Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
06/1993
06/10/1993WO1993011131A1 Cephalosporin compounds
06/10/1993WO1993011130A1 Rapamycin derivative and its medicinal use
06/08/1993US5217980 Oxazolyl and piperidinyl substituted benimidazolyl compounds
06/08/1993US5217972 Quinolonecarboxylic acid derivatives and their use as antiviral agents
06/08/1993US5217969 Antiinflammatory, antiulcer agent
06/08/1993US5217968 N-alkylbenzo(b)thieno [3,2-b]oxazin-2,4-diones
06/02/1993EP0544445A2 Furyl-substituted purines, oxazolopyrimidines and pteridines as adenosine antagonists
06/02/1993EP0543930A1 Arthropodicidal pyrazolines, pyrazolidines and hydrazines
06/02/1993EP0543879A1 Macrocyclic compounds
06/02/1993CN1072683A 水溶性喜树碱衍生物 Water-soluble derivative of camptothecin
06/01/1993US5215984 Antihypertensive spiro(piperidine- pyrrolidine- or hexahydroazepinyl substituted) pyrrolo(2,1-c)(1,4)benzoxazepines)
05/1993
05/27/1993WO1993010122A1 Rapamycin pyrazoles
05/27/1993WO1993010100A1 New substituted pyrazolylpyrazoles, processes for their preparation, as well as intermediates, and their use as herbicides
05/26/1993CN1020853C Tricyclic compounds, their preparation and pharmaceutical composition containing them
05/26/1993CA2082333A1 Heterocyclic compounds
05/25/1993US5214038 1-(pyrido[3,4-b]-1,4-oxazinyl-4-yl)-1H-indoles and intermediates for the preparation thereof
05/19/1993EP0542609A1 3-sulfonylamino-2-(1H)-quinolinones and 7-aza derivatives as excitatory amino acids antagonists
05/19/1993EP0542388A1 New substituted pyrazolylpyrazoles, processes for their preparation, as well as intermediates, and their use as herbicides
05/19/1993EP0541807A1 Novel benzopyran derivative
05/18/1993US5212305 Cyclization and forming a carbon-nitrogen bond
05/18/1993US5212186 Cardioactive pyrrolobenzimidazoles
05/15/1993CA2082856A1 3-sulfonylamino-2-(1h)-quinoleinone derivatives, process for their preparation and pharmaceutical compositions containing them
05/13/1993WO1993008809A1 Compositions containing k-252 compounds for potentiation of neurotrophin activity
05/13/1993CA2123096A1 Compositions containing k-252 compounds for potentiation of neurotrophin activity
05/12/1993EP0540625A1 Novel spiro-isoxazolidine derivatives as cholinergic agents
05/12/1993CN1071917A Quinalozine derivatives as inhibitors of hiv reverse transcriptase
05/12/1993CN1020612C Method for preparing antihypertensive tricyclic lactam derivs.
05/12/1993CN1020610C Process for preparation of substituted benzoxazine rifamycin
05/11/1993US5210227 Derivatives of macrolide FR-900506, which had previously been isolated from Streptomyces microorganisms
05/11/1993US5210082 Treating panic disorder
05/11/1993US5210030 Process for selectively acylating immunomycin
05/11/1993CA1317590C 2-substituted-e-fused-¬1,2,4|triazolo¬1,5- c|pyrimidines, pharmaceutical compositions, and uses thereof
05/05/1993EP0540185A1 4'-(N-substituted-N-oxide)staurosporine derivatives
05/05/1993EP0540099A1 Water soluble camptothecin derivatives
05/05/1993EP0539451A1 Vinylsulphonyl pristinamycin and preparation thereof.
