Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
01/2003
01/22/2003EP1277751A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277749A1 2- and 2,5-substituted phenylketo enols
01/22/2003EP1277738A1 Condensed heteroaryl derivatives
01/22/2003EP1277735A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277734A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1277733A1 2- and 2,5-substituted phenylketo-enols
01/22/2003EP1276741A1 Phenyl substituted 4-hydroxy tetrahydropyridone
01/22/2003EP1276740A2 Novel epothilone derivatives, method for the preparation thereof and their pharmaceutical use
01/22/2003EP0968213B1 Alkynyl-substituted camptothecins and process for their preparation
01/22/2003EP0646115B1 Heterocyclic-cyclic amine derivatives
01/22/2003CN1099420C Substituted spiroheterocyclic 1H-3-arylpyrrolidine-2-4,-dione derivatives, methods of preparing them and their use as pest-control agents
01/21/2003US6509346 Chemokine receptor antagonists and methods of use therefor
01/21/2003US6509345 For therapy of cancerous diseases
01/21/2003US6509344 Indenoisoquinolines as antineoplastic agents
01/21/2003US6509341 The invention relates to carboxylic acid derivatives of formula (I), wherein the substituents have the meaning as commented in the description. It also relates to the production and use of same as endothelin receptor antagonists.
01/21/2003US6509340 Amide and urea derivatives as 5-HT reuptake inhibitors and as 5-HT1B/1D ligands
01/16/2003WO2003004501A2 (hetero) aryl substituted benzofurans as 5-ht ligands
01/16/2003WO2003004495A1 Novel immunomodulating compounds
01/16/2003WO2003004488A1 Indazole benzimidazole compounds as tyrosine and serine/threonine kinase inhibitors
01/16/2003WO2003004467A2 Thiazole benzamide derivatives and pharmaceutical compositions for inhibiting cell proliferation, and methods for their use
01/16/2003WO2003004032A1 Oral administration of 6-hydroxy-oxymorphone for use as an analgesic
01/16/2003WO2003004031A1 Parenteral administration of 6-hydroxy-oxymorphone for use as an analgesic
01/16/2003WO2003004030A1 Oxymorphone controlled release formulations
01/16/2003WO2003004020A1 Heteroaryl carboxylic acid amides, the production thereof and the use of the same as inhibitors of the microsomal triglyceride transfer protein (mtp)
01/16/2003WO2002050062A3 Benzimidazole and pyridylimidazole derivatives as ligands for gaba receptors
01/16/2003WO2002046129A3 Inhibitors of histone deacetylase
01/16/2003US20030013757 Aromatic dicarboxylic acid derivatives
01/16/2003US20030013715 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
01/16/2003US20030013603 Catalyst for oxidation, carbonylation, nitration, sulfonation
01/16/2003US20030013041 Write-once optical data carrier
01/16/2003US20030012831 Liquid-liquid extraction being carried out in the first stage at a pH-value of about 4; treating narrow-angle glaucoma, Alzheimer's disease, as well as alcohol and nicotine dependence.
01/16/2003CA2452874A1 Oral administration of 6-hydroxy-oxymorphone for use as an analgesic
01/16/2003CA2452872A1 Parenteral administration of 6-hydroxy-oxymorphone for use as an analgesic
01/16/2003CA2452609A1 Thiazole benzamide derivatives and pharmaceutical compositions for inhibiting cell proliferation, and methods for their use
01/16/2003CA2451749A1 Novel immunomodulating compounds
01/16/2003CA2451606A1 (hetero) aryl substituted benzofurans as 5-ht ligands
01/15/2003EP1274713A1 Anti-viral pyrimidine nucleoside analogues
01/15/2003EP1274431A1 10,11-difluoromethylenedioxycamptothecin compounds with topoisomerase i inhibition
01/15/2003CN1391473A VLA-4 inhibitor compounds
01/15/2003CN1390834A Indenoindolone compounds, their preparation and medicinal compositions containing them
01/14/2003US6506876 LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use
01/14/2003US6506773 Hydroxamic and carboxylic acid derivatives
01/14/2003US6506769 Heterocyclic compounds useful as inhibitors of tyrosine kinases
01/14/2003US6506766 Glucocortiocoid-selective antinflammatory agents
01/14/2003US6506507 Methine compound, material for organic luminescence element, and organic luminescence element using the same
01/14/2003CA2217477C Tricyclic compounds useful for inhibition of farnesyl protein transferase
01/09/2003WO2003002715A2 Compositions and methods for labeling oligonucleotides
01/09/2003WO2003002561A1 N-aroyl cyclic amine derivatives as orexin receptor antagonists
01/09/2003WO2003002548A1 A process for the preparation of chiral glucocorticoid receptor agents
