17/1996CA2179403A1 Antifungal sordaridin derivatives
05/15/1996EP0711765A1 Immunosuppressive cyclolignan derivatives
05/15/1996EP0711557A1 Base for formulating pharmaceutical agents
05/15/1996EP0711556A1 Intravenous solutions containing staurosporine derivatives
05/15/1996EP0711298A1 Activated macrolactams having immunomodulatory activities
05/15/1996EP0711297A1 Rapamycin derivative with antimicrobial, anticancer and immunomodulation activity
05/15/1996EP0711296A1 IMIDAZOLYLALKYL DERIVATIVES OF IMIDAZOL(5,1-c)(1,4)BENZOXAZIN-1-ONE AND THEIR USE AS THERAPEUTIC AGENTS
05/15/1996EP0711292A1 Aza spiro compounds acting on the cholinergic system with muscarinic agonist activity
05/15/1996DE4440193A1 Verwendung von Dioxomorpholinen zur Bekämpfung von Endoparasiten, neue Dioxomorpholine und Verfahren zur ihrer Herstellung Use of Dioxomorpholinen for controlling endoparasites, new Dioxomorpholine and methods for their preparation
05/15/1996CA2162760A1 Immunosuppressive cyclolignan derivatives
05/14/1996US5516781 Method of treating restenosis with rapamycin
05/14/1996US5516780 Immunosuppressive, antiinflammatory, antifungal and antitumor agents
05/14/1996US5516772 K-252 derivatives which enhance neurotrophin-induced activity
05/14/1996US5516771 Use of indolocarbazole derivatives to treat a pathological condition of the prostate
05/14/1996US5516566 Cyclic oligomers for production of linear polyketones, polyphthalazines and polyisoquinolines
05/10/1996CA2162342A1 Intravenous solutions for a derivative of staurosporine
05/10/1996CA2162341A1 Pharmaceutical carriers
05/09/1996WO1996013506A1 Protein kinase inhibitors for treatment of neurological disorders
05/09/1996WO1996013505A1 PROCESSES AND INTERMEDIATES FOR PREPARING 5,7-DIHYDRO-3-[2-{1-BENZYLPIPERIDIN-4-YL}ETHYL]-6H-PYRROLO-[4,5-f]-1,2-BENZISOXAZOL-6-ONE
05/09/1996CA2203767A1 Protein kinase inhibitors for treatment of neurological disorders
05/08/1996EP0710231A1 Preparation of benzoxazine compounds in solventless systems
05/08/1996EP0710110A1 Rapamycin conjugates and antibodies
05/07/1996US5514813 Preparation of macrocyclic polyetherimide oligomers from substituted bisphthalimides
05/07/1996US5514686 Use of macrolide compounds for eye diseases
05/07/1996US5514685 Antiinflammatory antoproliferative agents, immunosuppressants
05/02/1996WO1996012722A1 5-ht4 receptor agonist
05/01/1996EP0709386A1 Fused benzazepine derivative and pharmaceutical composition containing the same
05/01/1996EP0691931A4 Embossed card package production system with modular inserters for multiple forms and card verification apparatus
05/01/1996CN1121710A Heterocyclic compounds, their use and preparation
04/1996
04/30/1996US5512579 Aminobenzoic acid derivatives
04/30/1996US5512566 Useful in treating diseases of central nervous system
04/30/1996US5512564 Tricyclic thiazole and oxazole derivatives and pharmaceutical agents containing them
04/30/1996US5512563 Tricyclic benzazepine vasopressin antagonists
04/30/1996US5512562 Tricyclic 2,3,4,5-tetrahydro-1H-3-benzapines
04/25/1996WO1996011926A1 Photochromic naphthoxazine compounds
04/24/1996EP0708105A1 5-HT4 receptor agonists
04/24/1996EP0708092A1 Process for the preparation of 3-aminopyridines from 3-nitropyridines
04/24/1996EP0707579A1 Piperidinyl substituted methanoanthracenes as d1/d2-antagonists and 5ht2-serotanin-antagonists
04/24/1996EP0689545A4 Macrocyclic amide and urea immunomodulators
04/24/1996EP0602097B1 Tricyclic thiazol and oxazol derivates with antiviral action
04/24/1996EP0450097B1 Benzoheterocyclic compounds
04/23/1996US5510374 3-aminochroman compounds
04/23/1996US5510319 Pyrrolo-2,3-b-pyridinyl derivatives
04/21/1996CA2160420A1 5-ht4 receptor agonists
04/17/1996CN1120541A New tetracyclic piperidine and 1,4-oxazine compounds, a process for their preparation and pharmaceutical compositions containing them
04/16/1996US5508428 Spiro compound
04/16/1996US5508399 Carbamates of rapamycin
04/16/1996US5508398 New extractive process for the recovery of naturally occurring macrolides
04/16/1996US5508397 Ascomycin immunosuppressant
04/16/1996US5508290 Hindered N-oxide esters of rapamycin
04/16/1996US5508286 Rapamycin amidino carbamates
04/16/1996US5508285 Hindered N-oxide esters of rapamycin
04/16/1996US5508278 Bactericides
04/16/1996US5508272 Compounds containing a fused bicycle ring and processes therefor
04/10/1996EP0705836A1 Polyalkylpiperidine compounds
04/10/1996EP0705835A1 Quinoxalic-2,3-diones with an oxa or thiaheterocyclic fused ring
04/10/1996EP0705828A1 Quinolone- and naphthyridone carboxylic acid derivatives as antibacterial agents
04/10/1996EP0705825A2 Diaminic compounds, preparation, use and intermediates
04/10/1996EP0705250A1 Bis-imide polycyclic and heterocyclic chromophores useful as tumoricidals