05/05/1993EP0539421A1 Novel oxazolyl derivatives
05/04/1993US5208241 N-heteroaryl, n-alkylheteroaryl, n-alkenylheteroaryl and n-alkynylheteroarylmacrolides having immunosuppressive activity
04/1993
04/30/1993CA2081580A1 Water soluble camptothecin derivatives
04/29/1993WO1993008191A1 Azabicyclo oxime and amine cholinergic agents and methods of treatment
04/29/1993WO1993008185A1 N-aryl-n1-azabicyclo-ureas as 5-ht3 antagonists
04/28/1993EP0538691A1 Substituted tetrahydrothiophenes, methods for their preparation, and their use in pharmaceutical compositions
04/28/1993EP0538477A1 Novel cyclic aminophenylacetic acid derivative, production thereof, and immune response modulator containing the same as active ingredient
04/27/1993US5206751 Process for the production of an impact-resistant liquid crystal switching and display device
04/27/1993US5206247 Spiro(4.5.)decane compounds
04/27/1993US5206240 Nitrogen-containing spirocycles
04/27/1993CA1316916C Hydroxide mediated fk-506 rearrangement product
04/23/1993CA2080863A1 Use of substituted tetrahydrothiophenes, some of which are known, as medicaments, new active substances and processes for their preparation
04/21/1993EP0537354A1 Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
04/21/1993EP0537353A1 Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
04/15/1993WO1993007153A1 4'-(n-substituted-n-oxide)staurosporine derivatives
04/15/1993WO1993007143A1 Methylpiperazinoazepine derivatives, their preparation and use
04/15/1993WO1993007129A1 Remedy for osteoporosis and diazepine compound
04/15/1993CA2120939A1 Therapeutic agent for osteoporosis and diazepine compound
04/14/1993EP0536896A1 Imidazolidyl macrolides having immunosuppressive activity
04/14/1993EP0536401A1 Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
04/13/1993US5202440 Cholinesterase inhibitors for treatment of alzheimer*s disease
04/13/1993US5202332 Rapamycin analog as immunosuppressant
04/13/1993US5202328 Substituted fused pyrimidinones
04/13/1993CA1316174C Process for the preparation of chromogenic cryptahemispherands
04/07/1993EP0535521A2 Condensed oxazole and thiazole derivatives as leukotriene biosynthesis inhibitors
04/07/1993EP0535377A2 Optically active benzopyran compound, process for producing it and optically active manganese complex
04/06/1993US5200407 Azole derivatives and anti-ulcerative composition containing same
04/01/1993WO1993006108A1 Pyrrolobenzoxazine derivatives as 5-ht agonists and antagonists
03/1993
03/31/1993EP0534492A2 Carboxyalkyl substituted inhibitors of enkephalinase and ACE
03/31/1993EP0534396A2 2-Substituted indane-2-carboxyalkyl derivatives useful as inhibitors of enkephalinase and ace
03/31/1993EP0534363A2 Novel 2-substituted indane-2-mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
03/31/1993EP0533930A1 Use of a macrolide compound such as fk 506 for manufacturing a medicament for treating idiopathic thrombocytopenic purpura and basedow's disease
03/31/1993EP0533837A1 Inhibition of 5-lipoxygenase and cyclooxygenase pathway mediated diseases
03/30/1993CA1315474C Pristinamycin ii b derivatives, their preparation, and pharmaceutical compositions containing them
03/25/1993CA2078810A1 Leukotriene biosynthesis inhibitors
03/24/1993EP0533433A1 Use of rapamycin for the manufacture of a medicament for the treatment of immunoinflammatory diseases
03/24/1993EP0532862A1 Use of rapamycin for the preparation of a medicament for the treatment of ocular inflammation
03/23/1993US5196425 Antihypertensive 3-piperidinyl-indazole derivatives
03/23/1993CA1314879C Anellated indole derivatives
03/23/1993CA1314878C Pristinamycin process
03/23/1993CA1314876C Azithromycin dihydrate
03/18/1993WO1993005059A1 Imidazolidyl macrolides
03/18/1993WO1993005058A1 O-heteroaryl, o-alkylheteroaryl, o-alkenylheteroaryl and o-alkynylheteroarylmacrolides
03/18/1993WO1993005049A1 Rare earth macrocyclic complexes and use thereof for reduction of disturbances in an assay using fluorescence
03/18/1993WO1993005047A1 New tricyclic thiazol and oxazol derivates with antiviral action
03/18/1993WO1993005046A1 Aminodiesters of rapamycin
03/18/1993WO1993005028A1 Receptor compounds based on 1,7-dioxa-4,10-diazacyclododecane
03/18/1993WO1993004680A1 Macrocyclic immunomodulators
03/18/1993CA2117062A1 New tricyclic thiazole and oxazole derivatives and pharmaceutical agents containing them
03/17/1993EP0532089A1 N-heteroaryl, N-alkylheteroaryl, N-alkenylheteroaryl & N-alkynylheteroarylmacrolides
03/17/1993EP0532088A1 O-Heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroaryl macrolides
03/17/1993EP0531883A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them
03/17/1993CN1020102C Preparation for bicyclic carboxylic ether and bicyclic carboxylic amide
03/16/1993US5194447 Sulfonylcarbamates of rapamycin
03/16/1993US5194378 Immunosuppressants
03/11/1993DE4129779A1 Neue tricyclische thiazol- und oxazol-derivate und diese enthaltende arzneimittel Thiazole and oxazole novel tricyclic derivatives and pharmaceutical compositions containing them
03/10/1993EP0530994A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase
03/10/1993EP0530888A1 Fluoromacrolides having immunosuppressive activity
03/10/1993EP0530198A1 Heterocyclic compounds as aldose reductase inhibitors
03/10/1993CN1069732A 1,7-Condensed 2-(piperazinealkyl)-indole derivatives and process for preparing same and intermediate and pharmaceutical containing same
03/10/1993CA2077638A1 N-heteroaryl, n-alkylheteroaryl, n-alkenylheteroaryl and n- alkynylheteroarylmacrolides having immunosuppressive activity
03/10/1993CA2077331A1 O-heteroaryl, o-alkylheteroaryl, o-alkenylheteroaryl and o-alkynylheteroaryl macrolides having immunosuppressive activity
03/09/1993US5192357 Acrylate fungicides
03/07/1993CA2077577A1 Condensed 5-membered heterocyclic compounds, processes for preparing them and pharmaceutical preparations containing these compounds
03/06/1993WO1993004679A1 Macrocyclic immunomodulators