01/09/2003WO2002080152A3 Optical data carrier that contains a heterocyclic azo dye as the light-absorbing compound in the information layer
01/09/2003WO2002059111A3 Pyrazole compounds useful as protein kinase inhibitors
01/09/2003US20030009031 Useful for the inhibition of polymerization
01/09/2003US20030008910 Use of proteasome inhibitors to treat dry eye disorders
01/09/2003US20030008898 Indole derivatives and their use for the treatment of malignant and other diseases based on pathological proliferation
01/09/2003US20030008848 Small molecules useful in the treatment of inflammatory disease
01/09/2003US20030008234 Optical data carrier comprising a cyanine dye as light-absorbent compound in the information layer
01/09/2003US20030007941 Method of treating hair loss using thyromimetic compounds
01/09/2003US20030006516 Radiation transparent subsrates; reflecting layer
01/09/2003CA2451464A1 N-aroyl cyclic amine derivatives as orexin receptor antagonists
01/08/2003EP1273584A1 2- or 4-Chromenyliden based merocyanines and use thereof
01/08/2003EP1272491A1 Perylene-derivative based crystallization modifiers
01/08/2003EP1272484A2 Benzoamide piperidine compounds as substance p antagonists
01/08/2003EP1272480A1 Method for the production of spirocyclic tetronic acid derivatives
01/08/2003EP1272192A2 A use of galantamine for the treatment of neuropsychiatric behaviour associated with alzheimer's disease
01/08/2003EP1272168A2 Small organic molecule regulators of cell proliferation
01/08/2003EP1095011A4 Novel fluorescent lanthanide chelates
01/08/2003EP1053239B1 Glucocorticoid-selective anti-inflammatory agents
01/08/2003EP0863878B1 Cyclic nitrones and pharmaceutical compositions containing them
01/08/2003CN1390221A Spiro (2H-1-benzopyran-2,4'-piperididine) derivates as glycine transport inhibitors
01/08/2003CN1389203A Method for treating hair-dropping using thyromimetic compound
01/08/2003CN1098266C Fused pyrrolo (2,3-c) carbazole-6-one which potentiate activity of gamma interferon
01/07/2003US6504036 2- and 2.5-substituted phenylketoenols
01/07/2003US6504029 Condensed-hexacyclic compounds and a process therefor
01/07/2003US6503926 Nitrogen heterocycle compounds
01/07/2003US6503919 Compounds of 7-oxo-2,3,7,14-tetrahydro-1H-benzo[b]pyrano[3,2-h]acridin carboxylate
01/07/2003US6503899 Azepino[4,5-b]pyrano[3,2-e]indoles
01/03/2003WO2003000697A1 Furoisoquinoline derivative, process for producing the same, and use
01/03/2003WO2003000691A1 Carboline derivatives as pdev inhibitors
01/03/2003WO2003000677A1 Spiropiperidine compounds as ligands for orl-1 receptor
01/03/2003WO2003000676A1 1,2,4-trioxolane antimalarials
01/03/2003WO2003000265A1 Crystalline anticholinergic, method for its production, and use thereof in the production of a drug
01/03/2003WO2003000240A2 Stable powder inhalation dosage formulation
01/03/2003WO2002046170A8 Anilinopyrimidine derivatives as jnk pathway inhibitors and compositions and methods related thereto
01/03/2003WO2001083800A8 Heterologous production of polyketides
01/03/2003CA2450550A1 Spiropiperidine compounds as ligands for orl-1 receptor
01/02/2003US20030004355 Regulating intracellular levels of cyclic guanosine-3*,5*-monophosphate by activiating soluble guanylate cyclase or inhibiting phosphodiesterases
01/02/2003US20030004351 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
01/02/2003US20030004344 Thrombin or factor Xa inhibitors
01/02/2003US20030004338 Antitumor, anticancer agents
01/02/2003US20030004208 Squalene synthetase inhibitors; antilipemic agents, anticholesterol agents
01/02/2003US20030004183 Quinoline-4-carboxamide derivatives as NK-2 and NK-3 receptor antagonists
01/02/2003US20030004172 Cardiovascular disorders, osteoporosis, multiple sclerosis, antiarthritic agents
01/02/2003US20030004166 Novel triazine compounds useful as sorbitol dehydrogenase inhibitors
01/02/2003US20030004164 Anticancer agents; autoimmune diseases
01/02/2003US20030004162 Antidiabetic agents; dietetics
01/02/2003US20030004161 Anticancer agents; autoimmune diseases
01/02/2003US20030004150 New analogues of camptothecin, their use as medicaments and the pharmaceutical compositions containing them
01/02/2003US20030003396 Reflection, protective or covering layers which can be written on or read by blue, red or infrared light
01/02/2003EP1270579A1 Process for producing camptothecin
01/02/2003EP1270578A1 Novel process for producing fused imidazopyridine derivative and novel crystal form